[1]JournalofMedicinalChemistry,2016,vol.59,p.4778-4789
[2]Patent:WO2015/188368,2015,A1.Locationinpatent:Page/Pagecolumn46
[1]CurrentPatentAssignee:MERCK&COINC-WO2015/188368,2015,A1Locationinpatent:Page/Pagecolumn144
[2]Walji,AbbasM.;Hostetler,EricD.;Selnick,Harold;Zeng,Zhizhen;Miller,Patricia;Bennacef,Idriss;Salinas,Cristian;Connolly,Brett;Gantert,Liza;Holahan,Marie;O'Malley,Stacey;Purcell,Mona;Riffel,Kerry;Li,Jing;Balsells,Jaume;Obrien,JulieA.;Melquist,Stacey;Soriano,Aileen;Zhang,Xiaoping;Ogawa,Aimie;Xu,Serena;Joshi,Elizabeth;DellaRocca,Joseph;Hess,FredJ.;Schachter,Joel;Hesk,David;Schenk,David;Struyk,Arie;Babaoglu,Kerim;Lohith,TalakadG.;Wang,Yaode;Yang,Kun;Fu,Jianmin;Evelhoch,JeffreyL.;Coleman,PaulJ.[JournalofMedicinalChemistry,2016,vol.59,#10,p.4778-4789]