Title: Design, facile synthesis, and antibacterial activity of hybrid 1,3,4-thiadiazole-1,3,5-triazine derivatives tethered via -S- bridge.
Journal: Chemical biology & drug design20121001
Title: Cell death features induced in Leishmania major by 1,3,4-thiadiazole derivatives.
Journal: Experimental parasitology20121001
Title: Novel immunomodulatory function of 1,3,4-thiadiazole derivatives with leishmanicidal activity.
Journal: The Journal of antimicrobial chemotherapy20120801
Title: Synthesis of new 1,3,4-thiadiazole and 1,2,3,4-oxathiadiazole derivatives from carbohydrate precursors and study of their effect on tyrosinase enzyme.
Journal: Molecules (Basel, Switzerland)20120711
Title: Synthesis and cytotoxicity of 3,4-disubstituted-5-(3,4,5-trimethoxyphenyl)-4H-1,2,4-triazoles and novel 5,6-dihydro-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole derivatives bearing 3,4,5-trimethoxyphenyl moiety.
Journal: Bioorganic & medicinal chemistry letters20120701
Title: Design, synthesis and preliminary bioactivity studies of 1,3,4-thiadiazole hydroxamic acid derivatives as novel histone deacetylase inhibitors.
Journal: Bioorganic & medicinal chemistry20120615
Title: Bis(2-amino-5-methyl-1,3,4-thia-diazole-κN(3))dichloridocobalt(II).
Journal: Acta crystallographica. Section E, Structure reports online20120601
Title: 2,5-Bis[(3-chloro-benz-yl)sulfan-yl]-1,3,4-thia-diazole.
Journal: Acta crystallographica. Section E, Structure reports online20120601
Title: Synthesis and biological evaluation of isoxazolo[4,5-d]pyridazin-4-(5H)-one analogues as potent anti-inflammatory agents.
Journal: Bioorganic & medicinal chemistry20120501
Title: Synthesis of novel nalidixic acid-based 1,3,4-thiadiazole and 1,3,4-oxadiazole derivatives as potent antibacterial agents.
Journal: Chemical biology & drug design20120401
Title: 1,3,4-Thiadiazole derivatives as selective inhibitors of iNOS versus nNOS: Synthesis and structure-activity dependence.
Journal: European journal of medicinal chemistry20120401
Title: Aqua-bis-[2,5-bis-(pyridin-2-yl)-1,3,4-thia-diazole-κ(2)N(2),N(3)](trifluoro-methane-sulfonato-κO)copper(II) trifluoro-methane-sulfonate.
Journal: Acta crystallographica. Section E, Structure reports online20120401
Title: 4-Bromo-benzoic acid-6-(4-bromo-phen-yl)-3-methyl-1,2,4-triazolo[3,4-b][1,3,4]thia-diazole (1/1).
Journal: Acta crystallographica. Section E, Structure reports online20120401
Title: 5-({3-[(5-Amino-1,3,4-thia-diazol-2-yl)sulfanylmeth-yl]benz-yl}sulfan-yl)-1,3,4-thia-diazol-2-amine.
Journal: Acta crystallographica. Section E, Structure reports online20120401
Title: Calix[4]arene based 1,3,4-oxadiazole and thiadiazole derivatives: design, synthesis, and biological evaluation.
Journal: Organic & biomolecular chemistry20120307
Title: New heterocyclic compounds from 1,2,4-triazole and 1,3,4-thiadiazole class bearing diphenylsulfone moieties. Synthesis, characterization and antimicrobial activity evaluation.
Journal: European journal of medicinal chemistry20120301
Title: Novel imidazo[2,1-b][1,3,4]thiadiazole carrying rhodanine-3-acetic acid as potential antitubercular agents.
Journal: Bioorganic & medicinal chemistry letters20120301
Title: 2-(4-Methyl-phen-yl)-5-[({[5-(4-methyl-phen-yl)-1,3,4-thia-diazol-2-yl]sulfan-yl}meth-yl)sulfan-yl]-1,3,4-thia-diazole.
Journal: Acta crystallographica. Section E, Structure reports online20120301
Title: Synthesis of novel sulfonamide-1,2,4-triazoles, 1,3,4-thiadiazoles and 1,3,4-oxadiazoles, as potential antibacterial and antifungal agents. Biological evaluation and conformational analysis studies.
Journal: Bioorganic & medicinal chemistry20120215
Title: Synthesis and evaluation of anti-inflammatory, analgesic, ulcerogenic and lipid peroxidation properties of new 2-(4-isobutylphenyl)propanoic acid derivatives.
Journal: Journal of enzyme inhibition and medicinal chemistry20120201
Title: Synthesis, biological evaluation, and molecular docking studies of cinnamic acyl 1,3,4-thiadiazole amide derivatives as novel antitubulin agents.
Journal: Bioorganic & medicinal chemistry20120201
Title: N-(5-Eth-oxy-1,3,4-thia-diazol-2-yl)benzamide.
Journal: Acta crystallographica. Section E, Structure reports online20120201
Title: Synthesis and antimicrobial studies of some novel bis-[1,3,4]thiadiazole and bis-thiazole pendant to thieno[2,3-b]thiophene moiety.
Journal: International journal of molecular sciences20120101
Title: Design and Microwave-assisted Synthesis of 1,3,4-Oxadiazole Derivatives for Analgesic and Anti-inflammatory Activity.
Journal: Journal of young pharmacists : JYP20120101
Title: Synthesis and antiepileptic activity of some novel semicarbazones containing 1,3,4-thiadiazole and quinazoline ring.
Journal: Acta poloniae pharmaceutica20120101
Title: Synthesis and evaluation of the anti-microbial activity of new heterocycles containing the 1,3,4-thiadiazole moiety.
Journal: Molecules (Basel, Switzerland)20111215
Title: Synthesis, biological evaluation and molecular docking studies of 1,3,4-thiadiazole derivatives containing 1,4-benzodioxan as potential antitumor agents.
Journal: Bioorganic & medicinal chemistry letters20111015
Title: Pro-oxidant and antiproliferative effects of the 1,3,4-thiadiazole-based Schiff base and its metal complexes.
Journal: Drug and chemical toxicology20111001
Title: Synthesis and anticancer evaluation of novel 2-cyclopropylimidazo[2,1-b][1,3,4]-thiadiazole derivatives.
Journal: European journal of medicinal chemistry20110901
Title: (E)-4-Phenyl-butan-2-one oxime.
Journal: Acta crystallographica. Section E, Structure reports online20110901
Title: The use of umbelliferone in the synthesis of new heterocyclic compounds.
Journal: Molecules (Basel, Switzerland)20110810
Title: Discovery of adamantyl heterocyclic ketones as potent 11β-hydroxysteroid dehydrogenase type 1 inhibitors.
Journal: ChemMedChem20110801
Title: trans-Diaqua-bis-[2,5-bis-(pyridin-2-yl)-1,3,4-thia-diazole]nickel(II) bis-(tetra-fluoridoborate).
Journal: Acta crystallographica. Section E, Structure reports online20110801
Title: Synthesis and biological activities on metal complexes of 2,5-diamino-1,3,4-thiadiazole derived from semicarbazide hydrochloride.
Journal: Molecules (Basel, Switzerland)20110712
Title: Synthesis of novel 1,2,4-oxadiazoles and analogues as potential anticancer agents.
Journal: European journal of medicinal chemistry20110701
Title: trans-Diaqua-bis-[2,5-bis-(pyridin-2-yl)-1,3,4-thia-diazole]cobalt(II) bis-(tetra-fluoridoborate).
Journal: Acta crystallographica. Section E, Structure reports online20110701
Title: Experimental and theoretical study on molecular aggregation and its effect on the photo-physical properties of the mesogenic bi-1,3,4-thiadiazole derivative.
Journal: Physical chemistry chemical physics : PCCP20110528
Title: NMR QSAR model for the analysis of 4-(5-arylamino-1,3,4-thiadiazol-2-yl)benzene-1,3-diols.
Journal: Archiv der Pharmazie20110501
Title: 3-Methyl-6-trichloro-methyl-1,2,4-triazolo[3,4-b][1,3,4]thia-diazole.
Journal: Acta crystallographica. Section E, Structure reports online20110501
Title: Synthesis, singlet oxygen photogeneration and DNA photocleavage of porphyrins with nitrogen heterocycle tails.
Journal: Molecules (Basel, Switzerland)20110426
Title: One-pot synthesis and anticancer studies of 2-arylamino-5-aryl-1,3,4-thiadiazoles.
Journal: Bioorganic & medicinal chemistry letters20110415
Title: Synthesis of 5-amino-1,3,4-thiadiazole-2-sulphonamide derivatives and their inhibition effects on human carbonic anhydrase isozymes.
Journal: Journal of enzyme inhibition and medicinal chemistry20110401
Title: Novel highly emissive non-proteinogenic amino acids: synthesis of 1,3,4-thiadiazolyl asparagines and evaluation as fluorimetric chemosensors for biologically relevant transition metal cations.
Journal: Amino acids20110401
Title: Synthesis and insecticidal activities of novel 1,3,4-thiadiazole 5-fluorouracil acetamides derivatives: an RNA interference insecticide.
Journal: Nucleosides, nucleotides & nucleic acids20110401
Title: Synthesis and antileishmanial activity of 5-(5-nitroaryl)-2-substituted-thio-1,3,4-thiadiazoles.
Journal: Journal of enzyme inhibition and medicinal chemistry20110201
Title: 2-Isobutyl-6-phenyl-imidazo[2,1-b][1,3,4]thia-diazole.
Journal: Acta crystallographica. Section E, Structure reports online20110201
Title: 1-(4-Chloro-phen-yl)-3-{5-[(E)-2-phenyl-ethen-yl]-1,3,4-thia-diazol-2-yl}urea.
Journal: Acta crystallographica. Section E, Structure reports online20110201
Title: Spectroscopic studies of intramolecular proton transfer in 2-(4-fluorophenylamino)-5-(2,4-dihydroxybenzeno)-1,3,4-thiadiazole.
Journal: Journal of fluorescence20110101
Title: Synthesis of new functionalized 3-substituted [1,2,4]triazolo [4,3-a]pyrimidine derivatives: potential antihypertensive agents.
Journal: Acta poloniae pharmaceutica20110101
Title: 5-[(4-Meth-oxy-benz-yl)sulfan-yl]-2-methyl-1,3,4-thia-diazole.
Journal: Acta crystallographica. Section E, Structure reports online20110101
Title: 2-Methyl-5-[(3-methyl-4-nitro-benz-yl)sulfan-yl]-1,3,4-thia-diazole.
Journal: Acta crystallographica. Section E, Structure reports online20110101
Title: 6-(4-Chloro-phen-yl)-2-isobutyl-imidazo[2,1-b][1,3,4]thia-diazole.
Journal: Acta crystallographica. Section E, Structure reports online20110101
Title: Inorganic base-catalyzed formation of antivirally active N-substituted benzamides from α-amido sulfones and N-nucleophile.
Journal: Chemistry Central journal20110101
Title: Antidepressant potential of nitrogen-containing heterocyclic moieties: An updated review.
Journal: Journal of pharmacy & bioallied sciences20110101
Title: Cytotoxicity of new 5-phenyl-4,5-dihydro-1,3,4-thiadiazole analogues.
Journal: Chemical & pharmaceutical bulletin20110101
Title: Synthesis and antimicrobial activity of pyrrolyl/pyrazolyl arylaminosulfonylmethyl 1,3,4-oxadiazoles, 1,3,4-thiadiazoles and 1,2,4-triazoles.
Journal: Chemical & pharmaceutical bulletin20110101
Title: Metal-based biologically active compounds: synthesis, spectral, and antimicrobial studies of cobalt, nickel, copper, and zinc complexes of triazole-derived schiff bases.
Journal: Bioinorganic chemistry and applications20110101
Title: Bis[(5-phenyl-1,3,4-thia-diazol-2-yl)sulfan-yl]methane.
Journal: Acta crystallographica. Section E, Structure reports online20101201
Title: Cyclization of some carbothioamide derivatives containing antipyrine and triazole moieties and investigation of their antimicrobial activities.
Journal: European journal of medicinal chemistry20101101
Title: Synthesis, antioxidant activities and urease inhibition of some new 1,2,4-triazole and 1,3,4-thiadiazole derivatives.
Journal: European journal of medicinal chemistry20101101
Title: 3-Ethyl-6-[3-(4-fluoro-phen-yl)-1H-pyrazol-4-yl]-1,2,4-triazolo[3,4-b][1,3,4]thia-diazole.
Journal: Acta crystallographica. Section E, Structure reports online20101101
Title: (14)N NQR, (1)H NMR and DFT/QTAIM study of hydrogen bonding and polymorphism in selected solid 1,3,4-thiadiazole derivatives.
Journal: Physical chemistry chemical physics : PCCP20101028
Title: Synthesis and anticancer activity of 5-(3-indolyl)-1,3,4-thiadiazoles.
Journal: European journal of medicinal chemistry20101001
Title: Investigation of the toxic functional group of cephalosporins by zebrafish embryo toxicity test.
Journal: Archiv der Pharmazie20101001
Title: Urea-type ligand-modified CdSe quantum dots as a fluorescence 'turn-on' sensor for CO3(2-) anions.
Journal: Photochemical & photobiological sciences : Official journal of the European Photochemistry Association and the European Society for Photobiology20100924
Title: Synthesis and evaluation of anti-Toxoplasma gondii and antimicrobial activities of thiosemicarbazides, 4-thiazolidinones and 1,3,4-thiadiazoles.
Journal: European journal of medicinal chemistry20100901
Title: Synthesis and bioassay of aminosulfonyl-1,3,4-oxadiazoles and their interconversion to 1,3,4-thiadiazoles.
Journal: European journal of medicinal chemistry20100901
Title: Synthesis and pharmacological evaluation of condensed heterocyclic 6-substituted 1,2,4-triazolo-[3,4-b]-1,3,4-thiadiazole and 1,3,4-oxadiazole derivatives of isoniazid.
Journal: Bioorganic & medicinal chemistry letters20100815
Title: Design and synthesis of thiadiazoles and thiazoles targeting the Bcr-Abl T315I mutant: from docking false positives to ATP-noncompetitive inhibitors.
Journal: ChemMedChem20100802
Title: Homology modeling and QSAR analysis of 1,3,4-thiadiazole and 1,3,4-triazole derivatives as carbonic anhydrase inhibitors.
Journal: Indian journal of biochemistry & biophysics20100801
Title: 2-(4-Fluoro-benzyl-idene)-N-(4-meth-oxy-benzylidene)-1,3,4-thia-diazol-2-amine.
Journal: Acta crystallographica. Section E, Structure reports online20100701
Title: Comparative studies of mercapto thiadiazoles self-assembled on gold nanoparticle as ionophores for Cu(II) carbon paste sensors.
Journal: Analytica chimica acta20100430
Title: Synthesis and anti-inflammatory evaluation of some condensed [4-(3,4-dimethylphenyl)-1(2H)-oxo-phthalazin-2-yl]acetic acid hydrazide.
Journal: European journal of medicinal chemistry20100401
Title: Novel C-aryl glucoside SGLT2 inhibitors as potential antidiabetic agents: 1,3,4-Thiadiazolylmethylphenyl glucoside congeners.
Journal: Bioorganic & medicinal chemistry20100315
Title: Synthesis and antimicrobial activity evaluation of new 1,2,4-triazoles and 1,3,4-thiadiazoles bearing imidazo[2,1-b]thiazole moiety.
Journal: European journal of medicinal chemistry20100101
Title: Synthesis and antimicrobial activity of 3-(1,3,4-Oxadiazol-2-yl)quinazolin-4(3H)-ones.
Journal: Scientia pharmaceutica20100101
Title: Synthesis and Antibacterial and Antifungal Studies of Novel Nitrogen Containing Heterocycles from 5-Ethylpyridin-2-ethanol.
Journal: Indian journal of pharmaceutical sciences20100101
Title: Vanadium-induced formation of thiadiazole and thiazoline compounds. Mononuclear and dinuclear oxovanadium(v) complexes with open-chain and cyclized thiosemicarbazone ligands.
Journal: Dalton transactions (Cambridge, England : 2003)20091128
Title: 2-Substituted-5-nitroheterocycles: in vitro anti-Helicobacter pylori activity and structure-activity relationship study.
Journal: Medicinal chemistry (Shariqah (United Arab Emirates))20091101
Title: N,N-Bis(2,6-difluoro-benz-yl)-1,3,4-thia-diazol-2-amine.
Journal: Acta crystallographica. Section E, Structure reports online20090901
Title: Methylsulfonylpyrazolyl oxadiazoles and thiadiazoles as potent, orally bioavailable cannabinoid-1 receptor antagonists for the treatment of obesity.
Journal: Future medicinal chemistry20090801
Title: Synthesis and biological activity of some new 1,3,4-thiadiazole and 1,2,4-triazole compounds containing a phenylalanine moiety.
Journal: Molecules (Basel, Switzerland)20090716
Title: A one-dimensional cadmium(II) complex supported by a sulfur-nitro-gen mixed-donor ligand.
Journal: Acta crystallographica. Section E, Structure reports online20090701
Title: 5-(3-Fluoro-phen-yl)-1,3,4-thia-diazol-2-amine.
Journal: Acta crystallographica. Section E, Structure reports online20090601
Title: 5-(2-Methyl-phen-yl)-1,3,4-thia-diazol-2-amine.
Journal: Acta crystallographica. Section E, Structure reports online20090501
Title: Nitroimidazolyl-1,3,4-thiadiazole-based anti-leishmanial agents: synthesis and in vitro biological evaluation.
Journal: European journal of medicinal chemistry20090401
Title: Selective leishmanicidal effect of 1,3,4-thiadiazole derivatives and possible mechanism of action against Leishmania species.
Journal: Experimental parasitology20090401
Title: Two bicyclic dinuclear complexes generated from 3,3'-[1,3,4-thiadiazole-2,5-diyldi(thiomethylene)]dibenzoic acid (L) and dimethylformamide (DMF): [Cu(L)(DMF)]2and [Zn(L)(DMF)]2.
Journal: Acta crystallographica. Section C, Crystal structure communications20090201
Title: Synthesis of 1,3,4-thiadiazole derivatives as aminopeptidase N inhibitors.
Journal: Die Pharmazie20090201
Title: 2-Benzoyl-amino-N-[5-(4-bromo-phen-yl)-1,3,4-thia-diazol-2-yl]ethanamide.
Journal: Acta crystallographica. Section E, Structure reports online20090201
Title: Synthesis, cytotoxicity and effects of some 1,2,4-triazole and 1,3,4-thiadiazole derivatives on immunocompetent cells.
Journal: European journal of medicinal chemistry20090101
Title: Ultrasound assisted synthesis of some new 1,3,4-thiadiazole and bi(1,3,4-thiadiazole) derivatives incorporating pyrazolone moiety.
Journal: Ultrasonics sonochemistry20090101
Title: 1-(4-Methyl-benzo-yl)-3-[5-(4-pyrid-yl)-1,3,4-thia-diazol-2-yl]urea.
Journal: Acta crystallographica. Section E, Structure reports online20081201
Title: 3,4,5-Trimethoxy-benzohydrazidium chloride.
Journal: Acta crystallographica. Section E, Structure reports online20081201
Title: N-[4-Acetyl-5-(3-methoxy-phen-yl)-4,5-dihydro-1,3,4-thia-diazol-2-yl]acetamide.
Journal: Acta crystallographica. Section E, Structure reports online20081101
Title: (2R)-2-Cinnamoylamino-N-[5-(4-methoxy-phen-yl)-1,3,4-thia-diazol-2-yl]propanamide.
Journal: Acta crystallographica. Section E, Structure reports online20081001
Title: (2R)-N-[5-(4-Chloro-phen-yl)-1,3,4-thia-diazol-2-yl]-2-(cinnamoylamino)propanamide.
Journal: Acta crystallographica. Section E, Structure reports online20081001
Title: 6-(4-Methyl-phen-yl)-3-(3,4,5-trimethoxy-phen-yl)-1,2,4-triazolo[3,4-b][1,3,4]thiadiazole.
Journal: Acta crystallographica. Section E, Structure reports online20081001
Title: Synthesis and cytotoxic evaluation of novel dimethyl [1,1'-biphenyl]-2,2'-dicarboxylates bearing 1,3,4-thiadiazole moieties.
Journal: Chemistry & biodiversity20080901
Title: Synthesis and in vitro anti-Helicobacter pylori activity of N-[5-(5-nitro-2-heteroaryl)-1,3,4-thiadiazol-2-yl]thiomorpholines and related compounds.
Journal: European journal of medicinal chemistry20080801
Title: 6-(3-Pyrid-yl)-3-(3,4,5-trimethoxy-phen-yl)-1,2,4-triazolo[3,4-b][1,3,4]thia-diazole.
Journal: Acta crystallographica. Section E, Structure reports online20080801
Title: 6-(2-Methyl-phen-yl)-3-(3,4,5-trimethoxy-phen-yl)-1,2,4-triazolo[3,4-b][1,3,4]thia-diazole.
Journal: Acta crystallographica. Section E, Structure reports online20080801
Title: 3,6-Bis(3,4,5-trimethoxy-phen-yl)-1,2,4-triazolo[3,4-b][1,3,4]thia-diazole.
Journal: Acta crystallographica. Section E, Structure reports online20080801
Title: 6-(4-Pyrid-yl)-3-(3,4,5-trimethoxy-phen-yl)-1,2,4-triazolo[3,4-b][1,3,4]thia-diazole.
Journal: Acta crystallographica. Section E, Structure reports online20080801
Title: Novel aminopeptidase N inhibitors derived from 1,3,4-thiadiazole scaffold.
Journal: Bioorganic & medicinal chemistry20080715
Title: Synthesis and anti-Helicobacter pylori activity of 5-(nitroaryl)-1,3,4-thiadiazoles with certain sulfur containing alkyl side chain.
Journal: Bioorganic & medicinal chemistry letters20080601
Title: 3-[1-(4-Isobutyl-phen-yl)eth-yl]-6-(4-methyl-phen-yl)-1,2,4-triazolo[3,4-b][1,3,4]thia-diazole.
Journal: Acta crystallographica. Section E, Structure reports online20080601
Title: Synthesis and antifungal activity of novel sulfoxide derivatives containing trimethoxyphenyl substituted 1,3,4-thiadiazole and 1,3,4-oxadiazole moiety.
Journal: Bioorganic & medicinal chemistry20080401
Title: Synthesis and antimicrobial activity of new 1,2,4-triazole and 1,3,4-thiadiazole derivatives.
Journal: Journal of enzyme inhibition and medicinal chemistry20080401
Title: 3-(2-Fluoro-phen-yl)-6-(phenoxy-meth-yl)-1,2,4-triazolo[3,4-b][1,3,4]thia-diazole.
Journal: Acta crystallographica. Section E, Structure reports online20080401
Title: Discovery and SAR of 1,3,4-thiadiazole derivatives as potent Abl tyrosine kinase inhibitors and cytodifferentiating agents.
Journal: Bioorganic & medicinal chemistry letters20080201
Title: Some QSAR studies for a group of sulfonamide Schiff base as carbonic anhydrase CA II inhibitors.
Journal: International journal of molecular sciences20080201
Title: 3,3-Dimethyl-1-[5-(1H-1,2,4-triazol-1-yl-meth-yl)-1,3,4-thia-diazol-2-ylsulfan-yl]butan-2-one.
Journal: Acta crystallographica. Section E, Structure reports online20080201
Title: Anti-hepatitis B virus activity of new 1,2,4-triazol-2-yl- and 1,3,4-oxadiazol-2-yl-2-pyridinone derivatives.
Journal: Zeitschrift fur Naturforschung. C, Journal of biosciences20080101
Title: A high throughput serum paraoxonase assay for discovery of small molecule modulators of PON1 activity.
Journal: Current chemical genomics20080101
Title: N-[1-(5-Acetamido-3-acetyl-2-methyl-2,3-dihydro-1,3,4-thia-diazol-2-yl)-2-phenyl-ethyl]acetamide.
Journal: Acta crystallographica. Section E, Structure reports online20080101
Title: Ethyl 5-[6-(furan-2-yl)-1,2,4-triazolo[3,4-b][1,3,4]thia-diazol-3-yl]-2,6-di-methylnicotinate.
Journal: Acta crystallographica. Section E, Structure reports online20080101
Title: Synthesis and Biological Screening of 5-{[(4,6-Disubstituted pyrimidine-2-yl)thio]methyl}-N-phenyl-1,3,4-thiadiazol-2-amines.
Journal: Indian journal of pharmaceutical sciences20080101
Title: Non-carboxylic analogues of naproxen: design, synthesis, and pharmacological evaluation of some 1,3,4-oxadiazole/thiadiazole and 1,2,4-triazole derivatives.
Journal: Archiv der Pharmazie20071101
Title: 1-Acylthiosemicarbazides, 1,2,4-triazole-5(4H)-thiones, 1,3,4-thiadiazoles and hydrazones containing 5-methyl-2-benzoxazolinones: synthesis, analgesic-anti-inflammatory and antimicrobial activities.
Journal: Bioorganic & medicinal chemistry20070901
Title: Evaluation of electronic, lipophilic and membrane affinity effects on antiproliferative activity of 5-substituted-2-(2,4-dihydroxyphenyl)-1,3,4-thiadiazoles against various human cancer cells.
Journal: European journal of medicinal chemistry20070701
Title: Synthesis of some novel heterocyclic compounds derived from diflunisal hydrazide as potential anti-infective and anti-inflammatory agents.
Journal: European journal of medicinal chemistry20070701
Title: Synthesis and biological evaluation of new 3-substituted indole derivatives as potential anti-inflammatory and analgesic agents.
Journal: Bioorganic & medicinal chemistry20070601
Title: Synthesis and antimicrobial activity of some new 1,3,4-thiadiazole and 1,2,4-triazole compounds having a D,L-methionine moiety.
Journal: Molecules (Basel, Switzerland)20070129
Title: Cyclization of thiosemicarbazide derivatives of 5-arylidene-2,4-dioxothiazolidine-3-acetic acids to 1,3,4-thiadiazoles and their pharmacological properties.
Journal: Acta poloniae pharmaceutica20070101
Title: Heterocyclic system containing bridgehead nitrogen atom: synthesis and pharmacological activities of some substituted 1,2,4-triazolo[3,4-b]-1,3,4-thiadiazoles.
Journal: European journal of medicinal chemistry20060901
Title: X-ray crystallographic studies reveal that the incorporation of spacer groups in carbonic anhydrase inhibitors causes alternate binding modes.
Journal: Acta crystallographica. Section F, Structural biology and crystallization communications20060701
Title: Synthesis, anticonvulsant, and anti-inflammatory evaluation of some new benzotriazole and benzofuran-based heterocycles.
Journal: Bioorganic & medicinal chemistry20060601
Title: New 1,3,4-thiadiazole derivatives endowed with analgesic and anti-inflammatory activities.
Journal: Bioorganic & medicinal chemistry20060315
Title: Synthesis of 1,3,4-thiadiazole, 1,3,4-thiadiazine, 1,3,6-thiadiazepane and quinoxaline derivatives from symmetrical dithiobiureas and thioureidoethylthiourea derivatives.
Journal: Molecules (Basel, Switzerland)20050831
Title: The synthesis and antimicrobial activity of some new methyl N-arylthiocarbamates, dimethyl N-aryldithiocarbonimidates and 2-arylamino-2-imidazolines.
Journal: European journal of medicinal chemistry20050701
Title: Carbonic anhydrase inhibitors. Inhibition of the cytosolic and tumor-associated carbonic anhydrase isozymes I, II, and IX with a series of 1,3,4-thiadiazole- and 1,2,4-triazole-thiols.
Journal: Bioorganic & medicinal chemistry letters20050502
Title: Solid-phase synthesis of 1,3,4-oxadiazole and 1,3,4-thiadiazole derivatives via selective, reagent-based cyclization of acyldithiocarbazate resins.
Journal: Journal of combinatorial chemistry20050101
Title: 1,3,4-thiadiazole derivatives. Synthesis, structure elucidation, and structure-antituberculosis activity relationship investigation.
Journal: Journal of medicinal chemistry20041230
Title: Synthesis and antitrypanosomal profile of new functionalized 1,3,4-thiadiazole-2-arylhydrazone derivatives, designed as non-mutagenic megazol analogues.
Journal: Bioorganic & medicinal chemistry letters20041220
Title: Synthesis and antimicrobial activities of some new 1-(5-phenylamino-[1,3,4]thiadiazol-2-yl)methyl-5-oxo-[1,2,4]triazole and 1-(4-phenyl-5-thioxo-[1,2,4]triazol-3-yl)methyl-5-oxo- [1,2,4]triazole derivatives.
Journal: European journal of medicinal chemistry20040901
Title: Antimelanoma activity of 1,3,4-thiadiazolium mesoionics: a structure-activity relationship study.
Journal: Anti-cancer drugs20040301
Title: Thiosugar nucleosides. Synthesis and biological activity of 1,3,4-thiadiazole, thiazoline and thiourea derivatives of 5-thio-D-glucose.
Journal: Nucleosides, nucleotides & nucleic acids20040101
Title: The synthesis and antibacterial activity of 1,3,4-thiadiazole phenyl oxazolidinone analogues.
Journal: Bioorganic & medicinal chemistry letters20031201
Title: Synthesis, fungicidal activity, and 3D-QSAR of pyridazinone-substituted 1,3,4-oxadiazoles and 1,3,4-thiadiazoles.
Journal: Journal of agricultural and food chemistry20020619
Title: Synthesis and antimicrobial activity of new substituted anilinobenzimidazoles.
Journal: Archives of pharmacal research20020601
Title: Thiadiazole-derived expanded heteroazaporphyrinoids.
Journal: Organic letters20010712
Title: [Synthesis and antibacterial activities of 3,6-disubstituted-5,6-dihydrogen-1,2,4-s-triazolo-[3,4-b]-1,3,4-thiadiazoles].
Journal: Yao xue xue bao = Acta pharmaceutica Sinica20010401
