Title: Evaluation of metabolism dependent inhibition of CYP2B6 mediated bupropion hydroxylation in human liver microsomes by monoamine oxidase inhibitors and prediction of potential as perpetrators of drug interaction.
Journal: Chemico-biological interactions20150325
Title: Kinetic resolution of propargylamines via a highly enantioselective non-enzymatic N-acylation process.
Journal: Chemical communications (Cambridge, England)20121104
Title: Chiral Brønsted acid catalyzed enantioselective allenylation of aldehydes.
Journal: Chemical communications (Cambridge, England)20120921
Title: Investigation of pyridine/propargyl bromide reaction and strong fluorescence enhancements of the resultant poly(propargyl pyridinium bromide).
Journal: The journal of physical chemistry. B20120920
Title: Low molecular weight amidoximes that act as potent inhibitors of lysine-specific demethylase 1.
Journal: Journal of medicinal chemistry20120913
Title: Stereoselective intermolecular C-H amination reactions.
Journal: Chemical communications (Cambridge, England)20120814
Title: Effects of diphenyl diselenide on depressive-like behavior in ovariectomized mice submitted to subchronic stress: involvement of the serotonergic system.
Journal: Psychopharmacology20120801
Title: The selective inhibition of the D₁ dopamine receptor results in an increase of metabolized dopamine in the rat striatum.
Journal: Neurochemical research20120801
Title: Site-specific protein propargylation using tissue transglutaminase.
Journal: Organic & biomolecular chemistry20120721
Title: Diastereoselective [4 + 1] cycloaddition of alkenyl propargyl acetates with CO catalyzed by [RhCl(CO)2]2.
Journal: The Journal of organic chemistry20120720
Title: 15N magnetic resonance hyperpolarization via the reaction of parahydrogen with 15N-propargylcholine.
Journal: Journal of the American Chemical Society20120711
Title: Behavioral effects of α,α,β,β-tetradeutero-5-MeO-DMT in rats: comparison with 5-MeO-DMT administered in combination with a monoamine oxidase inhibitor.
Journal: Psychopharmacology20120601
Title: Synthesis and crystal structure of hydroxyacetophenone Schiff bases containing propargyl moiety: solvent effects on UV-visible spectra.
Journal: Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy20120601
Title: Multipotent MAO and cholinesterase inhibitors for the treatment of Alzheimer's disease: synthesis, pharmacological analysis and molecular modeling of heterocyclic substituted alkyl and cycloalkyl propargyl amine.
Journal: European journal of medicinal chemistry20120601
Title: Cross-linked DNA: propargylated ribonucleosides as 'click' ligation sites for bifunctional azides.
Journal: The Journal of organic chemistry20120504
Title: Highly chemoselective calcium-catalyzed propargylic deoxygenation.
Journal: Chemistry (Weinheim an der Bergstrasse, Germany)20120410
Title: Efficient iron(III)-catalyzed three-component coupling reaction of alkynes, CH2Cl2 and amines to propargylamines.
Journal: Chemical communications (Cambridge, England)20120214
Title: Highly stereoselective synthesis of cis-β-enaminones mediated by diethyl azodicarboxylate.
Journal: Chemical communications (Cambridge, England)20120207
Title: Indium-mediated asymmetric Barbier-type propargylations: additions to aldehydes and ketones and mechanistic investigation of the organoindium reagents.
Journal: The Journal of organic chemistry20120120
Title: Over-expression of LSD1 promotes proliferation, migration and invasion in non-small cell lung cancer.
Journal: PloS one20120101
Title: The marriage of organocatalysis with metal catalysis: access to multisubstituted chiral 2,5-dihydropyrroles by cascade iminium/enamine-metal cooperative catalysis.
Journal: Chemistry (Weinheim an der Bergstrasse, Germany)20111209
Title: Pharmacokinetic study of six flavones in rat plasma and tissues after oral administration of 'JiangYaBiFeng' using SPE-HPLC-DAD.
Journal: Journal of pharmaceutical and biomedical analysis20111205
Title: Role of androgen receptor and associated lysine-demethylase coregulators, LSD1 and JMJD2A, in localized and advanced human bladder cancer.
Journal: Molecular carcinogenesis20111201
Title: Crystal structures of Candida albicans dihydrofolate reductase bound to propargyl-linked antifolates reveal the flexibility of active site loop residues critical for ligand potency and selectivity.
Journal: Chemical biology & drug design20111001
Title: Copper-mediated aerobic synthesis of 3-azabicyclo[3.1.0]hex-2-enes and 4-carbonylpyrroles from N-allyl/propargyl enamine carboxylates.
Journal: Journal of the American Chemical Society20110907
Title: 3-Iodothyronamine metabolism and functional effects in FRTL5 thyroid cells.
Journal: Journal of molecular endocrinology20110801
Title: Effects of the thyroid hormone derivatives 3-iodothyronamine and thyronamine on rat liver oxidative capacity.
Journal: Molecular and cellular endocrinology20110720
Title: Electrochemical impedance spectroscopy sensor for ascorbic acid based on copper(I) catalyzed click chemistry.
Journal: Biosensors & bioelectronics20110715
Title: A general copper-BINAP-catalyzed asymmetric propargylation of ketones with propargyl boronates.
Journal: Journal of the American Chemical Society20110713
Title: The effects of pargyline and 2-phenylethylamine on D1-like dopamine receptor binding.
Journal: Journal of neural transmission (Vienna, Austria : 1996)20110701
Title: Palladium-catalyzed coupling of propargylic carbonates with N-tosylhydrazones: highly selective synthesis of substituted propargylic N-sulfonylhydrazones and vinylallenes.
Journal: Chemistry (Weinheim an der Bergstrasse, Germany)20110614
Title: Simultaneous determination of eight active components in Chinese medicine 'JiangYaBiFeng' tablet by HPLC coupled with diode array detection.
Journal: Journal of pharmaceutical and biomedical analysis20110601
Title: Toward selective drug development for the human 5-hydroxytryptamine 1E receptor: a comparison of 5-hydroxytryptamine 1E and 1F receptor structure-affinity relationships.
Journal: The Journal of pharmacology and experimental therapeutics20110601
Title: Synthesis of 4-aminoquinoline analogues and their platinum(II) complexes as new antileishmanial and antitubercular agents.
Journal: Biomedicine & pharmacotherapy = Biomedecine & pharmacotherapie20110601
Title: Cyclization-carbonylation-cyclization coupling reactions of propargyl acetates and amides with palladium(II)-bisoxazoline catalysts.
Journal: Angewandte Chemie (International ed. in English)20110418
Title: Helical chiral 2,2'-bipyridine N-monoxides as catalysts in the enantioselective propargylation of aldehydes with allenyltrichlorosilane.
Journal: Organic letters20110401
Title: An image-based, high-throughput screening assay for molecules that induce excess DNA replication in human cancer cells.
Journal: Molecular cancer research : MCR20110301
Title: Pargyline reduces renal damage associated with ischaemia-reperfusion and cyclosporin.
Journal: Nephrology, dialysis, transplantation : official publication of the European Dialysis and Transplant Association - European Renal Association20110201
Title: Star polymers composed entirely of amino acid building blocks: a route towards stereospecific, biodegradable and hierarchically functionalized stars.
Journal: Chemical communications (Cambridge, England)20110128
Title: Hexaphenylbenzene as a rigid template for the straightforward syntheses of 'star-shaped' glycodendrimers.
Journal: The Journal of organic chemistry20110121
Title: Gold(I)-catalyzed formation of dihydroquinolines and indoles from N-aminophenyl propargyl malonates.
Journal: Chemical communications (Cambridge, England)20110107
Title: Domino gold-catalyzed rearrangement and fluorination of propargyl acetates.
Journal: Chemical communications (Cambridge, England)20110107
Title: Microdialysis with radiometric monitoring of L-[β-11C]DOPA to assess dopaminergic metabolism: effect of inhibitors of L-amino acid decarboxylase, monoamine oxidase, and catechol-O-methyltransferase on rat striatal dialysate.
Journal: Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism20110101
Title: Synthesis and SAR studies of 1,4-benzoxazine MenB inhibitors: novel antibacterial agents against Mycobacterium tuberculosis.
Journal: Bioorganic & medicinal chemistry letters20101101
Title: A simple method for the preparation of propargylamines using molecular sieve modified with copper(II).
Journal: Organic & biomolecular chemistry20101021
Title: Fine-tuning the morphology of self-assembled nanostructures of propargyl ammonium-based amphiphiles.
Journal: The journal of physical chemistry. B20101007
Title: Merging nucleophilic and hydrogen bonding catalysis: an anion binding approach to the kinetic resolution of propargylic amines.
Journal: Journal of the American Chemical Society20101006
Title: Highly diastereoselective synthesis of α-difluoromethyl amines from N-tert-butylsulfinyl ketimines and difluoromethyl phenyl sulfone.
Journal: Chemistry (Weinheim an der Bergstrasse, Germany)20101004
Title: Characterization of monoamine oxidases in mesenchymal stem cells: role in hydrogen peroxide generation and serotonin-dependent apoptosis.
Journal: Stem cells and development20101001
Title: Haloperidol, spiperone, pimozide and aripiprazole reduce intracellular dopamine content in PC12 cells and rat mesencephalic cultures: Implication of inhibition of vesicular transport.
Journal: European journal of pharmacology20100825
Title: Mechanistic insights into the one-pot synthesis of propargylamines from terminal alkynes and amines in chlorinated solvents catalyzed by gold compounds and nanoparticles.
Journal: Chemistry (Weinheim an der Bergstrasse, Germany)20100809
Title: Synthesis of fused and linked bicyclic nitrogen heterocycles by palladium-catalyzed domino cyclization of propargyl bromides.
Journal: Chemistry (Weinheim an der Bergstrasse, Germany)20100726
Title: Effects of monoamine oxidase inhibitor and cytochrome P450 2D6 status on 5-methoxy-N,N-dimethyltryptamine metabolism and pharmacokinetics.
Journal: Biochemical pharmacology20100701
Title: Enantioselective synthesis of 3-azabicyclo[4.1.0]heptenes and 3-azabicyclo[3.2.0]heptenes by Ir-catalyzed asymmetric allylic amination of N-tosyl propynylamine and Pt-catalyzed cycloisomerization.
Journal: Chemistry (Weinheim an der Bergstrasse, Germany)20100611
Title: Unprecedented Cu(I)-catalyzed microwave-assisted three-component coupling of a ketone, an alkyne, and a primary amine.
Journal: Organic letters20100604
Title: Comparative analysis of small molecules and histone substrate analogues as LSD1 lysine demethylase inhibitors.
Journal: Journal of the American Chemical Society20100310
Title: Chiral N-phosphonyl imine chemistry: an efficient asymmetric synthesis of chiral N-phosphonyl propargylamines.
Journal: Organic & biomolecular chemistry20100307
Title: Copper-catalyzed enantioselective three-component synthesis of optically active propargylamines from aldehydes, amines, and aliphatic alkynes.
Journal: Chemistry (Weinheim an der Bergstrasse, Germany)20100222
Title: A versatile synthetic platform based on strained propargyl amines.
Journal: Angewandte Chemie (International ed. in English)20100222
Title: Silver(I)-mediated highly enantioselective synthesis of axially chiral allenes under thermal and microwave-assisted conditions.
Journal: Chemical communications (Cambridge, England)20100114
Title: Zinc catalyzed and mediated propargylations with propargyl boronates.
Journal: Organic letters20100101
Title: Synthesis of 2-thio- and 2-oxoimidazoles via cascade addition-cycloisomerization reactions of propargylcyanamides.
Journal: The Journal of organic chemistry20100101
Title: Propargylamine containing compounds as modulators of proteolytic cleavage of amyloid-beta protein precursor: involvement of MAPK and PKC activation.
Journal: Journal of Alzheimer's disease : JAD20100101
Title: Inhibition of monoamine oxidase activity by antidepressants and mood stabilizers.
Journal: Neuro endocrinology letters20100101
Title: Highly selective fluorescent probe for Au3+ based on cyclization of propargylamide.
Journal: Chemical communications (Cambridge, England)20091214
Title: Acidic vesicles of the endo-exocytic pathways as targets for some anti-monoamine oxidase drugs.
Journal: Metabolic brain disease20091201
Title: Inhibition of the histone demethylase LSD1 blocks alpha-herpesvirus lytic replication and reactivation from latency.
Journal: Nature medicine20091101
Title: Genetic mapping of targets mediating differential chemical phenotypes in Plasmodium falciparum.
Journal: Nature chemical biology20091001
Title: Synthesis of enantioenriched homopropargylic sulfonamides by a three component reaction of aldehydes, sulfonamides, and chiral allenylsilanes.
Journal: Organic letters20091001
Title: Highly stereoselective intramolecular alpha-arylation of self-stabilized non-racemic enolates: synthesis of alpha-quaternary alpha-amino acid derivatives.
Journal: Chemical communications (Cambridge, England)20090907
Title: Zn(II)-Catalyzed synthesis of piperidines from propargyl amines and cyclopropanes.
Journal: Organic letters20090820
Title: Functional mechanism of neuroprotection by inhibitors of type B monoamine oxidase in Parkinson's disease.
Journal: Expert review of neurotherapeutics20090801
Title: In vitro biological activity and structural analysis of 2,4-diamino-5-(2'-arylpropargyl)pyrimidine inhibitors of Candida albicans.
Journal: Bioorganic & medicinal chemistry20090715
Title: Iron(III)-catalyzed and air-mediated tandem reaction of aldehydes, alkynes and amines: an efficient approach to substituted quinolines.
Journal: Chemistry (Weinheim an der Bergstrasse, Germany)20090622
Title: Three-component synthesis of N-Boc-4-iodopyrroles and sequential one-pot alkynylation.
Journal: Organic letters20090604
Title: Development of spin-labeled pargyline analogues as specific inhibitors of human monoamine oxidases A and B.
Journal: Biochemistry20090512
Title: Chemoselective C-H bond activation: ligand and solvent free iron-catalyzed oxidative C-C cross-coupling of tertiary amines with terminal alkynes. Reaction scope and mechanism.
Journal: Organic letters20090416
Title: Synthesis of diacetylene-containing peptide building blocks and amphiphiles, their self-assembly and topochemical polymerization in organic solvents.
Journal: Chemistry (Weinheim an der Bergstrasse, Germany)20090101
Title: Total synthesis of pentabromo- and pentachloropseudilin, and synthetic analogues--allosteric inhibitors of myosin ATPase.
Journal: Angewandte Chemie (International ed. in English)20090101
Title: Nickel-catalyzed asymmetric cross-couplings of racemic propargylic halides with arylzinc reagents.
Journal: Journal of the American Chemical Society20080924
Title: Neurotoxic catecholamine metabolite in nociceptors contributes to painful peripheral neuropathy.
Journal: The European journal of neuroscience20080901
Title: TVP1022 and propargylamine protect neonatal rat ventricular myocytes against doxorubicin-induced and serum starvation-induced cardiotoxicity.
Journal: Journal of cardiovascular pharmacology20080901
Title: Evidence for serotonin synthesis-dependent regulation of in vitro neuronal firing rates in the midbrain raphe complex.
Journal: European journal of pharmacology20080820
Title: Dopamine release in organotypic cultures of foetal mouse mesencephalon: effects of depolarizing agents, pargyline, nomifensine, tetrodotoxin and calcium.
Journal: The European journal of neuroscience20080801
Title: Clorgyline and other propargylamine derivatives as inhibitors of succinate-dependent H(2)O(2) release at NADH:UBIQUINONE oxidoreductase (Complex I) in brain mitochondria.
Journal: Journal of bioenergetics and biomembranes20080801
Title: Application of the 4-trifluoromethylbenzenepropargyl ether group as an unhindered, electron deficient protecting group for stereoselective glycosylation.
Journal: The Journal of organic chemistry20080704
Title: Synthesis and evaluation of homodimeric GnRHR antagonists having a rigid bis-propargylated benzene core.
Journal: Bioorganic & medicinal chemistry20080401
Title: Direct construction of bicyclic heterocycles by palladium-catalyzed domino cyclization of propargyl bromides.
Journal: Organic letters20080320
Title: The immobilization of proteins on biodegradable polymer fibers via click chemistry.
Journal: Biomaterials20080301
Title: [A comparison of the pharmacology of (-)-deprenyl to N-methylpropargylamine-1-aminoindane (J-508) and rasagiline, the desmethyl-analogue of J-508].
Journal: Neuropsychopharmacologia Hungarica : a Magyar Pszichofarmakologiai Egyesulet lapja = official journal of the Hungarian Association of Psychopharmacology20080301
Title: Gold-catalyzed highly enantioselective synthesis of axially chiral allenes.
Journal: Organic letters20080207
Title: Comparison of the structural properties of the active site cavities of human and rat monoamine oxidase A and B in their soluble and membrane-bound forms.
Journal: Biochemistry20080115
Title: Enantioselective copper-catalyzed propargylic amination.
Journal: Angewandte Chemie (International ed. in English)20080101
Title: Efficient synthesis of methylenetetrahydrofurans and methylenepyrrolidines by formal [3+2] cycloadditions of propargyl substrates.
Journal: Chemistry (Weinheim an der Bergstrasse, Germany)20080101
Title: A highly efficient and selective Au(I)-catalyzed tandem synthesis of diversely substituted pyrrolo[1,2-a]quinolines in aqueous media.
Journal: Angewandte Chemie (International ed. in English)20080101
Title: [Analysis of ubiquitin-dependent regulation of the monoamine oxidase sensitivity to proteolysis and specific inhibition by pargyline].
Journal: Biomeditsinskaia khimiia20080101
Title: Effect of endogenous catecholamines on apoptosis of Con A-activated lymphocytes of rats.
Journal: Journal of neuroimmunology20071201
Title: Reduction of fat deposition by combined inhibition of monoamine oxidases and semicarbazide-sensitive amine oxidases in obese Zucker rats.
Journal: Pharmacological research20071201
Title: The monoamine oxidase inhibitor phenelzine enhances the discriminative stimulus effect of nicotine in rats.
Journal: Behavioural pharmacology20071101
Title: Diastereoselective alkynylation of N-p-tolylsulfinylimines with aluminum acetylides.
Journal: The Journal of organic chemistry20071012
Title: Localization of L-DOPA uptake and decarboxylating neuronal structures in the cat brain using dopamine immunohistochemistry.
Journal: Brain research20070905
Title: MAO-A-induced mitogenic signaling is mediated by reactive oxygen species, MMP-2, and the sphingolipid pathway.
Journal: Free radical biology & medicine20070701
Title: Rapid, efficient synthesis of heterobifunctional biodegradable dendrimers.
Journal: Journal of the American Chemical Society20070606
Title: Pargyline effect on luteinizing hormone secretion throughout the rat estrous cycle: correlation with serotonin, catecholamines and nitric oxide in the medial preoptic area.
Journal: Brain research20070420
Title: Beta-silylated homopropargylic amines via the asymmetric allenylboration of aldimines.
Journal: Organic letters20070315
Title: Mapping the amphetamine-evoked changes in [11C]raclopride binding in living rat using small animal PET: modulation by MAO-inhibition.
Journal: NeuroImage20070301
Title: A RSK kinase inhibitor reporting its selectivity in vivo.
Journal: Nature chemical biology20070301
Title: Efficient ruthenium and copper cocatalzyed five-component coupling to form dipropargyl amines under mild conditions in water.
Journal: Organic & biomolecular chemistry20070207
Title: Fucosylated pentaerythrityl phosphodiester oligomers (PePOs): automated synthesis of DNA-based glycoclusters and binding to Pseudomonas aeruginosa lectin (PA-IIL).
Journal: Bioconjugate chemistry20070101
Title: Biotinylated anisomycin: a comparison of classical and 'click' chemistry approaches.
Journal: Bioconjugate chemistry20070101
Title: Neuroprotection by propargylamines in Parkinson's disease: intracellular mechanism underlying the anti-apoptotic function and search for clinical markers.
Journal: Journal of neural transmission. Supplementum20070101
Title: EPR studies of amine radical cations. Part 2. Thermal and photo-induced rearrangements of propargylamine and allylamine radical cations in low-temperature freon matrices.
Journal: The journal of physical chemistry. A20061228
Title: Crystallographic characterization of difluoropropargyl indium bromide, a reactive fluoroorganometallic reagent.
Journal: Angewandte Chemie (International ed. in English)20061106
Title: Direct addition of alkynes to imines and related C=N electrophiles: A convenient access to propargylamines.
Journal: Chemical communications (Cambridge, England)20061104
Title: Photoisomerization as a modulator of the DNA-cleaving efficiency of novel azo bispropargyl sulfones.
Journal: Chemical communications (Cambridge, England)20060928
Title: Synthesis of 3-miktoarm stars and 1st generation mikto dendritic copolymers by 'living' radical polymerization and 'click' chemistry.
Journal: Journal of the American Chemical Society20060906
Title: Asymmetric synthesis of alpha,alpha-dibranched propargylamines by acetylide additions to N-tert-butanesulfinyl ketimines.
Journal: The Journal of organic chemistry20060901
Title: [Molecular mechanisms of the neuroprotective effect of (-)-deprenyl].
Journal: Orvosi hetilap20060709
Title: Effect of monoamine oxidase inhibition on amphetamine-evoked changes in dopamine receptor availability in the living pig: a dual tracer PET study with [11C]harmine and [11C]raclopride.
Journal: Synapse (New York, N.Y.)20060601
Title: Highly enantioselective access to primary propargylamines: 4-piperidinone as a convenient protecting group.
Journal: Organic letters20060525
Title: Practical highly enantioselective synthesis of propargylamines through a copper-catalyzed one-pot three-component condensation reaction.
Journal: Chemistry (Weinheim an der Bergstrasse, Germany)20060524
Title: Rationale for considering that propargylamines might be neuroprotective in Parkinson's disease.
Journal: Neurology20060523
Title: Microsphere-based protease assays and screening application for lethal factor and factor Xa.
Journal: Cytometry. Part A : the journal of the International Society for Analytical Cytology20060501
Title: Zinc- and indium-promoted conjugate addition-cyclization reactions of ethenetricarboxylates with propargylamines and alcohol: novel methylenepyrrolidine and methylenetetrahydrofuran syntheses.
Journal: The Journal of organic chemistry20060428
Title: Enhanced diastereoselectivity in beta-mannopyranosylation through the use of sterically minimal propargyl ether protecting groups.
Journal: The Journal of organic chemistry20060414
Title: Gold(III) Salen complex-catalyzed synthesis of propargylamines via a three-component coupling reaction.
Journal: Organic letters20060413
Title: Antioxidant properties of propargylamine derivatives: assessment of their ability to scavenge peroxynitrite.
Journal: The Journal of pharmacy and pharmacology20060401
Title: Very mild, enantioselective synthesis of propargylamines catalyzed by copper(I)-bisimine complexes.
Journal: The Journal of organic chemistry20060303
Title: Effects of co-administration of a selective serotonin reuptake inhibitor and monoamine oxidase inhibitors on 5-HT-related behavior in rats.
Journal: European journal of pharmacology20060227
Title: Physical, chemical and environmental properties of selected chemical alternatives for the pre-plant use of methyl bromide as soil fumigant.
Journal: Pest management science20060201
Title: N-Propargylamine protects SH-SY5Y cells from apoptosis induced by an endogenous neurotoxin, N-methyl(R)salsolinol, through stabilization of mitochondrial membrane and induction of anti-apoptotic Bcl-2.
Journal: Journal of neural transmission (Vienna, Austria : 1996)20060101
Title: Involvement of multiple survival signal transduction pathways in the neuroprotective, neurorescue and APP processing activity of rasagiline and its propargyl moiety.
Journal: Journal of neural transmission. Supplementum20060101
Title: Difluoroallenyl bromide as a wide-ranging difluoromethylene cation equivalent: SN2 substitution of difluoropropargyl bromide through sequential SE2' and SN2' reactions.
Journal: Angewandte Chemie (International ed. in English)20051201
Title: Regulation of Bcl-2 family proteins, neurotrophic factors, and APP processing in the neurorescue activity of propargylamine.
Journal: FASEB journal : official publication of the Federation of American Societies for Experimental Biology20051101
Title: Glucose handling in streptozotocin-induced diabetic rats is improved by tyramine but not by the amine oxidase inhibitor semicarbazide.
Journal: European journal of pharmacology20051017
Title: Isoflurane anesthesia induces biphasic effect on dopamine release in the rat striatum.
Journal: Brain research bulletin20051015
Title: Effect of endogenous catecholamines in lymphocytes on lymphocyte function.
Journal: Journal of neuroimmunology20051001
Title: Halothane enhances dopamine metabolism at presynaptic sites in a calcium-independent manner in rat striatum.
Journal: British journal of anaesthesia20051001
Title: LSD1 demethylates repressive histone marks to promote androgen-receptor-dependent transcription.
Journal: Nature20050915
Title: Effects of manganese on extracellular levels of dopamine in rat striatum: an analysis in vivo by brain microdialysis.
Journal: Neurochemical research20050901
Title: The potential efficiency of irrigation management and propargyl bromide in controlling three soil pests: Tylenchulus semipenetrans, Fusarium oxysporum and Echinochloa crus-galli.
Journal: Pest management science20050801
Title: Eugenol and its structural analogs inhibit monoamine oxidase A and exhibit antidepressant-like activity.
Journal: Bioorganic & medicinal chemistry20050801
Title: Novel neuroprotective mechanism of action of rasagiline is associated with its propargyl moiety: interaction of Bcl-2 family members with PKC pathway.
Journal: Annals of the New York Academy of Sciences20050801
Title: Electrostatic stabilization in a pre-organized polar active site: the catalytic role of Lys-80 in Candida tenuis xylose reductase (AKR2B5) probed by site-directed mutagenesis and functional complementation studies.
Journal: The Biochemical journal20050715
Title: A Re(V)-catalyzed C-N bond-forming route to human lipoxygenase inhibitors.
Journal: Organic letters20050609
Title: Dopamine is metabolised by different enzymes along the rat nephron.
Journal: Pflugers Archiv : European journal of physiology20050601
Title: Incompatibility of metam sodium with halogenated fumigants.
Journal: Pest management science20050501
Title: Gastric pentadecapeptide BPC 157 effective against serotonin syndrome in rats.
Journal: European journal of pharmacology20050411
Title: A new hypertrophic mechanism of serotonin in cardiac myocytes: receptor-independent ROS generation.
Journal: FASEB journal : official publication of the Federation of American Societies for Experimental Biology20050401
Title: Directed evolution of an amine oxidase for the preparative deracemisation of cyclic secondary amines.
Journal: Chembiochem : a European journal of chemical biology20050401
Title: Synthesis of heterocyclic allenes via palladium-catalyzed hydride-transfer reaction of propargylic amines.
Journal: The Journal of organic chemistry20050318
Title: An efficient synthesis of propargylamines via C-H activation catalyzed by copper(I) in ionic liquids.
Journal: Chemical communications (Cambridge, England)20050314
Title: Diurnal variation in serotonin immunoreactivity in the dorsal raphe nucleus.
Journal: Brain research20050209
Title: Rasagiline: neurodegeneration, neuroprotection, and mitochondrial permeability transition.
Journal: Journal of neuroscience research20050101
Title: Effect of application variables on emissions and distribution of fumigants applied via subsurface drip irrigation.
Journal: Environmental science & technology20041101
Title: Preclinical evidence for neuroprotection with monoamine oxidase-B inhibitors in Parkinson's disease.
Journal: Neurology20041012
Title: Novel bifunctional drugs targeting monoamine oxidase inhibition and iron chelation as an approach to neuroprotection in Parkinson's disease and other neurodegenerative diseases.
Journal: Journal of neural transmission (Vienna, Austria : 1996)20041001
Title: The mechanism of nitrogenase. Computed details of the site and geometry of binding of alkyne and alkene substrates and intermediates.
Journal: Journal of the American Chemical Society20040929
Title: Differential inhibition of six copper amine oxidases by a family of 4-(aryloxy)-2-butynamines: evidence for a new mode of inactivation.
Journal: Biochemistry20040831
Title: Effect of surface tarp on emissions and distribution of drip-applied fumigants.
Journal: Environmental science & technology20040815
Title: D-amphetamine-induced hydrogen peroxide production in skeletal muscle is modulated by monoamine oxidase inhibition.
Journal: International journal of sports medicine20040801
Title: Selective inhibition of bovine plasma amine oxidase by homopropargylamine, a new inactivator motif.
Journal: Journal of the American Chemical Society20040630
Title: Helical polymer carrying helical grafts from peptide-based acetylene macromonomers: synthesis.
Journal: Macromolecular bioscience20040625
Title: L-type calcium channel blockers enhance 5-HTP-induced antinociception in mice.
Journal: Acta pharmacologica Sinica20040501
Title: Highly enantioselective addition of phenylacetylene to aldehydes catalyzed by a camphorsulfonamide ligand.
Journal: Organic letters20040415
Title: Fumigant combinations for Cyperus esculentum L control.
Journal: Pest management science20040401
Title: Protective effects of neuronal nitric oxide synthase inhibitor in mouse brain against MPTP neurotoxicity: an immunohistological study.
Journal: European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology20040301
Title: Neuroprotection by monoamine oxidase B inhibitors: a therapeutic strategy for Parkinson's disease?
Journal: BioEssays : news and reviews in molecular, cellular and developmental biology20040101
Title: Advances in neuroprotection research for neurodegenerative diseases.
Journal: Advances in experimental medicine and biology20040101
Title: Cytotoxicity, cytoprotection and neurotoxicity of novel deprenyl-related propargylamines, stable nitroxide free radicals, in vitro and in vivo.
Journal: In vivo (Athens, Greece)20040101
Title: The importance of propargylamine moiety in the anti-Parkinson drug rasagiline and its derivatives in MAPK-dependent amyloid precursor protein processing.
Journal: FASEB journal : official publication of the Federation of American Societies for Experimental Biology20031201
Title: TCH346 prevents motor symptoms and loss of striatal FDOPA uptake in bilaterally MPTP-treated primates.
Journal: Neurobiology of disease20031101
Title: Selegiline reduces N-methyl-D-aspartic acid induced perturbation of neurotransmission but it leaves NMDA receptor dependent long-term potentiation intact in the hippocampus.
Journal: Journal of neural transmission (Vienna, Austria : 1996)20031101
Title: Novel synthesis of carbapenam by intramolecular attack of lactam nitrogen toward eta1-allenyl and eta3-propargylpalladium complex.
Journal: The Journal of organic chemistry20031017
Title: Three-component enantioselective synthesis of propargylamines through Zr-catalyzed additions of alkyl zinc reagents to alkynylimines.
Journal: Angewandte Chemie (International ed. in English)20030915
Title: Enantioselective synthesis of propargylamines through Zr-catalyzed addition of mixed alkynylzinc reagents to arylimines.
Journal: Organic letters20030904
Title: Effects of reboxetine on sympathetic neuroeffector transmission in rabbit carotid artery.
Journal: The Journal of pharmacology and experimental therapeutics20030901
Title: Transient behavioral sensitization to nicotine becomes long-lasting with monoamine oxidases inhibitors.
Journal: Pharmacology, biochemistry, and behavior20030901
Title: Structural comparison of human monoamine oxidases A and B: mass spectrometry monitoring of cysteine reactivities.
Journal: The Journal of biological chemistry20030801
Title: 4-Methylthioamphetamine-induced hyperthermia in mice: influence of serotonergic and catecholaminergic pathways.
Journal: Toxicology and applied pharmacology20030801
Title: Intracellular patch electrochemistry: regulation of cytosolic catecholamines in chromaffin cells.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience20030702
Title: Synthesis of enantiomerically enriched propargylamines by copper-catalyzed addition of alkynes to enamines.
Journal: Chemistry (Weinheim an der Bergstrasse, Germany)20030616
Title: Highly potent propargylamine and allylamine inhibitors of bovine plasma amine oxidase.
Journal: Biochemical and biophysical research communications20030516
Title: Role of extracellular serotonin levels in the effect of 5-HT1B receptor blockade.
Journal: Psychopharmacology20030501
Title: High-frequency stimulation of the subthalamic nucleus enhances striatal dopamine release and metabolism in rats.
Journal: Journal of neurochemistry20030501
Title: Striatal formation of 6-hydroxydopamine in mice treated with pargyline, pyrogallol and methamphetamine.
Journal: Journal of neural transmission (Vienna, Austria : 1996)20030501
Title: Neuroprotection by deprenyl and other propargylamines: glyceraldehyde-3-phosphate dehydrogenase rather than monoamine oxidase B.
Journal: Journal of neural transmission (Vienna, Austria : 1996)20030501
Title: Inhibition of rat fat cell lipolysis by monoamine oxidase and semicarbazide-sensitive amine oxidase substrates.
Journal: European journal of pharmacology20030418
Title: Ovicide-induced serosa degeneration and its impact on embryonic development in Manduca sexta (Insecta: Lepidoptera).
Journal: Tissue & cell20030401
Title: Histamine antilipolytic action in rat adipocytes: comparison with the effect of tyramine.
Journal: Inflammation research : official journal of the European Histamine Research Society ... [et al.]20030401
Title: Iterative oxazole assembly via alpha-chloroglycinates: total synthesis of (-)-muscoride A.
Journal: Angewandte Chemie (International ed. in English)20030328
Title: Novel iminium ion equivalents prepared through C-H oxidation for the stereocontrolled synthesis of functionalized propargylic amine derivatives.
Journal: Journal of the American Chemical Society20030226
Title: Mechanism by which brain-derived neurotrophic factor increases dopamine release from the rabbit retina.
Journal: Investigative ophthalmology & visual science20030201
Title: In situ imaging of specific binding of [3H]isatin in rat brain.
Journal: Journal of neurochemistry20030201
Title: Proton magnetic resonance imaging and spectroscopy identify metabolic changes in the striatum in the MPTP feline model of parkinsonism.
Journal: Experimental neurology20030201
Title: Antioxidant properties of newly synthesized N-propargylamine derivatives of nitroxyl: a comparison with deprenyl.
Journal: Polish journal of pharmacology20030101
Title: Gas-phase sorption-desorption of propargyl bromide and 1,3-dichloropropene on plastic materials.
Journal: Journal of environmental quality20030101
Title: Novel dual inhibitors of AChE and MAO derived from hydroxy aminoindan and phenethylamine as potential treatment for Alzheimer's disease.
Journal: Journal of medicinal chemistry20021121
Title: Characterization of propargyl bromide transformation in soil.
Journal: Pest management science20021001
Title: Monoamine oxidase inhibitor-induced blockade of locomotor sensitization to quinpirole: role of striatal dopamine uptake inhibition.
Journal: Neuropharmacology20020901
Title: Therapeutic effect of neuronal nitric oxide synthase inhibitor (7-nitroindazole) against MPTP neurotoxicity in mice.
Journal: Metabolic brain disease20020901
Title: Synthesis of cyclophanetetrayne complexes from bis(propargyldicobalt) dication equivalents.
Journal: Chemical communications (Cambridge, England)20020721
Title: Tyramine and monoamine oxidase inhibitors as modulators of the mitochondrial membrane permeability transition.
Journal: The Journal of membrane biology20020701
Title: Progressive alteration of neuronal dopamine transporter activity in a rat injured by an intranigral injection of MPP+.
Journal: Brain research20020621
Title: Stable DNA triple helix formation using oligonucleotides containing 2'-aminoethoxy,5-propargylamino-U.
Journal: Biochemistry20020611
Title: Enantioselective direct-addition of terminal alkynes to imines catalyzed by copper(I)pybox complex in water and in toluene.
Journal: Journal of the American Chemical Society20020522
Title: Concise, stereoselective syntheses of cis-nemorensic acid and 4-hydroxy-cis-nemorensic acid via tandem carbonyl ylide formation-cycloaddition.
Journal: Organic letters20020516
Title: Propargylamines induce antiapoptotic new protein synthesis in serum- and nerve growth factor (NGF)-withdrawn, NGF-differentiated PC-12 cells.
Journal: The Journal of pharmacology and experimental therapeutics20020501
Title: 5-Hydroxytryptophan (5-HTP) uptake and decarboxylation in the kitten brain.
Journal: Journal of neural transmission (Vienna, Austria : 1996)20020501
Title: Pharmacological interventions in aging and age-associated disorders: potentials of propargylamines for human use.
Journal: Annals of the New York Academy of Sciences20020401
Title: N-methyl-norsalsolinol, a putative dopaminergic neurotoxin, passes through the blood-brain barrier in vivo.
Journal: Neuroreport20020121
Title: A dynamic two-dimensional system for measuring volatile organic compound volatilization and movement in soils.
Journal: Journal of environmental quality20020101
Title: Aliphatic propargylamines as symptomatic and neuroprotective treatments for neurodegenerative diseases.
Journal: Neurotoxicology and teratology20020101
Title: Neuroprotection by propargylamines in Parkinson's disease: suppression of apoptosis and induction of prosurvival genes.
Journal: Neurotoxicology and teratology20020101
Title: Dynamics of histamine H(3) receptor antagonists on brain histamine metabolism: do all histamine H(3) receptor antagonists act at a single site?
Journal: European journal of pharmacology20011116
Title: Novel intramolecular rearrangement of tertiary propargylamine N-oxides.
Journal: The Journal of organic chemistry20011019
Title: Oxidation products of polyamines induce mitochondrial uncoupling and cytochrome c release.
Journal: FEBS letters20011019
Title: Combinatorial synthesis of SSAO inhibitors using sonogashira coupling: SAR of aryl propargylic amines.
Journal: Bioorganic & medicinal chemistry letters20011008
Title: Oxygen dependency of monoamine oxidase activity in the intact lung.
Journal: American journal of physiology. Lung cellular and molecular physiology20011001
Title: Preparation of 2,5-disubstituted oxazoles from N-propargylamides.
Journal: Organic letters20010809
Title: Inhibition of rat liver microsomal CYP1A2 and CYP2B1 activity by N-(2-heptyl)-N-methyl-propargylamine and by N-(2-heptyl)-propargylamine.
Journal: Drug metabolism and disposition: the biological fate of chemicals20010801
Title: Oxygen inhalation enhances striatal dopamine metabolism and monoamineoxidase enzyme inhibition prevents it: a microdialysis study.
Journal: European journal of pharmacology20010622
Title: Inhibition of MAO-A activity enhances behavioural activity of rats assessed using water maze and open arena tasks.
Journal: Pharmacology & toxicology20010601
Title: Antiapoptotic properties of rasagiline, N-propargylamine-1(R)-aminoindan, and its optical (S)-isomer, TV1022.
Journal: Annals of the New York Academy of Sciences20010601
Title: Long-term impairment of anterograde axonal transport along fiber projections originating in the rostral raphe nuclei after treatment with fenfluramine or methylenedioxymethamphetamine.
Journal: Synapse (New York, N.Y.)20010501
Title: Maintaining mitochondrial membrane impermeability. an opportunity for new therapy in glaucoma?
Journal: Survey of ophthalmology20010501
Title: L-Deprenyl prevents the cell hypoxia induced by dopaminergic neurotoxins, MPP(+) and beta-carbolinium: a microdialysis study in rats.
Journal: Neuroscience letters20010420
Title: Pharmacological properties of the MPTP analog trans-1-methyl-4-[4-dimethylaminophenylethenyl]-1,2,3,6-tetrahydropyridine and its pyridinium metabolite in mouse brain synaptosomes: a potential visual marker for substrates of MPTP-induced neurotoxicity.
Journal: Progress in neuro-psychopharmacology & biological psychiatry20010401
Title: Dialysate dihydroxyphenylglycol as a window for in situ axoplasmic norepinephrine disposition.
Journal: Neurochemistry international20010301
Title: Vitreal dihydroxyphenylacetic acid (DOPAC) as an index of retinal dopamine release.
Journal: Journal of neurochemistry20010301
Title: Characterization of extracellular dopamine clearance in the medial prefrontal cortex: role of monoamine uptake and monoamine oxidase inhibition.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience20010101
Title: Different sensitivity of mitochondrial and cytosolic monoamine oxidases to in vivo but not in vitro inhibition by specific irreversible inhibitors.
Journal: Medical science monitor : international medical journal of experimental and clinical research20010101
Title: Glutamate regulates the spontaneous and evoked release of dopamine in the rat striatum.
Journal: Neuroscience20010101
Title: Novel propargylamine-linked nucleosides for high throughput SNP genotyping by MALDI-TOF MS.
Journal: Nucleosides, nucleotides & nucleic acids20010101
Title: Differential trace amine alterations in individuals receiving acetylenic inhibitors of MAO-A (clorgyline) or MAO-B (selegiline and pargyline).
Journal: Journal of neural transmission. Supplementum19980101
Title: Mechanism-based inactivation of porcine kidney diamine oxidase by 1,4-diamino-2-butene.
Journal: Biochimica et biophysica acta19951115
Title: The MAO-B inhibitor deprenyl, but not the MAO-A inhibitor clorgyline, potentiates the neurotoxicity of p-chloroamphetamine.
Journal: Brain research19940711
Title: The involvement of noradrenaline, 5-hydroxytryptamine and acetylcholine in imipramine-induced seizures in mice.
Journal: Experientia19931015
Title: Deprenyl (selegiline), a selective MAO-B inhibitor with active metabolites; effects on locomotor activity, dopaminergic neurotransmission and firing rate of nigral dopamine neurons.
Journal: The Journal of pharmacology and experimental therapeutics19911101
Title: Inhibition of human brain aromatic L-amino acid decarboxylase by cooked food-derived 3-amino-1-methyl-5H-pyrido[4,3-b]indole (Trp-P-2) and other heterocyclic amines.
Journal: Neuroscience letters19900824
Title: Synthesis and quantitative structure-activity relationship analysis of N-triiodoallyl- and N-iodopropargylazoles. New antifungal agents.
Journal: Journal of medicinal chemistry19870301
Title: Pargyline reduces/prevents neuroleptic-induced acute dystonia in monkeys.
Journal: Psychopharmacology19870101
Title: SR 95191, a selective inhibitor of type A monoamine oxidase with dopaminergic properties. I. Psychopharmacological profile in rodents.
Journal: The Journal of pharmacology and experimental therapeutics19870101
Title: Diazepam-induced decrease in histamine turnover in mouse brain.
Journal: European journal of pharmacology19860527
Title: [Effects of pentoxifylline on 5-hydroxytryptamine in the mouse brain].
Journal: Nihon yakurigaku zasshi. Folia pharmacologica Japonica19851101
Title: Chronic but not acute treatment with antidepressants enhances the electroconvulsive seizure response in rats.
Journal: Neuropharmacology19851001
Title: Treatment with clorgyline and pargyline differentially decreases clonidine-induced hypotension and bradycardia.
Journal: Naunyn-Schmiedeberg's archives of pharmacology19840901
Title: Testicular toxicity produced by ethylene glycol monomethyl and monoethyl ethers in the rat.
Journal: Environmental health perspectives19840801
Title: Brain monoamine oxidase in suckling rabbits treated with organophosphorus compound. I. Acute intoxication.
Journal: Acta physiologica Polonica19840101
Title: Pargyline-induced mania in primary affective disorder: case report.
Journal: The Journal of clinical psychiatry19830101
Title: The nature of the inhibition of rat liver monoamine oxidase types A and B by the acetylenic inhibitors clorgyline, l-deprenyl and pargyline.
Journal: Biochemical pharmacology19821115
Title: Selective and nonselective monoamine oxidase inhibitors: behavioral disturbances during their administration to depressed patients.
Journal: Archives of general psychiatry19820501
Title: Testosterone-attenuated stereotype and hyperactivity induced by beta-phenylethylamine in pargyline-pretreated rats.
Journal: Biological psychiatry19780801
Title: Role of the sympathetic nervous system in daunomycin-induced arrhythmia in the monkey.
Journal: British journal of pharmacology19700701
Title: Effect of certain monoamine oxidase inhibitors on isoproterenol-induced cardiac necrosis in rats.
Journal: Proceedings of the Western Pharmacology Society19660101
