Title: Medicinal chemistry of A₃ adenosine receptor modulators: pharmacological activities and therapeutic implications.
Journal: Journal of medicinal chemistry 20120628
Title: Pharmacophore elucidation for a new series of 2-aryl-pyrazolo-triazolo-pyrimidines as potent human A3 adenosine receptor antagonists.
Journal: Bioorganic & medicinal chemistry letters 20110515
Title: Antagonist selective modulation of adenosine A1 and A3 receptor pharmacology by the food dye Brilliant Black BN: evidence for allosteric interactions.
Journal: Molecular pharmacology 20100401
Title: Synthesis of theophylline derivatives and study of their activity as antagonists at adenosine receptors.
Journal: Bioorganic & medicinal chemistry 20100315
Title: The role of adenosine receptors in regulating production of tumour necrosis factor-alpha and chemokines by human lung macrophages.
Journal: British journal of pharmacology 20100301
Title: Adenosine blocks IFN-gamma-induced phosphorylation of STAT1 on serine 727 to reduce macrophage activation.
Journal: Journal of immunology (Baltimore, Md. : 1950) 20091115
Title: Multiple receptor subtypes and multiple mechanisms of dilation are involved in vascular network dilation caused by adenosine.
Journal: Microvascular research 20090501
Title: Caffeine modulates TNF-alpha production by cord blood monocytes: the role of adenosine receptors.
Journal: Pediatric research 20090201
Title: Adenosine receptor subtypes in the airways responses to 5'-adenosine monophosphate inhalation of sensitized guinea-pigs.
Journal: Clinical and experimental allergy : journal of the British Society for Allergy and Clinical Immunology 20080901
Title: Inosine and equilibrative nucleoside transporter 2 contribute to hypoxic preconditioning in the murine cardiomyocyte HL-1 cell line.
Journal: American journal of physiology. Heart and circulatory physiology 20080601
Title: Dual purinergic synaptic transmission in the human enteric nervous system.
Journal: American journal of physiology. Gastrointestinal and liver physiology 20080201
Title: Indomethacin stimulates activity and expression of ecto-5'-nucleotidase/CD73 in glioma cell lines.
Journal: European journal of pharmacology 20070813
Title: Stimulation of adenosine A1 and A2A receptors by AMP in the submucosal plexus of guinea pig small intestine.
Journal: American journal of physiology. Gastrointestinal and liver physiology 20070201
Title: Inhibitory responses to exogenous adenosine in murine proximal and distal colon.
Journal: British journal of pharmacology 20060801
Title: Pharmacophore based receptor modeling: the case of adenosine A3 receptor antagonists. An approach to the optimization of protein models.
Journal: Journal of medicinal chemistry 20060713
Title: Inosine released after hypoxia activates hepatic glucose liberation through A3 adenosine receptors.
Journal: American journal of physiology. Endocrinology and metabolism 20060501
Title: Radioligand binding and functional responses of ligands for human recombinant adenosine A(3) receptors.
Journal: Autonomic & autacoid pharmacology 20060401
Title: A3 adenosine receptor antagonists delay irreversible synaptic failure caused by oxygen and glucose deprivation in the rat CA1 hippocampus in vitro.
Journal: British journal of pharmacology 20060301
Title: Antiinflammatory effect of A3 adenosine receptor agonists in murine autoimmune arthritis models.
Journal: The Journal of rheumatology 20050301
Title: Modulation of seizures and synaptic plasticity by adenosinergic receptors in an experimental model of temporal lobe epilepsy induced by pilocarpine in rats.
Journal: Epilepsia 20050101
Title: [3H]OSIP339391, a selective, novel, and high affinity antagonist radioligand for adenosine A2B receptors.
Journal: Biochemical pharmacology 20040715
Title: Inosine stimulates chemotaxis, Ca2+-transients and actin polymerization in immature human dendritic cells via a pertussis toxin-sensitive mechanism independent of adenosine receptors.
Journal: Journal of cellular physiology 20040401
Title: A2A and A3 receptors mediate the adenosine-induced relaxation in spontaneously active possum duodenum in vitro.
Journal: British journal of pharmacology 20030401
Title: Positive coupling of atypical adenosine A3 receptors on human eosinophils to adenylyl cyclase.
Journal: Biochemical and biophysical research communications 20030117
Title: Activation of A(3) receptors by endogenous adenosine inhibits synaptic transmission during hypoxia in rat cortical neurons.
Journal: Restorative neurology and neuroscience 20030101
Title: Structural determinants of A(3) adenosine receptor activation: nucleoside ligands at the agonist/antagonist boundary.
Journal: Journal of medicinal chemistry 20020926
Title: 1,2,4-Triazolo[5,1-i]purine derivatives as highly potent and selective human adenosine A(3) receptor ligands.
Journal: Journal of medicinal chemistry 20020815
Title: Targeted deletion of adenosine A(3) receptors augments adenosine-induced coronary flow in isolated mouse heart.
Journal: American journal of physiology. Heart and circulatory physiology 20020601
Title: 2-Chloro-N(6)-cyclopentyladenosine, adenosine A(1) receptor agonist, antagonizes the adenosine A(3) receptor.
Journal: European journal of pharmacology 20020517
Title: p53-Independent induction of Fas and apoptosis in leukemic cells by an adenosine derivative, Cl-IB-MECA.
Journal: Biochemical pharmacology 20020301
Title: Effects of A(3) adenosine receptor activation and gene knock-out in ischemic-reperfused mouse heart.
Journal: Cardiovascular research 20020101
Title: A3 receptors mediate rapid inflammatory cell influx into the lungs of sensitized guinea-pigs.
Journal: Clinical and experimental allergy : journal of the British Society for Allergy and Clinical Immunology 20010601
Title: Cyclic AMP-dependent inhibition of human neutrophil oxidative activity by substituted 2-propynylcyclohexyl adenosine A(2A) receptor agonists.
Journal: British journal of pharmacology 20010301
Title: Adenosine A(1) and A(3) receptors mediate inhibition of synaptic transmission in rat cortical neurons.
Journal: Neuropharmacology 20010101
Title: Activation of the A3 adenosine receptor affects cell cycle progression and cell growth.
Journal: Naunyn-Schmiedeberg's archives of pharmacology 20000301
Title: Pharmacological characterization of novel A3 adenosine receptor-selective antagonists.
Journal: Neuropharmacology 19970901
Title: Derivatives of the triazoloquinazoline adenosine antagonist (CGS15943) are selective for the human A3 receptor subtype.
Journal: Journal of medicinal chemistry 19961011
