[1]Castaldi,Graziano;Cavicchioli,Silvia;Giordano,Claudio;Uggeri,Fulvio[JournalofOrganicChemistry,1987,vol.52,#14,p.3018-3027]
[1]Zhang,Kun;Rombach,David;Nötel,NicolasYannick;Jeschke,Gunnar;Katayev,Dmitry[AngewandteChemie-InternationalEdition,2021,vol.60,#41,p.22487-22495][Angew.Chem.,2021,vol.133,#41,p.22661-22669]
[2]Locationinpatent:experimentalpartHuang,Zhangjian;Velázquez,CarlosA.;Abdellatif,KhaledR.A.;Chowdhury,MorshedA.;Reisz,JulieA.;Dumond,JennaF.;King,S.Bruce;Knaus,EdwardE.[JournalofMedicinalChemistry,2011,vol.54,#5,p.1356-1364]
[3]Kariofillis,StavrosK.;Shields,BenjaminJ.;Tekle-Smith,MakedaA.;Zacuto,MichaelJ.;Doyle,AbigailG.[JournaloftheAmericanChemicalSociety,2020,vol.142,#16,p.7683-7689]
[4]Capim,SauloL.;Goncalves,GabrielaM.;DosSantos,GabrielaC.M.;Marinho,BrunoG.;Vasconcellos,MarioL.A.A.[BioorganicandMedicinalChemistry,2013,vol.21,#19,p.6003-6010]
[5]CurrentPatentAssignee:LONZAGROUPAG-WO2012/69423,2012,A1Locationinpatent:Page/Pagecolumn11
[6]Chaturvedi,Devdutt;Dwivedi,ParmeshKumar;Chaturvedi,AmitK.;Mishra,Nisha;Siddiqui;Mishra,Vorenda[MedicinalChemistryResearch,2015,vol.24,#7,p.2799-2812]
[7]Levit;Koroleva;Krasnov[RussianJournalofOrganicChemistry,1998,vol.34,#3,p.346-350]
[8]CurrentPatentAssignee:NICOXS.A.-WO2009/723,2008,A1Locationinpatent:Page/Pagecolumn28-29
[9]CurrentPatentAssignee:PRECIGENINC-WO2008/153801,2008,A1Locationinpatent:Page/Pagecolumn112-113
[10]Helal,MohamedH.;Abbas,SamirY.;Salem,MohamedA.;Farag,AwatefA.;Ammar,YousryA.[MedicinalChemistryResearch,2013,vol.22,#11,p.5598-5609]
[11]Castaldi,Graziano;Cavicchioli,Silvia;Giordano,Claudio;Uggeri,Fulvio[JournalofOrganicChemistry,1987,vol.52,#14,p.3018-3027]
[12]Spahn[ArchivderPharmazie,1988,vol.321,#12,p.847-850]
[13]Shan,Daxian;Zheng,Ailian;Ballard,C.Eric;Wang,Wei;Borchardt,RonaldT.;Wang,Binghe[ChemicalandPharmaceuticalBulletin,2000,vol.48,#2,p.238-244]
[14]Lin,Man-Yuan;Lay,Eddy;Wen,Wen-Yen;Dewi,Hamza;Cheng,Yu-Chi;Tsai,Shau-Wei[JournalofPhysicalOrganicChemistry,2004,vol.17,#5,p.387-392]
[15]Huang,Jian;Hsung,RichardP.[JournaloftheAmericanChemicalSociety,2005,vol.127,#1,p.50-51]
[16]Anilkumar,Gopinathan;Bhor,Santosh;Tse,ManKin;Klawonn,Markus;Bitterlich,Bianca;Beller,Matthias[TetrahedronAsymmetry,2005,vol.16,#21,p.3536-3561]
[17]Doulgkeris,ChristosM.;Galanakis,Dimitrios;Kourounakis,AngelikiP.;Tsiakitzis,KaryofyllisC.;Gavalas,AntoniosM.;Eleftheriou,PhaedraT.;Victoratos,Panagiotis;Rekka,EleniA.;Kourounakis,PanosN.[BioorganicandMedicinalChemistryLetters,2006,vol.16,#4,p.825-829]
[18]Reid;Stobaugh;Sternson[AnalyticalChemistry,1989,vol.61,#5,p.441-446]
[19]Weber;Meyer-Trumpener[ArchivderPharmazie,1994,vol.327,#5,p.337-345]
[20]Hyun,MyungHo;Hwang,Seung-Ryul;Ryoo,Jae-Jeong[ChemistryLetters,1994,#6,p.1021-1024]
[21]Georgiadis,TaxiarchisM.;Georgiadis,MillieM.;Diederich,Francois[JournalofOrganicChemistry,1991,vol.56,#10,p.3362-3369]
[22]Kerdesky,FrancisA.J.;Brooks,ClintD.W.;Hulkower,KerenI.;Bouska,JenniferB.;Bell,RandyL.[BioorganicandMedicinalChemistry,1997,vol.5,#2,p.393-396]
[23]Madhavan,G.V.Bindu;Martin,JohnC.[JournalofOrganicChemistry,1986,vol.51,#8,p.1287-1293]
[24]Brown,RichardJ.;Annis,Gary;Casalnuovo,Albert;Chan,Dominic;Shapiro,Rafael;Marshall,WilliamJ.[Tetrahedron,2004,vol.60,#20,p.4361-4375]
[25]Pischel,Uwe;Abad,Sergio;Miranda,MiguelA.[ChemicalCommunications,2003,#9,p.1088-1089]
[26]Yadav,MangeRam;Nimekar,DattaM.;Ananthakrishnan;Brahmkshatriya,PathikS.;Shirude,ShrikantT.;Giridhar,Rajani;Parmar,Arvind;Balaraman[BioorganicandMedicinalChemistry,2006,vol.14,#24,p.8701-8706]
[27]CurrentPatentAssignee:PIRAMALENTERPRISESLIMITED-US2006/46967,2006,A1Locationinpatent:Page/Pagecolumn114-115;145
[28]Wang;Chiang;Chen[JournalofPharmacyandPharmacology,2002,vol.54,#8,p.1129-1135]
[29]CurrentPatentAssignee:JIANGSUPUXINPHARMACEUTICALS-EP2161267,2010,A1Locationinpatent:Page/Pagecolumn11
[30]Duong,HungA.;Gilligan,RuthE.;Cooke,MichaelL.;Phipps,RobertJ.;Gaunt,MatthewJ.[AngewandteChemie-InternationalEdition,2011,vol.50,#2,p.463-466]
[31]Locationinpatent:experimentalpartVanPelt;Zhang;Otten;Holt;Sorokin;VanRantwijk;Black;Perry;Sheldon[OrganicandBiomolecularChemistry,2011,vol.9,#8,p.3011-3019]
[32]CurrentPatentAssignee:PIRAMALENTERPRISESLIMITED-US2011/263526,2011,A1Locationinpatent:Page/Pagecolumn77
[33]Locationinpatent:schemeortableMukhlall,JoshuaA.;Noll,BruceC.;Hersh,WilliamH.[JournalofSulfurChemistry,2011,vol.32,#3,p.199-212]
[34]Locationinpatent:experimentalpartSharma,PrabodhChander;Yadav,Sonia;Pahwa,Rakesh;Kaushik,Dhirender;Jain,Sandeep[MedicinalChemistryResearch,2011,vol.20,#5,p.648-655]
[35]Locationinpatent:experimentalpartBorhade,Namdev;Pathan,AsifRahimkhan;Halder,Somnath;Karwa,Manoj;Dhiman,Mini;Pamidiboina,Venu;Gund,Machhindra;Deshattiwar,JagannathJanardhan;Mali,SunilVasantrao;Deshmukh,NitinJanardanrao;Senthilkumar,SubrayanPalanisamy;Gaikwad,Parikshit;Tipparam,SanthoshGoud;Mudgal,Jayesh;Dutta,MilanChandra;Burhan,AslamUsmangani;Thakre,Gajanan;Sharma,Ankur;Deshpande,Shubhada;Desai,DattatrayaChandrakant;Dubash,NauzerPervez;Jain,ArunKumar;Sharma,Somesh;Nemmani,KumarVenkataSubrahmanya;Satyam,Apparao[ChemicalandPharmaceuticalBulletin,2012,vol.60,#4,p.465-481]
[36]Doulgkeris,ChristosM.;Siskou,IoannaC.;Xanthopoulou,Nikoletta;Lagouri,Vassiliki;Kravaritou,Constantina;Eleftheriou,Phaedra;Kourounakis,PanosN.;Rekka,EleniA.[MedicinalChemistryResearch,2012,vol.21,#9,p.2280-2291]
[37]Bhardwaj,Atul;Kaur,Jatinder;Sharma,SaiKiran;Huang,Zhangjian;Wuest,Frank;Knaus,EdwardE.[BioorganicandMedicinalChemistryLetters,2013,vol.23,#1,p.163-168]
[38]Yosef;Elmasry;Ismael,EmanH.I.;Mahran[EgyptianJournalofChemistry,2010,vol.53,#5,p.745-755]Yosef,HishamAbdallahA.;Elmasry;Ibrahim,NabilaM.;Ismael,EmanH.I.;Mahran[EgyptianJournalofChemistry,2017,vol.60,#2,p.301-328]
[39]Jain,ArunK.;Gund,MachhindraG.;Desai,DattatrayaC.;Borhade,Namdev;Senthilkumar,SubrayanP.;Dhiman,Mini;Mangu,NaveenK.;Mali,SunilV.;Dubash,NauzerP.;Halder,Somnath;Satyam,Apparao[BioorganicChemistry,2013,vol.49,p.40-48]
[40]Gruzdev,DmitryA.;Chulakov,EvgenyN.;Levit,GalinaL.;Ezhikova,MarinaA.;Kodess,MikhailI.;Krasnov,VictorP.[TetrahedronAsymmetry,2013,vol.24,#19,p.1240-1246]
[41]Yamagami,Takafumi;Hatsuda,Masanori;Utsugi,Masayuki;Kobayashi,Ryo;Moritani,Yasunori[EuropeanJournalofOrganicChemistry,2013,#33,p.7467-7470]
[42]Reddy,G.Prashanth;Bandichhor,Rakeshwar[AsianJournalofChemistry,2013,vol.25,#15,p.8701-8707]
[43]Raghavendra,NulgumnalliManjunathaiah;Ramakrishna,Kota;Sirisha,Vippula;Divya,Pingli;Rao,AlapatiVenkateswara[MedicinalChemistry,2013,vol.9,#4,p.553-559]
[44]Conda-Sheridan,Martin;Lee,SungsooS.;Preslar,AdamT.;Stupp,SamuelI.[ChemicalCommunications,2014,vol.50,#89,p.13757-13760]
[45]Gund,Machhindra;Gaikwad,Parikshit;Borhade,Namdev;Burhan,Aslam;Desai,DattatrayaC.;Sharma,Ankur;Dhiman,Mini;Patil,Mohan;Sheikh,Javed;Thakre,Gajanan;Tipparam,SanthoshG.;Sharma,Somesh;Nemmani,KumarV.S.;Satyam,Apparao[BioorganicandMedicinalChemistryLetters,2014,vol.24,#24,p.5587-5592]
[46]Xiong,Heng-Ying;Besset,Tatiana;Cahard,Dominique;Pannecoucke,Xavier[JournalofOrganicChemistry,2015,vol.80,#8,p.4204-4212]
[47]Scheidt,Thomas;Land,Henrik;Anderson,Mattias;Chen,Yujie;Berglund,Per;Yi,Dong;Fessner,Wolf-Dieter[AdvancedSynthesisandCatalysis,2015,vol.357,#8,p.1721-1731]
[48]Eissa;Farrag;Galeel[DrugResearch,2014,vol.64,#9,p.485-492]
[49]Yosef;Shaker,NihalO.;Morsy,NesrinM.;Mahran[EgyptianJournalofChemistry,2014,vol.57,#5-6,p.387-410]
[50]Montoya-Balbás,IrisJ.;Valentín-Guevara,Berenice;López-Mendoza,Estefanía;Linzaga-Elizalde,Irma;Ordoñez,Mario;Román-Bravo,Perla[Molecules,2015,vol.20,#12,p.22028-22043]
[51]Ullah,Nasir;Huang,Zhangjian;Sanaee,Forough;Rodriguez-Dimitrescu,Alexandra;Aldawsari,Fahad;Jamali,Fakhreddin;Bhardwaj,Atul;Islam,NazarUl;Velázquez-Martínez,CarlosA.[JournalofEnzymeInhibitionandMedicinalChemistry,2016,vol.31,#6,p.1018-1028]
[52]Theodosis-Nobelos,Panagiotis;Politou,TheodoraC.;Athanasekou,Chrysoula;Rekka,EleniA.[Lettersindrugdesignanddiscovery,2016,vol.14,#4,p.464-475]
[53]González-Trujano,MaríaEva;Uribe-Figueroa,Gerardo;Hidalgo-Figueroa,Sergio;Martínez,AnaLaura;Déciga-Campos,Myrna;Navarrete-Vazquez,Gabriel[BiomedicineandPharmacotherapy,2018,vol.101,p.553-562]
[54]CurrentPatentAssignee:ZHEJIANGUNIVERSITY-CN108250008,2018,ALocationinpatent:Paragraph0014
[55]CurrentPatentAssignee:WU,Yong-Qian;HAMILTON,Gregory,S.;BELYAKOV,Sergei;WALDON,Daniel-WO2006/138187,2006,A1Locationinpatent:Page/Pagecolumn33
[56]Elhenawy,AhmedA.;Al-Harbi;Moustafa,GaberO.;El-Gazzar;Abdel-Rahman,RehabF.;Salim,AbdElhamid[DrugDesign,DevelopmentandTherapy,2019,vol.13,p.1773-1790]
[57]Chen,Guojun;Wang,Liling;Liu,Xiaozu;Liu,Peijun[AdvancedSynthesisandCatalysis,2020,vol.362,#14,p.2990-2996]
[58]Cai,Jin;Duan,Yanbing;Yu,Jia;Chen,Junqing;Chao,Meng;Ji,Min[EuropeanJournalofMedicinalChemistry,2012,vol.55,p.409-419,11]
[59]Chulakov,E.N.;Levit,G.L.;Tumashov,A.A.;Sadretdinova,L.Sh.;Krasnov,V.P.[ChemistryofHeterocyclicCompounds,2012,vol.48,#5,p.724-732,9]
[60]Chen,Jin-Yang;Zhong,Chun-Tao;Gui,Qing-Wen;Zhou,Yuan-Ming;Fang,Yang-Yang;Liu,Kai-Jian;Lin,Ying-Wu;Cao,Zhong;He,Wei-Min[ChineseChemicalLetters,2021,vol.32,#1,p.475-479]
[1]Otevrel,Jan;Svestka,David;Bobal,Pavel[OrganicandBiomolecularChemistry,2019,vol.17,#21,p.5244-5248]
[2]Scheidt,Thomas;Land,Henrik;Anderson,Mattias;Chen,Yujie;Berglund,Per;Yi,Dong;Fessner,Wolf-Dieter[AdvancedSynthesisandCatalysis,2015,vol.357,#8,p.1721-1731]
[3]Kerdesky,FrancisA.J.;Brooks,ClintD.W.;Hulkower,KerenI.;Bouska,JenniferB.;Bell,RandyL.[BioorganicandMedicinalChemistry,1997,vol.5,#2,p.393-396]
[4]Locationinpatent:experimentalpartVanPelt;Zhang;Otten;Holt;Sorokin;VanRantwijk;Black;Perry;Sheldon[OrganicandBiomolecularChemistry,2011,vol.9,#8,p.3011-3019]
[5]Locationinpatent:experimentalpartBorhade,Namdev;Pathan,AsifRahimkhan;Halder,Somnath;Karwa,Manoj;Dhiman,Mini;Pamidiboina,Venu;Gund,Machhindra;Deshattiwar,JagannathJanardhan;Mali,SunilVasantrao;Deshmukh,NitinJanardanrao;Senthilkumar,SubrayanPalanisamy;Gaikwad,Parikshit;Tipparam,SanthoshGoud;Mudgal,Jayesh;Dutta,MilanChandra;Burhan,AslamUsmangani;Thakre,Gajanan;Sharma,Ankur;Deshpande,Shubhada;Desai,DattatrayaChandrakant;Dubash,NauzerPervez;Jain,ArunKumar;Sharma,Somesh;Nemmani,KumarVenkataSubrahmanya;Satyam,Apparao[ChemicalandPharmaceuticalBulletin,2012,vol.60,#4,p.465-481]
[6]Reddy,G.Prashanth;Bandichhor,Rakeshwar[AsianJournalofChemistry,2013,vol.25,#15,p.8701-8707]
[1]Sakai,Takashi;Miki,Yasushi;Tsuboi,Masashi;Takeuchi,Hiroaki;Ema,Tadashi;Uneyama,Kenji;Utaka,Masanori[JournalofOrganicChemistry,2000,vol.65,#9,p.2740-2747]
[2]Sakai,Takashi;Miki,Yasushi;Tsuboi,Masashi;Takeuchi,Hiroaki;Ema,Tadashi;Uneyama,Kenji;Utaka,Masanori[JournalofOrganicChemistry,2000,vol.65,#9,p.2740-2747]
[3]Sakai,Takashi;Miki,Yasushi;Nakatani,Mayumi;Ema,Tadashi;Uneyama,Kenji;Utaka,Masanori[TetrahedronLetters,1998,vol.39,#29,p.5233-5236]
[1]EuropeanJournalofPharmaceuticalSciences,2000,vol.11,p.157-163