[1]Smith,BrianM.;Smith,JeffreyM.;Tsai,JamesH.;Schultz,JeffreyA.;Gilson,CharlesA.;Estrada,ScottA.;Chen,RitaR.;Park,DouglasM.;Prieto,EmilyB.;Gallardo,CharlemagneS.;Sengupta,Dipanjan;Thomsen,WilliamJ.;Saldana,HazelR.;Whelan,KevinT.;Menzaghi,Frederique;Webb,RobertR.;Beeley,NigelR.A.[BioorganicandMedicinalChemistryLetters,2005,vol.15,#5,p.1467-1470]
[2]CurrentPatentAssignee:C.H.BoehringerSohnAG&Co.KG-WO2008/80891,2008,A2Locationinpatent:Page/Pagecolumn121
[3]CurrentPatentAssignee:SYGNATUREDISCOVERYLTD;OTSUKAHOLDINGSCOLTD-WO2017/68412,2017,A1Locationinpatent:Page/Pagecolumn240
[1]Smith,BrianM.;Smith,JeffreyM.;Tsai,JamesH.;Schultz,JeffreyA.;Gilson,CharlesA.;Estrada,ScottA.;Chen,RitaR.;Park,DouglasM.;Prieto,EmilyB.;Gallardo,CharlemagneS.;Sengupta,Dipanjan;Thomsen,WilliamJ.;Saldana,HazelR.;Whelan,KevinT.;Menzaghi,Frederique;Webb,RobertR.;Beeley,NigelR.A.[BioorganicandMedicinalChemistryLetters,2005,vol.15,#5,p.1467-1470]
[2]CurrentPatentAssignee:SYGNATUREDISCOVERYLTD;OTSUKAHOLDINGSCOLTD-WO2017/68412,2017,A1
[1]Smith,BrianM.;Smith,JeffreyM.;Tsai,JamesH.;Schultz,JeffreyA.;Gilson,CharlesA.;Estrada,ScottA.;Chen,RitaR.;Park,DouglasM.;Prieto,EmilyB.;Gallardo,CharlemagneS.;Sengupta,Dipanjan;Thomsen,WilliamJ.;Saldana,HazelR.;Whelan,KevinT.;Menzaghi,Frederique;Webb,RobertR.;Beeley,NigelR.A.[BioorganicandMedicinalChemistryLetters,2005,vol.15,#5,p.1467-1470]
[1]CurrentPatentAssignee:C.H.BoehringerSohnAG&Co.KG-WO2008/80891,2008,A2Locationinpatent:Page/Pagecolumn121
Title: Discovery and structure-activity relationship of (1R)-8-chloro-2,3,4,5-tetrahydro-1-methyl-1H-3-benzazepine (Lorcaserin), a selective serotonin 5-HT2C receptor agonist for the treatment of obesity.
Journal: Journal of medicinal chemistry 20080124
Title: Discovery and SAR of new benzazepines as potent and selective 5-HT(2C) receptor agonists for the treatment of obesity.
Journal: Bioorganic & medicinal chemistry letters 20050301