Title: Betulinyl Sulfamates as Anticancer Agents and Radiosensitizers in Human Breast Cancer Cells.
Journal: International journal of molecular sciences 20151101
Title: Synthesis and carbonic anhydrase inhibitory properties of sulfamides structurally related to dopamine.
Journal: Bioorganic & medicinal chemistry 20130601
Title: Ethylenediammonium dication: H-bonded complexes with terephthalate, chloroacetate, phosphite, selenite and sulfamate anions. Detailed vibrational spectroscopic and theoretical studies of ethylenediammonium terephthalate.
Journal: Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy 20121201
Title: Efficacious N-protection of O-aryl sulfamates with 2,4-dimethoxybenzyl groups.
Journal: Organic & biomolecular chemistry 20121007
Title: A modular synthesis of dithiocarbamate pendant unnatural α-amino acids.
Journal: Chemical communications (Cambridge, England) 20120914
Title: Measurement of nitrosamine and nitramine formation from NOx reactions with amines during amine-based carbon dioxide capture for postcombustion carbon sequestration.
Journal: Environmental science & technology 20120904
Title: Sulfamate proton solvent exchange in heparin oligosaccharides: evidence for a persistent hydrogen bond in the antithrombin-binding pentasaccharide Arixtra.
Journal: Glycobiology 20120901
Title: Anion inhibition studies of an α-carbonic anhydrase from the thermophilic bacterium Sulfurihydrogenibium yellowstonense YO3AOP1.
Journal: Bioorganic & medicinal chemistry letters 20120901
Title: Acyl-sulfamates target the essential glycerol-phosphate acyltransferase (PlsY) in Gram-positive bacteria.
Journal: Bioorganic & medicinal chemistry 20120815
Title: Comparison of arylboron-based nucleophiles in Ni-catalyzed Suzuki-Miyaura cross-coupling with aryl mesylates and sulfamates.
Journal: The Journal of organic chemistry 20120720
Title: Ureido-substituted sulfamates show potent carbonic anhydrase IX inhibitory and antiproliferative activities against breast cancer cell lines.
Journal: Bioorganic & medicinal chemistry letters 20120715
Title: Modular functionalization of allenes to aminated stereotriads.
Journal: Journal of the American Chemical Society 20120704
Title: Palladium-catalysed aminosulfonylation of aryl-, alkenyl- and heteroaryl halides: scope of the three-component synthesis of N-aminosulfonamides.
Journal: Organic & biomolecular chemistry 20120528
Title: Proton-in-flight mechanism for the spontaneous hydrolysis of N-methyl O-phenyl sulfamate: implications for the design of steroid sulfatase inhibitors.
Journal: The Journal of organic chemistry 20120504
Title: Hydrolysis of N-alkyl sulfamates and the catalytic efficiency of an S-N cleaving sulfamidase.
Journal: The Journal of organic chemistry 20120316
Title: Total synthesis of (-)-kaitocephalin based on a Rh-catalyzed C-H amination.
Journal: Organic letters 20120316
Title: Cloning, characterization and sulfonamide inhibition studies of an α-carbonic anhydrase from the living fossil sponge Astrosclera willeyana.
Journal: Bioorganic & medicinal chemistry 20120215
Title: Mechanistic studies of substrate-assisted inhibition of ubiquitin-activating enzyme by adenosine sulfamate analogues.
Journal: The Journal of biological chemistry 20111125
Title: Promiscuity of carbonic anhydrase II. Unexpected ester hydrolysis of carbohydrate-based sulfamate inhibitors.
Journal: Journal of the American Chemical Society 20111116
Title: Detection of the 1H and 15N NMR resonances of sulfamate groups in aqueous solution: a new tool for heparin and heparan sulfate characterization.
Journal: Analytical chemistry 20111015
Title: Aziridines from intramolecular alkene aziridination of sulfamates: reactivity toward carbon nucleophiles. application to the synthesis of spisulosine and its fluoro analogue.
Journal: The Journal of organic chemistry 20110916
Title: Inhibition studies of the β-carbonic anhydrases from the bacterial pathogen Salmonella enterica serovar Typhimurium with sulfonamides and sulfamates.
Journal: Bioorganic & medicinal chemistry 20110815
Title: Aromatase and dual aromatase-steroid sulfatase inhibitors from the letrozole and vorozole templates.
Journal: ChemMedChem 20110801
Title: Structure-activity relationships of C-17-substituted estratriene-3-O-sulfamates as anticancer agents.
Journal: Journal of medicinal chemistry 20110714
Title: Development of steroid sulfatase inhibitors.
Journal: Molecular and cellular endocrinology 20110704
Title: Inhibition studies with anions and small molecules of two novel β-carbonic anhydrases from the bacterial pathogen Salmonella enterica serovar Typhimurium.
Journal: Bioorganic & medicinal chemistry letters 20110615
Title: Rapid nickel-catalyzed Suzuki-Miyaura cross-couplings of aryl carbamates and sulfamates utilizing microwave heating.
Journal: The Journal of organic chemistry 20110304
Title: Nickel-catalyzed amination of aryl sulfamates.
Journal: Angewandte Chemie (International ed. in English) 20110225
Title: A new β-carbonic anhydrase from Brucella suis, its cloning, characterization, and inhibition with sulfonamides and sulfamates, leading to impaired pathogen growth.
Journal: Bioorganic & medicinal chemistry 20110201
Title: Mechanisms of hydrolysis of phenyl- and benzyl 4-nitrophenyl-sulfamate esters.
Journal: Organic & biomolecular chemistry 20110121
Title: Carbonic anhydrase inhibitors. Inhibition studies with anions and sulfonamides of a new cytosolic enzyme from the scleractinian coral Stylophora pistillata.
Journal: Bioorganic & medicinal chemistry letters 20110115
Title: Characterization and anions inhibition studies of an α-carbonic anhydrase from the teleost fish Dicentrarchus labrax.
Journal: Bioorganic & medicinal chemistry 20110115
Title: Inhibition of the β-carbonic anhydrase from Streptococcus pneumoniae by inorganic anions and small molecules: Toward innovative drug design of antiinfectives?
Journal: Bioorganic & medicinal chemistry 20110101
Title: Design and synthesis of cyclic sulfonamides and sulfamates as new calcium sensing receptor agonists.
Journal: Bioorganic & medicinal chemistry letters 20101215
Title: Sulfamic acid catalyzed solvent-free synthesis of 10-aryl-7,7-dimethyl-6,7,8,10-tetrahydro-9H-[1,3]-dioxolo [4,5- b]xanthen-9-ones and 12-aryl-9,9-dimethyl-8,9,10,12-tetrahydro-11H-benzo[a]xanthen-11-ones.
Journal: Molecular diversity 20101101
Title: The effect of aminosulfonate buffers on the light responses and intracellular pH of goldfish retinal horizontal cells.
Journal: Journal of neurochemistry 20101001
Title: Bicyclic derivatives of the potent dual aromatase-steroid sulfatase inhibitor 2-bromo-4-{[(4-cyanophenyl)(4h-1,2,4-triazol-4-yl)amino]methyl}phenylsulfamate: synthesis, SAR, crystal structure, and in vitro and in vivo activities.
Journal: ChemMedChem 20100903
Title: Inhibition of the R1 fragment of the cadmium-containing zeta-class carbonic anhydrase from the diatom Thalassiosira weissflogii with anions.
Journal: Bioorganic & medicinal chemistry letters 20100815
Title: Affinity of sulfamates and sulfamides to carbonic anhydrase II isoform: experimental and molecular modeling approaches.
Journal: Journal of chemical information and modeling 20100628
Title: Carbonic anhydrase inhibitors: crystallographic and solution binding studies for the interaction of a boron-containing aromatic sulfamide with mammalian isoforms I-XV.
Journal: Bioorganic & medicinal chemistry letters 20100615
Title: Brucella carbonic anhydrases: new targets for designing anti-infective agents.
Journal: Current pharmaceutical design 20100101
Title: Suzuki-Miyaura coupling of aryl carbamates, carbonates, and sulfamates.
Journal: Journal of the American Chemical Society 20091216
Title: Design and synthesis of carbon-11-labeled dual aromatase-steroid sulfatase inhibitors as new potential PET agents for imaging of aromatase and steroid sulfatase expression in breast cancer.
Journal: Steroids 20091101
Title: Carbonic anhydrase inhibitors. Comparison of aliphatic sulfamate/bis-sulfamate adducts with isozymes II and IX as a platform for designing tight-binding, more isoform-selective inhibitors.
Journal: Journal of medicinal chemistry 20091008
Title: Carbonic anhydrase inhibitors; fluorinated phenyl sulfamates show strong inhibitory activity and selectivity for the inhibition of the tumor-associated isozymes IX and XII over the cytosolic ones I and II.
Journal: Bioorganic & medicinal chemistry letters 20090901
Title: Which carbonic anhydrases are targeted by the antiepileptic sulfonamides and sulfamates?
Journal: Chemical biology & drug design 20090901
Title: One-pot three-component Mannich-type reactions using sulfamic acid catalyst under ultrasound irradiation.
Journal: Ultrasonics sonochemistry 20090801
Title: Identification of new 2-amino-3-methylimidazo[4,5-f]quinoline urinary metabolites from beta-naphthoflavone-treated mice.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20090801
Title: Development of structure-taste relationships for thiazolyl-, benzothiazolyl-, and thiadiazolylsulfamates.
Journal: Journal of agricultural and food chemistry 20090624
Title: Carbonic anhydrase inhibitors. Cloning, characterization, and inhibition studies of a new beta-carbonic anhydrase from Mycobacterium tuberculosis.
Journal: Journal of medicinal chemistry 20090514
Title: Molecular cloning, characterization, and inhibition studies of the Rv1284 beta-carbonic anhydrase from Mycobacterium tuberculosis with sulfonamides and a sulfamate.
Journal: Journal of medicinal chemistry 20090423
Title: Copper(II) sulfamate: an efficient catalyst for the one-pot synthesis of 3,4-dihydropyrimidine-2(1H)-ones and thiones.
Journal: Molecules (Basel, Switzerland) 20090213
Title: Carbonic anhydrase inhibitors: inhibition studies of a coral secretory isoform with inorganic anions.
Journal: Bioorganic & medicinal chemistry letters 20090201
Title: Carbonic anhydrase inhibitors: inhibition of the beta-class enzyme from the yeast Saccharomyces cerevisiae with sulfonamides and sulfamates.
Journal: Bioorganic & medicinal chemistry 20090201
Title: Structure and inhibition of the CO2-sensing carbonic anhydrase Can2 from the pathogenic fungus Cryptococcus neoformans.
Journal: Journal of molecular biology 20090130
Title: N,N-Dichloroaminosulfonic acids as novel topical antimicrobial agents.
Journal: Bioorganic & medicinal chemistry letters 20090101
Title: A stereoselective synthesis of the bromopyrrole natural product (-)-agelastatin A.
Journal: Angewandte Chemie (International ed. in English) 20090101
Title: Synthesis of aryl sulfamate and phenol small peptide derivatives using a multidetachable sulfamate linker strategy.
Journal: Advances in experimental medicine and biology 20090101
Title: Carbonic anhydrase inhibitors. Inhibition of the beta-class enzyme from the yeast Saccharomyces cerevisiae with anions.
Journal: Bioorganic & medicinal chemistry letters 20081215
Title: Effects of C-17 heterocyclic substituents on the anticancer activity of 2-ethylestra-1,3,5(10)-triene-3-O-sulfamates: synthesis, in vitro evaluation and computational modelling.
Journal: Organic & biomolecular chemistry 20081121
Title: Mouse Ae1 E699Q mediates SO42-i/anion-o exchange with [SO42-]i-dependent reversal of wild-type pHo sensitivity.
Journal: American journal of physiology. Cell physiology 20080801
Title: A chiral rhodium carboxamidate catalyst for enantioselective C-H amination.
Journal: Journal of the American Chemical Society 20080723
Title: Poly(amidosulfonic acid) modified glassy carbon electrode for determination of isoniazid in pharmaceuticals.
Journal: Bioelectrochemistry (Amsterdam, Netherlands) 20080601
Title: Enantioselective silica-based monoliths modified with a novel aminosulfonic acid-derived strong cation exchanger for electrically driven and pressure-driven capillary chromatography.
Journal: Electrophoresis 20080401
Title: Carboxylic acid bioisosteres acylsulfonamides, acylsulfamides, and sulfonylureas as novel antagonists of the CXCR2 receptor.
Journal: Bioorganic & medicinal chemistry letters 20080315
Title: Direct evidence for ArO-S bond cleavage upon inactivation of Pseudomonas aeruginosa arylsulfatase by aryl sulfamates.
Journal: Chembiochem : a European journal of chemical biology 20080303
Title: Catalytic enantioselective addition of organometallic reagents to N-formylimines using monodentate phosphoramidite ligands.
Journal: The Journal of organic chemistry 20080201
Title: Anticonvulsant sulfonamides/sulfamates/sulfamides with carbonic anhydrase inhibitory activity: drug design and mechanism of action.
Journal: Current pharmaceutical design 20080101
Title: Three-component one-pot synthesis of 4,6-diarylpyrimidin- 2(1H)-ones under solvent-free conditions in the presence of sulfamic acid as a green and reusable catalyst.
Journal: Molecular diversity 20080101
Title: Carbonic anhydrase inhibitors: cloning, characterization, and inhibition studies of the cytosolic isozyme III with sulfonamides.
Journal: Bioorganic & medicinal chemistry 20071201
Title: Carbonic anhydrase inhibitors: the inhibition profiles of the human mitochondrial isoforms VA and VB with anions are very different.
Journal: Bioorganic & medicinal chemistry 20071101
Title: Aminosulfonate modulated pH-induced conformational changes in connexin26 hemichannels.
Journal: The Journal of biological chemistry 20070323
Title: Carbonic anhydrase inhibitors. Inhibition of transmembrane isozymes XII (cancer-associated) and XIV with anions.
Journal: Bioorganic & medicinal chemistry letters 20070315
Title: Stereospecific construction of substituted piperidines. Synthesis of (-)-paroxetine and (+)-laccarin.
Journal: Chemical communications (Cambridge, England) 20070221
Title: Carbonic anhydrase inhibitors. DNA cloning, characterization, and inhibition studies of the human secretory isoform VI, a new target for sulfonamide and sulfamate inhibitors.
Journal: Journal of medicinal chemistry 20070125
Title: Antitubercular nucleosides that inhibit siderophore biosynthesis: SAR of the glycosyl domain.
Journal: Journal of medicinal chemistry 20061228
Title: 2-substituted estradiol bis-sulfamates, multitargeted antitumor agents: synthesis, in vitro SAR, protein crystallography, and in vivo activity.
Journal: Journal of medicinal chemistry 20061228
Title: Synthesis and evaluation of general mechanism-based inhibitors of sulfatases based on (difluoro)methyl phenyl sulfate and cyclic phenyl sulfamate motifs.
Journal: Bioorganic & medicinal chemistry 20061215
Title: Inhibitory effects of sulfamic acid on three thiosulfate-oxidizing chemolithotrophs.
Journal: FEMS microbiology letters 20061101
Title: New zinc binding motifs in the design of selective carbonic anhydrase inhibitors.
Journal: Mini reviews in medicinal chemistry 20060801
Title: Examination of two independent kinetic assays for determining the inhibition of carbonic anhydrases I and II: structure-activity comparison of sulfamates and sulfamides.
Journal: Chemical biology & drug design 20060801
Title: Carbonic anhydrase inhibitors: inhibition of the cytosolic human isozyme VII with anions.
Journal: Bioorganic & medicinal chemistry letters 20060615
Title: Reactivity of cyclic sulfamidates towards sulfur-stabilised enolates. Stereocontrolled synthesis of functionalised lactams.
Journal: Organic & biomolecular chemistry 20060521
Title: Carbonic anhydrase inhibitors: DNA cloning and inhibition studies of the alpha-carbonic anhydrase from Helicobacter pylori, a new target for developing sulfonamide and sulfamate gastric drugs.
Journal: Journal of medicinal chemistry 20060323
Title: 1,2,3,4-Tetrahydroisoquinolinyl sulfamic acids as phosphatase PTP1B inhibitors.
Journal: Bioorganic & medicinal chemistry letters 20060315
Title: Synthesis and biological properties of new phosmidosine analogs having an N-acylsulfamate linkage.
Journal: Nucleosides, nucleotides & nucleic acids 20060101
Title: Carbonic anhydrase inhibitors. The mitochondrial isozyme VB as a new target for sulfonamide and sulfamate inhibitors.
Journal: Journal of medicinal chemistry 20051201
Title: Inhibition of MDA-MB-231 cell cycle progression and cell proliferation by C-2-substituted oestradiol mono- and bis-3-O-sulphamates.
Journal: International journal of cancer 20051020
Title: Exploring new uses for C-H amination: Ni-catalyzed cross-coupling of cyclic sulfamates.
Journal: Organic letters 20051013
Title: Cyclic sulfamide gamma-secretase inhibitors.
Journal: Bioorganic & medicinal chemistry letters 20051001
Title: Synthesis of an N-acyl sulfamate analog of luciferyl-AMP: a stable and potent inhibitor of firefly luciferase.
Journal: Bioorganic & medicinal chemistry letters 20050901
Title: A-ring-substituted estrogen-3-O-sulfamates: potent multitargeted anticancer agents.
Journal: Journal of medicinal chemistry 20050811
Title: Inhibition of laccase activity from Trametes versicolor by heavy metals and organic compounds.
Journal: Chemosphere 20050801
Title: Carbonic anhydrase inhibitors. Synthesis and inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, and IX with boron-containing sulfonamides, sulfamides, and sulfamates: toward agents for boron neutron capture therapy of hypoxic tumors.
Journal: Bioorganic & medicinal chemistry letters 20050701
Title: Comparison of sulfamate and sulfamide groups for the inhibition of carbonic anhydrase-II by using topiramate as a structural platform.
Journal: Journal of medicinal chemistry 20050324
Title: Sulfamates and their therapeutic potential.
Journal: Medicinal research reviews 20050301
Title: Catabolism of sulfamate by Mycobacterium sp. CF1.
Journal: Environmental microbiology 20050301
Title: Tethered aminohydroxylation using acyclic homo-allylic sulfamate esters and sulfonamides as substrates.
Journal: Organic & biomolecular chemistry 20050221
Title: Identification of nonpeptidic small-molecule inhibitors of interleukin-2.
Journal: Bioorganic & medicinal chemistry letters 20050215
Title: Carbonic anhydrase inhibitors. Inhibition of the membrane-bound human and bovine isozymes IV with sulfonamides.
Journal: Bioorganic & medicinal chemistry letters 20050215
Title: Cyclic sulfamide HIV-1 protease inhibitors, with sidechains spanning from P2/P2' to P1/P1'.
Journal: Bioorganic & medicinal chemistry 20050201
Title: Carbonic anhydrase inhibitors. Inhibition of isozymes I, II, IV, V, and IX with anions isosteric and isoelectronic with sulfate, nitrate, and carbonate.
Journal: Bioorganic & medicinal chemistry letters 20050201
Title: Carbonic anhydrase inhibitors: synthesis and inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, and IX with bis-sulfamates.
Journal: Bioorganic & medicinal chemistry letters 20050201
Title: Carbonic anhydrase inhibitors. Inhibition of the prokariotic beta and gamma-class enzymes from Archaea with sulfonamides.
Journal: Bioorganic & medicinal chemistry letters 20041220
Title: Carbonic anhydrase inhibitors: inhibition of the membrane-bound human isozyme IV with anions.
Journal: Bioorganic & medicinal chemistry letters 20041206
Title: Carbonic anhydrase inhibitors. Inhibition of the newly isolated murine isozyme XIII with anions.
Journal: Bioorganic & medicinal chemistry letters 20041101
Title: The role of steroid sulphatase in regulating the oestrogenicity of oestrogen sulphamates.
Journal: Biochemical and biophysical research communications 20040910
Title: Carbonic anhydrase inhibitors. Inhibition of the beta-class enzyme from the methanoarchaeon Methanobacterium thermoautotrophicum (Cab) with anions.
Journal: Bioorganic & medicinal chemistry letters 20040906
Title: Carbonic anhydrase inhibitors: aliphatic N-phosphorylated sulfamates--a novel zinc-anchoring group leading to nanomolar inhibitors.
Journal: Journal of enzyme inhibition and medicinal chemistry 20040601
Title: Sulfamide derivatives as transition state analogue inhibitors for carboxypeptidase A.
Journal: Bioorganic & medicinal chemistry 20040501
Title: Inhibition of in vitro angiogenesis by 2-methoxy- and 2-ethyl-estrogen sulfamates.
Journal: International journal of cancer 20040420
Title: 2-phenylindole sulfamates: inhibitors of steroid sulfatase with antiproliferative activity in MCF-7 breast cancer cells.
Journal: The Journal of steroid biochemistry and molecular biology 20040401
Title: Inhibition of estrone sulfatase (ES) by alkyl and cycloalkyl ester derivatives of 4-[(aminosulfonyl)oxy] benzoic acid.
Journal: Bioorganic & medicinal chemistry letters 20040209
Title: Carbonic anhydrase inhibitors: inhibition of transmembrane, tumor-associated isozyme IX, and cytosolic isozymes I and II with aliphatic sulfamates.
Journal: Journal of medicinal chemistry 20031204
Title: Development of novel steroid sulfatase inhibitors. I. Synthesis and biological evaluation of biphenyl-4-O-sulfamates.
Journal: The Journal of steroid biochemistry and molecular biology 20031101
Title: Measurement of physiological S-nitrosothiols: a problem child and a challenge.
Journal: Nitric oxide : biology and chemistry 20030801
Title: The effects of 2-methoxy oestrogens and their sulphamoylated derivatives in conjunction with TNF-alpha on endothelial and fibroblast cell growth, morphology and apoptosis.
Journal: The Journal of steroid biochemistry and molecular biology 20030801
Title: Carbonic anhydrase inhibitors. Inhibition of cytosolic isozymes I and II and transmembrane, tumor-associated isozyme IX with sulfamates including EMATE also acting as steroid sulfatase inhibitors.
Journal: Journal of medicinal chemistry 20030522
Title: Is the negative charge on RNHSO3-M+ an essential requirement for sulfamate sweetness?
Journal: Journal of agricultural and food chemistry 20030507
Title: Carbonic anhydrase inhibitors: SAR and X-ray crystallographic study for the interaction of sugar sulfamates/sulfamides with isozymes I, II and IV.
Journal: Bioorganic & medicinal chemistry letters 20030310
Title: Structure-activity relationship determination within a group of substituted phenyl sulfamate based compounds against the enzyme oestrone sulfatase.
Journal: The Journal of pharmacy and pharmacology 20030201
Title: Growth inhibition of multi-drug-resistant breast cancer cells by 2-methoxyoestradiol-bis-sulphamate and 2-ethyloestradiol-bis-sulphamate.
Journal: The Journal of steroid biochemistry and molecular biology 20030201
Title: 3Beta-sulfamate derivatives of C19 and C21 steroids bearing a t-butylbenzyl or a benzyl group: synthesis and evaluation as non-estrogenic and non-androgenic steroid sulfatase inhibitors.
Journal: Journal of enzyme inhibition and medicinal chemistry 20030201
Title: Solid-phase parallel synthesis of 17alpha-substituted estradiol sulfamate and phenol libraries using the multidetachable sulfamate linker.
Journal: Journal of combinatorial chemistry 20030101
Title: Sulfamoyloxy-substituted 2-phenylindoles: antiestrogen-based inhibitors of the steroid sulfatase in human breast cancer cells.
Journal: Bioorganic & medicinal chemistry 20021201
Title: A multidetachable sulfamate linker successfully used in a solid-phase strategy to generate libraries of sulfamate and phenol derivatives.
Journal: Bioorganic & medicinal chemistry letters 20021021
Title: Application of the U and gamma' models in binary sweet taste mixtures.
Journal: Chemical senses 20020701
Title: The mechanism of the irreversible inhibition of estrone sulfatase (ES) through the consideration of a range of methane- and amino-sulfonate-based compounds.
Journal: Bioorganic & medicinal chemistry letters 20020506
Title: Evidence for the mechanism of the irreversible inhibition of oestrone sulphatase (ES) by aminosulphonate based compounds.
Journal: The Journal of steroid biochemistry and molecular biology 20020401
Title: Nonsteroidal compounds designed to mimic potent steroid sulfatase inhibitors.
Journal: The Journal of steroid biochemistry and molecular biology 20020301
Title: Crystal structure of human carbonic anhydrase II complexed with an anti-convulsant sugar sulphamate.
Journal: The Biochemical journal 20020201
Title: Carbonic anhydrase activity modulators: synthesis of inhibitors and activators incorporating 2-substituted-thiazol-4-yl-methyl scaffolds.
Journal: Journal of enzyme inhibition 20011001
Title: Change in rate-determining step in an E1cB mechanism during aminolysis of sulfamate esters in acetonitrile.
Journal: The Journal of organic chemistry 20010921
Title: Antitumour benzothiazoles. Part 15: The synthesis and physico-chemical properties of 2-(4-aminophenyl)benzothiazole sulfamate salt derivatives.
Journal: Bioorganic & medicinal chemistry letters 20010423
Title: Acid dissociation constant, a potential physicochemical factor in the inhibition of the enzyme estrone sulfatase (ES).
Journal: Bioorganic & medicinal chemistry letters 20010409
Title: Novel inhibitors of the enzyme estrone sulfatase (ES).
Journal: Bioorganic & medicinal chemistry letters 20010326
Title: Sulfonylated aminothiazoles as new small molecule inhibitors of protein phosphatases.
Journal: Bioorganic & medicinal chemistry letters 20010212
Title: Non-steroidal and steroidal sulfamates: new drugs for cancer therapy.
Journal: Molecular and cellular endocrinology 20010122
Title: Alternative splicing of a Drosophila GABA receptor subunit gene identifies determinants of agonist potency.
Journal: Neuroscience 20010101
Title: Nonpeptidic HIV protease inhibitors: 6-alkyl-5,6-dihydropyran-2-ones possessing a novel and achiral 3-(2-t-butyl-5-methyl-4-sulfamate)phenylthio moiety.
Journal: Bioorganic & medicinal chemistry letters 19990802
Title: Aromatic sulfonic acids as viral inhibitors. Structure-activity study using rhino, adeno 3, herpes simplex, and influenza viruses.
Journal: Journal of medicinal chemistry 19710701
