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63074-08-8,MFCD00941408
Catalog No.:AA00IB2K

63074-08-8 | Terazosin hydrochloride

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Purity
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1g
98%
in stock  
$24.00   $17.00
- +
5g
98%
in stock  
$61.00   $43.00
- +
10g
98%
in stock  
$120.00   $84.00
- +
25g
98%
in stock  
$202.00   $142.00
- +
100g
98%
in stock  
$760.00   $532.00
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  • Technical Information
  • Properties
  • Downstream Synthesis Route
  • Literature
  • Request for Quotation
  • Download SDS
  • Technical Information
  • Properties
  • Downstream Synthesis Route
  • Literature
Technical Information
Catalog Number:
AA00IB2K
Chemical Name:
Terazosin hydrochloride
CAS Number:
63074-08-8
Molecular Formula:
C19H26ClN5O4
Molecular Weight:
423.8938
MDL Number:
MFCD00941408
SMILES:
COc1cc2nc(nc(c2cc1OC)N)N1CCN(CC1)C(=O)C1CCCO1.Cl
NSC Number:
759168
Properties
Computed Properties
 
Complexity:
544  
Covalently-Bonded Unit Count:
2  
Heavy Atom Count:
29  
Hydrogen Bond Acceptor Count:
8  
Hydrogen Bond Donor Count:
2  
Rotatable Bond Count:
4  
Undefined Atom Stereocenter Count:
1  

Downstream Synthesis Route

[1]CurrentPatentAssignee:SKCAPITALPARTNERSLP-US2006/205944,2006,A1Locationinpatent:Page/Pagecolumn3

[2]CurrentPatentAssignee:AUROBINDOPHARMALIMITED-US2007/161791,2007,A1Locationinpatent:Page/Pagecolumn4

23680-84-4   
terazosinhydrochloride 

[1]CurrentPatentAssignee:H.LUNDBECKA/S-US5990128,1999,A

[2]CurrentPatentAssignee:H.LUNDBECKA/S-US5508306,1996,A

[3]CurrentPatentAssignee:H.LUNDBECKA/S-US5578611,1996,ACurrentPatentAssignee:H.LUNDBECKA/S-US5861309,1999,ACurrentPatentAssignee:H.LUNDBECKA/S-US6015819,2000,A

23680-84-4    63074-07-7   
1-(4-amino-6,7-dimethoxy-2-quinaolinyl)-4-(2-tetrahydrofuroyl)piperazinehydrochloride 
 
terazosinhydrochloride 

[1]CurrentPatentAssignee:ABBOTTLABORATORIESINC-US5504207,1996,A

Literature

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Title: Amlodipine alone or combined with terazosin improves lower urinary tract disorder in rat models of benign prostatic hyperplasia or detrusor instability: focus on detrusor overactivity.

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Title: Role of alpha adrenergic blocker in the management of posterior urethral valves.

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Title: Fluorescent quantification of terazosin hydrochloride content in human plasma and tablets using second-order calibration based on both parallel factor analysis and alternating penalty trilinear decomposition.

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Title: Effects of four different alpha(1)-adrenoceptor antagonists on alpha-adrenoceptor agonist-induced contractions in isolated mouse and hamster ureters.

Journal: Journal of smooth muscle research = Nihon Heikatsukin Gakkai kikanshi 20090801

Title: [Retrospective analysis of the combined therapy of terazosin with chlormezanone for chronic prostatitis/chronic pelvic pain syndrome].

Journal: Zhonghua nan ke xue = National journal of andrology 20090801

Title: Tamsulosin versus terazosin for benign prostatic hyperplasia: a systematic review.

Journal: Systems biology in reproductive medicine 20090801

Title: Direct high-performance liquid chromatography enantioseparation of terazosin on an immobilised polysaccharide-based chiral stationary phase under polar organic and reversed-phase conditions.

Journal: Journal of chromatography. A 20090710

Title: A multicomponent behavioural and drug intervention for nocturia in elderly men: rationale and pilot results.

Journal: BJU international 20090701

Title: Efficacy of combined amlodipine/terazosin therapy in male hypertensive patients with lower urinary tract symptoms: a randomized, double-blind clinical trial.

Journal: Urology 20090701

Title: Iris morphologic changes related to alpha(1)-adrenergic receptor antagonists implications for intraoperative floppy iris syndrome.

Journal: Ophthalmology 20090501

Title: [Amlodipine combined with terazosin reduces postvoid residual and the risk of acute urinary retention].

Journal: Zhonghua nan ke xue = National journal of andrology 20090501

Title: Combined effects of terazosin and genistein on a metastatic, hormone-independent human prostate cancer cell line.

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Title: Functional screening of adrenergic receptors by measuring intracellular calcium using the FlexStation scanning fluorimeter.

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Title: Terazosin treatment suppresses basic fibroblast growth factor expression in the rat ventral prostate.

Journal: Clinical and investigative medicine. Medecine clinique et experimentale 20090201

Title: Adjunctive medical therapy with an alpha-1A-specific blocker after shock wave lithotripsy of lower ureteral stones.

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Title: [Using setegis (terasosine) in early postoperative period after transurethral prostate resection].

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Title: Effects of alpha-adrenoceptor antagonist doxazosin on MDR1-mediated multidrug resistance and transcellular transport.

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Title: Noradrenaline triggers muscle tone by amplifying glutamate-driven excitation of somatic motoneurones in anaesthetized rats.

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Title: [Efficacy of electroacupuncture in treating 93 patients with benign prostatic hyperplasia].

Journal: Zhongguo Zhong xi yi jie he za zhi Zhongguo Zhongxiyi jiehe zazhi = Chinese journal of integrated traditional and Western medicine 20081101

Title: Fabrication of terazocin-loaded poly(D,L-lactide) microspheres by an ultrasonic spray drying method and their release behaviors.

Journal: Journal of nanoscience and nanotechnology 20081001

Title: Combined use of melatonin and terazosin restores bladder contractility in rabbits with partial outlet obstruction.

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Title: Cardio-protective role of terazosin is possibly mediated through alteration in thyroid function.

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Title: The effect of terazosin on functional bladder outlet obstruction in women: a pilot study.

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Title: More effects of extracorporeal magnetic innervation and terazosin therapy than terazosin therapy alone for non-inflammatory chronic pelvic pain syndrome: a pilot study.

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Journal: Psychopharmacology 20051101

Title: Effects of different alpha-1 adrenoceptor blockers on proximal urethral function using in vivo isovolumetric pressure changes.

Journal: Journal of smooth muscle research = Nihon Heikatsukin Gakkai kikanshi 20051001

Title: Efficacy of terazosin and finasteride in symptomatic benign prostatic hyperplasia: A comparative study.

Journal: Bangladesh Medical Research Council bulletin 20050801

Title: Initial, long-term, and durable responses to terazosin, placebo, or other therapies for chronic prostatitis/chronic pelvic pain syndrome.

Journal: Urology 20050701

Title: The risk of overanticoagulation with antibiotic use in outpatients on stable warfarin regimens.

Journal: Journal of general internal medicine 20050701

Title: Evidence of roles of central alpha1-adrenoceptors and epinephrine in orexin A-induced hyperactivity in mice.

Journal: Neuroscience letters 20050624

Title: The comparison and efficacy of 3 different alpha1-adrenergic blockers for distal ureteral stones.

Journal: The Journal of urology 20050601

Title: Effect of terazosin on tissue vascularity and apoptosis in transitional cell carcinoma of bladder.

Journal: Urology 20050501

Title: High prevalence of orthostatic hypotension and its correlation with potentially causative medications among elderly veterans.

Journal: Journal of clinical pharmacy and therapeutics 20050401

Title: Comparative evaluation of Prostina and terazosin in the treatment of benign prostatic hyperplasia.

Journal: Journal of the Indian Medical Association 20050201

Title: Sympathetic modulation of activity in Adelta- and C-primary nociceptive afferents after intradermal injection of capsaicin in rats.

Journal: Journal of neurophysiology 20050101

Title: alpha1-Adrenergic receptor antagonists induce production of IL-18 and expression of ICAM-1 and CD40 in human monocytes.

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Title: [Double-blind placebo-controlled trial of terazosine efficacy in patients with chronic abacterial prostatitis].

Journal: Urologiia (Moscow, Russia : 1999) 20050101

Title: [Clinical efficacy and safety of terazosine (setegis) in patients with benign prostatic hyperplasia with concomitant cardiovascular diseases].

Journal: Urologiia (Moscow, Russia : 1999) 20050101

Title: [Kornam in the treatment of imperative urine incontinence in females].

Journal: Urologiia (Moscow, Russia : 1999) 20050101

Title: Terazosin in the treatment of premature ejaculation: a short-term follow-up.

Journal: International urology and nephrology 20050101

Title: Sympathetic and angiotensin-dependent hypertension during cage-switch stress in mice.

Journal: American journal of physiology. Regulatory, integrative and comparative physiology 20041201

Title: Role of locus coeruleus alpha1-adrenoceptors in motor activity in rats.

Journal: Synapse (New York, N.Y.) 20041201

Title: Visceral afferent bias on cortical processing: role of adrenergic afferents to the basal forebrain cholinergic system.

Journal: Behavioral neuroscience 20041201

Title: Effects of alpha-1 adrenergic receptor antagonist, terazosin, on cardiovascular functions in anaesthetised dogs.

Journal: Indian journal of experimental biology 20041201

Title: Initial, long-term, and durable responses to terazosin, placebo, or other therapies for chronic prostatitis/chronic pelvic pain syndrome.

Journal: Urology 20041101

Title: Sympathetic influence on capsaicin-evoked enhancement of dorsal root reflexes in rats.

Journal: Journal of neurophysiology 20041001

Title: Baroreceptor mediated blood pressure regulation is not affected during dose dependent inhibition of prostatic contractions by terazosin.

Journal: Indian journal of physiology and pharmacology 20041001

Title: Gross mapping of alpha1-adrenoceptors that regulate behavioral activation in the mouse brain.

Journal: Behavioural brain research 20040709

Title: Meta-analysis: creating a level playing field for the patient with symptomatic benign prostatic hyperplasia?

Journal: BJU international 20040701

Title: The role of alpha-blockers in the management of prostate cancer.

Journal: Expert opinion on pharmacotherapy 20040601

Title: [The growth inhibition effect of alpha-adrenoceptor antagonists on androgen- independent prostate cancer cell line].

Journal: Zhonghua wai ke za zhi [Chinese journal of surgery] 20040522

Title: Inhibition of human ether-a-go-go-related gene potassium channels by alpha 1-adrenoceptor antagonists prazosin, doxazosin, and terazosin.

Journal: Naunyn-Schmiedeberg's archives of pharmacology 20040501

Title: Combination of finasteride and doxazosin for the treatment of benign prostatic hyperplasia.

Journal: Expert opinion on pharmacotherapy 20040501

Title: Apoptotic impact of alpha1-blockers on prostate cancer growth: a myth or an inviting reality?

Journal: The Prostate 20040401

Title: Measurement of low-dose active pharmaceutical ingredient in a pharmaceutical blend using frequency-domain photon migration.

Journal: Journal of pharmaceutical sciences 20040301

Title: Regulatory considerations of pharmaceutical solid polymorphism in Abbreviated New Drug Applications (ANDAs).

Journal: Advanced drug delivery reviews 20040223

Title: [Effect of nitric oxide donor and alpha1-receptor antagonist on proliferation/apoptosis of hyperplastic prostatic stromal cells in vitro].

Journal: Zhonghua wai ke za zhi [Chinese journal of surgery] 20040222

Title: Herbal and vitamin supplement use in a prostate cancer screening population.

Journal: Urology 20040201

Title: A current review of medical therapy for benign prostatic hyperplasia.

Journal: The Journal of the American Osteopathic Association 20040201

Title: Validated specific HPLC methods for determination of prazosin, terazosin and doxazosin in the presence of degradation products formed under ICH-recommended stress conditions.

Journal: Journal of pharmaceutical and biomedical analysis 20040127

Title: [Combined treatment of voiding disorders in women with m-cholinolytic and alpha 1-adrenoblocker].

Journal: Urologiia (Moscow, Russia : 1999) 20040101

Title: Terazosin and doxazosin in the treatment of BPH: results of a randomized study with crossover in non-responders.

Journal: Urologia internationalis 20040101

Title: Cost-effectiveness of tamsulosin, doxazosin, and terazosin in the treatment of benign prostatic hyperplasia.

Journal: Journal of managed care pharmacy : JMCP 20040101

Title: The use and rationale of selective alpha blockade in children with non-neurogenic neurogenic bladder dysfunction.

Journal: International braz j urol : official journal of the Brazilian Society of Urology 20040101

Title: A comparison of four different alpha1-blockers in benign prostatic hyperplasia patients with and without diabetes.

Journal: Scandinavian journal of urology and nephrology 20040101

Title: Immobility from administration of the alpha1-adrenergic antagonist, terazosin, in the IVth ventricle in rats.

Journal: Neuroscience letters 20031226

Title: Hormonal and morphologic evaluation of the effects of antiandrogens on the blood supply of the rat prostate.

Journal: Urology 20031101

Title: Influence of hypertension on lower urinary tract symptoms in benign prostatic hyperplasia.

Journal: International journal of urology : official journal of the Japanese Urological Association 20031101

Title: Growth inhibiting effects of terazosin on androgen-independent prostate cancer cell lines.

Journal: Chinese medical journal 20031101

Title: [Pharmacologic treatment of benign prostatic hyperplasia].

Journal: Orvosi hetilap 20030914

Title: The role of combination therapy for lower urinary tract symptoms secondary to benign prostatic hyperplasia.

Journal: Current urology reports 20030801

Title: [Serum nitric oxide and D-dimer before and after administering antihypertensive drugs in essential hypertension].

Journal: Hunan yi ke da xue xue bao = Hunan yike daxue xuebao = Bulletin of Hunan Medical University 20030801

Title: Role of epinephrine stimulation of CNS alpha1-adrenoceptors in motor activity in mice.

Journal: Synapse (New York, N.Y.) 20030701

Title: Changes in nocturia from medical treatment of benign prostatic hyperplasia: secondary analysis of the Department of Veterans Affairs Cooperative Study Trial.

Journal: The Journal of urology 20030701

Title: Effects of intravenous and infravesical administration of suramin, terazosin and BMY 7378 on bladder instability in conscious rats with bladder outlet obstruction.

Journal: BJU international 20030701

Title: Doxazosin and terazosin suppress prostate growth by inducing apoptosis: clinical significance.

Journal: The Journal of urology 20030401

Title: Anoikis induction by quinazoline based alpha 1-adrenoceptor antagonists in prostate cancer cells: antagonistic effect of bcl-2.

Journal: The Journal of urology 20030301

Title: Effect of terazosin on clinical benign prostatic hyperplasia in older adults.

Journal: Journal of the American Geriatrics Society 20030301

Title: Terazosin therapy for chronic prostatitis/chronic pelvic pain syndrome: a randomized, placebo controlled trial.

Journal: The Journal of urology 20030201

Title: Identification of apoptotic and antiangiogenic activities of terazosin in human prostate cancer and endothelial cells.

Journal: The Journal of urology 20030201

Title: Nitric oxide opposes glucose-induced hypertension by suppressing sympathetic activity.

Journal: Hypertension (Dallas, Tex. : 1979) 20030201

Title: [Hepatotoxicity induced by terazosin].

Journal: Medicina clinica 20030201

Title: Doxazosin induces apoptosis in cardiomyocytes cultured in vitro by a mechanism that is independent of alpha1-adrenergic blockade.

Journal: Circulation 20030107

Title: [Results of treatment of irritative symptoms and urinary retention in patients 1 year after radical retropubic prostatectomy].

Journal: Urologiia (Moscow, Russia : 1999) 20030101

Title: Plasma atrial natriuretic peptide in essential hypertension after treatment with terazocin.

Journal: European journal of drug metabolism and pharmacokinetics 20030101

Title: The alpha1-adrenoceptor antagonist terazosin induces prostate cancer cell death through a p53 and Rb independent pathway.

Journal: Oncology reports 20030101

Title: Comparison of finasteride and alpha-blockers as independent risk factors for erectile dysfunction.

Journal: International journal of clinical practice 20030101

Title: Mice expressing the alpha(1B)-adrenergic receptor induces a synucleinopathy with excessive tyrosine nitration but decreased phosphorylation.

Journal: Journal of neurochemistry 20021101

Title: Prophylactic versus therapeutic alpha-blockers after permanent prostate brachytherapy.

Journal: Urology 20021001

Title: [Comparison of prazosin, terazosin and tramsulosin: functional and binding studies in isolated prostatic and vascular human tissues].

Journal: Minerva urologica e nefrologica = The Italian journal of urology and nephrology 20020901

Title: [Effects of terazosine and atenolol on serum lipids in essential hypertension].

Journal: Zeitschrift fur Kardiologie 20020901

Title: Prior iontophoresis of saline enhances vasoconstriction to phenylephrine and clonidine in the skin of the human forearm.

Journal: British journal of clinical pharmacology 20020701

Title: Urodynamic effects of terazosin treatment for Japanese patients with symptomatic benign prostatic hyperplasia.

Journal: The Journal of urology 20020601

Title: [Chiral separation and preparation of three new antagonists of alpha 1-adrenoceptors by chiral mobile phase HPLC].

Journal: Yao xue xue bao = Acta pharmaceutica Sinica 20020601

Title: The efficacy of terazosin for treating benign prostatic hyperplasia: a multicentre clinical trial.

Journal: BJU international 20020501

Title: Hypertension in L-NAME-treated diabetic rats depends on an intact sympathetic nervous system.

Journal: American journal of physiology. Regulatory, integrative and comparative physiology 20020401

Title: Long-term risk of re-treatment of patients using alpha-blockers for lower urinary tract symptoms.

Journal: The Journal of urology 20020401

Title: Role of supraspinal alpha1-adrenoceptors for voiding in conscious rats with and without bladder outlet obstruction.

Journal: The Journal of urology 20020401

Title: Effect of fiduxosin, an antagonist selective for alpha(1A)- and alpha(1D)-adrenoceptors, on intraurethral and arterial pressure responses in conscious dogs.

Journal: The Journal of pharmacology and experimental therapeutics 20020201

Title: Quinazoline-derived alpha1-adrenoceptor antagonists induce prostate cancer cell apoptosis via an alpha1-adrenoceptor-independent action.

Journal: Cancer research 20020115

Title: Impact of alpha1-blockers in men with spinal cord injury and upper tract stasis.

Journal: The journal of spinal cord medicine 20020101

Title: Alpha1-adrenoceptor antagonists radiosensitize prostate cancer cells via apoptosis induction.

Journal: Anticancer research 20020101

Title: Apoptotic and proliferative index after Alpha-1-adrenoceptor antagonist and/or finasteride treatment in benign prostatic hyperplasia.

Journal: Urologia internationalis 20020101

Title: [Treatment of external RF hyperthermia combining with alpha 1-adrenergic receptor blocker for patients with prostatodynia and chronic non-bacterial prostatitis].

Journal: Zhonghua nan ke xue = National journal of andrology 20020101

Title: [Comparative evaluation of the efficacy of using terazosin and tamsulosin in patients with benign prostatic hyperplasia].

Journal: Urologiia (Moscow, Russia : 1999) 20020101

Title: [Results of monotherapy with terazosin (kornam) in chronic infectious prostatitis patients].

Journal: Urologiia (Moscow, Russia : 1999) 20020101

Title: [Use of alpha1-adrenergic blockaders in voiding disorders in women].

Journal: Urologiia (Moscow, Russia : 1999) 20020101

Title: Terazosin for benign prostatic hyperplasia.

Journal: The Cochrane database of systematic reviews 20020101

Title: Terazosin, doxazosin, and prazosin: current clinical experience.

Journal: Urology 20011201

Title: 5alpha-reductase inhibitors: what role should they play?

Journal: Urology 20011201

Title: Meta-analysis of randomized trials of terazosin in the treatment of benign prostatic hyperplasia.

Journal: Urology 20011101

Title: Reduction of human prostate tumor vascularity by the alpha1-adrenoceptor antagonist terazosin.

Journal: The Prostate 20010701

Title: Structure-activity studies for a novel series of bicyclic substituted hexahydrobenz[e]isoindole alpha1A adrenoceptor antagonists as potential agents for the symptomatic treatment of benign prostatic hyperplasia.

Journal: Journal of medicinal chemistry 20010607

Title: Comparison of prazosin, terazosin and tamsulosin: functional and binding studies in isolated prostatic and vascular human tissues.

Journal: The Prostate 20010601

Title: Pharmacological blockade of brain alpha1-adrenoceptors as measured by ex vivo [3H]prazosin binding is correlated with behavioral immobility.

Journal: European journal of pharmacology 20010525

Title: Evaluating adverse cardiovascular effects of drug treatment for benign prostatic hyperplasia (BPH): methodological considerations.

Journal: Journal of clinical epidemiology 20010501

Title: Initiation of nonselective alpha1-antagonist therapy and occurrence of hypotension-related adverse events among men with benign prostatic hyperplasia: a retrospective cohort study.

Journal: Clinical therapeutics 20010501

Title: The short-term effects of terazosin in Japanese men with benign prostatic hyperplasia.

Journal: Journal of Nippon Medical School = Nippon Ika Daigaku zasshi 20010401

Title: Overstimulation of the alpha1B-adrenergic receptor causes a 'seizure plus' syndrome.

Journal: Nature medicine 20010201

Title: Magnetic resonance imaging and morphometric histologic analysis of prostate tissue composition in predicting the clinical outcome of terazosin therapy in benign prostatic hyperplasia.

Journal: International journal of urology : official journal of the Japanese Urological Association 20010201

Title: [A randomized comparative study assessing once versus twice a day treatment of benign prostatic hyperplasia with terazosin].

Journal: Hinyokika kiyo. Acta urologica Japonica 20010201

Title: alpha-Blockade improves symptoms suggestive of bladder outlet obstruction but fails to relieve it.

Journal: The Journal of urology 20010101

Title: Targeted transurethral microwave thermotherapy versus alpha-blockade in benign prostatic hyperplasia: outcomes at 18 months.

Journal: Urology 20010101

Title: Combined effect of terazosin and finasteride on apoptosis, cell proliferation, and transforming growth factor-beta expression in benign prostatic hyperplasia.

Journal: The Prostate 20010101

Title: A quantitative analysis of antagonism and inverse agonism at wild-type and constitutively active hamster alpha1B-adrenoceptors.

Journal: Naunyn-Schmiedeberg's archives of pharmacology 20010101

Title: [The efficacy and safety of terazosin and tamsulosin in patients with urinary disturbance accompanying prostatic hypertrophy].

Journal: Hinyokika kiyo. Acta urologica Japonica 20010101

Title: Effect of terazosin on the lipid profile in patients with symptomatic benign prostatic hyperplasia.

Journal: Urologia internationalis 20010101

Title: Use of terazosine in patients with chronic pelvic pain syndrome and evaluation by prostatitis symptom score index.

Journal: International urology and nephrology 20010101

Title: High-performance liquid chromatographic analysis and pharmacokinetics of terazosin in healthy volunteers.

Journal: Research communications in molecular pathology and pharmacology 20010101

Title: Suppression of human prostate cancer cell growth by alpha1-adrenoceptor antagonists doxazosin and terazosin via induction of apoptosis.

Journal: Cancer research 20000815

Title: Alpha 1-adrenoceptor antagonists terazosin and doxazosin induce prostate apoptosis without affecting cell proliferation in patients with benign prostatic hyperplasia.

Journal: The Journal of urology 19990601

Title: A meta-analysis on the efficacy and tolerability of alpha1-adrenoceptor antagonists in patients with lower urinary tract symptoms suggestive of benign prostatic obstruction.

Journal: European urology 19990101

Title: Terazosin in benign prostatic hyperplasia: effects on blood pressure in normotensive and hypertensive men.

Journal: British journal of urology 19980901

Title: Effects of oral and intravenous terazosin and head-up tilt on blood pressure responses in patients with hypertension.

Journal: Journal of clinical pharmacology 19980601

Title: 4-Amino-2-[4-[1-(benzyloxycarbonyl)-2(S)- [[(1,1-dimethylethyl)amino]carbonyl]-piperazinyl]-6, 7-dimethoxyquinazoline (L-765,314): a potent and selective alpha1b adrenergic receptor antagonist.

Journal: Journal of medicinal chemistry 19980409

Title: A double-blind comparison of terazosin and tamsulosin on their differential effects on ambulatory blood pressure and nocturnal orthostatic stress testing.

Journal: European urology 19980101

Title: Clinical comparison of selective and non-selective alpha 1A-adrenoceptor antagonists for bladder outlet obstruction associated with benign prostatic hyperplasia: studies on tamsulosin and terazosin in Chinese patients. The Chinese Tamsulosin Study Group.

Journal: Journal of medicine 19980101

Title: Synthesis and pharmacological characterization of 3-[2-((3aR,9bR)-cis-6-methoxy-2,3,3a,4,5,9b-hexahydro-1H-benz[e] isoindol-2-yl)ethyl]pyrido-[3',4':4,5]thieno[3,2-d]pyrimidine-2,4 (1H,3H)-dione (A-131701): a uroselective alpha 1A adrenoceptor antagonist for the symptomatic treatment of benign prostatic hyperplasia.

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Title: Side effects of terazosin in the treatment of symptomatic benign prostatic hyperplasia.

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Title: Prostatic alpha 1-adrenoceptors and uroselectivity.

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Title: A multicenter, randomized, double-blind, placebo-controlled study to evaluate the safety and efficacy of terazosin in the treatment of benign prostatic hyperplasia.

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Title: Effect of alpha 1 adrenoceptor antagonists on prostatic pressure and blood pressure in the anesthetized dog.

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Title: Effects of ANG-converting enzyme and alpha 1-adrenoceptor inhibition on intrarenal hemodynamics in SHR.

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Title: [Use of terazosin and alfuzosin in the treatment of benign prostatic hypertrophy (BPH): our experience].

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Title: Intraoperative hypotension in a patient treated with terazosin, a new alpha-adrenergic receptor antagonist.

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Title: [Comparison of selective alpha-1 blockades for alpha-receptors in human hypertrophied prostatic adenomas].

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Title: Ju M, et al. Efficacy of combination terazosin and nifedipine therapy in postoperative treatment of distal ureteral stones after transurethral ureteroscopic lithotripsy. J Int Med Res. 2020 Apr;48(4):300060520904851.

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Tags:63074-08-8 Molecular Formula|63074-08-8 MDL|63074-08-8 SMILES|63074-08-8 Terazosin hydrochloride