Title: Discovery of potent small-molecule inhibitors of multidrug-resistant Plasmodium falciparum using a novel miniaturized high-throughput luciferase-based assay.
Journal: Antimicrobial agents and chemotherapy 20100901
Title: Histamine excites neonatal rat sympathetic preganglionic neurons in vitro via activation of H1 receptors.
Journal: Journal of neurophysiology 20060401
Title: Mechanisms of inverse agonism at histamine H(2) receptors - potential benefits and concerns.
Journal: Inflammopharmacology 20060301
Title: Alteration of intracellular histamine H2 receptor cycling precedes antagonist-induced upregulation.
Journal: American journal of physiology. Gastrointestinal and liver physiology 20051101
Title: Effects of cimetidine-like drugs on recombinant GABAA receptors.
Journal: Life sciences 20041008
Title: Tiotidine, a histamine H2 receptor inverse agonist that binds with high affinity to an inactive G-protein-coupled form of the receptor. Experimental support for the cubic ternary complex model.
Journal: Molecular pharmacology 20030801
Title: Extremely early onset of ranitidine action on human histamine H2 receptors expressed in HEK293 cells.
Journal: Digestion 20030101
Title: Histamine H1 receptors in rat dorsal raphe nucleus: pharmacological characterisation and linking to increased neuronal activity.
Journal: Brain research 20021108
Title: Effects of N-alpha-methyl-histamine on human H(2) receptors expressed in CHO cells.
Journal: Gut 20020601
Title: Histamine H(2) -like receptors in chick cerebral cortex: effects on cyclic AMP synthesis and characterization by [(3) H]tiotidine binding.
Journal: Journal of neurochemistry 20020601
Title: Regulation of phospholipase C activation by the number of H(2) receptors during Ca(2+)-induced differentiation of mouse keratinocytes.
Journal: Biochemical pharmacology 20020515
Title: Mouse mammary epithelial cells bear histamine receptors.
Journal: Inflammation research : official journal of the European Histamine Research Society ... [et al.] 20020401
Title: The initial inositol 1,4,5-trisphosphate response induced by histamine is strongly amplified by Ca(2+) release from internal stores in smooth muscle.
Journal: Cell calcium 20020401
Title: Characterization of histamine H(2)-like receptors in duck cerebral cortical membranes by [(3)H]tiotidine binding.
Journal: Neuroscience letters 20020222
Title: Similar apparent constitutive activity of human histamine H(2)-receptor fused to long and short splice variants of G(salpha).
Journal: The Journal of pharmacology and experimental therapeutics 20011201
Title: Distinct interaction of human and guinea pig histamine H2-receptor with guanidine-type agonists.
Journal: Molecular pharmacology 20011201
Title: Histamine deficiency induces tissue-specific down-regulation of histamine H2 receptor expression in histidine decarboxylase knockout mice.
Journal: FEBS letters 20011116
Title: ElogD(oct): a tool for lipophilicity determination in drug discovery. 2. Basic and neutral compounds.
Journal: Journal of medicinal chemistry 20010719
Title: Inhibition of effects of endogenously synthesized histamine disturbs in vitro human dendritic cell differentiation.
Journal: Immunology letters 20010402
Title: Potent and long-lasting action of lafutidine on the human histamine H(2) receptor.
Journal: Digestion 20010101
Title: G649, an allelic variant of the human H2 receptor with low basal activity, is resistant to upregulation upon antagonist exposure.
Journal: The pharmacogenomics journal 20010101
Title: Heterologous expression of rat epitope-tagged histamine H2 receptors in insect Sf9 cells.
Journal: British journal of pharmacology 19971101
Title: Barth H, et al. Structural requirements of imidazole compounds to be inhibitors or activators of histaminemethyltransferase: investigation of histamine analogues and H2-receptor antagonists.
Title: Trzeciakowski JP, et al. The cardiac pharmacology of tiotidine (LCL 125, 211): a new histamine H2-receptor antagonist. J Pharmacol Exp Ther. 1980 Sep;214(3):629-34.
Title: Monczor F, et al. Tiotidine, a histamine H2 receptor inverse agonist that binds with high affinity to an inactive G-protein-coupled form of the receptor. Experimental support for the cubic ternary complex model. Mol Pharmacol. 2003 Aug;64(2):512-20.
