[1]Locationinpatent:experimentalpartNegoro,Kenji;Yonetoku,Yasuhiro;Maruyama,Tatsuya;Yoshida,Shigeru;Takeuchi,Makoto;Ohta,Mitsuaki[BioorganicandMedicinalChemistry,2012,vol.20,#7,p.2369-2375]
[1]Negoro,Kenji;Yonetoku,Yasuhiro;Maruyama,Tatsuya;Yoshida,Shigeru;Takeuchi,Makoto;Ohta,Mitsuaki[BioorganicandMedicinalChemistry,2012,vol.20,#7,p.2369-2375]
[1]Negoro,Kenji;Yonetoku,Yasuhiro;Maruyama,Tatsuya;Yoshida,Shigeru;Takeuchi,Makoto;Ohta,Mitsuaki[BioorganicandMedicinalChemistry,2012,vol.20,#7,p.2369-2375]
[1]Negoro,Kenji;Yonetoku,Yasuhiro;Maruyama,Tatsuya;Yoshida,Shigeru;Takeuchi,Makoto;Ohta,Mitsuaki[BioorganicandMedicinalChemistry,2012,vol.20,#7,p.2369-2375]
Title: Synthesis and structure-activity relationship of 4-amino-2-phenylpyrimidine derivatives as a series of novel GPR119 agonists.
Journal: Bioorganic & medicinal chemistry 20120401
Title: Synthesis and SAR studies of 1,4-benzoxazine MenB inhibitors: novel antibacterial agents against Mycobacterium tuberculosis.
Journal: Bioorganic & medicinal chemistry letters 20101101
Title: Identification of a novel GPR119 agonist, AS1269574, with in vitro and in vivo glucose-stimulated insulin secretion.
Journal: Biochemical and biophysical research communications 20100924
Title: Yoshida S, et al. Identification of a novel GPR119 agonist, AS1269574, with in vitro and in vivo glucose-stimulated insulin secretion. Biochem Biophys Res Commun. 2010;400(3):437-441.
Title: Chepurny OG, et al. GPR119 Agonist AS1269574 Activates TRPA1 Cation Channels to Stimulate GLP-1 Secretion. Mol Endocrinol. 2016;30(6):614-629.