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Home Other Building Blocks 1971920-73-6
1971920-73-6,MFCD32710277
Catalog No.:AA01V791

1971920-73-6 | Tolebrutinib

Pack Size
Purity
Availability
Price(USD)
Quantity
  
5mg
≥95%
in stock  
$96.00   $67.00
- +
10mg
≥95%
in stock  
$172.00   $120.00
- +
  • Technical Information
  • Properties
  • Downstream Synthesis Route
  • Literature
  • Request for Quotation
  • Download SDS
  • Technical Information
  • Properties
  • Downstream Synthesis Route
  • Literature
Technical Information
Catalog Number:
AA01V791
Chemical Name:
Tolebrutinib
CAS Number:
1971920-73-6
Molecular Formula:
C26H25N5O3
Molecular Weight:
455.5084
MDL Number:
MFCD32710277
SMILES:
C=CC(=O)N1CCC[C@H](C1)n1c(=O)n(c2c1ccnc2N)c1ccc(cc1)Oc1ccccc1
Properties

Downstream Synthesis Route

[1]CurrentPatentAssignee:SANOFI-WO2016/196840,2016,A1

[1]CurrentPatentAssignee:SANOFI-WO2016/196840,2016,A1

[1]CurrentPatentAssignee:SANOFI-WO2016/196840,2016,A1

[1]CurrentPatentAssignee:SANOFI-WO2016/196840,2016,A1

[1]CurrentPatentAssignee:SANOFI-WO2016/196840,2016,A1

Literature

Title: Dahl K, et, al. Radiosynthesis of a Bruton's tyrosine kinase inhibitor, [ 11 CTolebrutinib, via palladium-NiXantphos-mediated carbonylation. J Labelled Comp Radiopharm. 2020 Sep;63(11):482-487.

Title: Francesco MR, et, al. PRN2246, a potent and selective blood brain barrier penetrating BTK inhibitor, exhibits efficacy in central nervous system immunity. Multiple Sclerosis Journal. 2017;Poster Session 2:P989.

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SDS
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