Title: Radiofluorinated histamine H₃ receptor antagonist as a potential probe for in vivo PET imaging: radiosynthesis and pharmacological evaluation.
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Title: Novel and highly potent histamine H3 receptor ligands. Part 2: exploring the cyclohexylamine-based series.
Journal: Bioorganic & medicinal chemistry letters 20110915
Title: Histamine H3 receptor as a drug discovery target.
Journal: Journal of medicinal chemistry 20110113
Title: Indole- and benzothiophene-based histamine H3 antagonists.
Journal: Bioorganic & medicinal chemistry letters 20101101
Title: Novel substituted pyrrolidines are high affinity histamine H3 receptor antagonists.
Journal: Bioorganic & medicinal chemistry letters 20100501
Title: Acidic elements in histamine H(3) receptor antagonists.
Journal: Bioorganic & medicinal chemistry letters 20100301
Title: Heterocyclic replacement of the central phenyl core of diamine-based histamine H3 receptor antagonists.
Journal: European journal of medicinal chemistry 20091101
Title: 5-hydroxyindole-2-carboxylic acid amides: novel histamine-3 receptor inverse agonists for the treatment of obesity.
Journal: Journal of medicinal chemistry 20090709
Title: Fluorinated non-imidazole histamine H3 receptor antagonists.
Journal: Bioorganic & medicinal chemistry letters 20090415
Title: 2-Aryloxymethylmorpholine histamine H(3) antagonists.
Journal: Bioorganic & medicinal chemistry letters 20081101
Title: Diamine derivatives containing imidazolidinylidene propanedinitrile as a new class of histamine H3 receptor antagonists. Part I.
Journal: Bioorganic & medicinal chemistry letters 20080401
Title: Lead identification of acetylcholinesterase inhibitors-histamine H3 receptor antagonists from molecular modeling.
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Title: Benzylamine histamine H(3) antagonists and serotonin reuptake inhibitors.
Journal: Bioorganic & medicinal chemistry letters 20070901
Title: A new class of histamine H3 receptor antagonists derived from ligand based design.
Journal: Bioorganic & medicinal chemistry letters 20070701
Title: Histamine H3 receptor antagonists: from target identification to drug leads.
Journal: Biochemical pharmacology 20070415
Title: 4-[6-(2-Aminoethyl)naphthalen-2-yl]benzonitriles are potent histamine H3 receptor antagonists with high CNS penetration.
Journal: Bioorganic & medicinal chemistry letters 20070301
Title: Microsphere-based protease assays and screening application for lethal factor and factor Xa.
Journal: Cytometry. Part A : the journal of the International Society for Analytical Cytology 20060501
Title: Effects of histamine H(3) antagonists and donepezil on learning and mnemonic deficits induced by pentylenetetrazol kindling in weanling mice.
Journal: Neuropharmacology 20060301
Title: Aplysamine-1 and related analogs as histamine H3 receptor antagonists.
Journal: Bioorganic & medicinal chemistry letters 20060215
Title: 4-phenoxypiperidines: potent, conformationally restricted, non-imidazole histamine H3 antagonists.
Journal: Journal of medicinal chemistry 20050324
Title: 2-(4-alkylpiperazin-1-yl)quinolines as a new class of imidazole-free histamine H3 receptor antagonists.
Journal: Journal of medicinal chemistry 20050113
Title: Acute wake-promoting actions of JNJ-5207852, a novel, diamine-based H3 antagonist.
Journal: British journal of pharmacology 20041101
Title: A new class of diamine-based human histamine H3 receptor antagonists: 4-(aminoalkoxy)benzylamines.
Journal: Journal of medicinal chemistry 20030828
Title: Barbier AJ, et al. Acute wake-promoting actions of JNJ-5207852, a novel, diamine-based H3 antagonist. Br J Pharmacol. 2004 Nov;143(5):649-61.
Title: Abuhamdah RM, et al. Effects of methimepip and JNJ-5207852 in Wistar rats exposed to an open-field with and without object and in Balb/c mice exposed to a radial-arm maze. Front Syst Neurosci. 2012 Jul 16;6:54.