Title: Molecular cloning, characterization, and inhibition studies of a β-carbonic anhydrase from Malassezia globosa, a potential antidandruff target.
Journal: Journal of medicinal chemistry 20120412
Title: Design and synthesis of thiourea compounds that inhibit transmembrane anchored carbonic anhydrases.
Journal: Bioorganic & medicinal chemistry 20120401
Title: Mutation of active site residues Asn67 to Ile, Gln92 to Val and Leu204 to Ser in human carbonic anhydrase II: influences on the catalytic activity and affinity for inhibitors.
Journal: Bioorganic & medicinal chemistry 20120401
Title: Cloning, characterization and sulfonamide inhibition studies of an α-carbonic anhydrase from the living fossil sponge Astrosclera willeyana.
Journal: Bioorganic & medicinal chemistry 20120215
Title: Inhibition studies of the β-carbonic anhydrases from the bacterial pathogen Salmonella enterica serovar Typhimurium with sulfonamides and sulfamates.
Journal: Bioorganic & medicinal chemistry 20110815
Title: Inhibition of hypoxia-inducible carbonic anhydrase-IX enhances hexokinase II inhibitor-induced hepatocellular carcinoma cell apoptosis.
Journal: Acta pharmacologica Sinica 20110701
Title: A new β-carbonic anhydrase from Brucella suis, its cloning, characterization, and inhibition with sulfonamides and sulfamates, leading to impaired pathogen growth.
Journal: Bioorganic & medicinal chemistry 20110201
Title: Carbonic anhydrase inhibitors. Inhibition studies with anions and sulfonamides of a new cytosolic enzyme from the scleractinian coral Stylophora pistillata.
Journal: Bioorganic & medicinal chemistry letters 20110115
Title: Synthesis and SAR studies of 1,4-benzoxazine MenB inhibitors: novel antibacterial agents against Mycobacterium tuberculosis.
Journal: Bioorganic & medicinal chemistry letters 20101101
Title: Mutation of Phe91 to Asn in human carbonic anhydrase I unexpectedly enhanced both catalytic activity and affinity for sulfonamide inhibitors.
Journal: Bioorganic & medicinal chemistry 20100801
Title: Low noise detection of biomolecular interactions with signal-locking surface plasmon resonance.
Journal: Analytical chemistry 20100715
Title: Synthesis and biological evaluation of a 99mTc-labelled sulfonamide conjugate for in vivo visualization of carbonic anhydrase IX expression in tumor hypoxia.
Journal: Nuclear medicine and biology 20100701
Title: 3D-QSAR study of benzene sulfonamide analogs as carbonic anhydrase II inhibitors.
Journal: Bioorganic & medicinal chemistry letters 20100515
Title: Cloning, characterization, and inhibition studies of a beta-carbonic anhydrase from Brucella suis.
Journal: Journal of medicinal chemistry 20100311
Title: Probing protein binding spectra with Fourier microfluidics.
Journal: Conference proceedings : ... Annual International Conference of the IEEE Engineering in Medicine and Biology Society. IEEE Engineering in Medicine and Biology Society. Annual Conference 20100101
Title: Carbonic anhydrase inhibitors. Characterization and inhibition studies of the most active beta-carbonic anhydrase from Mycobacterium tuberculosis, Rv3588c.
Journal: Bioorganic & medicinal chemistry letters 20091201
Title: 4-{2-[(5-Bromo-2-hydroxy-benzyl-idene)amino]eth-yl}benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20091001
Title: Carbonic anhydrase inhibitors. Inhibition of the Rv1284 and Rv3273 beta-carbonic anhydrases from Mycobacterium tuberculosis with diazenylbenzenesulfonamides.
Journal: Bioorganic & medicinal chemistry letters 20090901
Title: Carbonic anhydrase inhibitors. Inhibition studies of a coral secretory isoform by sulfonamides.
Journal: Bioorganic & medicinal chemistry 20090715
Title: Carbonic anhydrase inhibitors. Inhibition and homology modeling studies of the fungal beta-carbonic anhydrase from Candida albicans with sulfonamides.
Journal: Bioorganic & medicinal chemistry 20090701
Title: Carbonic anhydrase inhibitors. Cloning, characterization, and inhibition studies of a new beta-carbonic anhydrase from Mycobacterium tuberculosis.
Journal: Journal of medicinal chemistry 20090514
Title: Molecular cloning, characterization, and inhibition studies of the Rv1284 beta-carbonic anhydrase from Mycobacterium tuberculosis with sulfonamides and a sulfamate.
Journal: Journal of medicinal chemistry 20090423
Title: Carbonic anhydrase inhibitors. Biphenylsulfonamides with inhibitory action towards the transmembrane, tumor-associated isozymes IX possess cytotoxic activity against human colon, lung and breast cancer cell lines.
Journal: Journal of enzyme inhibition and medicinal chemistry 20090401
Title: Carbonic anhydrase inhibitors: inhibition of the beta-class enzyme from the yeast Saccharomyces cerevisiae with sulfonamides and sulfamates.
Journal: Bioorganic & medicinal chemistry 20090201
Title: LC and LC-MS study on establishment of degradation pathway of glipizide under forced decomposition conditions.
Journal: Journal of chromatographic science 20080701
Title: 4-{2-[(5-Chloro-2-hydroxy-benzyl-idene)amino]eth-yl}benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20080401
Title: The alpha-carbonic anhydrase from the malaria parasite and its inhibition.
Journal: Current pharmaceutical design 20080101
Title: Carbonic anhydrase inhibitors: cloning, characterization, and inhibition studies of the cytosolic isozyme III with sulfonamides.
Journal: Bioorganic & medicinal chemistry 20071201
Title: Carbonic anhydrase inhibitors: the beta-carbonic anhydrase from Helicobacter pylori is a new target for sulfonamide and sulfamate inhibitors.
Journal: Bioorganic & medicinal chemistry letters 20070701
Title: Carbonic anhydrase inhibitors. DNA cloning, characterization, and inhibition studies of the human secretory isoform VI, a new target for sulfonamide and sulfamate inhibitors.
Journal: Journal of medicinal chemistry 20070125
Title: Malarial parasite carbonic anhydrase and its inhibitors.
Journal: Current topics in medicinal chemistry 20070101
Title: Microsphere-based protease assays and screening application for lethal factor and factor Xa.
Journal: Cytometry. Part A : the journal of the International Society for Analytical Cytology 20060501
Title: Carbonic anhydrase inhibitors: cloning and sulfonamide inhibition studies of a carboxyterminal truncated alpha-carbonic anhydrase from Helicobacter pylori.
Journal: Bioorganic & medicinal chemistry letters 20060415
Title: QSAR study on topically acting sulfonamides incorporating GABA moieties: a molecular connectivity approach.
Journal: Bioorganic & medicinal chemistry letters 20060401
Title: Antibacterial, antifungal and cytotoxic properties of some sulfonamide-derived chromones.
Journal: Journal of enzyme inhibition and medicinal chemistry 20060401
Title: Carbonic anhydrase inhibitors: DNA cloning and inhibition studies of the alpha-carbonic anhydrase from Helicobacter pylori, a new target for developing sulfonamide and sulfamate gastric drugs.
Journal: Journal of medicinal chemistry 20060323
Title: Carbonic anhydrase inhibitors. The mitochondrial isozyme VB as a new target for sulfonamide and sulfamate inhibitors.
Journal: Journal of medicinal chemistry 20051201
Title: Carbonic anhydrase inhibitors: inhibition of the human transmembrane isozyme XIV with a library of aromatic/heterocyclic sulfonamides.
Journal: Bioorganic & medicinal chemistry 20051115
Title: Carbonic anhydrase inhibitors: inhibition of the tumor-associated isozymes IX and XII with a library of aromatic and heteroaromatic sulfonamides.
Journal: Bioorganic & medicinal chemistry letters 20051101
Title: Carbonic anhydrase inhibitors: inhibition of the transmembrane isozyme XIV with sulfonamides.
Journal: Bioorganic & medicinal chemistry letters 20050901
Title: Carbonic anhydrase inhibitors. Inhibition of red blood cell ostrich (Struthio camelus) carbonic anhydrase with a series of aromatic and heterocyclic sulfonamides.
Journal: Journal of enzyme inhibition and medicinal chemistry 20050801
Title: Carbonic anhydrase inhibitors. Design of fluorescent sulfonamides as probes of tumor-associated carbonic anhydrase IX that inhibit isozyme IX-mediated acidification of hypoxic tumors.
Journal: Journal of medicinal chemistry 20050728
Title: Carbonic anhydrase inhibitors: novel sulfonamides incorporating 1,3,5-triazine moieties as inhibitors of the cytosolic and tumour-associated carbonic anhydrase isozymes I, II and IX.
Journal: Bioorganic & medicinal chemistry letters 20050615
Title: Carbonic anhydrase inhibitors. Inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, IX, and XII with Schiff's bases incorporating chromone and aromatic sulfonamide moieties, and their zinc complexes.
Journal: Bioorganic & medicinal chemistry letters 20050615
Title: Carbonic anhydrase inhibitors: synthesis and inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, and IX with sulfonamides incorporating thioureido-sulfanilyl scaffolds.
Journal: Bioorganic & medicinal chemistry letters 20050502
Title: Carbonic anhydrase inhibitors. Inhibition of the transmembrane isozyme XII with sulfonamides-a new target for the design of antitumor and antiglaucoma drugs?
Journal: Bioorganic & medicinal chemistry letters 20050215
Title: Carbonic anhydrase inhibitors. Inhibition of the human cytosolic isozyme VII with aromatic and heterocyclic sulfonamides.
Journal: Bioorganic & medicinal chemistry letters 20050215
Title: Carbonic anhydrase inhibitors. Inhibition of the membrane-bound human and bovine isozymes IV with sulfonamides.
Journal: Bioorganic & medicinal chemistry letters 20050215
Title: Carbonic anhydrase inhibitors. Inhibition of the prokariotic beta and gamma-class enzymes from Archaea with sulfonamides.
Journal: Bioorganic & medicinal chemistry letters 20041220
Title: Carbonic anhydrase inhibitors: inhibition of human cytosolic isozyme II and mitochondrial isozyme V with a series of benzene sulfonamide derivatives.
Journal: Bioorganic & medicinal chemistry letters 20041115
Title: Carbonic anhydrase inhibitors: synthesis and inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, and IX with sulfonamides incorporating 1,2,4-triazine moieties.
Journal: Bioorganic & medicinal chemistry letters 20041101
Title: Carbonic anhydrase inhibitors. Inhibition of cytosolic isozyme XIII with aromatic and heterocyclic sulfonamides: a novel target for the drug design.
Journal: Bioorganic & medicinal chemistry letters 20040716
Title: Carbonic anhydrase inhibitors: the first QSAR study on inhibition of tumor-associated isoenzyme IX with aromatic and heterocyclic sulfonamides.
Journal: Bioorganic & medicinal chemistry letters 20040621
Title: Carbonic anhydrase inhibitors: Schiff's bases of aromatic and heterocyclic sulfonamides and their metal complexes.
Journal: Journal of enzyme inhibition and medicinal chemistry 20040601
Title: Carbonic anhydrase inhibitors. Inhibition of mitochondrial isozyme V with aromatic and heterocyclic sulfonamides.
Journal: Journal of medicinal chemistry 20040226
Title: Carbonic anhydrase inhibitors: the first selective, membrane-impermeant inhibitors targeting the tumor-associated isozyme IX.
Journal: Bioorganic & medicinal chemistry letters 20040223
Title: Carbonic anhydrase inhibitors: X-ray crystallographic structure of the adduct of human isozyme II with a bis-sulfonamide-two heads are better than one?
Journal: Bioorganic & medicinal chemistry letters 20030818
Title: Carbonic anhydrase inhibitors: inhibition of the tumor-associated isozyme IX with aromatic and heterocyclic sulfonamides.
Journal: Bioorganic & medicinal chemistry letters 20030324
Title: A simple LC method with UV detection for the analysis of creatine and creatinine and its application to several creatine formulations.
Journal: Journal of pharmaceutical and biomedical analysis 20020731
Title: Carbonic anhydrase inhibitors. A general approach for the preparation of water-soluble sulfonamides incorporating polyamino-polycarboxylate tails and of their metal complexes possessing long-lasting, topical intraocular pressure-lowering properties.
Journal: Journal of medicinal chemistry 20020328
Title: Carbonic anhydrase inhibitors: synthesis of sulfonamides incorporating dtpa tails and of their zinc complexes with powerful topical antiglaucoma properties.
Journal: Bioorganic & medicinal chemistry letters 20010226
