[1]BioorganicandMedicinalChemistryLetters,2010,vol.20,#9,p.2958-2963
Title: Alleviation of behavioral hypersensitivity in mouse models of inflammatory pain with two structurally different casein kinase 1 (CK1) inhibitors.
Journal: Molecular pain 20140101
Title: Aryl hydrocarbon receptor-mediated disruption of contact inhibition is associated with connexin43 downregulation and inhibition of gap junctional intercellular communication.
Journal: Archives of toxicology 20130301
Title: IC261 induces cell cycle arrest and apoptosis of human cancer cells via CK1δ/ɛ and Wnt/β-catenin independent inhibition of mitotic spindle formation.
Journal: Oncogene 20110602
Title: Kinase inhibitors modulate huntingtin cell localization and toxicity.
Journal: Nature chemical biology 20110529
Title: Inhibition of gamma-secretase by the CK1 inhibitor IC261 does not depend on CK1delta.
Journal: Bioorganic & medicinal chemistry letters 20100501
Title: CK1epsilon is required for breast cancers dependent on beta-catenin activity.
Journal: PloS one 20100101
Title: Anti-apoptotic and growth-stimulatory functions of CK1 delta and epsilon in ductal adenocarcinoma of the pancreas are inhibited by IC261 in vitro and in vivo.
Journal: Gut 20080601
Title: Phosphorylation of nm23-H1 by CKI induces its complex formation with h-prune and promotes cell motility.
Journal: Oncogene 20080320
Title: Inhibition of casein kinase 1-epsilon induces cancer-cell-selective, PERIOD2-dependent growth arrest.
Journal: Genome biology 20080101
Title: Casein kinase 1 is a novel negative regulator of E-cadherin-based cell-cell contacts.
Journal: Molecular and cellular biology 20070501
Title: Posttranslational regulation of Neurospora circadian clock by CK1a-dependent phosphorylation.
Journal: Cold Spring Harbor symposia on quantitative biology 20070101
Title: Mono-(2-ethylhexyl) phthalate rapidly increases celsr2 protein phosphorylation in HeLa cells via protein kinase C and casein kinase 1.
Journal: Toxicological sciences : an official journal of the Society of Toxicology 20060501
Title: Inhibition of casein kinase I delta alters mitotic spindle formation and induces apoptosis in trophoblast cells.
Journal: Oncogene 20051201
Title: Protein kinase CK1alpha regulates mRNA binding by heterogeneous nuclear ribonucleoprotein C in response to physiologic levels of hydrogen peroxide.
Journal: The Journal of biological chemistry 20050415
Title: Circadian regulation of GABAA receptor function by CKI epsilon-CKI delta in the rat suprachiasmatic nuclei.
Journal: Nature neuroscience 20040501
Title: Casein kinase 1 delta phosphorylates tau and disrupts its binding to microtubules.
Journal: The Journal of biological chemistry 20040416
Title: Casein kinase 1 regulates connexin-43 gap junction assembly.
Journal: The Journal of biological chemistry 20021122
Title: Sustained ER Ca2+ depletion suppresses protein synthesis and induces activation-enhanced cell death in mast cells.
Journal: The Journal of biological chemistry 20020419
Title: Crystal structure of a conformation-selective casein kinase-1 inhibitor.
Journal: The Journal of biological chemistry 20000630
Title: Mashhoon N, et al. Crystal structure of a conformation-selective casein kinase-1 inhibitor. J Biol Chem. 2000 Jun 30;275(26):20052-60.
Title: Stöter M, et al. Inhibition of casein kinase I delta alters mitotic spindle formation and induces apoptosis in trophoblast cells. Oncogene. 2005 Dec 1;24(54):7964-75.
Title: Brockschmidt C, et al. Anti-apoptotic and growth-stimulatory functions of CK1 delta and epsilon in ductal adenocarcinoma of the pancreas are inhibited by IC261 in vitro and in vivo. Gut. 2008 Jun;57(6):799-806.