Title: Discovery of a selective allosteric M1 receptor modulator with suitable development properties based on a quinolizidinone carboxylic acid scaffold.
Journal: Journal of medicinal chemistry 20110714
Title: Quinolizidinone carboxylic acid selective M1 allosteric modulators: SAR in the piperidine series.
Journal: Bioorganic & medicinal chemistry letters 20110315
Title: Heterocyclic fused pyridone carboxylic acid M(1) positive allosteric modulators.
Journal: Bioorganic & medicinal chemistry letters 20100415
Title: N-heterocyclic derived M1 positive allosteric modulators.
Journal: Bioorganic & medicinal chemistry letters 20100215
Title: Pyridine containing M(1) positive allosteric modulators with reduced plasma protein binding.
Journal: Bioorganic & medicinal chemistry letters 20100115
Title: Parallel synthesis of N-biaryl quinolone carboxylic acids as selective M(1) positive allosteric modulators.
Journal: Bioorganic & medicinal chemistry letters 20100115
Title: Microsphere-based protease assays and screening application for lethal factor and factor Xa.
Journal: Cytometry. Part A : the journal of the International Society for Analytical Cytology 20060501
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