Home Fluorides 5002-47-1
5002-47-1,MFCD00798504
Catalog No.:AA006WP8

5002-47-1 | 2-(4-{3-[2-(trifluoromethyl)-10H-phenothiazin-10-yl]propyl}piperazin-1-yl)ethyl decanoate

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Purity
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5mg
98%(HPLC)
in stock  
$81.00   $57.00
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25mg
98%(HPLC)
in stock  
$161.00   $113.00
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100mg
98%
in stock  
$278.00   $195.00
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250mg
98%
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$544.00   $381.00
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1g
98%
in stock  
$1,424.00   $997.00
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  • Technical Information
  • Properties
  • Literature
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  • Technical Information
  • Properties
  • Literature
Technical Information
Catalog Number:
AA006WP8
Chemical Name:
2-(4-{3-[2-(trifluoromethyl)-10H-phenothiazin-10-yl]propyl}piperazin-1-yl)ethyl decanoate
CAS Number:
5002-47-1
Molecular Formula:
C32H44F3N3O2S
Molecular Weight:
591.7709
MDL Number:
MFCD00798504
SMILES:
CCCCCCCCCC(=O)OCCN1CCN(CC1)CCCN1c2ccccc2Sc2c1cc(cc2)C(F)(F)F
NSC Number:
169510
Properties
Properties
 
BP:
658.1±55.0 °C(Predicted)  
Form:
Solid  
MP:
30-32°  
Solubility:
Practically insoluble in water, very soluble in ethanol and in methylene chloride, freely soluble in methanol.  
Storage:
Keep in dry area;Room Temperature;  

Computed Properties
 
Complexity:
765  
Covalently-Bonded Unit Count:
1  
Heavy Atom Count:
41  
Hydrogen Bond Acceptor Count:
9  
Rotatable Bond Count:
16  
XLogP3:
9  

Literature

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Journal: American journal of hospital pharmacy 19940401

Title: Two cases of long term dopamine D2 receptor blockade after depot neuroleptics.

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Title: Positive and negative symptoms, depression and social disability in chronic schizophrenia: a comparative trial of bromperidol and fluphenazine decanoates.

Journal: International clinical psychopharmacology 19921101

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Title: Unusual treatment response of a severe dystonia to diphenhydramine.

Journal: Annals of emergency medicine 19870601

Title: A case of neuroleptic malignant syndrome in a mentally retarded adolescent.

Journal: Journal of adolescent health care : official publication of the Society for Adolescent Medicine 19861101

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Title: Catatonia associated with phenylpropanolamine overdose and fluphenazine treatment: case report.

Journal: The Journal of clinical psychiatry 19850701

Title: Costs and benefits of two doses of fluphenazine.

Journal: Archives of general psychiatry 19841101

Title: Fluphenazine decanoate-induced cholestatic jaundice and thrombocytopenia.

Journal: Pharmacotherapy 19840101

Title: Management of a case of neuroleptic malignant syndrome with bromocriptine.

Journal: The American journal of psychiatry 19831201

Title: Treatment of the neuroleptic malignant syndrome with bromocriptine.

Journal: JAMA 19830701

Title: Neuroleptic malignant syndrome: successful treatment with dantrolene and bromocriptine.

Journal: Annals of neurology 19830701

Title: Psychotropic-induced sexual inhibition.

Journal: The American journal of psychiatry 19830401

Title: Variation in oro-facial tardive dyskinesia during depot antipsychotic drug treatment.

Journal: Psychopharmacology 19830101

Title: Lithium carbonate/fluphenazine decanoate producing irreversible brain damage.

Journal: Lancet (London, England) 19820731

Title: Catatonic-like syndrome during neuroleptic therapy.

Journal: Psychosomatics 19820701

Title: Fluphenazine enanthate and fluphenazine decanoate in the treatment of schizophrenic outpatients: extrapyramidal symptoms and therapeutic effect.

Journal: The American journal of psychiatry 19820301

Title: Development and prediction of postpsychotic depression in neuroleptic-treated schizophrenics.

Journal: Archives of general psychiatry 19820201

Title: Neurotoxicity in patients with schizophrenia during lithium therapy.

Journal: Comprehensive psychiatry 19820101

Title: Catalepsy produced by long-acting neuroleptics, fluphenazine enanthate and fluphenazine decanoate, in mice.

Journal: Pharmacology 19820101

Title: Extrapyramidal reaction to fluphenazine potentiated by thyrotoxicosis.

Journal: The American journal of psychiatry 19810201

Title: Neuroleptic-induced syndrome mimicking myasthenia gravis.

Journal: Psychosomatics 19810101

Title: behavior of rats and mice administered active metabolites of fluphenazine, 7-hydroxy-fluphenazine and fluphenazine-sulfoxide.

Journal: Archives internationales de pharmacodynamie et de therapie 19801101

Title: Patients at risk of developing severe side effects from depot fluphenazine treatment.

Journal: The American journal of psychiatry 19800201

Title: Depressive and extrapyramidal symptoms and clinical effects: a trial of fluphenazine versus flupenthixol in maintenance of schizophrenic out-patients.

Journal: The British journal of psychiatry : the journal of mental science 19791201

Title: Endocrinological changes in patients with sexual dysfunction under long-term neuroleptic treatment.

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Title: Iatrogenic morbidity in patients taking depot fluphenazine.

Journal: The American journal of psychiatry 19790701

Title: Unwanted effects of fluphenazine enanthate and decanoate.

Journal: Lancet (London, England) 19790210

Title: Acute extrapyramidal reactions with fluphenazine hydrochloride and fluphenazine decanoate.

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Title: Neuroleptic malignant syndrome due to depot fluphenazine.

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Title: Comparison of the incidence and severity of extrapyramidal side effects with fluphenazine enanthate and fluphenazine decanoate.

Journal: The American journal of psychiatry 19781201

Title: Depot injections and tardive dyskinesia.

Journal: The British journal of psychiatry : the journal of mental science 19781001

Title: Double-blind therapeutic evaluation of fluspirilene compared with fluphenazine decanoate in chronic schizophrenics.

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Title: A comparison of piribedil, procyclidine and placebo in the control of phenothiazine-induced parkinsonism.

Journal: The British journal of psychiatry : the journal of mental science 19770601

Title: Comparison of antipsychotic depot injections in the maintenance treatment of schizophrenia.

Journal: The British journal of psychiatry : the journal of mental science 19761101

Title: Letter: Parkinsonism induced by fluphenazine decanoate.

Journal: Lancet (London, England) 19760227

Title: A comparative trial of orphenadrine and tofenacin in the control of depression and extrapyramidal side-effects associated with fluphenazine decanoate therapy.

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Title: [Complications of the treatment with long-acting neuroleptic preparations. Brain disease due to fluphenazine decanoate].

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Title: Antiparkinsonian agents and fluphenazine decanoate.

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Title: Letter: Potentiation of tardive dyskinesia: possible drug interaction.

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Title: A comparative trail of fluphenazine decanoate and flupenthixol decanoate.

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Title: Fluphenazine enanthate and fluphenazine decanoate: a comparison of their duration of action and motor side effects.

Journal: The American journal of psychiatry 19730701

Title: Institutional management of chronic schizophrenics with fluphenazine decanoate.

Journal: Diseases of the nervous system 19700901

Title: Severe depressive mood changes following slow-release intramuscular fluphenazine injection.

Journal: British medical journal 19690906

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Tags:5002-47-1 Molecular Formula|5002-47-1 MDL|5002-47-1 SMILES|5002-47-1 2-(4-{3-[2-(trifluoromethyl)-10H-phenothiazin-10-yl]propyl}piperazin-1-yl)ethyl decanoate