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Journal: Bioorganic & medicinal chemistry letters 20121201
Title: Pharmacokinetic benefits of 3,4-dimethoxy substitution of a phenyl ring and design of isosteres yielding orally available cathepsin K inhibitors.
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Title: New hypotheses for the binding mode of 4- and 7-substituted indazoles in the active site of neuronal nitric oxide synthase.
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Title: Distribution of primary and specialized metabolites in Nigella sativa seeds, a spice with vast traditional and historical uses.
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Title: Osmium(IV) complexes with 1H- and 2H-indazoles: tautomer identity versus spectroscopic properties and antiproliferative activity.
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Title: Discovery of a novel azaindole class of antibacterial agents targeting the ATPase domains of DNA gyrase and Topoisomerase IV.
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Title: The synthesis and SAR of calcitonin gene-related peptide (CGRP) receptor antagonists derived from tyrosine surrogates. Part 1.
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Title: Discovery and structure-activity relationship of 2,6-disubstituted pyrazines, potent and selective inhibitors of protein kinase CK2.
Journal: Bioorganic & medicinal chemistry letters 20120701
Title: Highly efficient redox isomerisation of allylic alcohols catalysed by pyrazole-based ruthenium(IV) complexes in water: mechanisms of bifunctional catalysis in water.
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Title: Tris[2-(2H-indazol-2-yl)eth-yl]amine.
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Title: 2-(1H-Pyrrolo-[2,3-b]pyridin-2-yl)pyridine.
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Title: Synthesis, antimicrobial and anti-cancer activities of some new N-ethyl, N-benzyl and N-benzoyl-3-indolyl heterocycles.
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Title: Diazaheterocycle analogues of tetracene: synthesis and properties of a naphtho-fused cinnoline and a naphtho-fused isoindazole.
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Title: A convenient approach to β-heteroarylated (C-N bond) ketones from Cs2CO3 promoted reaction between propargyl alcohols and nitrogen-heterocycles.
Journal: Organic & biomolecular chemistry 20120507
Title: YC-1 exerts inhibitory effects on MDA-MB-468 breast cancer cells by targeting EGFR in vitro and in vivo under normoxic condition.
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Title: 1,3-Dimethyl-1H-indazol-6-amine.
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Title: Synthesis of substituted 1H-indazoles from arynes and hydrazones.
Journal: The Journal of organic chemistry 20120406
Title: Synthesis of new α aminophosphonate system bearing Indazole moiety and their biological activity.
Journal: European journal of medicinal chemistry 20120401
Title: Ethyl 3-[7-eth-oxy-6-(4-meth-oxy-benzene-sulfonamido)-2H-indazol-2-yl]propano-ate.
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Title: HS-116, a novel phosphatidylinositol 3-kinase inhibitor induces apoptosis and suppresses angiogenesis of hepatocellular carcinoma through inhibition of the PI3K/AKT/mTOR pathway.
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Title: Synthesis of fused indazole ring systems and application to nigeglanine hydrobromide.
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Title: Highly fluorinated aryl-substituted tris(indazolyl)borate thallium complexes: diverse regiochemistry at the B-N bond.
Journal: Inorganic chemistry 20120305
Title: Design, synthesis and biological evaluation of Trypanosoma brucei trypanothione synthetase inhibitors.
Journal: ChemMedChem 20120102
Title: Pyrrolo[3,2-d]pyrimidine derivatives as type II kinase insert domain receptor (KDR) inhibitors: CoMFA and CoMSIA studies.
Journal: International journal of molecular sciences 20120101
Title: Investigation of indazole unbinding pathways in CYP2E1 by molecular dynamics simulations.
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Title: Genomics of Dementia: APOE- and CYP2D6-Related Pharmacogenetics.
Journal: International journal of Alzheimer's disease 20120101
Title: Third generation tyrosine kinase inhibitors and their development in advanced renal cell carcinoma.
Journal: Frontiers in oncology 20120101
Title: Design and synthesis of pyridone inhibitors of non-nucleoside reverse transcriptase.
Journal: Bioorganic & medicinal chemistry letters 20111215
Title: (WO2011057959) indole and indazole derivatives as glycogen synthase activators: a patent evaluation.
Journal: Expert opinion on therapeutic patents 20111201
Title: Discovery of novel anti-inflammatory drug-like compounds by aligning in silico and in vivo screening: the nitroindazolinone chemotype.
Journal: European journal of medicinal chemistry 20111201
Title: Experimental and theoretical electron-density study of three isoindole derivatives: topological and Hirshfeld surface analysis of weak intermolecular interactions.
Journal: Acta crystallographica. Section B, Structural science 20111201
Title: N-[7-Eth-oxy-2-(prop-2-en-1-yl)-2H-indazol-6-yl]-4-methyl-benzene-sulfonamide.
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Title: 3-Bromo-6-nitro-1-(prop-2-yn-yl)-1H-indazole.
Journal: Acta crystallographica. Section E, Structure reports online 20111201
Title: Design and synthesis of conformationally constrained inhibitors of non-nucleoside reverse transcriptase.
Journal: Journal of medicinal chemistry 20111124
Title: Discovery of a potent, selective, and orally available class I phosphatidylinositol 3-kinase (PI3K)/mammalian target of rapamycin (mTOR) kinase inhibitor (GDC-0980) for the treatment of cancer.
Journal: Journal of medicinal chemistry 20111110
Title: Design, synthesis and insight into the structure-activity relationship of 1,3-disubstituted indazoles as novel HIF-1 inhibitors.
Journal: Bioorganic & medicinal chemistry letters 20111101
Title: Design, synthesis and SAR of indazole and benzoisoxazole containing 4-azetidinyl-1-aryl-cyclohexanes as CCR2 antagonists.
Journal: Bioorganic & medicinal chemistry letters 20111015
Title: Synthesis, evaluation and application of polycyclic fluorescent analogues as N-methyl-D-aspartate receptor and voltage gated calcium channel ligands.
Journal: European journal of medicinal chemistry 20111001
Title: Lead generation of heat shock protein 90 inhibitors by a combination of fragment-based approach, virtual screening, and structure-based drug design.
Journal: Bioorganic & medicinal chemistry letters 20111001
Title: Novel indole and azaindole (pyrrolopyridine) cannabinoid (CB) receptor agonists: design, synthesis, structure-activity relationships, physicochemical properties and biological activity.
Journal: European journal of medicinal chemistry 20111001
Title: Synthesis and SAR optimization of diketo acid pharmacophore for HCV NS5B polymerase inhibition.
Journal: European journal of medicinal chemistry 20111001
Title: A general and efficient approach to 2H-indazoles and 1H-pyrazoles through copper-catalyzed intramolecular N-N bond formation under mild conditions.
Journal: Chemical communications (Cambridge, England) 20110928
Title: Structure-based design and optimization of potent renin inhibitors on 5- or 7-azaindole-scaffolds.
Journal: Bioorganic & medicinal chemistry letters 20110915
Title: Benzotriazoles and indazoles are scaffolds with biological activity against Entamoeba histolytica.
Journal: Journal of biomolecular screening 20110901
Title: [Evaluation of the retention properties of two cyclodextrin stationary phases with different spacers].
Journal: Se pu = Chinese journal of chromatography 20110901
Title: En route to osmium analogues of KP1019: synthesis, structure, spectroscopic properties and antiproliferative activity of trans-[Os(IV)Cl4(Hazole)2].
Journal: Inorganic chemistry 20110815
Title: Discovery of indazoles as inhibitors of Tpl2 kinase.
Journal: Bioorganic & medicinal chemistry letters 20110815
Title: Insights into the structural requirements of PKCβII inhibitors based on HQSAR and CoMSIA analyses.
Journal: Chemical biology & drug design 20110801
Title: 2,2'-(Propane-1,3-di-yl)bis-(2H-indazole).
Journal: Acta crystallographica. Section E, Structure reports online 20110801
Title: Selectivity of kinase inhibitor fragments.
Journal: Journal of medicinal chemistry 20110728
Title: Rapid preparation of triazolyl substituted NH-heterocyclic kinase inhibitors via one-pot Sonogashira coupling-TMS-deprotection-CuAAC sequence.
Journal: Organic & biomolecular chemistry 20110721
Title: Synthesis and antitumor activity of 3-(2-phenyl-1,3-thiazol-4-yl)-1H-indoles and 3-(2-phenyl-1,3-thiazol-4-yl)-1H-7-azaindoles.
Journal: ChemMedChem 20110704
Title: Consecutive condensation, C-N and N-N bond formations: a copper- catalyzed one-pot three-component synthesis of 2H-indazole.
Journal: Organic letters 20110701
Title: N-[7-Eth-oxy-1-(prop-2-en-1-yl)-1H-indazol-4-yl]-4-methyl-benzene-sulfonamide.
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Title: The Davis-Beirut reaction: N1,N2-disubstituted-1H-indazolones via 1,6-electrophilic addition to 3-alkoxy-2H-indazoles.
Journal: Organic letters 20110617
Title: Understanding the binding mode and function of BMS-488043 against HIV-1 viral entry.
Journal: Proteins 20110601
Title: Progress in the preclinical discovery and clinical development of class I and dual class I/IV phosphoinositide 3-kinase (PI3K) inhibitors.
Journal: Current medicinal chemistry 20110601
Title: Axitinib for the management of metastatic renal cell carcinoma.
Journal: Drugs in R&D 20110601
Title: 4,6-Bis(4-fluoro-phen-yl)-2-phenyl-1H-indazol-3(2H)-one.
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Title: N-(7-Eth-oxy-1H-indazol-4-yl)-4-methyl-benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20110601
Title: N-(2-Chloro-pyrimidin-4-yl)-2-methyl-2H-indazol-6-amine methanol monosolvate.
Journal: Acta crystallographica. Section E, Structure reports online 20110601
Title: 2-Methyl-6-nitro-2H-indazole.
Journal: Acta crystallographica. Section E, Structure reports online 20110601
Title: 3D-QSAR and molecular docking studies of azaindole derivatives as Aurora B kinase inhibitors.
Journal: Journal of molecular modeling 20110501
Title: Synthesis and biological evaluation of indazole derivatives.
Journal: European journal of medicinal chemistry 20110401
Title: Atomic force microscopy-based screening of drug-excipient miscibility and stability of solid dispersions.
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Title: Non-oxime inhibitors of B-Raf(V600E) kinase.
Journal: Bioorganic & medicinal chemistry letters 20110215
Title: Ethyl 3,6-dihy-droxy-6-methyl-4-phenyl-4,5,6,7-tetra-hydro-1H-indazole-5-carboxyl-ate monohydrate.
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Title: Preparation and evaluation of trisubstituted pyrimidines as phosphatidylinositol 3-kinase inhibitors. 3-Hydroxyphenol analogues and bioisosteric replacements.
Journal: Bioorganic & medicinal chemistry 20110115
Title: Organometallic anticancer compounds.
Journal: Journal of medicinal chemistry 20110113
Title: Chemical and biological evaluation of 153 Sm and 46/47 Sc complexes of indazolebisphosphonates for targeted radiotherapy.
Journal: Applied radiation and isotopes : including data, instrumentation and methods for use in agriculture, industry and medicine 20110101
Title: Synthesis of substituted 3-amino-N-phenyl-1H-indazole-1-carboxamides endowed with antiproliferative activity.
Journal: European journal of medicinal chemistry 20110101
Title: Fragment-based discovery of 6-substituted isoquinolin-1-amine based ROCK-I inhibitors.
Journal: Bioorganic & medicinal chemistry letters 20110101
Title: Novel serotonin type 3 receptor partial agonists for the potential treatment of irritable bowel syndrome.
Journal: Bioorganic & medicinal chemistry letters 20110101
Title: Nanoscaled carborane ruthenium(II)-arene complex inducing lung cancer cells apoptosis.
Journal: Journal of nanobiotechnology 20110101
Title: Identification of human IKK-2 inhibitors of natural origin (part I): modeling of the IKK-2 kinase domain, virtual screening and activity assays.
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Title: Interpreting linear support vector machine models with heat map molecule coloring.
Journal: Journal of cheminformatics 20110101
Title: Inhibition of reactive gliosis prevents neovascular growth in the mouse model of oxygen-induced retinopathy.
Journal: PloS one 20110101
Title: Lucanthone and its derivative hycanthone inhibit apurinic endonuclease-1 (APE1) by direct protein binding.
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Title: Investigation of the structure requirement for 5-HT₆ binding affinity of arylsulfonyl derivatives: a computational study.
Journal: International journal of molecular sciences 20110101
Title: Neurochemical architecture of the central complex related to its function in the control of grasshopper acoustic communication.
Journal: PloS one 20110101
Title: ROCKing Regeneration: Rho Kinase Inhibition as Molecular Target for Neurorestoration.
Journal: Frontiers in molecular neuroscience 20110101
Title: Studies on the influence of host plants and effect of chemical stimulants on the feeding behavior in the muga silkworm, Antheraea assamensis.
Journal: Journal of insect science (Online) 20110101
Title: Azaindole N-methyl hydroxamic acids as HIV-1 integrase inhibitors-II. The impact of physicochemical properties on ADME and PK.
Journal: Bioorganic & medicinal chemistry letters 20101215
Title: Discovery of new azaindole-based PI3Kα inhibitors: apoptotic and antiangiogenic effect on cancer cells.
Journal: Bioorganic & medicinal chemistry letters 20101215
Title: The indazole derivative YD-3 specifically inhibits thrombin-induced angiogenesis in vitro and in vivo.
Journal: Shock (Augusta, Ga.) 20101201
Title: Indazole derivatives as novel bradykinin B1 receptor antagonists.
Journal: Bioorganic & medicinal chemistry letters 20101201
Title: PHD3 regulates differentiation, tumour growth and angiogenesis in pancreatic cancer.
Journal: British journal of cancer 20101109
Title: Inhibitors of the tyrosine kinase EphB4. Part 3: identification of non-benzodioxole-based kinase inhibitors.
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Title: 2-(4-Methyl-phen-yl)-2H-indazole.
Journal: Acta crystallographica. Section E, Structure reports online 20101101
Title: N-(2-Chloro-pyrimidin-4-yl)-N,2-di-methyl-2H-indazol-6-amine.
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Title: Palladium-catalyzed amination of unprotected halo-7-azaindoles.
Journal: Organic letters 20101015
Title: Expanding the diversity of allosteric bcr-abl inhibitors.
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Title: Nonsteroidal dissociated glucocorticoid agonists containing azaindoles as steroid A-ring mimetics.
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Title: Structural studies of some push-pull N-arylbenzazoles.
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Title: Design of potent IGF1-R inhibitors related to bis-azaindoles.
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Title: Synthesis and evaluation of indazole based analog sensitive Akt inhibitors.
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Title: Benzydamine as a useful substrate of hepatic flavin-containing monooxygenase activity in veterinary species.
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Title: Synthesis and characterization of selective dopamine D2 receptor antagonists. 2. Azaindole, benzofuran, and benzothiophene analogs of L-741,626.
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Title: Synthesis of quinazolines from N-(2-nitrophenylsulfonyl)iminodiacetate and alpha-(2-nitrophenylsulfonyl)amino ketones via 2H-indazole 1-oxides.
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Title: Mode of action of nifurtimox and N-oxide-containing heterocycles against Trypanosoma cruzi: is oxidative stress involved?
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Title: Discovery of GSK1070916, a potent and selective inhibitor of Aurora B/C kinase.
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Title: 5-Functionalized indazoles as glucocorticoid receptor agonists.
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Title: One-step conversion of azine N-oxides to alpha-1,2,4-triazolo-, 1,2,3-triazolo, imidazolo-, and pyrazoloheteroarenes.
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Title: 4-Chloro-7-methoxy-methyl-2-phenyl-7H-pyrrolo[2,3-b]pyridine.
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Title: Integrated in silico-in vitro strategy for addressing cytochrome P450 3A4 time-dependent inhibition.
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Title: Discovery of 4-amino-1-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)piperidine-4-carboxamides as selective, orally active inhibitors of protein kinase B (Akt).
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Title: Blue fluorescent amino acids as in vivo building blocks for proteins.
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Title: Cu-catalyzed N-alkynylation of imidazoles, benzimidazoles, indazoles, and pyrazoles using PEG as solvent medium.
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Title: Serum-protein interactions with anticancer Ru(III) complexes KP1019 and KP418 characterized by EPR.
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Title: Discovery of biaryl inhibitors of H+/K+ ATPase.
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Title: Luminescent platinum complexes with terdentate ligands forming 6-membered chelate rings: advantageous and deleterious effects in N--N--N and N--C--N-coordinated complexes.
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Title: 2,3,5-Trisubstituted pyridines as selective AKT inhibitors. Part II: Improved drug-like properties and kinase selectivity from azaindazoles.
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Title: Heterocyclic indazole derivatives as SGK1 inhibitors, WO2008138448.
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Title: Secondary metabolites of Volvariella bombycina and their inhibitory effects on melanogenesis.
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Title: Expression genetics identifies spinal mechanisms supporting formalin late phase behaviors.
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Title: A role for nitric oxide-driven retrograde signaling in the consolidation of a fear memory.
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Title: Effects of TLR agonists on the hypoxia-regulated transcription factor HIF-1alpha and dendritic cell maturation under normoxic conditions.
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Title: Nigella sativa L. seed extract modulates the neurotransmitter amino acids release in cultured neurons in vitro.
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Title: Synthesis and Characterization of Novel Ruthenium(III) Complexes with Histamine.
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Title: Studies of the Antiproliferative Activity of Ruthenium (II) Cyclopentadienyl-Derived Complexes with Nitrogen Coordinated Ligands.
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Title: Novel HTS strategy identifies TRAIL-sensitizing compounds acting specifically through the caspase-8 apoptotic axis.
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Title: Janus kinase 2 inhibitors. Synthesis and characterization of a novel polycyclic azaindole.
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Title: Aza-tryptamine substrates in monoterpene indole alkaloid biosynthesis.
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Title: Novel pyrazolopyrimidines as highly potent B-Raf inhibitors.
Journal: Bioorganic & medicinal chemistry letters 20091215
Title: Inhibitors of human immunodeficiency virus type 1 (HIV-1) attachment. 5. An evolution from indole to azaindoles leading to the discovery of 1-(4-benzoylpiperazin-1-yl)-2-(4,7-dimethoxy-1H-pyrrolo[2,3-c]pyridin-3-yl)ethane-1,2-dione (BMS-488043), a drug candidate that demonstrates antiviral activity in HIV-1-infected subjects.
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Title: Theoretical calculations of a model of NOS indazole inhibitors: interaction of aromatic compounds with Zn-porphyrins.
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Title: Effect of fish oils containing different amounts of EPA, DHA, and antioxidants on plasma and brain fatty acids and brain nitric oxide synthase activity in rats.
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Title: Marine pyrrolocarbazoles and analogues: synthesis and kinase inhibition.
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Title: Mutual prodrug of cephazolin and benzydamin: 3-[(1-benzyl-1H-indazol-3-yl)-oxy]-N,N-dimethyl-propan-1-aminium 3-{[(5-methyl-1,3,4-thia-diazol-2-yl)sulfan-yl]meth-yl}-8-oxo-7-[(1H-tetra-zol-1-yl)acetamido]-5-thia-1-aza-bicyclo-[4.2.0]octane-2-carboxyl-ate (benzydaminium cephazolinate).
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Title: [Os(IV)Cl(5)(Hazole)](-) complexes: synthesis, structure, spectroscopic properties, and antiproliferative activity.
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Title: Dissecting the essentiality of the bifunctional trypanothione synthetase-amidase in Trypanosoma brucei using chemical and genetic methods.
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Title: Recent developments in ruthenium anticancer drugs.
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Title: Fluorinated indazoles as novel selective inhibitors of nitric oxide synthase (NOS): synthesis and biological evaluation.
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Title: Electronic structural investigations of ruthenium compounds and anticancer prodrugs.
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Title: 2,3-Dimethyl-6-nitro-2H-indazole.
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Title: N-[(E)-Quinoxalin-2-ylmethyl-idene]-1H-indazol-5-amine.
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Title: Heterobiaryl human immunodeficiency virus entry inhibitors.
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Title: Investigation of various N-heterocyclic substituted piperazine versions of 5/7-{[2-(4-aryl-piperazin-1-yl)-ethyl]-propyl-amino}-5,6,7,8-tetrahydro-naphthalen-2-ol: effect on affinity and selectivity for dopamine D3 receptor.
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Title: Structure-activity relationships and X-ray structures describing the selectivity of aminopyrazole inhibitors for c-Jun N-terminal kinase 3 (JNK3) over p38.
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Title: IRAK-4 inhibitors for inflammation.
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Title: Discovery of potent and selective DP1 receptor antagonists in the azaindole series.
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Title: 1-(5-Carboxyindol-1-yl)propan-2-ones as inhibitors of human cytosolic phospholipase A2alpha: synthesis and properties of bioisosteric benzimidazole, benzotriazole and indazole analogues.
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Title: Study of 5-nitroindazoles' anti-Trypanosoma cruzi mode of action: electrochemical behaviour and ESR spectroscopic studies.
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Title: Selective P2X(7) receptor antagonists for chronic inflammation and pain.
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Title: 2-(6-Phenyl-1H-indazol-3-yl)-1H-benzo[d]imidazoles: design and synthesis of a potent and isoform selective PKC-zeta inhibitor.
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Title: Structure-activity relationship (SAR): effort towards blocking N-glucuronidation of indazoles (PF-03376056) by human UGT1A enzymes.
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Title: Inhibitory Effects of the Ruthenium Complex KP1019 in Models of Mammary Cancer Cell Migration and Invasion.
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Title: Fragment-based discovery of inhibitors of protein kinase B.
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Title: Targeted treatment of imatinib-resistant chronic myeloid leukemia: Focus on dasatinib.
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Title: Thermodynamic characterization of pyrazole and azaindole derivatives binding to p38 mitogen-activated protein kinase using Biacore T100 technology and van't Hoff analysis.
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Title: Synthesis, spectral analysis, antibacterial and antifungal activities of some 4,6-diaryl-4,5-dihydro-3-hydroxy-2[H]-indazole-a novel fused indazole derivative.
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Title: Design and synthesis of potent and selective azaindole-based Rho kinase (ROCK) inhibitors.
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Title: 3-(4-Pyrid-yl)-4,5-dihydro-1H-benzo[g]indazole.
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Title: Structures of human cytochrome P-450 2E1. Insights into the binding of inhibitors and both small molecular weight and fatty acid substrates.
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Title: GdCl(3) catalysed Grieco condensation: a facile approach for the synthesis of novel pyrimidine and annulated pyrimidine fused indazole derivatives in single pot under mild conditions and their anti-microbial activity.
Journal: European journal of medicinal chemistry 20080201
Title: 7-fluoroindazoles as potent and selective inhibitors of factor Xa.
Journal: Journal of medicinal chemistry 20080124
Title: Drug design with Cdc7 kinase: a potential novel cancer therapy target.
Journal: Drug design, development and therapy 20080101
Title: Dibromidotetra-kis(1H-indazole-κN)copper(II).
Journal: Acta crystallographica. Section E, Structure reports online 20080101
Title: A planar carboxylate-rich tetraironII complex and its conversion to linear triironII and paddlewheel diironII complexes.
Journal: Inorganic chemistry 20071210
Title: Synthesis and evaluation of novel 17-indazole androstene derivatives designed as CYP17 inhibitors.
Journal: Steroids 20071201
Title: Cardiovascular effects of a novel potent and highly selective azaindole-based inhibitor of Rho-kinase.
Journal: British journal of pharmacology 20071201
Title: Electrophilic chemistry of thia-PAHs: stable carbocations (NMR and DFT), S-alkylated onium salts, model electrophilic substitutions (nitration and bromination), and mutagenicity assay.
Journal: The Journal of organic chemistry 20071026
Title: Addition reactions and redox esterifications of carbonyl compounds by N-heterocyclic carbenes of indazole.
Journal: Organic letters 20070830
Title: Luminescent platinum(II) complexes containing isoquinolinyl indazolate ligands: synthetic reaction pathway and photophysical properties.
Journal: Inorganic chemistry 20070820
Title: In vitro structure-activity relationship and in vivo characterization of 1-(aryl)-3-(4-(amino)benzyl)urea transient receptor potential vanilloid 1 antagonists.
Journal: Journal of medicinal chemistry 20070726
Title: Alpha-methylation at benzylic fragment of N-aryl-N'-benzyl ureas provides TRPV1 antagonists with better pharmacokinetic properties and higher efficacy in inflammatory pain model.
Journal: Bioorganic & medicinal chemistry letters 20070715
Title: A general modular method of azaindole and thienopyrrole synthesis via Pd-catalyzed tandem couplings of gem-dichloroolefins.
Journal: The Journal of organic chemistry 20070706
Title: Synthesis and antifungal activities of new fluconazole analogues with azaheterocycle moiety.
Journal: Bioorganic & medicinal chemistry letters 20070701
Title: Organometallic methods for the synthesis and functionalization of azaindoles.
Journal: Chemical Society reviews 20070701
Title: QSAR analysis of indazole estrogens as selective beta-estrogen receptor ligands: rationalization of physicochemical properties.
Journal: Medicinal chemistry (Shariqah (United Arab Emirates)) 20070701
Title: Discovery of novel indazole-linked triazoles as antifungal agents.
Journal: Bioorganic & medicinal chemistry letters 20070615
Title: Osmium NAMI-A analogues: synthesis, structural and spectroscopic characterization, and antiproliferative properties.
Journal: Inorganic chemistry 20070611
Title: 4-substituted indazoles as new inhibitors of neuronal nitric oxide synthase.
Journal: Bioorganic & medicinal chemistry letters 20070601
Title: Structure-activity relationships for NAMI-A-type complexes (HL)[trans-RuCl4L(S-dmso)ruthenate(III)] (L = imidazole, indazole, 1,2,4-triazole, 4-amino-1,2,4-triazole, and 1-methyl-1,2,4-triazole): aquation, redox properties, protein binding, and antiproliferative activity.
Journal: Journal of medicinal chemistry 20070503
Title: Pyrazole complexes as anion receptors: effects of changing the metal, the pyrazole substitution pattern, and the number of pyrazole ligands.
Journal: Inorganic chemistry 20070416
Title: Design and synthesis of pyridine-pyrazolopyridine-based inhibitors of protein kinase B/Akt.
Journal: Bioorganic & medicinal chemistry 20070315
Title: Development of dihydropyridone indazole amides as selective Rho-kinase inhibitors.
Journal: Journal of medicinal chemistry 20070111
Title: Design and synthesis of Rho kinase inhibitors (II).
Journal: Bioorganic & medicinal chemistry 20070101
Title: Synthesis of a library of 2-alkyl-3-alkyloxy-2H-indazole-6-carboxamides.
Journal: Journal of combinatorial chemistry 20070101
Title: DNA-metallodrugs interactions signaled by electrochemical biosensors: an overview.
Journal: Bioinorganic chemistry and applications 20070101
Title: 3-(Indol-2-yl)indazoles as Chek1 kinase inhibitors: Optimization of potency and selectivity via substitution at C6.
Journal: Bioorganic & medicinal chemistry letters 20061201
Title: Synthesis of heterocyclic compounds via nucleophilic aroylation catalyzed by imidazolidenyl carbene.
Journal: Chemical & pharmaceutical bulletin 20061201
Title: Metabolism-dependent mutagenicity of a compound containing a piperazinyl indazole motif: Role of a novel p450-mediated metabolic reaction involving a putative oxaziridine intermediate.
Journal: Chemical research in toxicology 20061001
Title: On the illusive nature of o-formylazobenzenes: exploiting the nucleophilicity of the azo group for cyclization to indazole derivatives.
Journal: The Journal of organic chemistry 20060929
Title: Synthesis of 2H-indazoles via Lewis acid promoted cyclization of 2-(phenylazo)benzonitriles.
Journal: The Journal of organic chemistry 20060818
Title: Structure-activity studies of a novel series of 5,6-fused heteroaromatic ureas as TRPV1 antagonists.
Journal: Bioorganic & medicinal chemistry 20060715
Title: Regioselective protection at N-2 and derivatization at C-3 of indazoles.
Journal: The Journal of organic chemistry 20060707
Title: Redox behavior of tumor-inhibiting ruthenium(III) complexes and effects of physiological reductants on their binding to GMP.
Journal: Dalton transactions (Cambridge, England : 2003) 20060414
Title: Prediction of the binding mode between BMS-378806 and HIV-1 gp120 by docking and molecular dynamics simulation.
Journal: Biochimica et biophysica acta 20060401
Title: Identification of a buried pocket for potent and selective inhibition of Chk1: prediction and verification.
Journal: Bioorganic & medicinal chemistry 20060315
Title: Platinum group metallodrug-protein binding studies by capillary electrophoresis - inductively coupled plasma-mass spectrometry: a further insight into the reactivity of a novel antitumor ruthenium(III) complex toward human serum proteins.
Journal: Electrophoresis 20060301
Title: Synthesis and biological evaluation of novel heterocyclic quinones as inhibitors of the dual specificity protein phosphatase CDC25C.
Journal: Bioorganic & medicinal chemistry letters 20060101
Title: Recent advances in the solid-phase combinatorial synthetic strategies for the quinoxaline, quinazoline and benzimidazole based privileged structures.
Journal: Mini reviews in medicinal chemistry 20060101
Title: Relaxant effects of the soluble guanylate cyclase activator and NO sensitizer YC-1 in piglet pulmonary arteries.
Journal: Biology of the neonate 20060101
Title: Inhibitive properties and surface morphology of a group of heterocyclic diazoles as inhibitors for acidic iron corrosion.
Journal: Langmuir : the ACS journal of surfaces and colloids 20051220
Title: Excited state tautomerization of azaindole.
Journal: Organic & biomolecular chemistry 20051021
Title: YC-1 suppresses constitutive nuclear factor-kappaB activation and induces apoptosis in human prostate cancer cells.
Journal: Molecular cancer therapeutics 20051001
Title: Pharmacological properties of indazole derivatives: recent developments.
Journal: Mini reviews in medicinal chemistry 20051001
Title: Tuning of redox properties for the design of ruthenium anticancer drugs: part 2. Syntheses, crystal structures, and electrochemistry of potentially antitumor [Ru III/II Cl6-n(Azole)n]z(n = 3, 4, 6) complexes.
Journal: Inorganic chemistry 20050919
Title: High resolution electronic spectra of 7-azaindole and its Ar atom van der Waals complex.
Journal: The Journal of chemical physics 20050901
Title: Spatial orientation of the antagonist granisetron in the ligand-binding site of the 5-HT3 receptor.
Journal: Molecular pharmacology 20050801
Title: Isomeric [RuCl2(dmso)2(indazole)2] complexes: ruthenium(II)-mediated coupling reaction of acetonitrile with 1H-indazole.
Journal: Dalton transactions (Cambridge, England : 2003) 20050721
Title: Comparative binding of antitumor indazolium [trans-tetrachlorobis(1H-indazole)ruthenate(III)] to serum transport proteins assayed by capillary zone electrophoresis.
Journal: Analytical biochemistry 20050615
Title: Modification and structure-activity relationship of a small molecule HIV-1 inhibitor targeting the viral envelope glycoprotein gp120.
Journal: Organic & biomolecular chemistry 20050507
Title: Metabolism of the calmodulin antagonist DY-9760e in animals and humans.
Journal: Xenobiotica; the fate of foreign compounds in biological systems 20050501
Title: Redox-active antineoplastic ruthenium complexes with indazole: correlation of in vitro potency and reduction potential.
Journal: Journal of medicinal chemistry 20050421
Title: Indazole estrogens: highly selective ligands for the estrogen receptor beta.
Journal: Journal of medicinal chemistry 20050224
Title: Dopamine D1/D5 receptor antagonists with improved pharmacokinetics: design, synthesis, and biological evaluation of phenol bioisosteric analogues of benzazepine D1/D5 antagonists.
Journal: Journal of medicinal chemistry 20050210
Title: Claimed 2,1-benzisoxazoles are indazalones.
Journal: The Journal of organic chemistry 20050204
Title: From model compounds to protein binding: syntheses, characterizations and fluorescence studies of [RuII(bipy)(terpy)L]2+ complexes (bipy = 2,2'-bipyridine; terpy = 2,2':6',2''-terpyridine; L = imidazole, pyrazole and derivatives, cytochrome c).
Journal: Dalton transactions (Cambridge, England : 2003) 20050121
Title: Reactions of potent antitumor complex trans-[Ru(III)Cl4(indazole)2]- with a DNA-relevant nucleobase and thioethers: insight into biological action.
Journal: Inorganic chemistry 20050110
Title: Electrospray ionization mass spectrometric studies of nucleophilic carbenes derived from pyrazolium and indazolium carboxylates.
Journal: Rapid communications in mass spectrometry : RCM 20050101
Title: Design, synthesis and evaluation of bicyclic benzamides as novel 5-HT1F receptor agonists.
Journal: Bioorganic & medicinal chemistry letters 20041220
Title: The indazole derivative YD-3 inhibits thrombin-induced vascular smooth muscle cell proliferation and attenuates intimal thickening after balloon injury.
Journal: Thrombosis and haemostasis 20041201
Title: Tuning of redox potentials for the design of ruthenium anticancer drugs -- an electrochemical study of [trans-RuCl(4)L(DMSO)](-) and [trans-RuCl(4)L(2)](-) complexes, where L = imidazole, 1,2,4-triazole, indazole.
Journal: Inorganic chemistry 20041101
Title: A flexible, palladium-catalyzed indole and azaindole synthesis by direct annulation of chloroanilines and chloroaminopyridines with ketones.
Journal: Angewandte Chemie (International ed. in English) 20040827
Title: The effect of a newly synthesized indazole compound, TAS-3-124, on experimental autoimmune disease.
Journal: Biological & pharmaceutical bulletin 20040801
Title: Design, synthesis and structure-activity relationship studies of novel indazole analogues as DNA gyrase inhibitors with Gram-positive antibacterial activity.
Journal: Bioorganic & medicinal chemistry letters 20040607
Title: New antithrombotics with an indazole structure.
Journal: Archiv der Pharmazie 20040601
Title: Design and synthesis of Rho kinase inhibitors (I).
Journal: Bioorganic & medicinal chemistry 20040501
Title: The isoindazole nucleus as a donor in fullerene-based dyads. Evidence for electron transfer.
Journal: The Journal of organic chemistry 20040416
Title: Inhibition studies with rationally designed inhibitors of the human low molecular weight protein tyrosine phosphatase.
Journal: Bioorganic & medicinal chemistry 20040415
Title: A new alkaloid and its artificial derivative with an indazole ring from Nigella glandulifera.
Journal: Chemical & pharmaceutical bulletin 20040401
Title: Regioselective synthesis of indazole N1- and N2-(beta-D-ribonucleosides).
Journal: Nucleosides, nucleotides & nucleic acids 20040101
Title: Possible mechanism(s) for relaxant effect of aqueous and macerated extracts from Nigella sativa on tracheal chains of guinea pig.
Journal: BMC pharmacology 20040101
Title: Soluble guanylyl cyclase activator YC-1 inhibits human neutrophil functions through a cGMP-independent but cAMP-dependent pathway.
Journal: Molecular pharmacology 20031201
Title: Initial evaluation of novel selective ligands for imidazoline(2) receptors in rat whole brain.
Journal: Annals of the New York Academy of Sciences 20031201
Title: Inhibitory effects and spectral interactions of isomeric methoxyindazoles on recombinant nitric oxide synthases.
Journal: Nitric oxide : biology and chemistry 20030901
Title: A parallel synthesis demonstration library of tri-substituted indazoles containing new antimutagenic/antioxidant hits related to benzydamine.
Journal: Combinatorial chemistry & high throughput screening 20030801
Title: Syntheses and antiproliferative activities of rebeccamycin analogues bearing two 7-azaindole moieties.
Journal: Bioorganic & medicinal chemistry 20030306
Title: Discovery of an orally efficacious inhibitor of coagulation factor Xa which incorporates a neutral P1 ligand.
Journal: Journal of medicinal chemistry 20030227
Title: Syntheses and antiproliferative activities of 7-azarebeccamycin analogues bearing one 7-azaindole moiety.
Journal: Journal of medicinal chemistry 20030213
Title: Rebeccamycin analogues as anti-cancer agents.
Journal: European journal of medicinal chemistry 20030201
Title: Indazole inhibition of cystic fibrosis transmembrane conductance regulator Cl(-) channels in rat epididymal epithelial cells.
Journal: Biology of reproduction 20021201
Title: New N-pyridinyl(methyl)-indole-2- and 3-(alkyl)carboxamides and derivatives acting as systemic and topical inflammation inhibitors.
Journal: Journal of enzyme inhibition and medicinal chemistry 20021201
Title: Deciphering the mechanistic dichotomy in the cyclization of 1-(2-ethynylphenyl)-3,3-dialkyltriazenes: competition between pericyclic and pseudocoarctate pathways.
Journal: Journal of the American Chemical Society 20021113
Title: Mechanism of lonidamine inhibition of the CFTR chloride channel.
Journal: British journal of pharmacology 20021101
Title: 7-Methoxy-1H-indazole, a new inhibitor of neuronal nitric oxide synthase.
Journal: Acta crystallographica. Section C, Crystal structure communications 20021101
Title: Cyclization of 1-(2-alkynylphenyl)-3,3-dialkyltriazenes: a convenient, high-yield synthesis of substituted cinnolines and isoindazoles.
Journal: The Journal of organic chemistry 20020906
Title: Fused azaindole derivatives: molecular design, synthesis and in vitro pharmacology leading to the preferential dopamine D3 receptor agonist FAUC 725.
Journal: Bioorganic & medicinal chemistry letters 20020902
Title: Male fertility: core chemical structure in pharmacological research.
Journal: Contraception 20020401
Title: Two unusual, competitive mechanisms for (2-ethynylphenyl)triazene cyclization: pseudocoarctate versus pericyclic reactivity.
Journal: Journal of the American Chemical Society 20020227
Title: Inhibition of superoxide anion generation by YC-1 in rat neutrophils through cyclic GMP-dependent and -independent mechanisms.
Journal: Biochemical pharmacology 20020215
Title: Azole. 47. Uber 3-thiomorpholino- und 3-(4-methylpiperazino)-5-nitroindazole.
Journal: Acta crystallographica. Section C, Crystal structure communications 20011001
Title: Rationally based efficacy tuning of selective dopamine d4 receptor ligands leading to the complete antagonist 2-[4-(4-chlorophenyl)piperazin-1-ylmethyl]pyrazolo[1,5-a]pyridine (FAUC 213).
Journal: Journal of medicinal chemistry 20010816
Title: Investigations into the interaction between tumor-inhibiting ruthenium(III) complexes and nucleotides by capillary electrophoresis.
Journal: Journal of chromatography. B, Biomedical sciences and applications 20010805
Title: Studies on synthetic approaches to 1H- and 2H-indazolyl derivatives.
Journal: The Journal of organic chemistry 20010615
Title: Topoisomerase II poisoning by indazole and imidazole complexes of ruthenium.
Journal: Journal of biosciences 20010601
Title: The design of competitive, small-molecule inhibitors of coagulation factor Xa.
Journal: Current topics in medicinal chemistry 20010601
Title: Inhibition of neuronal nitric oxide synthase by 7-methoxyindazole and related substituted indazoles.
Journal: Bioorganic & medicinal chemistry letters 20010507
Title: Surface enhanced Raman spectroscopic studies of 1H-indazole on silver sols.
Journal: Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy 20010501
Title: Biophysical analysis of natural, double-helical DNA modified by anticancer heterocyclic complexes of ruthenium(III) in cell-free media.
Journal: Journal of biological inorganic chemistry : JBIC : a publication of the Society of Biological Inorganic Chemistry 20010401
Title: Discovery and optimization of a novel series of thrombin receptor (par-1) antagonists: potent, selective peptide mimetics based on indole and indazole templates.
Journal: Journal of medicinal chemistry 20010329
Title: Hydrolysis of the tumor-inhibiting ruthenium(III) complexes HIm trans-[RuCl4(im)2] and HInd trans-[RuCl4(ind)2] investigated by means of HPCE and HPLC-MS.
Journal: Journal of biological inorganic chemistry : JBIC : a publication of the Society of Biological Inorganic Chemistry 20010301
Title: Synthesis and biological evaluation of novel pyrazoles and indazoles as activators of the nitric oxide receptor, soluble guanylate cyclase.
Journal: Journal of medicinal chemistry 20010104
Title: Synthesis and in vitro LTD4 antagonist activity of bicyclic and monocyclic cyclopentylurethane and cyclopentylacetamide N-arylsulfonyl amides.
Journal: Journal of medicinal chemistry 19900901
