Title: Structural insights from binding poses of CCR2 and CCR5 with clinically important antagonists: a combined in silico study.
Journal: PloS one 20120101
Title: Synthesis and biological evaluation of 3-aminopyrrolidine derivatives as CC chemokine receptor 2 antagonists.
Journal: Bioorganic & medicinal chemistry letters 20100401
Title: Elucidation of binding sites of dual antagonists in the human chemokine receptors CCR2 and CCR5.
Journal: Molecular pharmacology 20090601
Title: Potent antagonists of the CCR2b receptor. Part 3: SAR of the (R)-3-aminopyrrolidine series.
Journal: Bioorganic & medicinal chemistry letters 20080315
Title: Moree WJ, et al. Potent antagonists of the CCR2b receptor. Part 3: SAR of the (R)-3-aminopyrrolidine series. Bioorg Med Chem Lett. 2008 Mar 15;18(6):1869-73.
Title: Hall SE, et al. Elucidation of binding sites of dual antagonists in the human chemokine receptors CCR2 and CCR5. Mol Pharmacol. 2009 Jun;75(6):1325-36.
Title: Calin M, et al. VCAM-1 directed target-sensitive liposomes carrying CCR2 antagonists bind to activated endothelium and reduce adhesion and transmigration of monocytes. Eur J Pharm Biopharm. 2015 Jan;89:18-29.
