Title: Peripheral antinociceptive effect of anandamide and drugs that affect the endocannabinoid system on the formalin test in normal and streptozotocin-diabetic rats.
Journal: Neuropharmacology 20121201
Title: Inhibition of fatty acid amide hydrolase by URB597 attenuates the anxiolytic-like effect of acetaminophen in the mouse elevated plus-maze test.
Journal: Behavioural pharmacology 20120801
Title: Effects of alterations in cannabinoid signaling, alone and in combination with morphine, on pain-elicited and pain-suppressed behavior in mice.
Journal: The Journal of pharmacology and experimental therapeutics 20120701
Title: The anandamide transport inhibitor AM404 reduces the rewarding effects of nicotine and nicotine-induced dopamine elevations in the nucleus accumbens shell in rats.
Journal: British journal of pharmacology 20120401
Title: Medial prefrontal cortex endocannabinoid system modulates baroreflex activity through CB(1) receptors.
Journal: American journal of physiology. Regulatory, integrative and comparative physiology 20120401
Title: Endocannabinoid analogues exacerbate marble-burying behavior in mice via TRPV1 receptor.
Journal: Neuropharmacology 20120401
Title: Effects of the anandamide uptake blocker AM404 on food intake depend on feeding status and route of administration.
Journal: Pharmacology, biochemistry, and behavior 20120301
Title: A catalytically silent FAAH-1 variant drives anandamide transport in neurons.
Journal: Nature neuroscience 20120101
Title: Novel bioactive metabolites of dipyrone (metamizol).
Journal: Bioorganic & medicinal chemistry 20120101
Title: Involvement of the endocannabinoid system in ethanol-induced corticostriatal synaptic depression.
Journal: Journal of pharmacological sciences 20120101
Title: Hippocampal endocannabinoids play an important role in induction of long-term potentiation and regulation of contextual fear memory formation.
Journal: Brain research bulletin 20111010
Title: Involvement of endocannabinoids in antidepressant and anti-compulsive effect of fluoxetine in mice.
Journal: Behavioural brain research 20110930
Title: Paracetamol-induced hypothermia is independent of cannabinoids and transient receptor potential vanilloid-1 and is not mediated by AM404.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20110901
Title: Endogenously generated 2-arachidonoylglycerol plays an inhibitory role in bombesin-induced activation of central adrenomedullary outflow in rats.
Journal: European journal of pharmacology 20110511
Title: Cannabinoid receptor activation modifies NMDA receptor mediated release of intracellular calcium: implications for endocannabinoid control of hippocampal neural plasticity.
Journal: Neuropharmacology 20110501
Title: Cannabinoid transmission in the basolateral amygdala modulates fear memory formation via functional inputs to the prelimbic cortex.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience 20110406
Title: Interactions between endocannabinoid and serotonergic systems in mood disorders caused by nicotine withdrawal.
Journal: Nicotine & tobacco research : official journal of the Society for Research on Nicotine and Tobacco 20110401
Title: Facilitation of CB1 receptor-mediated neurotransmission decreases marble burying behavior in mice.
Journal: Progress in neuro-psychopharmacology & biological psychiatry 20110330
Title: Pharmacological elevation of anandamide impairs short-term memory by altering the neurophysiology in the hippocampus.
Journal: Neuropharmacology 20110101
Title: Inhibition of monoacylglycerol lipase by troglitazone, N-arachidonoyl dopamine and the irreversible inhibitor JZL184: comparison of two different assays.
Journal: British journal of pharmacology 20101201
Title: Cannabinoid CB1 receptors in the medial prefrontal cortex modulate the expression of contextual fear conditioning.
Journal: The international journal of neuropsychopharmacology 20101001
Title: Regulation of subthalamic neuron activity by endocannabinoids.
Journal: Synapse (New York, N.Y.) 20100901
Title: Possible inhibitory roles of endogenous 2-arachidonoylglycerol during corticotropin-releasing factor-induced activation of central sympatho-adrenomedullary outflow in anesthetized rats.
Journal: European journal of pharmacology 20100901
Title: The effects of anandamide transport inhibitor AM404 on voltage-dependent calcium channels.
Journal: European journal of pharmacology 20100525
Title: Reduction in endocannabinoid tone is a homeostatic mechanism for specific inhibitory synapses.
Journal: Nature neuroscience 20100501
Title: Olvanil: a non-pungent TRPV1 activator has anti-emetic properties in the ferret.
Journal: Neuropharmacology 20100201
Title: Quantitative analyses of aggregation, autofluorescence, and reactivity artifacts in a screen for inhibitors of a thiol protease.
Journal: Journal of medicinal chemistry 20100114
Title: Cannabinoids and their interactions with diazepam on modulation of serum corticosterone concentration in male mice.
Journal: Neurochemical research 20100101
Title: Characterization of an AM404 analogue, N-(3-hydroxyphenyl)arachidonoylamide, as a substrate and inactivator of prostaglandin endoperoxide synthase.
Journal: Biochemistry 20091229
Title: Effects of the endocannabinoid transport inhibitors AM404 and UCM707 on diabetic neuropathy in rats.
Journal: Clinical and experimental pharmacology & physiology 20091101
Title: The endocannabinoid transport inhibitor AM404 modulates nociception in cholestasis.
Journal: Neuroscience letters 20091025
Title: Differential endocannabinoid regulation of baroreflex-evoked sympathoinhibition in normotensive versus hypertensive rats.
Journal: Autonomic neuroscience : basic & clinical 20091005
Title: Chronic ethanol treatment potentiates ethanol-induced increases in interstitial nucleus accumbens endocannabinoid levels in rats.
Journal: Journal of neurochemistry 20091001
Title: Role of anandamide transporter in regulating calcitonin gene-related peptide production and blood pressure in hypertension.
Journal: Journal of hypertension 20090601
Title: Divergent effects of anandamide transporter inhibitors with different target selectivity on social play behavior in adolescent rats.
Journal: The Journal of pharmacology and experimental therapeutics 20090101
Title: New analgesics synthetically derived from the paracetamol metabolite N-(4-hydroxyphenyl)-(5Z,8Z,11Z,14Z)-icosatetra-5,8,11,14-enamide.
Journal: Journal of medicinal chemistry 20081225
Title: Facilitation of contextual fear memory extinction and anti-anxiogenic effects of AM404 and cannabidiol in conditioned rats.
Journal: European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology 20081201
Title: Enhancement of endocannabinoid neurotransmission through CB1 cannabinoid receptors counteracts the reinforcing and psychostimulant effects of cocaine.
Journal: The international journal of neuropsychopharmacology 20081101
Title: Evaluation of interactions between cannabinoid compounds and diazepam in electroshock-induced seizure model in mice.
Journal: Journal of neural transmission (Vienna, Austria : 1996) 20081101
Title: Augmentation of endogenous cannabinoid tone modulates lipopolysaccharide-induced alterations in circulating cytokine levels in rats.
Journal: Immunology 20081001
Title: Pro-drugs for indirect cannabinoids as therapeutic agents.
Journal: Current drug delivery 20081001
Title: Activation of cannabinoid CB1 receptors in the dorsolateral periaqueductal gray induces anxiolytic effects in rats submitted to the Vogel conflict test.
Journal: European journal of pharmacology 20080928
Title: Endocannabinoid- and mGluR5-dependent short-term synaptic depression in an isolated neuron/bouton preparation from the hippocampal CA1 region.
Journal: Journal of neurophysiology 20080801
Title: Endocannabinoid modulation of male rat sexual behavior.
Journal: Psychopharmacology 20080701
Title: RNA interference-mediated knockdown of dynamin 2 reduces endocannabinoid uptake into neuronal dCAD cells.
Journal: Molecular pharmacology 20080701
Title: Short- and long-term effects of cannabinoids on the extinction of contextual fear memory in rats.
Journal: Neurobiology of learning and memory 20080701
Title: TRPV2 is activated by cannabidiol and mediates CGRP release in cultured rat dorsal root ganglion neurons.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience 20080611
Title: Mechanisms of AM404-induced [Ca(2+)](i) rise and death in human osteosarcoma cells.
Journal: Toxicology letters 20080610
Title: Expression and function of CB1 receptor in the rat striatum: localization and effects on D1 and D2 dopamine receptor-mediated motor behaviors.
Journal: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20080601
Title: Activation of CB1 cannabinoid receptors in the dorsolateral periaqueductal gray reduces the expression of contextual fear conditioning in rats.
Journal: Psychopharmacology 20080601
Title: Activation of endocannabinoid transmission induces antidepressant-like effects in rats.
Journal: Journal of physiology and pharmacology : an official journal of the Polish Physiological Society 20080601
Title: Differential involvement of opioidergic and serotonergic systems in the antinociceptive activity of N-arachidonoyl-phenolamine (AM404) in the rat: comparison with paracetamol.
Journal: Naunyn-Schmiedeberg's archives of pharmacology 20080501
Title: AM404, an anandamide transport inhibitor, reduces plasma extravasation in a model of neuropathic pain in rat: role for cannabinoid receptors.
Journal: Neuropharmacology 20080301
Title: Interaction between cannabinoid compounds and diazepam on anxiety-like behaviour of mice.
Journal: Pharmacology, biochemistry, and behavior 20080301
Title: Differential stimulatory effects of cannabinoids on VIP release and NO synthase activity in synaptosomal fractions from rat ileum.
Journal: Neuropeptides 20080101
Title: Delta9-tetrahydrocannabinol (THC) and AM 404 protect against cerebral ischaemia in gerbils through a mechanism involving cannabinoid and opioid receptors.
Journal: British journal of pharmacology 20071201
Title: The local antinociceptive effects of paracetamol in neuropathic pain are mediated by cannabinoid receptors.
Journal: European journal of pharmacology 20071114
Title: Characterization of the vasorelaxant mechanisms of the endocannabinoid anandamide in rat aorta.
Journal: British journal of pharmacology 20071101
Title: Actions of the endocannabinoid transport inhibitor AM404 in neuropathic and inflammatory pain models.
Journal: Clinical and experimental pharmacology & physiology 20071101
Title: Studies of anandamide accumulation inhibitors in cerebellar granule neurons: comparison to inhibition of fatty acid amide hydrolase.
Journal: Journal of molecular neuroscience : MN 20070901
Title: The anandamide transport inhibitor AM404 reduces ethanol self-administration.
Journal: The European journal of neuroscience 20070701
Title: AM404 decreases Fos-immunoreactivity in the spinal cord in a model of inflammatory pain.
Journal: Brain research 20070604
Title: The acetaminophen-derived bioactive N-acylphenolamine AM404 inhibits NFAT by targeting nuclear regulatory events.
Journal: Biochemical pharmacology 20070401
Title: The endogenous cannabinoid anandamide produces delta-9-tetrahydrocannabinol-like discriminative and neurochemical effects that are enhanced by inhibition of fatty acid amide hydrolase but not by inhibition of anandamide transport.
Journal: The Journal of pharmacology and experimental therapeutics 20070401
Title: Anxiolytic-like effect of cannabinoids injected into the rat dorsolateral periaqueductal gray.
Journal: Neuropharmacology 20070301
Title: Evaluation of the neuroprotective effect of cannabinoids in a rat model of Parkinson's disease: importance of antioxidant and cannabinoid receptor-independent properties.
Journal: Brain research 20070223
Title: 5-HT1A receptors are involved in the anxiolytic effect of Delta9-tetrahydrocannabinol and AM 404, the anandamide transport inhibitor, in Sprague-Dawley rats.
Journal: European journal of pharmacology 20070126
Title: Cannabinoid (CB1) receptor activation inhibits trigeminovascular neurons.
Journal: The Journal of pharmacology and experimental therapeutics 20070101
Title: Anxiolytic-like properties of the anandamide transport inhibitor AM404.
Journal: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20061201
Title: Acyl-based anandamide uptake inhibitors cause rapid toxicity to C6 glioma cells at pharmacologically relevant concentrations.
Journal: Journal of neurochemistry 20061001
Title: Neuropathic pain and the endocannabinoid system in the dorsal raphe: pharmacological treatment and interactions with the serotonergic system.
Journal: The European journal of neuroscience 20061001
Title: Endocannabinoids modulate stress-induced suppression of hippocampal cell proliferation and activation of defensive behaviours.
Journal: The European journal of neuroscience 20061001
Title: Differential effect of cannabinoid agonists and endocannabinoids on histamine release from distinct regions of the rat brain.
Journal: The European journal of neuroscience 20060901
Title: AM404, an inhibitor of anandamide uptake, prevents pain behaviour and modulates cytokine and apoptotic pathways in a rat model of neuropathic pain.
Journal: British journal of pharmacology 20060801
Title: Endocannabinoid system in frog and rodent testis: type-1 cannabinoid receptor and fatty acid amide hydrolase activity in male germ cells.
Journal: Biology of reproduction 20060701
Title: Modulation of neuropathic and inflammatory pain by the endocannabinoid transport inhibitor AM404 [N-(4-hydroxyphenyl)-eicosa-5,8,11,14-tetraenamide].
Journal: The Journal of pharmacology and experimental therapeutics 20060601
Title: Cannabinoid modulation of electrically evoked pH and oxygen transients in the nucleus accumbens of awake rats.
Journal: Journal of neurochemistry 20060501
Title: Effects of intra-amygdala infusion of CB1 receptor agonists on the reconsolidation of fear-potentiated startle.
Journal: Learning & memory (Cold Spring Harbor, N.Y.) 20060501
Title: Role of TRPV1 and cannabinoid CB1 receptors in AM 404-evoked hypothermia in rats.
Journal: Pharmacology, biochemistry, and behavior 20060401
Title: Endocannabinoids activate transient receptor potential vanilloid 1 receptors to reduce hyperdopaminergia-related hyperactivity: therapeutic implications.
Journal: Biological psychiatry 20060315
Title: New metabolically stable fatty acid amide ligands of cannabinoid receptors: Synthesis and receptor affinity studies.
Journal: Bioorganic & medicinal chemistry letters 20060101
Title: Effects of cannabinoids on the anxiety-like response in mice.
Journal: Pharmacological reports : PR 20060101
Title: Activity-dependent release and actions of endocannabinoids in the rat hypothalamic supraoptic nucleus.
Journal: The Journal of physiology 20051215
Title: Pharmacological enhancement of cannabinoid CB1 receptor activity elicits an antidepressant-like response in the rat forced swim test.
Journal: European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology 20051201
Title: Cannabinoid agonists but not inhibitors of endogenous cannabinoid transport or metabolism enhance the reinforcing efficacy of heroin in rats.
Journal: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20051101
Title: Decreased endocannabinoid levels in the brain and beneficial effects of agents activating cannabinoid and/or vanilloid receptors in a rat model of multiple sclerosis.
Journal: Neurobiology of disease 20051101
Title: Uptake blockade of endocannabinoids in the NTS modulates baroreflex-evoked sympathoinhibition.
Journal: Brain research 20051019
Title: Role of endocannabinoids in the pathogenesis of cirrhotic cardiomyopathy in bile duct-ligated rats.
Journal: British journal of pharmacology 20051001
Title: Conversion of acetaminophen to the bioactive N-acylphenolamine AM404 via fatty acid amide hydrolase-dependent arachidonic acid conjugation in the nervous system.
Journal: The Journal of biological chemistry 20050909
Title: Dual modulation of endocannabinoid transport and fatty acid amide hydrolase protects against excitotoxicity.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience 20050824
Title: The endocannabinoid system: drug targets, lead compounds, and potential therapeutic applications.
Journal: Journal of medicinal chemistry 20050811
Title: Inhibition of fatty acid amide hydrolase and monoacylglycerol lipase by the anandamide uptake inhibitor VDM11: evidence that VDM11 acts as an FAAH substrate.
Journal: British journal of pharmacology 20050801
Title: A role for endocannabinoids in viral-induced dyskinetic and convulsive phenomena.
Journal: Experimental neurology 20050801
Title: Effects of endocannabinoids on discharge of baroreceptive NTS neurons.
Journal: Neuroscience letters 20050624
Title: Accumulation of anandamide: evidence for cellular diversity.
Journal: Neuropharmacology 20050601
Title: Functional role of the endocannabinoid system and AMPA/kainate receptors in 5-HT2A receptor-mediated wet dog shakes.
Journal: European journal of pharmacology 20050523
Title: Synergistic interactions between cannabinoids and environmental stress in the activation of the central amygdala.
Journal: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20050301
Title: AM404, an inhibitor of anandamide reuptake decreases Fos-immunoreactivity in the spinal cord of neuropathic rats after non-noxious stimulation.
Journal: European journal of pharmacology 20050131
Title: Endocannabinoids in the intact retina: 3 H-anandamide uptake, fatty acid amide hydrolase immunoreactivity and hydrolysis of anandamide.
Journal: Visual neuroscience 20050101
Title: Endocannabinoids acting at cannabinoid-1 receptors regulate cardiovascular function in hypertension.
Journal: Circulation 20041005
Title: Sensorimotor gating in mice is disrupted after AM404, an anandamide reuptake and degradation inhibitor.
Journal: Psychopharmacology 20040901
Title: AM404 enhances the spontaneous release of L-glutamate in a manner sensitive to capsazepine in adult rat substantia gelatinosa neurones.
Journal: Brain research 20040827
Title: Anandamide transport inhibitor AM404 and structurally related compounds inhibit synaptic transmission between rat hippocampal neurons in culture independent of cannabinoid CB1 receptors.
Journal: European journal of pharmacology 20040802
Title: Cannabinoids enhance N-methyl-D-aspartate-induced excitation of locus coeruleus neurons by CB1 receptors in rat brain slices.
Journal: Neuroscience letters 20040603
Title: Experimental parkinsonism alters anandamide precursor synthesis, and functional deficits are improved by AM404: a modulator of endocannabinoid function.
Journal: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20040601
Title: Reversible, temperature-dependent, and AM404-inhibitable adsorption of anandamide to cell culture wells as a confounding factor in release experiments.
Journal: European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences 20040601
Title: Endocannabinoid transport tightly controls 2-arachidonoyl glycerol actions in the hippocampus: effects of low temperature and the transport inhibitor AM404.
Journal: The European journal of neuroscience 20040601
Title: Vanilloid receptor TRPV1 antagonists as the next generation of painkillers. Are we putting the cart before the horse?
Journal: Journal of medicinal chemistry 20040520
Title: Selective inhibition of anandamide cellular uptake versus enzymatic hydrolysis--a difficult issue to handle.
Journal: European journal of pharmacology 20040510
Title: Disruption of endocannabinoid release and striatal long-term depression by postsynaptic blockade of endocannabinoid membrane transport.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience 20040218
Title: Differential effects of the sleep-inducing lipid oleamide and cannabinoids on the induction of long-term potentiation in the CA1 neurons of the rat hippocampus in vitro.
Journal: Brain research 20040130
Title: Mediation of amphetamine-induced long-term depression of synaptic transmission by CB1 cannabinoid receptors in the rat amygdala.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience 20031112
Title: Sodium channel inhibition by anandamide and synthetic cannabimimetics in brain.
Journal: Brain research 20030718
Title: Design, synthesis, and biological evaluation of new inhibitors of the endocannabinoid uptake: comparison with effects on fatty acid amidohydrolase.
Journal: Journal of medicinal chemistry 20030410
Title: The actions of anandamide on rat superficial medullary dorsal horn neurons in vitro.
Journal: The Journal of physiology 20030401
Title: AM404 and VDM 11 non-specifically inhibit C6 glioma cell proliferation at concentrations used to block the cellular accumulation of the endocannabinoid anandamide.
Journal: Archives of toxicology 20030401
Title: Compounds acting at the endocannabinoid and/or endovanilloid systems reduce hyperkinesia in a rat model of Huntington's disease.
Journal: Journal of neurochemistry 20030301
Title: Modulation of anxiety through blockade of anandamide hydrolysis.
Journal: Nature medicine 20030101
Title: Prenatal elevation of endocannabinoids corrects the unbalance between dopamine systems and reduces activity in the Naples High Excitability rats.
Journal: Neuroscience and biobehavioral reviews 20030101
Title: Modulation of electrically evoked acetylcholine release through cannabinoid CB1 receptors: evidence for an endocannabinoid tone in the human neocortex.
Journal: Neuroscience 20030101
Title: Comparison of effects of anandamide at recombinant and endogenous rat vanilloid receptors.
Journal: British journal of anaesthesia 20021201
Title: Attenuation of spontaneous opiate withdrawal in mice by the anandamide transport inhibitor AM404.
Journal: European journal of pharmacology 20021101
Title: Experimental parkinsonism alters endocannabinoid degradation: implications for striatal glutamatergic transmission.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience 20020815
Title: Alleviation of motor hyperactivity and neurochemical deficits by endocannabinoid uptake inhibition in a rat model of Huntington's disease.
Journal: Synapse (New York, N.Y.) 20020401
Title: Design, synthesis and biological evaluation of novel arachidonic acid derivatives as highly potent and selective endocannabinoid transporter inhibitors.
Journal: Journal of medicinal chemistry 20011220
Title: Anandamide-induced relaxation of sheep coronary arteries: the role of the vascular endothelium, arachidonic acid metabolites and potassium channels.
Journal: British journal of pharmacology 20011101
Title: Long-term inhibition of nitric oxide synthase potentiates effects of anandamide in the rat mesenteric bed.
Journal: European journal of pharmacology 20010921
Title: Cannabinoid activation of recombinant and endogenous vanilloid receptors.
Journal: European journal of pharmacology 20010727
Title: Mechanisms of endocannabinoid inactivation: biochemistry and pharmacology.
Journal: The Journal of pharmacology and experimental therapeutics 20010701
Title: The activity of anandamide at vanilloid VR1 receptors requires facilitated transport across the cell membrane and is limited by intracellular metabolism.
Journal: The Journal of biological chemistry 20010420
Title: The uptake by cells of 2-arachidonoylglycerol, an endogenous agonist of cannabinoid receptors.
Journal: European journal of biochemistry 20010401
Title: Effects of topical anandamide-transport inhibitors, AM404 and olvanil, on intraocular pressure in normotensive rabbits.
Journal: Pharmaceutical research 20010401
Title: Cannabinoids and pain.
Journal: Current opinion in investigational drugs (London, England : 2000) 20010301
Title: Endocannabinoids control spasticity in a multiple sclerosis model.
Journal: FASEB journal : official publication of the Federation of American Societies for Experimental Biology 20010201
Title: Human platelets bind and degrade 2-arachidonoylglycerol, which activates these cells through a cannabinoid receptor.
Journal: European journal of biochemistry 20010201
Title: AM-404 elevates renal intracellular Ca(2+), questioning its selectivity as a pharmacological tool for investigating the anandamide transporter.
Journal: Journal of pharmacological and toxicological methods 20010101
Title: The anandamide transport inhibitor AM404 activates vanilloid receptors.
Journal: European journal of pharmacology 20000512
Title: Head group analogs of arachidonylethanolamide, the endogenous cannabinoid ligand.
Journal: Journal of medicinal chemistry 19961025
