Home Amines 192132-77-7
192132-77-7,MFCD28506265
Catalog No.:AA01JWMJ

192132-77-7 | 2-(2-((tert-Butoxycarbonyl)amino)ethoxy)-ethyl 4-methylbenzenesulfonate

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250mg
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  • Technical Information
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  • Downstream Synthesis Route
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  • Technical Information
  • Properties
  • Downstream Synthesis Route
  • Literature
Technical Information
Catalog Number:
AA01JWMJ
Chemical Name:
2-(2-((tert-Butoxycarbonyl)amino)ethoxy)-ethyl 4-methylbenzenesulfonate
CAS Number:
192132-77-7
Molecular Formula:
C16H25NO6S
Molecular Weight:
359.4378
MDL Number:
MFCD28506265
SMILES:
O=C(OC(C)(C)C)NCCOCCOS(=O)(=O)c1ccc(cc1)C
Properties

Downstream Synthesis Route
192132-77-7    294-90-6   
1,4,7,10-tetra-N-(tert-butoxycarbonyl)-2-(aminoethoxy(ethyl))-1,4,7,10-tetraazacyclododecane 

[1]Cruz-Morales,JorgeA.;Guadarrama,Patricia[JournalofMolecularStructure,2005,vol.779,#1-3,p.1-10]

[1]Tamura,Tomonori;Tsukiji,Shinya;Hamachi,Itaru[JournaloftheAmericanChemicalSociety,2012,vol.134,#4,p.2216-2226]

[2]CurrentPatentAssignee:KOREARESEARCHINSTITUTEOFCHEMICALTECHNOLOGY;KOREARESEARCHINSTITUTEOFBIOSCIENCEANDBIOTECHNOLOGY-EP3922632,2021,A1Locationinpatent:Paragraph0415-0417

[3]CurrentPatentAssignee:KOREARESEARCHINSTITUTEOFCHEMICALTECHNOLOGY;KOREARESEARCHINSTITUTEOFBIOSCIENCEANDBIOTECHNOLOGY-EP3922632,2021,A1Locationinpatent:Paragraph0415-0417

[4]Comeo,Eleonora;Kindon,NicholasD.;Soave,Mark;Stoddart,LeighA.;Kilpatrick,LauraE.;Scammells,PeterJ.;Hill,StephenJ.;Kellam,Barrie[JournalofMedicinalChemistry,2020,vol.63,#5,p.2656-2672]

[5]Matsusaki,Motonori;Muraoka,Takahiro;Okada,Shunsuke;Okumura,Masaki[Molecules,2021,vol.26,#4]

[6]Locationinpatent:schemeortableChang,Sung-Youn;Bae,SuJung;Lee,MyungYun;Baek,Seung-Hwa;Chang,Sukbok;Kim,SeongHwan[BioorganicandMedicinalChemistryLetters,2011,vol.21,#2,p.727-729]

[7]CurrentPatentAssignee:UNIVERSITYOFURBINO;THEUNIVERSITYOFBOLOGNA-WO2021/137134,2021,A1Locationinpatent:Page/Pagecolumn58

[8]Nosiglia,MarkA.;Colley,NathanD.;Danielson,MaryK.;Palmquist,MarkS.;Delawder,AbigailO.;Tran,SheilaL.;Harlan,GrayH.;Barnes,JonathanC.[JournaloftheAmericanChemicalSociety,2022,vol.144,#22,p.9990-9996]

[9]Cruz-Morales,JorgeA.;Guadarrama,Patricia[JournalofMolecularStructure,2005,vol.779,#1-3,p.1-10]

[10]Mori,Ryota;Kato,Asako;Komenoi,Kousuke;Kurasaki,Haruaki;Iijima,Touru;Kawagoshi,Masashi;Kiran;Takeda,Sho;Sakai,Norio;Konakahara,Takeo[EuropeanJournalofMedicinalChemistry,2014,vol.82,p.16-35]

[11]CurrentPatentAssignee:SSPharmaceuticalCo.,Ltd.-US6171520,2001,B2

[12]Söveges;Imre;Póti;Sok;Kele,Zs.;Alexa;Kele;Németh[OrganicandBiomolecularChemistry,2018,vol.16,#32,p.5756-5763]

[13]CurrentPatentAssignee:ENLIVENTHERAPEUTICS-WO2022/76973,2022,A1Locationinpatent:Paragraph0623

[14]Géraldy,Magalie;Morgen,Michael;Sehr,Peter;Steimbach,RaphaelR.;Moi,Davide;Ridinger,Johannes;Oehme,Ina;Witt,Olaf;Malz,Mona;Nogueira,MauroS.;Koch,Oliver;Gunkel,Nikolas;Miller,AubryK.[JournalofMedicinalChemistry,2019,vol.62,#9,p.4426-4443]

[15]CurrentPatentAssignee:UPPTHERA-WO2021/201577,2021,A1Locationinpatent:Paragraph544;550-551

[16]CurrentPatentAssignee:CIDARATHERAPEUTICSINC-WO2020/51498,2020,A1Locationinpatent:Page/Pagecolumn465;502

[17]Li,Haiwei;Wang,Shouxin;Ma,Wenxiao;Cheng,Boyang;Yi,Yanliang;Ma,Xinyuan;Xiao,Sulong;Zhang,Lihe;Zhou,Demin[JournalofMedicinalChemistry,2022,vol.65,#10,p.7154-7169]

[18]CurrentPatentAssignee:GLAXOSMITHKLINEPLC-WO2006/50941,2006,A1Locationinpatent:Page/Pagecolumn44

[19]Moon,JoongHo;McDaniel,William;MacLean,Paul;Hancock,LawrenceF.[AngewandteChemie-InternationalEdition,2007,vol.46,#43,p.8223-8225]

[20]CurrentPatentAssignee:HAINANHAILINGCHEMIPHARMA-EP2123283,2009,A1Locationinpatent:Page/Pagecolumn14

[21]CurrentPatentAssignee:HAINANHAILINGCHEMIPHARMA-US2009/325894,2009,A1Locationinpatent:Page/Pagecolumn9

[22]CurrentPatentAssignee:GLAXOSMITHKLINEPLC;GALAPAGOS-WO2006/50942,2006,A1Locationinpatent:Page/Pagecolumn68

[23]CurrentPatentAssignee:GLAXOSMITHKLINEPLC;GALAPAGOS-WO2006/50943,2006,A1Locationinpatent:Page/Pagecolumn49

[24]Welle,Alexandre;Billard,Francois;Marchand-Brynaert,Jacqueline[Synthesis,2012,vol.44,#14,p.2249-2254]

[25]El-Gendy,BahaaEl-DienM.;GhazviniZadeh,EbrahimH.;Sotuyo,AniaC.;Pillai,GirinathG.;Katritzky,AlanR.[ChemicalBiologyandDrugDesign,2013,vol.81,#5,p.577-582]

[26]Mendez,Eladio;Moon,JoongHo[ChemicalCommunications,2013,vol.49,#54,p.6048-6050]

[27]CurrentPatentAssignee:HEMAY(HONGKONG)INVESTMENTLIMITED-EP2824108,2015,A1Locationinpatent:Paragraph0107

[28]CurrentPatentAssignee:ROCHEHOLDINGAG-US2015/31674,2015,A1Locationinpatent:Paragraph0266;0268

[29]CurrentPatentAssignee:HEMAY(HONGKONG)INVESTMENTLIMITED-US2015/166595,2015,A1Locationinpatent:Paragraph0225

[30]CurrentPatentAssignee:CHONNAMNATIONALUNIVERSITY-KR2018/1250,2018,ALocationinpatent:Paragraph0060-0061

[31]CurrentPatentAssignee:MERCK&COINC-WO2018/57409,2018,A1Locationinpatent:Page/Pagecolumn86

[32]CurrentPatentAssignee:DANA-FARBERCANCERINSTITUTE-WO2019/165229,2019,A1Locationinpatent:Paragraph00534;00535

[33]CurrentPatentAssignee:SERVIERMONDE-WO2021/155006,2021,A1Locationinpatent:Page/Pagecolumn62;65

[1]Cruz-Morales,JorgeA.;Guadarrama,Patricia[JournalofMolecularStructure,2005,vol.779,#1-3,p.1-10]

[1]Matsusaki,Motonori;Muraoka,Takahiro;Okada,Shunsuke;Okumura,Masaki[Molecules,2021,vol.26,#4]

[2]CurrentPatentAssignee:GLAXOSMITHKLINEPLC-WO2006/50941,2006,A1Locationinpatent:Page/Pagecolumn44

[3]CurrentPatentAssignee:GLAXOSMITHKLINEPLC;GALAPAGOS-WO2006/50942,2006,A1Locationinpatent:Page/Pagecolumn68

[4]CurrentPatentAssignee:GLAXOSMITHKLINEPLC;GALAPAGOS-WO2006/50943,2006,A1Locationinpatent:Page/Pagecolumn49

[1]CurrentPatentAssignee:SSPharmaceuticalCo.,Ltd.-US6171520,2001,B2

Literature

Title: An S, et al. Small-molecule PROTACs: An emerging and promising approach for the development of targeted therapy drugs. EBioMedicine. 2018 Oct;36:553-562.

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Tags:192132-77-7 Molecular Formula|192132-77-7 MDL|192132-77-7 SMILES|192132-77-7 2-(2-((tert-Butoxycarbonyl)amino)ethoxy)-ethyl 4-methylbenzenesulfonate