[1]BioorganicandMedicinalChemistryLetters,2011,vol.21,#20,p.6031-6035
[2]Patent:EP1889836,2008,A1,
[1]Patent:WO2004/112793,2004,A1,.Locationinpatent:Page/Pagecolumn126
[1]Patent:US2005/54697,2005,A1,.Locationinpatent:Page/Pagecolumn78
[2]BioorganicandMedicinalChemistryLetters,2009,vol.19,#4,p.1084-1088
[3]Patent:WO2011/61214,2011,A1,.Locationinpatent:Page/Pagecolumn85-86
[4]Patent:US2014/288045,2014,A1,.Locationinpatent:Paragraph0605
[5]Patent:WO2016/44772,2016,A1,.Locationinpatent:Paragraph319
[6]Patent:US2016/207883,2016,A1,.Locationinpatent:Paragraph0394-0396
[7]Patent:WO2013/14448,2013,A1,.Locationinpatent:Page/Pagecolumn95;96
[8]Patent:WO2016/30310,2016,A1,.Locationinpatent:Page/Pagecolumn49
[9]Patent:WO2013/10453,2013,A1,.Locationinpatent:Page/Pagecolumn135
[10]MedicinalChemistryResearch,2013,vol.22,#12,p.5982-5989
[11]JournalofChemicalResearch-PartS,1996,#9,p.430-431
[12]Patent:WO2006/72353,2006,A1,.Locationinpatent:Page/Pagecolumn51-52
[13]Patent:WO2012/101654,2012,A2,.Locationinpatent:Page/Pagecolumn63
[14]Patent:EP1889836,2008,A1,.Locationinpatent:Page/Pagecolumn79
[15]Patent:US2008/214815,2008,A1,.Locationinpatent:Page/Pagecolumn13-14
[16]Patent:EP2119706,2009,A1,.Locationinpatent:Page/Pagecolumn47-48
[17]JournalofOrganicChemistry,1991,vol.56,#24,p.6729-6730
[18]JournalofMedicinalChemistry,1993,vol.36,#7,p.801-810
[19]JournalofChemicalResearch,2006,#7,p.478-480
[20]Patent:US2001/27193,2001,A1,
[21]Patent:US5846965,1998,A,
[22]Patent:US6242438,2001,B1,
[23]Patent:US6262075,2001,B1,
[24]Patent:WO2007/26207,2007,A1,.Locationinpatent:Page/Pagecolumn3
[25]Patent:EP1813610,2007,A1,.Locationinpatent:Page/Pagecolumn10
[26]Patent:US2007/254892,2007,A1,.Locationinpatent:Page/Pagecolumn38
[27]Patent:EP1918284,2008,A1,.Locationinpatent:Page/Pagecolumn33
[28]Patent:WO2008/60767,2008,A2,.Locationinpatent:Page/Pagecolumn122-123
[29]Patent:US2009/233904,2009,A1,.Locationinpatent:Page/Pagecolumn78
[30]BioorganicandMedicinalChemistryLetters,2009,vol.19,#5,p.1517-1521
[31]Patent:US2010/249399,2010,A1,.Locationinpatent:Page/Pagecolumn21
[32]BioorganicandMedicinalChemistryLetters,2011,vol.21,#20,p.6031-6035
[33]Patent:WO2012/76063,2012,A1,.Locationinpatent:Page/Pagecolumn44-45
[34]OrganicProcessResearchandDevelopment,2012,vol.16,#5,p.788-797
[35]Patent:US2013/261100,2013,A1,.Locationinpatent:Paragraph0314-0315
[36]OrganicLetters,2014,vol.16,#10,p.2744-2747
[37]Patent:EP2805946,2014,A1,.Locationinpatent:Paragraph0115;0116
[38]Patent:US2014/357613,2014,A1,.Locationinpatent:Paragraph0151;0152
[39]Patent:WO2008/107368,2008,A1,.Locationinpatent:Page/Pagecolumn40
[1]Patent:US2010/190771,2010,A1,.Locationinpatent:Page/Pagecolumn28-29
[2]JournalofMedicinalChemistry,2012,vol.55,#21,p.9055-9068
[1]Patent:EP1591443,2005,A1,.Locationinpatent:Page/Pagecolumn67
[1]CurrentPatentAssignee:EISAICOLTD-EP1889836,2008,A1Locationinpatent:Page/Pagecolumn79
[2]Frigola;Pares;Corbera;Vano;Merce;Torrens;Mas;Valenti[JournalofMedicinalChemistry,1993,vol.36,#7,p.801-810]
[1]Phosphorus,SulfurandSiliconandtheRelatedElements,1991,vol.56,p.1-4
[1]Heterocycles,1986,vol.24,p.2467-2470
[1]Patent:US2005/54697,2005,A1.Locationinpatent:Page/Pagecolumn78
[2]BioorganicandMedicinalChemistryLetters,2009,vol.19,p.1084-1088
[3]Patent:WO2011/61214,2011,A1.Locationinpatent:Page/Pagecolumn85-86
[4]Patent:US2014/288045,2014,A1.Locationinpatent:Paragraph0605
[5]Patent:WO2016/44772,2016,A1.Locationinpatent:Paragraph319
[6]Patent:US2016/207883,2016,A1.Locationinpatent:Paragraph0394-0396
[7]Patent:WO2019/238633,2019,A1.Locationinpatent:Page/Pagecolumn129
[8]Patent:WO2013/14448,2013,A1.Locationinpatent:Page/Pagecolumn95;96
[9]JournalofOrganicChemistry,2019,vol.84,p.1363-1371
[10]Patent:WO2016/30310,2016,A1.Locationinpatent:Page/Pagecolumn49
[11]Patent:WO2013/10453,2013,A1.Locationinpatent:Page/Pagecolumn135
[12]MedicinalChemistryResearch,2013,vol.22,p.5982-5989
[13]JournalofChemicalResearch-PartS,1996,p.430-431
[14]Patent:WO2006/72353,2006,A1.Locationinpatent:Page/Pagecolumn51-52
[15]Patent:WO2012/101654,2012,A2.Locationinpatent:Page/Pagecolumn63
[16]Patent:EP1889836,2008,A1.Locationinpatent:Page/Pagecolumn79
[17]Patent:US2008/214815,2008,A1.Locationinpatent:Page/Pagecolumn13-14
[18]Patent:EP2119706,2009,A1.Locationinpatent:Page/Pagecolumn47-48
[19]JournalofOrganicChemistry,1991,vol.56,p.6729-6730
[20]JournalofMedicinalChemistry,1993,vol.36,p.801-810
[21]JournalofChemicalResearch,2006,p.478-480
[22]Patent:US2001/27193,2001,A1
[23]Patent:US5846965,1998,A
[24]Patent:US6242438,2001,B1
[25]Patent:US6262075,2001,B1
[26]Patent:WO2007/26207,2007,A1.Locationinpatent:Page/Pagecolumn3
[27]Patent:EP1813610,2007,A1.Locationinpatent:Page/Pagecolumn10
[28]Patent:US2007/254892,2007,A1.Locationinpatent:Page/Pagecolumn38
[29]Patent:EP1918284,2008,A1.Locationinpatent:Page/Pagecolumn33
[30]Patent:WO2008/60767,2008,A2.Locationinpatent:Page/Pagecolumn122-123
[31]Patent:US2009/233904,2009,A1.Locationinpatent:Page/Pagecolumn78
[32]BioorganicandMedicinalChemistryLetters,2009,vol.19,p.1517-1521
[33]Patent:US2010/249399,2010,A1.Locationinpatent:Page/Pagecolumn21
[34]BioorganicandMedicinalChemistryLetters,2011,vol.21,p.6031-6035
[35]Patent:WO2012/76063,2012,A1.Locationinpatent:Page/Pagecolumn44-45
[36]OrganicProcessResearchandDevelopment,2012,vol.16,p.788-797
[37]Patent:US2013/261100,2013,A1.Locationinpatent:Paragraph0314-0315
[38]OrganicLetters,2014,vol.16,p.2744-2747
[39]Patent:EP2805946,2014,A1.Locationinpatent:Paragraph0115;0116
[40]Patent:US2014/357613,2014,A1.Locationinpatent:Paragraph0151;0152
[41]Patent:WO2008/107368,2008,A1.Locationinpatent:Page/Pagecolumn40
[42]Patent:WO2019/118612,2019,A1.Locationinpatent:Paragraph0226
[1]Patent:WO2013/14448,2013,A1.Locationinpatent:Page/Pagecolumn95
[2]ChemicalandPharmaceuticalBulletin,1993,vol.41,p.126-131
[3]JournalofMedicinalChemistry,1993,vol.36,p.801-810
[4]Patent:CN106810553,2017,A.Locationinpatent:Paragraph0093-0094