1884712-47-3 | Cpi-637

865156-34-9    1884712-47-3 

[1]Taylor,AlexanderM.;Côté,Alexandre;Hewitt,MichaelC.;Pastor,Richard;Leblanc,Yves;Nasveschuk,ChristopherG.;Romero,F.Anthony;Crawford,TerryD.;Cantone,Nico;Jayaram,Hariharan;Setser,Jeremy;Murray,Jeremy;Beresini,MaureenH.;DeLeonBoenig,Gladys;Chen,Zhongguo;Conery,AndrewR.;Cummings,RichardT.;Dakin,LeslieA.;Flynn,E.Megan;Huang,OscarW.;Kaufman,Susan;Keller,PatriciaJ.;Kiefer,JamesR.;Lai,Tommy;Li,Yingjie;Liao,Jiangpeng;Liu,Wenfeng;Lu,Henry;Pardo,Eneida;Tsui,Vickie;Wang,Jian;Wang,Yongyun;Xu,Zhaowu;Yan,Fen;Yu,Dong;Zawadzke,Laura;Zhu,Xiaoqin;Zhu,Xiaoyu;Sims,RobertJ.;Cochran,AndreaG.;Bellon,Steve;Audia,JamesE.;Magnuson,Steven;Albrecht,BrianK.[ACSMedicinalChemistryLetters,2016,vol.7,#5,p.531-536]

[2]CurrentPatentAssignee:MORPHOSYSAG;WUXIAPPTECCO.,LTD.;ROCHEHOLDINGAG-WO2016/55028,2016,A1

1884712-70-2    1884712-47-3 

[1]Taylor,AlexanderM.;Côté,Alexandre;Hewitt,MichaelC.;Pastor,Richard;Leblanc,Yves;Nasveschuk,ChristopherG.;Romero,F.Anthony;Crawford,TerryD.;Cantone,Nico;Jayaram,Hariharan;Setser,Jeremy;Murray,Jeremy;Beresini,MaureenH.;DeLeonBoenig,Gladys;Chen,Zhongguo;Conery,AndrewR.;Cummings,RichardT.;Dakin,LeslieA.;Flynn,E.Megan;Huang,OscarW.;Kaufman,Susan;Keller,PatriciaJ.;Kiefer,JamesR.;Lai,Tommy;Li,Yingjie;Liao,Jiangpeng;Liu,Wenfeng;Lu,Henry;Pardo,Eneida;Tsui,Vickie;Wang,Jian;Wang,Yongyun;Xu,Zhaowu;Yan,Fen;Yu,Dong;Zawadzke,Laura;Zhu,Xiaoqin;Zhu,Xiaoyu;Sims,RobertJ.;Cochran,AndreaG.;Bellon,Steve;Audia,JamesE.;Magnuson,Steven;Albrecht,BrianK.[ACSMedicinalChemistryLetters,2016,vol.7,#5,p.531-536]

[2]CurrentPatentAssignee:MORPHOSYSAG;WUXIAPPTECCO.,LTD.;ROCHEHOLDINGAG-WO2016/55028,2016,A1

1884712-71-3    1884712-55-3    1884712-47-3 

[1]Taylor,AlexanderM.;Côté,Alexandre;Hewitt,MichaelC.;Pastor,Richard;Leblanc,Yves;Nasveschuk,ChristopherG.;Romero,F.Anthony;Crawford,TerryD.;Cantone,Nico;Jayaram,Hariharan;Setser,Jeremy;Murray,Jeremy;Beresini,MaureenH.;DeLeonBoenig,Gladys;Chen,Zhongguo;Conery,AndrewR.;Cummings,RichardT.;Dakin,LeslieA.;Flynn,E.Megan;Huang,OscarW.;Kaufman,Susan;Keller,PatriciaJ.;Kiefer,JamesR.;Lai,Tommy;Li,Yingjie;Liao,Jiangpeng;Liu,Wenfeng;Lu,Henry;Pardo,Eneida;Tsui,Vickie;Wang,Jian;Wang,Yongyun;Xu,Zhaowu;Yan,Fen;Yu,Dong;Zawadzke,Laura;Zhu,Xiaoqin;Zhu,Xiaoyu;Sims,RobertJ.;Cochran,AndreaG.;Bellon,Steve;Audia,JamesE.;Magnuson,Steven;Albrecht,BrianK.[ACSMedicinalChemistryLetters,2016,vol.7,#5,p.531-536]

[2]CurrentPatentAssignee:MORPHOSYSAG;WUXIAPPTECCO.,LTD.;ROCHEHOLDINGAG-WO2016/55028,2016,A1Locationinpatent:Page/Pagecolumn114

3970-37-4   

(R)-4-methyl-6-(1-methyl-3-(1-methyl-1H-pyrazol-4-yl)-1H-indazol-5-yl)-1,3,4,5-tetrahydro-2Hbenzob1,4diazepin-2-one 

[1]ACSMedicinalChemistryLetters,2016,vol.7,p.531-536

1884712-53-1    1884712-47-3 

[1]Taylor,AlexanderM.;Côté,Alexandre;Hewitt,MichaelC.;Pastor,Richard;Leblanc,Yves;Nasveschuk,ChristopherG.;Romero,F.Anthony;Crawford,TerryD.;Cantone,Nico;Jayaram,Hariharan;Setser,Jeremy;Murray,Jeremy;Beresini,MaureenH.;DeLeonBoenig,Gladys;Chen,Zhongguo;Conery,AndrewR.;Cummings,RichardT.;Dakin,LeslieA.;Flynn,E.Megan;Huang,OscarW.;Kaufman,Susan;Keller,PatriciaJ.;Kiefer,JamesR.;Lai,Tommy;Li,Yingjie;Liao,Jiangpeng;Liu,Wenfeng;Lu,Henry;Pardo,Eneida;Tsui,Vickie;Wang,Jian;Wang,Yongyun;Xu,Zhaowu;Yan,Fen;Yu,Dong;Zawadzke,Laura;Zhu,Xiaoqin;Zhu,Xiaoyu;Sims,RobertJ.;Cochran,AndreaG.;Bellon,Steve;Audia,JamesE.;Magnuson,Steven;Albrecht,BrianK.[ACSMedicinalChemistryLetters,2016,vol.7,#5,p.531-536]

[2]CurrentPatentAssignee:MORPHOSYSAG;WUXIAPPTECCO.,LTD.;ROCHEHOLDINGAG-WO2016/55028,2016,A1

Title: Taylor AM, et al. Fragment-Based Discovery of a Selective and Cell-Active Benzodiazepinone CBP/EP300 Bromodomain Inhibitor (CPI-637). ACS Med Chem Lett. 2016 Mar 15;7(5):531-6.