Title: Efficacious N-protection of O-aryl sulfamates with 2,4-dimethoxybenzyl groups.
Journal: Organic & biomolecular chemistry 20121007
Title: Molecular cloning, characterization, and inhibition studies of a β-carbonic anhydrase from Malassezia globosa, a potential antidandruff target.
Journal: Journal of medicinal chemistry 20120412
Title: Aromatase and dual aromatase-steroid sulfatase inhibitors from the letrozole and vorozole templates.
Journal: ChemMedChem 20110801
Title: Carbonic anhydrase inhibitors; fluorinated phenyl sulfamates show strong inhibitory activity and selectivity for the inhibition of the tumor-associated isozymes IX and XII over the cytosolic ones I and II.
Journal: Bioorganic & medicinal chemistry letters 20090901
Title: Recent developments of steroid sulfatase inhibitors as anti-cancer agents.
Journal: Anti-cancer agents in medicinal chemistry 20081001
Title: Dual aromatase-sulfatase inhibitors based on the anastrozole template: synthesis, in vitro SAR, molecular modelling and in vivo activity.
Journal: Organic & biomolecular chemistry 20071021
Title: Dual aromatase-sulfatase inhibitors based on the anastrozole template: synthesis, in vitro SAR, molecular modelling and in vivo activity.
Journal: Organic & biomolecular chemistry 20070921
Title: Synthesis and evaluation of general mechanism-based inhibitors of sulfatases based on (difluoro)methyl phenyl sulfate and cyclic phenyl sulfamate motifs.
Journal: Bioorganic & medicinal chemistry 20061215
Title: Microsphere-based protease assays and screening application for lethal factor and factor Xa.
Journal: Cytometry. Part A : the journal of the International Society for Analytical Cytology 20060501
Title: Carbonic anhydrase inhibitors: inhibition of the human isozymes I, II, VA, and IX with a library of substituted difluoromethanesulfonamides.
Journal: Bioorganic & medicinal chemistry letters 20051201
Title: Steroid sulfatase: molecular biology, regulation, and inhibition.
Journal: Endocrine reviews 20050401
Title: A letrozole-based dual aromatase-sulphatase inhibitor with in vivo activity.
Journal: The Journal of steroid biochemistry and molecular biology 20050201
Title: Carbonic anhydrase inhibitors. Inhibition of cytosolic isozymes I and II and transmembrane, tumor-associated isozyme IX with sulfamates including EMATE also acting as steroid sulfatase inhibitors.
Journal: Journal of medicinal chemistry 20030522
Title: Structure-activity relationship determination within a group of substituted phenyl sulfamate based compounds against the enzyme oestrone sulfatase.
Journal: The Journal of pharmacy and pharmacology 20030201
Title: The mechanism of the irreversible inhibition of estrone sulfatase (ES) through the consideration of a range of methane- and amino-sulfonate-based compounds.
Journal: Bioorganic & medicinal chemistry letters 20020506
Title: Acid dissociation constant, a potential physicochemical factor in the inhibition of the enzyme estrone sulfatase (ES).
Journal: Bioorganic & medicinal chemistry letters 20010409
