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749-02-0,MFCD00055099
Catalog No.:AA003UC9

749-02-0 | Spiperone

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5mg
95%
1 week  
$102.00   $72.00
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10mg
95%
1 week  
$124.00   $87.00
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50mg
95%
1 week  
$289.00   $202.00
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100mg
95%
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$431.00   $302.00
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  • Technical Information
  • Properties
  • Literature
Technical Information
Catalog Number:
AA003UC9
Chemical Name:
Spiperone
CAS Number:
749-02-0
Molecular Formula:
C23H26FN3O2
Molecular Weight:
395.4698
MDL Number:
MFCD00055099
SMILES:
Fc1ccc(cc1)C(=O)CCCN1CCC2(CC1)C(=O)NCN2c1ccccc1
Properties
Properties
 
Form:
Solid  
MP:
190-196℃  
Storage:
2-8℃;  

Computed Properties
 
Complexity:
577  
Covalently-Bonded Unit Count:
1  
Heavy Atom Count:
29  
Hydrogen Bond Acceptor Count:
5  
Hydrogen Bond Donor Count:
1  
Rotatable Bond Count:
6  
XLogP3:
3  

Literature

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Journal: Toxicology and applied pharmacology 20180315

Title: The herbicide glyphosate causes behavioral changes and alterations in dopaminergic markers in male Sprague-Dawley rat.

Journal: Neurotoxicology 20150101

Title: Role of somatodendritic and postsynaptic 5-HT₁A receptors on learning and memory functions in rats.

Journal: Neurochemical research 20121001

Title: Syntheses and in vitro evaluation of decalinvesamicol analogues as potential imaging probes for vesicular acetylcholine transporter (VAChT).

Journal: Bioorganic & medicinal chemistry 20120815

Title: Design, synthesis, and pharmacological evaluation of novel tetrahydroprotoberberine derivatives: selective inhibitors of dopamine D₁ receptor.

Journal: Bioorganic & medicinal chemistry 20120801

Title: Pharmacokinetic-pharmacodynamic modeling of the D₂ and 5-HT (2A) receptor occupancy of risperidone and paliperidone in rats.

Journal: Pharmaceutical research 20120701

Title: The restructuring of dopamine receptor subtype gene transcripts in c-fos KO mice.

Journal: Brain research bulletin 20120410

Title: A novel G protein-coupled receptor of Schistosoma mansoni (SmGPR-3) is activated by dopamine and is widely expressed in the nervous system.

Journal: PLoS neglected tropical diseases 20120201

Title: Synthesis, biological activities and bioavailability of moschamine, a safflomide-type phenylpropenoic acid amide found in Centaurea cyanus.

Journal: Natural product research 20120101

Title: The influence of dopamine receptor d4 polymorphism on resting EEG in healthy young females.

Journal: The open neuroimaging journal 20120101

Title: Distinct neurobehavioural effects of cannabidiol in transmembrane domain neuregulin 1 mutant mice.

Journal: PloS one 20120101

Title: Dopamine D(2) Receptor-Mediated Heterologous Sensitization of AC5 Requires Signalosome Assembly.

Journal: Journal of signal transduction 20120101

Title: Serotonin receptors in hippocampus.

Journal: TheScientificWorldJournal 20120101

Title: Studies of olfactory system neural plasticity: the contribution of the unilateral naris occlusion technique.

Journal: Neural plasticity 20120101

Title: Development of a bivalent dopamine D₂ receptor agonist.

Journal: Journal of medicinal chemistry 20111124

Title: Dopamine as an anorectic neuromodulator in the cockroach Rhyparobia maderae.

Journal: The Journal of experimental biology 20111115

Title: Involvement of the first transmembrane segment of human α(2) -adrenoceptors in the subtype-selective binding of chlorpromazine, spiperone and spiroxatrine.

Journal: British journal of pharmacology 20111101

Title: Dopamine antagonists and brief vision distinguish lens-induced- and form-deprivation-induced myopia.

Journal: Experimental eye research 20111101

Title: Roles of Non-cholinergic Intrapancreatic Nerves, Serotonergic Nerves, on Pancreatic Exocrine Secretion in the Isolated Perfused Rat Pancreas.

Journal: The Korean journal of physiology & pharmacology : official journal of the Korean Physiological Society and the Korean Society of Pharmacology 20111001

Title: Absolute abundances and affinity states of dopamine receptors in mammalian brain: A review.

Journal: Synapse (New York, N.Y.) 20110901

Title: Profiling of a prescription drug library for potential renal drug-drug interactions mediated by the organic cation transporter 2.

Journal: Journal of medicinal chemistry 20110714

Title: Postnatal manganese exposure alters the expression of D2L and D2S receptor isoforms: relationship to PKA activity and Akt levels.

Journal: Synapse (New York, N.Y.) 20110701

Title: Participation of cyclooxygenase pathway in the vasoconstriction induced by 5-HT in the in situ autoperfused kidney of long-term diabetic rats.

Journal: European journal of pharmacology 20110520

Title: Wnt5a-dopamine D2 receptor interactions regulate dopamine neuron development via extracellular signal-regulated kinase (ERK) activation.

Journal: The Journal of biological chemistry 20110506

Title: Melittin stimulates fatty acid release through non-phospholipase-mediated mechanisms and interacts with the dopamine transporter and other membrane-spanning proteins.

Journal: European journal of pharmacology 20110115

Title: In vitro effects of both dopaminergic and enkephalinergic antagonists on the ovarian growth of Cherax quadricarinatus (Decapoda, Parastacidae), at different periods of the reproductive cycle.

Journal: Comparative biochemistry and physiology. Part A, Molecular & integrative physiology 20110101

Title: Decreased striatal dopamine receptor binding in primary focal dystonia: a D2 or D3 defect?

Journal: Movement disorders : official journal of the Movement Disorder Society 20110101

Title: Synthesis and SAR study of diphenylbutylpiperidines as cell autophagy inducers.

Journal: Bioorganic & medicinal chemistry letters 20110101

Title: Molecular characterization of novel sulfotransferases from the tick, Ixodes scapularis.

Journal: BMC biochemistry 20110101

Title: A novel role of protein tyrosine kinase2 in mediating chloride secretion in human airway epithelial cells.

Journal: PloS one 20110101

Title: Serotonin and dopamine protect from hypothermia/rewarming damage through the CBS/H2S pathway.

Journal: PloS one 20110101

Title: No evidence for strong recent positive selection favoring the 7 repeat allele of VNTR in the DRD4 gene.

Journal: PloS one 20110101

Title: Dopamine and octopamine influence avoidance learning of honey bees in a place preference assay.

Journal: PloS one 20110101

Title: Inverse agonism and its therapeutic significance.

Journal: Indian journal of pharmacology 20110101

Title: Honey bee dopamine and octopamine receptors linked to intracellular calcium signaling have a close phylogenetic and pharmacological relationship.

Journal: PloS one 20110101

Title: Inhibition of experimental myopia by a dopamine agonist: different effectiveness between form deprivation and hyperopic defocus in guinea pigs.

Journal: Molecular vision 20110101

Title: Sequential mechanisms underlying concentration invariance in biological olfaction.

Journal: Frontiers in neuroengineering 20110101

Title: Development of a microfluidic confocal fluorescence detection system for the hyphenation of nano-LC to on-line biochemical assays.

Journal: Analytical and bioanalytical chemistry 20101201

Title: Dopaminergic agonists that result in ocular growth inhibition also elicit transient increases in choroidal thickness in chicks.

Journal: Experimental eye research 20101101

Title: Synthesis and SAR studies of 1,4-benzoxazine MenB inhibitors: novel antibacterial agents against Mycobacterium tuberculosis.

Journal: Bioorganic & medicinal chemistry letters 20101101

Title: The effect of bright light on lens compensation in chicks.

Journal: Investigative ophthalmology & visual science 20101001

Title: Amphetamine regulates NR2B expression in Go2α knockout mice and thereby sustains behavioral sensitization.

Journal: Journal of neurochemistry 20101001

Title: [(3)H]-F13640, a novel, selective and high-efficacy serotonin 5-HT(1A) receptor agonist radioligand.

Journal: Naunyn-Schmiedeberg's archives of pharmacology 20101001

Title: Pharmacological profile of 5-hydroxytryptamine-induced inhibition on the pressor effect elicited by sympathetic stimulation in long-term diabetic pithed rats.

Journal: European journal of pharmacology 20100915

Title: Dopamine beta-hydroxylase-deficient mice have normal densities of D(2) dopamine receptors in the high-affinity state based on in vivo PET imaging and in vitro radioligand binding.

Journal: Synapse (New York, N.Y.) 20100901

Title: Dopamine inhibition of glycine release in the rat trigeminal nucleus pars caudalis: possible involvement of trace amine receptors.

Journal: Journal of neurochemistry 20100901

Title: Inhibition of aldehyde dehydrogenase-2 suppresses cocaine seeking by generating THP, a cocaine use-dependent inhibitor of dopamine synthesis.

Journal: Nature medicine 20100901

Title: Haloperidol, spiperone, pimozide and aripiprazole reduce intracellular dopamine content in PC12 cells and rat mesencephalic cultures: Implication of inhibition of vesicular transport.

Journal: European journal of pharmacology 20100825

Title: Further delineation of hydrophobic binding sites in dopamine D(2)/D(3) receptors for N-4 substituents on the piperazine ring of the hybrid template 5/7-{[2-(4-aryl-piperazin-1-yl)-ethyl]-propyl-amino}-5,6,7,8-tetrahydro-naphthalen-2-ol.

Journal: Bioorganic & medicinal chemistry 20100801

Title: Dopamine receptor alterations in female rats with diet-induced decreased brain docosahexaenoic acid (DHA): interactions with reproductive status.

Journal: Nutritional neuroscience 20100801

Title: Increased 5-HT2A receptors in the temporal cortex of parkinsonian patients with visual hallucinations.

Journal: Movement disorders : official journal of the Movement Disorder Society 20100730

Title: Leptin increases striatal dopamine D2 receptor binding in leptin-deficient obese (ob/ob) mice.

Journal: Synapse (New York, N.Y.) 20100701

Title: Non-competitive interaction between raclopride and spiperone on human D-receptors in intact Chinese hamster ovary cells.

Journal: Fundamental & clinical pharmacology 20100601

Title: Antagonist-D2S-dopamine receptor interactions in intact recombinant Chinese hamster ovary cells [corrected].

Journal: Fundamental & clinical pharmacology 20100601

Title: A 5-HT1A-like receptor is involved in the regulation of the embryonic rotation of Lymnaea stagnalis L.

Journal: Comparative biochemistry and physiology. Toxicology & pharmacology : CBP 20100601

Title: Concentration of receptor and ligand revisited in a modified receptor binding protocol for high-affinity radioligands: [3H]Spiperone binding to D2 and D3 dopamine receptors.

Journal: Journal of neuroscience methods 20100430

Title: Discovery of 4-(4-(2-((5-Hydroxy-1,2,3,4-tetrahydronaphthalen-2-yl)(propyl)amino)ethyl)piperazin-1-yl)quinolin-8-ol and its analogues as highly potent dopamine D2/D3 agonists and as iron chelator: in vivo activity indicates potential application in symptomatic and neuroprotective therapy for Parkinson's disease.

Journal: Journal of medicinal chemistry 20100311

Title: Development of (S)-N6-(2-(4-(isoquinolin-1-yl)piperazin-1-yl)ethyl)-N6-propyl-4,5,6,7-tetrahydrobenzo[d]-thiazole-2,6-diamine and its analogue as a D3 receptor preferring agonist: potent in vivo activity in Parkinson's disease animal models.

Journal: Journal of medicinal chemistry 20100211

Title: Effects of SCH23390 and spiperone administered into medial striatum and intermediate medial mesopallium on rewarding effects of morphine in day-old chicks.

Journal: European journal of pharmacology 20100210

Title: JL13 has clozapine-like actions on thermoregulatory cutaneous blood flow in rats: Involvement of serotonin 5-HT1A and 5-HT2A receptor mechanisms.

Journal: Progress in neuro-psychopharmacology & biological psychiatry 20100201

Title: Evidence for dopamine involvement in ambulation promoted by pulegone in mice.

Journal: Pharmacology, biochemistry, and behavior 20100201

Title: Competition between 11C-raclopride and endogenous dopamine in Parkinson's disease.

Journal: Nuclear medicine communications 20100201

Title: Serotonin regulates an acyl-CoA-binding protein (ACBP) gene expression in the midgut of Rhodnius prolixus.

Journal: Insect biochemistry and molecular biology 20100201

Title: MDMA-evoked changes in the binding of dopamine D(2) receptor ligands in striatum of rats with unilateral serotonin depletion.

Journal: Synapse (New York, N.Y.) 20100101

Title: Serotonin receptors are involved in the spinal mediation of descending facilitation of surgical incision-induced increase of Fos-like immunoreactivity in rats.

Journal: Molecular pain 20100101

Title: Altered ratio of D1 and D2 dopamine receptors in mouse striatum is associated with behavioral sensitization to cocaine.

Journal: PloS one 20100101

Title: Identification of a circadian clock-controlled neural pathway in the rabbit retina.

Journal: PloS one 20100101

Title: Impact of RNA editing on functions of the serotonin 2C receptor in vivo.

Journal: Frontiers in neuroscience 20100101

Title: Roles of aminergic neurons in formation and recall of associative memory in crickets.

Journal: Frontiers in behavioral neuroscience 20100101

Title: Adverse drug effects in hospitalized elderly: data from the healthcare cost and utilization project.

Journal: Clinical pharmacology : advances and applications 20100101

Title: Neuroprotective effects of pramipexole against tunicamycin-induced cell death in PC12 cells.

Journal: Clinical and experimental pharmacology & physiology 20091201

Title: Microglial responses to dopamine in a cell culture model of Parkinson's disease.

Journal: Neurobiology of aging 20091101

Title: Investigation of a dopamine receptor in Schistosoma mansoni: functional studies and immunolocalization.

Journal: Molecular and biochemical parasitology 20091101

Title: Characterization of the contractile 5-hydroxytryptamine receptor in the autoperfused kidney of L-NAME hypertensive rats.

Journal: European journal of pharmacology 20091012

Title: Physical binding pocket induction for affinity prediction.

Journal: Journal of medicinal chemistry 20091008

Title: Mutant 5-hydroxytryptamine 1A receptor D116A is a receptor activated solely by synthetic ligands with a rich pharmacology.

Journal: The Journal of pharmacology and experimental therapeutics 20091001

Title: Dopamine D2, D3, and D4 selective phenylpiperazines as molecular probes to explore the origins of subtype specific receptor binding.

Journal: Journal of medicinal chemistry 20090813

Title: Rats self-administer intravenous nicotine delivered in a novel smoking-relevant procedure: effects of dopamine antagonists.

Journal: The Journal of pharmacology and experimental therapeutics 20090801

Title: Overexpression of 5-HT2C receptors in forebrain leads to elevated anxiety and hypoactivity.

Journal: The European journal of neuroscience 20090701

Title: Automated on-line in-tube solid-phase microextraction coupled with HPLC/MS/MS for the determination of butyrophenone derivatives in human plasma.

Journal: Analytical and bioanalytical chemistry 20090601

Title: Platelet dopamine: D2 receptor binding in patients with migraine.

Journal: Cephalalgia : an international journal of headache 20090501

Title: Role of the serotoninergic system in the development of diseases of the intestinal and biliferous tracts.

Journal: Bulletin of experimental biology and medicine 20090501

Title: Early deprivation leads to long-term reductions in motivation for reward and 5-HT1A binding and both effects are reversed by fluoxetine.

Journal: Neuropharmacology 20090301

Title: Pulp and paper mill effluents contain neuroactive substances that potentially disrupt neuroendocrine control of fish reproduction.

Journal: Environmental science & technology 20090301

Title: Activation of serotonin 5-HT1-receptors decreased gripping-induced immobility episodes in taiep rats.

Journal: Neuroscience letters 20090109

Title: Evidence for dopamine involvement in ambulation promoted by menthone in mice.

Journal: Pharmacology, biochemistry, and behavior 20090101

Title: Spiperone, identified through compound screening, activates calcium-dependent chloride secretion in the airway.

Journal: American journal of physiology. Cell physiology 20090101

Title: Species differences in the relative densities of D1- and D2-like dopamine receptor subtypes in the Japanese quail and rats: an in vitro quantitative receptor autoradiography study.

Journal: Brain, behavior and evolution 20090101

Title: The importance of brain banks for molecular neuropathological research: The New South Wales Tissue Resource Centre experience.

Journal: International journal of molecular sciences 20090101

Title: 5-HT-induced depression of the spinal monosynaptic reflex potential utilizes different types of 5-HT receptors depending on Mg2+ availability.

Journal: Pharmacological reports : PR 20090101

Title: The role of dopamine in Drosophila larval classical olfactory conditioning.

Journal: PloS one 20090101

Title: Roles of octopaminergic and dopaminergic neurons in appetitive and aversive memory recall in an insect.

Journal: BMC biology 20090101

Title: Selective deletion of PTEN in dopamine neurons leads to trophic effects and adaptation of striatal medium spiny projecting neurons.

Journal: PloS one 20090101

Title: Spiperone enhances intracellular calcium level and inhibits the Wnt signaling pathway.

Journal: BMC pharmacology 20090101

Title: Serotomide and safflomide modulate forskolin-stimulated cAMP formation via 5-HT1 receptor.

Journal: Phytomedicine : international journal of phytotherapy and phytopharmacology 20081201

Title: The antipsychotic spiperone attenuates inflammatory response in cultured microglia via the reduction of proinflammatory cytokine expression and nitric oxide production.

Journal: Journal of neurochemistry 20081201

Title: Targeting liver myofibroblasts: a novel approach in anti-fibrogenic therapy.

Journal: Hepatology international 20081201

Title: Chemical substructures that enrich for biological activity.

Journal: Bioinformatics (Oxford, England) 20081101

Title: Effects of selective serotonin2 ligands on behaviors evoked by stress in the rat.

Journal: Pharmacology, biochemistry, and behavior 20081001

Title: Dopamine D1 receptor inhibition of NMDA receptor currents mediated by tyrosine kinase-dependent receptor trafficking in neonatal rat striatum.

Journal: The Journal of physiology 20081001

Title: Altered dopamine D2-like receptor binding in rats with behavioral sensitization to quinpirole: effects of pre-treatment with Ro 41-1049.

Journal: European journal of pharmacology 20080911

Title: Characterization of contractile 5-hydroxytryptamine receptor subtypes in the in situ autoperfused kidney in the anaesthetized rat.

Journal: European journal of pharmacology 20080911

Title: Serotonin receptors contribute to the promnesic effects of P. olacoides (Marapuama).

Journal: Physiology & behavior 20080903

Title: 11C-NMSP/ 18F-FDG microPET to monitor neural stem cell transplantation in a rat model of traumatic brain injury.

Journal: European journal of nuclear medicine and molecular imaging 20080901

Title: Selective alterations of brain dopamine D(2) receptor binding in cirrhotic patients: results of a (11)C-N-methylspiperone PET study.

Journal: Metabolic brain disease 20080901

Title: Induction of ovarian growth in Aegla platensis (Crustacea, Aeglidae) by means of neuroregulators incorporated to food.

Journal: Revista de biologia tropical 20080901

Title: Increased dopamine after mating impairs olfaction and prevents odor interference with pregnancy.

Journal: Nature neuroscience 20080801

Title: Serotoninergic system in the development of pyloric stenosis and pancreatitis.

Journal: Bulletin of experimental biology and medicine 20080801

Title: When administered to rats in a cold environment, 3,4-methylenedioxymethamphetamine reduces brown adipose tissue thermogenesis and increases tail blood flow: effects of pretreatment with 5-HT1A and dopamine D2 antagonists.

Journal: Neuroscience 20080717

Title: Synthesis and pharmacological investigation of novel 2-aminothiazole-privileged aporphines.

Journal: Bioorganic & medicinal chemistry 20080715

Title: Dopamine receptors in the anterior insular cortex modulate long-term nociception in the rat.

Journal: European journal of pain (London, England) 20080701

Title: Mechanisms for metoclopramide-mediated sensitization and haloperidol-induced catalepsy in rats.

Journal: European journal of pharmacology 20080610

Title: Antagonist-radioligand binding to D2L-receptors in intact cells.

Journal: Biochemical pharmacology 20080601

Title: Bioisosteric heterocyclic versions of 7-{[2-(4-phenyl-piperazin-1-yl)ethyl]propylamino}-5,6,7,8-tetrahydronaphthalen-2-ol: identification of highly potent and selective agonists for dopamine D3 receptor with potent in vivo activity.

Journal: Journal of medicinal chemistry 20080522

Title: Dopamine determines the vulnerability of striatal neurons to the N-terminal fragment of mutant huntingtin through the regulation of mitochondrial complex II.

Journal: Human molecular genetics 20080515

Title: Dopamine D4 receptors regulate intracellular calcium concentration in cultured chicken cone photoreceptor cells: relationship to dopamine receptor-mediated inhibition of cAMP formation.

Journal: Brain research 20080501

Title: Dopamine D2(High) receptors on intact cells.

Journal: Synapse (New York, N.Y.) 20080401

Title: Characterization of functional roles of DRY motif in the 2nd intracellular loop of dopamine D2 and D3 receptors.

Journal: Archives of pharmacal research 20080401

Title: PET analysis of the 5-HT2A receptor inverse agonist ACP-103 in human brain.

Journal: The international journal of neuropsychopharmacology 20080301

Title: Pergolide protects CA1 neurons from apoptosis in a gerbil model of global cerebral ischemia.

Journal: Neurological research 20080201

Title: Further structure-activity relationships study of hybrid 7-{[2-(4-phenylpiperazin-1-yl)ethyl]propylamino}-5,6,7,8-tetrahydronaphthalen-2-ol analogues: identification of a high-affinity D3-preferring agonist with potent in vivo activity with long duration of action.

Journal: Journal of medicinal chemistry 20080110

Title: Food restriction markedly increases dopamine D2 receptor (D2R) in a rat model of obesity as assessed with in-vivo muPET imaging ([11C] raclopride) and in-vitro ([3H] spiperone) autoradiography.

Journal: Synapse (New York, N.Y.) 20080101

Title: A review of imaging techniques for systems biology.

Journal: BMC systems biology 20080101

Title: The neuropharmacology of (-)-stepholidine and its potential applications.

Journal: Current neuropharmacology 20071201

Title: Possible involvement of endogenous 5-HT in aggravation of cerulein-induced acute pancreatitis in mice.

Journal: Journal of pharmacological sciences 20071101

Title: Chronic SKF83959 induced less severe dyskinesia and attenuated L-DOPA-induced dyskinesia in 6-OHDA-lesioned rat model of Parkinson's disease.

Journal: Neuropharmacology 20070701

Title: Dopamine D2 receptor stimulation inhibits cold-initiated thermogenesis in brown adipose tissue in conscious rats.

Journal: Neuroscience 20070615

Title: Frontal-subcortical circuitry and behavior.

Journal: Dialogues in clinical neuroscience 20070601

Title: Dopamine stimulates 45Ca2+ uptake through cAMP, PLC/PKC, and MAPKs in renal proximal tubule cells.

Journal: Journal of cellular physiology 20070501

Title: Activation of dopamine D2 receptors in the CNS inhibits sympathetic cutaneous vasomotor alerting responses (SCVARs), contributing to clozapine's SCVAR-inhibiting action.

Journal: Progress in neuro-psychopharmacology & biological psychiatry 20070330

Title: Acute and chronic administration of the cannabinoid receptor agonist CP 55,940 attenuates tumor-evoked hyperalgesia.

Journal: European journal of pharmacology 20070308

Title: Native rat hippocampal 5-HT1A receptors show constitutive activity.

Journal: Molecular pharmacology 20070301

Title: Screening of 5-HT1A receptor antagonists using molecularly imprinted polymers.

Journal: Journal of the American Chemical Society 20070214

Title: Striatal serotonin depletion facilitates rat egocentric learning via dopamine modulation.

Journal: European journal of pharmacology 20070205

Title: Changes in levels of D1, D2, or NMDA receptors during withdrawal from brief or extended daily access to IV cocaine.

Journal: Brain research 20070202

Title: Aversive learning in honeybees revealed by the olfactory conditioning of the sting extension reflex.

Journal: PloS one 20070101

Title: [Implication of serotonin in the regulation of hemostasis in the experiment].

Journal: Anesteziologiia i reanimatologiia 20070101

Title: Tracer coupling between fish rod horizontal cells: modulation by light and dopamine but not the retinal circadian clock.

Journal: Visual neuroscience 20070101

Title: Synthesis of two potential NK1-receptor ligands using [1-11C]ethyl iodide and [1-11C]propyl iodide and initial PET-imaging.

Journal: BMC medical imaging 20070101

Title: [The role of the serotoninergic system in the pathogenesis of experimental ulcerous colitis].

Journal: Vestnik Rossiiskoi akademii meditsinskikh nauk 20070101

Title: A positron emission tomography study on the role of nigral lesions in parkinsonism in patients with amyotrophic lateral sclerosis.

Journal: Archives of neurology 20061201

Title: Ptychodiscus brevis toxin-induced depression of spinal reflexes involves 5-HT via 5-HT3 receptors modulated by NMDA receptor.

Journal: Neuroscience letters 20061127

Title: Naloxone-blocked depriming effect of anxiolytic selank on apomorphine-induced behavioral manifestations of hyperfunction of dopamine system.

Journal: Bulletin of experimental biology and medicine 20061101

Title: Perospirone is a new generation antipsychotic: evidence from a positron emission tomography study of serotonin 2 and D2 receptor occupancy in the living human brain.

Journal: Journal of clinical psychopharmacology 20061001

Title: Roles of octopaminergic and dopaminergic neurons in mediating reward and punishment signals in insect visual learning.

Journal: The European journal of neuroscience 20061001

Title: Dopamine D2 receptor-mediated G protein activation assessed by agonist-stimulated [35S]guanosine 5'-O-(gamma-thiotriphosphate) binding in rat striatal membranes.

Journal: Progress in neuro-psychopharmacology & biological psychiatry 20060930

Title: Association of caffeine to MDMA does not increase antinociception but potentiates adverse effects of this recreational drug.

Journal: Brain research 20060921

Title: Sympathetic neurotransmission in the rat testicular capsule: functional characterization and identification of mRNA encoding alpha1-adrenoceptor subtypes.

Journal: European journal of pharmacology 20060814

Title: Fluorescence studies reveal heterodimerization of dopamine D1 and D2 receptors in the plasma membrane.

Journal: Biochemistry 20060725

Title: Dopaminergic regulation of ion transport in gills of the euryhaline semiterrestrial crab Chasmagnathus granulatus: interaction between D1- and D2-like receptors.

Journal: The Journal of experimental biology 20060701

Title: Effects of dopamine D1-like receptor agonists on food-maintained operant behavior in rats.

Journal: Behavioural pharmacology 20060601

Title: Comparison of rat dopamine D2 receptor occupancy for a series of antipsychotic drugs measured using radiolabeled or nonlabeled raclopride tracer.

Journal: Life sciences 20060522

Title: Microsphere-based protease assays and screening application for lethal factor and factor Xa.

Journal: Cytometry. Part A : the journal of the International Society for Analytical Cytology 20060501

Title: Serotonin receptor antagonists discriminate between PKA- and PKC-mediated plasticity in aplysia sensory neurons.

Journal: Journal of neurophysiology 20060401

Title: Pharmacological characterization of 5-hydroxytryptamine-induced contraction in the chicken gastrointestinal tract.

Journal: Autonomic & autacoid pharmacology 20060401

Title: Dopamine D(2) receptor activation modulates perceived odor intensity.

Journal: Behavioral neuroscience 20060401

Title: Potential vascular alpha1-adrenoceptor blocking properties of an array of 5-HT receptor ligands in the rat.

Journal: European journal of pharmacology 20060327

Title: Transient and selective overexpression of dopamine D2 receptors in the striatum causes persistent abnormalities in prefrontal cortex functioning.

Journal: Neuron 20060216

Title: Dopamine, oxytocin, and vasopressin receptor binding in the medial prefrontal cortex of monogamous and promiscuous voles.

Journal: Neuroscience letters 20060213

Title: Simultaneous analysis of haloperidol, its three metabolites and two other butyrophenone-type neuroleptics by high performance liquid chromatography with dual ultraviolet detection.

Journal: Biomedical chromatography : BMC 20060201

Title: D2-like receptors mediate the expulsion phase of ejaculation elicited by 8-hydroxy-2-(di-N-propylamino)tetralin in rats.

Journal: The Journal of pharmacology and experimental therapeutics 20060201

Title: Synthesis and binding profile of constrained analogues of N-[4-(4-arylpiperazin-1-yl)butyl]-3-methoxybenzamides, a class of potent dopamine D3 receptor ligands.

Journal: The Journal of pharmacy and pharmacology 20060201

Title: Differential effects of cocaine-induced seizures and lethality on M(1)-like muscarinic and dopaminergic D (1)- and D (2)-like binding receptors in mice brain.

Journal: Cellular and molecular neurobiology 20060201

Title: Investigation of the alternatively spliced insert region of the D2L dopamine receptor by epitope substitution.

Journal: Neuroscience letters 20060130

Title: Investigation of cooperativity in the binding of ligands to the D(2) dopamine receptor.

Journal: Molecular pharmacology 20060101

Title: Structural determinants of pharmacological specificity between D(1) and D(2) dopamine receptors.

Journal: Molecular pharmacology 20060101

Title: Pramipexole protects against H2O2-induced PC12 cell death.

Journal: Naunyn-Schmiedeberg's archives of pharmacology 20060101

Title: Influence of human B-casomorphin-7 on specific binding of 3H-spiperone to the 5-HT2-receptors of rat brain frontal cortex.

Journal: Protein and peptide letters 20060101

Title: Serotonin 5-HT2A and 5-HT6 receptors in the prefrontal cortex of Alzheimer and normal aging patients.

Journal: BMC neuroscience 20060101

Title: Dopamine presynaptically and heterogeneously modulates nucleus accumbens medium-spiny neuron GABA synapses in vitro.

Journal: BMC neuroscience 20060101

Title: Interaction between different parts of the autonomic nervous system in the regulation of smooth muscles in the femoral artery and trachea.

Journal: Bulletin of experimental biology and medicine 20060101

Title: Dibenzazecine compounds with a novel dopamine/5HT2A receptor profile and 3D-QSAR analysis.

Journal: BMC pharmacology 20060101

Title: Review of F-FDG Synthesis and Quality Control.

Journal: Biomedical imaging and intervention journal 20060101

Title: Modifications in muscarinic, dopaminergic and serotonergic receptors concentrations in the hippocampus and striatum of epileptic rats.

Journal: Life sciences 20051205

Title: Reactions between beta-casomorphins-7 and 5-HT2-serotonin receptors.

Journal: Bulletin of experimental biology and medicine 20051101

Title: 8-(Heteroaryl)phenalkyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-ones as opioid receptor modulators.

Journal: Medicinal chemistry (Shariqah (United Arab Emirates)) 20051101

Title: Differential in vivo inhibition of [3H]nemonapride binding by atypical antipsychotics in rat striatum, olfactory lobes, and frontal cortex.

Journal: Pharmacology 20051001

Title: Competitive MS binding assays for dopamine D2 receptors employing spiperone as a native marker.

Journal: Chembiochem : a European journal of chemical biology 20051001

Title: KKHA-761, a potent D3 receptor antagonist with high 5-HT1A receptor affinity, exhibits antipsychotic properties in animal models of schizophrenia.

Journal: Pharmacology, biochemistry, and behavior 20051001

Title: Participation of octopaminergic reward system and dopaminergic punishment system in insect olfactory learning revealed by pharmacological study.

Journal: The European journal of neuroscience 20050901

Title: Cognitive effects of dopaminergic and glutamatergic blockade in nucleus accumbens in pigeons.

Journal: Pharmacology, biochemistry, and behavior 20050801

Title: N1/P2 component of auditory evoked potential reflect changes of the brain serotonin biosynthesis in rats.

Journal: Nutritional neuroscience 20050801

Title: 2-[4-(3,4-Dimethylphenyl)piperazin-1-ylmethyl]-1H benzoimidazole (A-381393), a selective dopamine D4 receptor antagonist.

Journal: Neuropharmacology 20050701

Title: Reciprocal mutations in TM2/TM3 in a D2 dopamine receptor background confirms the importance of this microdomain as a selective determinant of para-halogenated 1,4-disubstituted aromatic piperazines.

Journal: Archiv der Pharmazie 20050601

Title: Chirospecific and subtype selective dopamine receptor binding of heterocyclic methoxynaphthamide analogs.

Journal: Archiv der Pharmazie 20050601

Title: Effects of mercury on neurochemical receptors in wild river otters (Lontra canadensis).

Journal: Environmental science & technology 20050515

Title: Enhanced binding of dopamine D1 receptors in caudate-putamen subregions in High-Yawning Sprague-Dawley rats.

Journal: Synapse (New York, N.Y.) 20050501

Title: Mechanisms of inverse agonist action at D2 dopamine receptors.

Journal: British journal of pharmacology 20050501

Title: Dopamine D2 receptor stimulation of mitogen-activated protein kinases mediated by cell type-dependent transactivation of receptor tyrosine kinases.

Journal: Journal of neurochemistry 20050501

Title: Dopamine receptor activation in bovine pinealocyte via a cAMP-dependent transcription pathway.

Journal: Journal of pineal research 20050401

Title: The role of the phosphatidyinositol-linked D1 dopamine receptor in the pharmacology of SKF83959.

Journal: Pharmacology, biochemistry, and behavior 20050401

Title: Estrogen mediated inhibition of dopamine transport in the striatum: regulation by G alpha i/o.

Journal: European journal of pharmacology 20050328

Title: Stimulation of 5-HT1A receptor with 8-OH-DPAT inhibits hydrogen peroxide-induced neurotoxicity in cultured rat cortical cells.

Journal: Pharmacological research 20050301

Title: Modeling the similarity and divergence of dopamine D2-like receptors and identification of validated ligand-receptor complexes.

Journal: Journal of medicinal chemistry 20050210

Title: Developmental neurotoxicity of pyrethroid insecticides: critical review and future research needs.

Journal: Environmental health perspectives 20050201

Title: Distribution of D1-like and D2-like dopamine receptors in the brain of genetic epileptic WAG/Rij rats.

Journal: Epilepsy research 20050201

Title: Effect of dopamine injection into caudate nucleus on immune responsiveness in rats: a pilot study.

Journal: Immunology letters 20050115

Title: Synthesis and structure-activity relationships of 1-aralkyl-4-benzylpiperidine and 1-aralkyl-4-benzylpiperazine derivatives as potent sigma ligands.

Journal: Journal of medicinal chemistry 20050113

Title: Effects of long-term biogenic amine transporter blockade on receptor/G-protein coupling in rat brain.

Journal: Neuropharmacology 20050101

Title: Prenatal ethanol preferentially enhances reactivity of the dopamine D1 but not D2 or D3 receptors in offspring.

Journal: Neurotoxicology and teratology 20050101

Title: Evidence for 5-HT2B and 5-HT7 receptor-mediated relaxation in pulmonary arteries of weaned pigs.

Journal: Naunyn-Schmiedeberg's archives of pharmacology 20050101

Title: Behavioral and neurochemical effects on rat offspring after prenatal exposure to ethanol.

Journal: Neurotoxicology and teratology 20050101

Title: Biphasic firing response of nucleus accumbens neurons elicited by THPB-18 and its correlation with DA receptor subtypes.

Journal: Acta pharmacologica Sinica 20041201

Title: Aglycemia and ischemia depress monosynaptic and polysynaptic reflexes in neonatal rat spinal cord in vitro by involving different types of 5-hydroxytryptamine receptors.

Journal: Neuroscience letters 20041130

Title: Atypical properties of several classes of antipsychotic drugs on the basis of differential induction of Fos-like immunoreactivity in the rat brain.

Journal: Life sciences 20041126

Title: Targeted mutation of CCK(2) receptor gene antagonises behavioural changes induced by social isolation in female, but not in male mice.

Journal: Behavioural brain research 20041105

Title: The influence of G protein subtype on agonist action at D2 dopamine receptors.

Journal: Neuropharmacology 20041101

Title: Reduced hypophagic effects of d-fenfluramine and the 5-HT2C receptor agonist mCPP in 5-HT1B receptor knockout mice.

Journal: Psychopharmacology 20041001

Title: Cloned human 5-HT1A receptor pharmacology determined using agonist binding and measurement of cAMP accumulation.

Journal: The Journal of pharmacy and pharmacology 20041001

Title: MDMA-evoked changes in [11C]raclopride and [11C]NMSP binding in living pig brain.

Journal: Synapse (New York, N.Y.) 20040915

Title: Cerebral D2 and 5-HT2 receptor occupancy in Schizophrenic patients treated with olanzapine or clozapine.

Journal: Journal of psychopharmacology (Oxford, England) 20040901

Title: Pharmacological characterisation of the agonist radioligand binding site of 5-HT(2A), 5-HT(2B) and 5-HT(2C) receptors.

Journal: Naunyn-Schmiedeberg's archives of pharmacology 20040801

Title: Novel regulatory properties of human type 9 adenylate cyclase.

Journal: The Journal of pharmacology and experimental therapeutics 20040701

Title: Electrostatic surface potential calculation on several new halogenated benzimidazole-like dopaminergic ligands.

Journal: Archiv der Pharmazie 20040701

Title: Early administration of tiapride to young rats without long-lasting changes in the development of the dopaminergic system.

Journal: Pharmacopsychiatry 20040701

Title: Lack of restraint-induced increases of brain serotonin metabolism in rats treated with spiperone: relationship with restraint-induced behavioral deficits.

Journal: Pakistan journal of pharmaceutical sciences 20040701

Title: Vasoconstrictor responses to 5-hydroxytryptamine in the autoperfused hindquarters of spontaneously hypertensive rats.

Journal: Pharmacology 20040601

Title: Measurement of dopamine D2-like receptors in postmortem CNS and pituitary: differential regional changes in schizophrenia.

Journal: Life sciences 20040507

Title: Investigation of the mechanism of agonist and inverse agonist action at D2 dopamine receptors.

Journal: Biochemical pharmacology 20040501

Title: Antipsychotic drugs influence transport of the beta-adrenergic antagonist [3H]-dihydroalprenolol into neuronal and blood cells.

Journal: The world journal of biological psychiatry : the official journal of the World Federation of Societies of Biological Psychiatry 20040401

Title: Micro-positron emission tomography imaging of cardiac gene expression in rats using bicistronic adenoviral vector-mediated gene delivery.

Journal: Circulation 20040323

Title: Evidence that alpha(1B)-adrenoceptors are involved in noradrenaline-induced contractions of rat tail artery.

Journal: European journal of pharmacology 20040319

Title: Pharmacological properties of serotonin receptor subtypes mediating contraction of bovine inferior alveolar arteries.

Journal: Archives of oral biology 20040301

Title: Opposing effects of D1 and D2 receptor activation on odor discrimination learning.

Journal: Behavioral neuroscience 20040201

Title: Cocaine treatment causes early and long-lasting changes in muscarinic and dopaminergic receptors.

Journal: Cellular and molecular neurobiology 20040201

Title: A circadian clock in the fish retina regulates dopamine release via activation of melatonin receptors.

Journal: The Journal of physiology 20040115

Title: Sensitization of neuronal A2A adenosine receptors after persistent D2 dopamine receptor activation.

Journal: The Journal of pharmacology and experimental therapeutics 20040101

Title: Postnatal haloperidol eliminates the deficit in circling behavior produced by prenatal exposure to the same drug.

Journal: Neurotoxicology and teratology 20040101

Title: Comparison of brain activity between dopamine D2 receptor-knockout and wild mice in response to dopamine agonist and antagonist assessed by fMRI.

Journal: Neuro-Signals 20040101

Title: Optimization of the pharmacophore model for 5-HT7R antagonism. Design and synthesis of new naphtholactam and naphthosultam derivatives.

Journal: Journal of medicinal chemistry 20031218

Title: Direct activation by dopamine of recombinant human 5-HT1A receptors: comparison with human 5-HT2C and 5-HT3 receptors.

Journal: Synapse (New York, N.Y.) 20031215

Title: Absence of circadian clock regulation of horizontal cell gap junctional coupling reveals two dopamine systems in the goldfish retina.

Journal: The Journal of comparative neurology 20031208

Title: Elevated neuronal nitric oxide synthase expression in chronic haloperidol-treated rats.

Journal: Neuropharmacology 20031201

Title: Pharmacological characterization of a serotonin receptor (5-HT7) stimulating cAMP production in human corneal epithelial cells.

Journal: Investigative ophthalmology & visual science 20031101

Title: Human umbilical vein vasoconstriction induced by epinephrine acting on alpha1B-adrenoceptor subtype.

Journal: American journal of obstetrics and gynecology 20031101

Title: [Effects of D1 and D2 dopamine receptor agonists and antagonists on cerebral ischemia/reperfusion injury].

Journal: Sheng li xue bao : [Acta physiologica Sinica] 20031025

Title: Molecular modeling of the three-dimensional structure of dopamine 3 (D3) subtype receptor: discovery of novel and potent D3 ligands through a hybrid pharmacophore- and structure-based database searching approach.

Journal: Journal of medicinal chemistry 20031009

Title: Effects of D1- and D2-dopamine receptor activation on melatonin synthesis in bovine pinealocytes.

Journal: Journal of pineal research 20031001

Title: Pilocarpine-induced seizures in adult rats: monoamine content and muscarinic and dopaminergic receptor changes in the striatum.

Journal: Comparative biochemistry and physiology. Toxicology & pharmacology : CBP 20031001

Title: Dopamine displaces [3H]domperidone from high-affinity sites of the dopamine D2 receptor, but not [3H]raclopride or [3H]spiperone in isotonic medium: Implications for human positron emission tomography.

Journal: Synapse (New York, N.Y.) 20030915

Title: Comparison of hippocampal G protein activation by 5-HT(1A) receptor agonists and the atypical antipsychotics clozapine and S16924.

Journal: Naunyn-Schmiedeberg's archives of pharmacology 20030901

Title: Pharmacologic identification of putative D1 dopamine receptors in feline kidneys.

Journal: Journal of veterinary pharmacology and therapeutics 20030801

Title: Higher-end serotonin receptors: 5-HT(5), 5-HT(6), and 5-HT(7).

Journal: Journal of medicinal chemistry 20030703

Title: Characterization of dopamine D2 receptor gene expression and binding sites in human placenta amniotic epithelial cells.

Journal: Placenta 20030701

Title: Pharmacological analysis of a dopamine D(2Short):G(alphao) fusion protein expressed in Sf9 cells.

Journal: FEBS letters 20030619

Title: Distinct effects of amantadine and memantine on dopaminergic transmission in the rat striatum.

Journal: Neuroscience letters 20030612

Title: Pharmacological and functional characterisation of dopamine D4 receptors in the rat retina.

Journal: Neuropharmacology 20030601

Title: Sigma1 and dopamine D2 receptor occupancy in the mouse brain after a single administration of haloperidol and two dopamine D2-like receptor ligands.

Journal: Nuclear medicine and biology 20030501

Title: 5-HT(2A) receptor binding is reduced in drug-naive and unchanged in SSRI-responder depressed patients compared to healthy controls: a PET study.

Journal: Psychopharmacology 20030401

Title: Interaction of the D2short dopamine receptor with G proteins: analysis of receptor/G protein selectivity.

Journal: Biochemical pharmacology 20030401

Title: Photic regulation of heme oxygenase activity in the golden hamster retina: involvement of dopamine.

Journal: Journal of neurochemistry 20030401

Title: Effect of sabcomeline on muscarinic and dopamine receptor binding in intact mouse brain.

Journal: Annals of nuclear medicine 20030401

Title: Biphasic role of dopamine on female sexual behaviour via D2 receptors in the mediobasal hypothalamus.

Journal: Neuropharmacology 20030301

Title: Pharmacological characterization of an adenylyl cyclase-coupled 5-HT receptor in aplysia: comparison with mammalian 5-HT receptors.

Journal: Journal of neurophysiology 20030301

Title: 5-HT7 receptor-mediated relaxation of the oviduct in nonpregnant proestrus pigs.

Journal: European journal of pharmacology 20030214

Title: In vivo evidence for dopamine-mediated internalization of D2-receptors after amphetamine: differential findings with [3H]raclopride versus [3H]spiperone.

Journal: Molecular pharmacology 20030201

Title: GABA(A) alpha 1 subunit knock-out mice do not show a hyperlocomotor response following amphetamine or cocaine treatment.

Journal: Neuropharmacology 20030201

Title: CCK2 receptor-deficient mice have increased sensitivity of dopamine D2 receptors.

Journal: Neuropeptides 20030201

Title: 5-HT(2) receptor-mediated phosphoinositide hydrolysis in bovine ciliary epithelium.

Journal: Journal of ocular pharmacology and therapeutics : the official journal of the Association for Ocular Pharmacology and Therapeutics 20030201

Title: Evidence for the involvement of dopamine in ambulation promoted by menthol in mice.

Journal: Journal of pharmacological sciences 20030201

Title: Characterization of the 5-hydroxytryptamine receptors mediating contraction in the pig isolated intravesical ureter.

Journal: British journal of pharmacology 20030101

Title: Corticotropin-releasing factor as well as opioid and dopamine are involved in tail-pinch-induced food intake of rats.

Journal: Neuroscience 20030101

Title: Behavioral response profiles following drug challenge with dopamine receptor subtype agonists and antagonists in developing rat.

Journal: Neurotoxicology and teratology 20030101

Title: Axonal degeneration and progressive neurologic disability in multiple sclerosis.

Journal: Neurotoxicity research 20030101

Title: Kinetics of synaptic transfer from rods and cones to horizontal cells in the salamander retina.

Journal: Neuroscience 20030101

Title: Targeted molecular imaging.

Journal: Korean journal of radiology 20030101

Title: The role of catecholamines in retention performance of a partially baited radial eight-arm maze for rats.

Journal: The Chinese journal of physiology 20021231

Title: Novel (bisarylmethoxy)butylpiperidine analogues as neurotransmitter transporter inhibitors with activity at dopamine receptor sites.

Journal: Bioorganic & medicinal chemistry 20021201

Title: Inhibition of protein tyrosine/mitogen-activated protein kinase phosphatase activity is associated with D2 dopamine receptor supersensitivity in a rat model of Parkinson's disease.

Journal: Molecular pharmacology 20021201

Title: Characterization of 5-HT receptor subtypes mediating contraction in human umbilical vein. 1. Evidence of involvement of 5-HT2A receptors using functional and radioligand binding assays.

Journal: Naunyn-Schmiedeberg's archives of pharmacology 20021201

Title: Functional cooperation between neurosteroids and D2 dopamine antagonists on KCl-evoked [3H]noradrenaline release: modulation by calcium channel blockers.

Journal: Journal of neuroendocrinology 20021201

Title: Serotonin-induced MMP-13 production is mediated via phospholipase C, protein kinase C, and ERK1/2 in rat uterine smooth muscle cells.

Journal: The Journal of biological chemistry 20021108

Title: Dopamine mediates circadian clock regulation of rod and cone input to fish retinal horizontal cells.

Journal: The Journal of physiology 20021101

Title: In vivo serotonin 5HT(2A) receptor binding and personality traits in healthy subjects: a positron emission tomography study.

Journal: NeuroImage 20021101

Title: Changes in electrophysiological properties of lamprey spinal motoneurons during fictive swimming.

Journal: Journal of neurophysiology 20021101

Title: Spreading depression: imaging and blockade in the rat neocortical brain slice.

Journal: Journal of neurophysiology 20021101

Title: Apomorphine induces trophic factors that support fetal rat mesencephalic dopaminergic neurons in cultures.

Journal: The European journal of neuroscience 20021101

Title: Effect of nooglutil on benzodiazepine withdrawal syndrome and binding of 3H-spiperone with D2 receptors in rat striatum.

Journal: Bulletin of experimental biology and medicine 20021101

Title: Synthesis and structure-activity relationship of the isoindolinyl benzisoxazolpiperidines as potent, selective, and orally active human dopamine D4 receptor antagonists.

Journal: Chembiochem : a European journal of chemical biology 20021004

Title: Antibody capture assay reveals bell-shaped concentration-response isotherms for h5-HT(1A) receptor-mediated Galpha(i3) activation: conformational selection by high-efficacy agonists, and relationship to trafficking of receptor signaling.

Journal: Molecular pharmacology 20020901

Title: Development of an automated system for synthesizing 18F-labeled compounds using [18F]fluoroethyl bromide as a synthetic precursor.

Journal: Applied radiation and isotopes : including data, instrumentation and methods for use in agriculture, industry and medicine 20020901

Title: Effects of rolipram on in vivo dopamine receptor binding.

Journal: Journal of neural transmission (Vienna, Austria : 1996) 20020901

Title: Metachlorophenylpiperazine (m-CPP) induced intracavernous pressure responses in anaesthetized rats.

Journal: International journal of impotence research 20020801

Title: Aripiprazole, a novel antipsychotic, is a high-affinity partial agonist at human dopamine D2 receptors.

Journal: The Journal of pharmacology and experimental therapeutics 20020701

Title: Effects of intrathecal injection of diatrizoate on dopamine receptors.

Journal: Academic radiology 20020701

Title: Ketanserin and spiperone as templates for novel serotonin 5-HT(2A) antagonists.

Journal: Current topics in medicinal chemistry 20020601

Title: Effect of dopamine receptor agonists on sensory nerve activity: possible therapeutic targets for the treatment of asthma and COPD.

Journal: British journal of pharmacology 20020601

Title: Adenosinergic modulation of the discriminative-stimulus effects of methamphetamine in rats.

Journal: Psychopharmacology 20020601

Title: Functional screening of G protein-coupled receptors by measuring intracellular calcium with a fluorescence microplate reader.

Journal: Journal of biomolecular screening 20020601

Title: Serotonin antagonist profiling on 5HT2A and 5HT2C receptors by nonequilibrium intracellular calcium response using an automated flow-through fluorescence analysis system, HT-PS 100.

Journal: Journal of biomolecular screening 20020601

Title: Design and synthesis of a piperazinylalkylisoxazole library for subtype selective dopamine receptor ligands.

Journal: Bioorganic & medicinal chemistry letters 20020520

Title: Hemiparkinsonism associated with a mesencephalic tumor.

Journal: Journal of the neurological sciences 20020515

Title: Contrasting effects of dopamine antagonists and frequency reduction on Fos expression induced by lateral hypothalamic stimulation.

Journal: Behavioural brain research 20020514

Title: Enhanced detection of receptor constitutive activity in the presence of regulators of G protein signaling: applications to the detection and analysis of inverse agonists and low-efficacy partial agonists.

Journal: Molecular pharmacology 20020501

Title: Brain neurotransmitter receptor binding and nootropic studies on Indian Hypericum perforatum Linn.

Journal: Phytotherapy research : PTR 20020501

Title: Sustained ER Ca2+ depletion suppresses protein synthesis and induces activation-enhanced cell death in mast cells.

Journal: The Journal of biological chemistry 20020419

Title: Physiologically identified 5-HT2-like receptors at the crayfish neuromuscular junction.

Journal: Brain research 20020405

Title: Hypothalamic paraventricular 5-hydroxytryptamine: receptor-specific inhibition of NPY-stimulated eating and energy metabolism.

Journal: Pharmacology, biochemistry, and behavior 20020401

Title: Neuropharmacological profile of a novel potential atypical antipsychotic drug Y-931 (8-fluoro-12-(4-methylpiperazin-1-yl)- 6H-[1]benzothieno[2,3-b][1,5] benzodiazepine maleate).

Journal: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20020401

Title: (+)-[76Br]A-69024: a non-benzazepine radioligand for studies of dopamine D1 receptors using PET.

Journal: Nuclear medicine and biology 20020401

Title: Positron emission tomography and ex vivo and in vitro autoradiography studies on dopamine D2-like receptor degeneration in the quinolinic acid-lesioned rat striatum: comparison of [11C]raclopride, [11C]nemonapride and [11C]N-methylspiperone.

Journal: Nuclear medicine and biology 20020401

Title: Timing is everything: the effects of putative dopamine antagonists on metamorphosis vary with larval age and experimental duration in the prosobranch gastropod Crepidula fornicata.

Journal: The Biological bulletin 20020401

Title: The atypical 5-HT2 receptor mediating tachycardia in pithed rats: pharmacological correlation with the 5-HT2A receptor subtype.

Journal: British journal of pharmacology 20020301

Title: The human 5-HT7 serotonin receptor splice variants: constitutive activity and inverse agonist effects.

Journal: British journal of pharmacology 20020301

Title: A novel series of hybrid compounds derived by combining 2-aminotetralin and piperazine fragments: binding activity at D2 and D3 receptors.

Journal: Bioorganic & medicinal chemistry letters 20020225

Title: In vitro evidence that 5-hydroxytryptamine increases efflux of glial glutamate via 5-HT(2A) receptor activation.

Journal: Journal of neuroscience research 20020201

Title: Effects of some steroids and other compounds on ovarian growth of the red swamp crayfish, Procambarus clarkii, during early vitellogenesis.

Journal: The Journal of experimental zoology 20020101

Title: Implementation and evaluation of a 3D one-step late reconstruction algorithm for 3D positron emission tomography brain studies using median root prior.

Journal: European journal of nuclear medicine and molecular imaging 20020101

Title: Atmospheric pressure laser desorption/chemical ionization mass spectrometry: a new ionization method based on existing themes.

Journal: Rapid communications in mass spectrometry : RCM 20020101

Title: Decreased [(3)H]spiperone binding in the anterior cingulate cortex of schizophrenia patients: an autoradiographic study.

Journal: Neuroscience 20020101

Title: [Dopamine antibodies as neuromodulators of behavioral reactions in mice of different genotypes].

Journal: Zhurnal vysshei nervnoi deiatelnosti imeni I P Pavlova 20020101

Title: The effects of dopamine synthesis inhibitors and dopamine antagonists on regeneration in the hydra Hydra attenuata.

Journal: Neuroscience and behavioral physiology 20020101

Title: Occurrence of dopaminergic (D(2)) receptors within the rabbit pulmonary circulation.

Journal: Pulmonary pharmacology & therapeutics 20020101

Title: Nad-299 antagonises 5-HT-stimulated and spiperone-inhibited [35S]GTPgammaS binding in cloned 5-HT1A receptors.

Journal: Journal of receptor and signal transduction research 20020101

Title: (-)S amisulpride binds with high affinity to cloned dopamine D(3) and D(2) receptors.

Journal: European journal of pharmacology 20011207

Title: Expression of catecholaminergic mRNAs in the hyperactive mouse mutant coloboma.

Journal: Brain research. Molecular brain research 20011130

Title: Modulation of [3H]quinpirole binding at striatal D2 dopamine receptors by a monoamine oxidaseA-like site: evidence from radioligand binding studies and D2 receptor- and MAO(A)-deficient mice.

Journal: Life sciences 20011130

Title: Effects of endogenous neurotransmitters on the in vivo binding of dopamine and 5-HT radiotracers in mice.

Journal: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20011101

Title: Modulation of dopamine uptake in rat nucleus accumbens: effect of specific dopamine receptor antagonists and sigma ligands.

Journal: Neuroscience letters 20011026

Title: Noninvasive, quantitative imaging in living animals of a mutant dopamine D2 receptor reporter gene in which ligand binding is uncoupled from signal transduction.

Journal: Gene therapy 20011001

Title: Benzamide bioisosteres incorporating dihydroheteroazole substructures: EPC synthesis and SAR leading to a selective dopamine D4 receptor partial agonist (FAUC 179).

Journal: Bioorganic & medicinal chemistry letters 20010917

Title: Determination of dopamine D(4) receptor density in rat striatum using PB12 as a probe.

Journal: European journal of pharmacology 20010907

Title: New 1-aryl-4-(biarylmethylene)piperazines as potential atypical antipsychotics sharing dopamine D(2)-receptor and serotonin 5-HT(1A)-receptor affinities.

Journal: Bioorganic & medicinal chemistry letters 20010903

Title: Dosing time-dependent tolerance of catalepsy by repetitive administration of haloperidol in mice.

Journal: The Journal of pharmacology and experimental therapeutics 20010901

Title: Dopamine inhibits vasopressin action in the rat inner medullary collecting duct via alpha(2)-adrenoceptors.

Journal: The Journal of pharmacology and experimental therapeutics 20010901

Title: Agonist regulation of D(2) dopamine receptor/G protein interaction. Evidence for agonist selection of G protein subtype.

Journal: The Journal of biological chemistry 20010803

Title: Direct correlation between positron emission tomographic images of two reporter genes delivered by two distinct adenoviral vectors.

Journal: Gene therapy 20010701

Title: Pharmacological evaluation of (+)-2- [123I]A-69024: a radioligand for in vivo studies of dopamine D1 receptors.

Journal: Life sciences 20010629

Title: Dopamine D2 receptor dimer formation: evidence from ligand binding.

Journal: The Journal of biological chemistry 20010622

Title: Hypericum perforatum as a nootropic drug: enhancement of retrieval memory of a passive avoidance conditioning paradigm in mice.

Journal: Journal of ethnopharmacology 20010601

Title: The cloned human 5-HT7 receptor splice variants: a comparative characterization of their pharmacology, function and distribution.

Journal: Naunyn-Schmiedeberg's archives of pharmacology 20010601

Title: Stimulation of sodium-dependent inorganic phosphate transport by activation of Gi/o-protein-coupled receptors by epinephrine in MC3T3-E1 osteoblast-like cells.

Journal: Bone 20010601

Title: Affinity of serotonin receptor antagonists and agonists to recombinant and native alpha1-adrenoceptor subtypes.

Journal: Japanese journal of pharmacology 20010601

Title: Pharmacological characterization of the D1- and D2-like dopamine receptors from the brain of the leopard frog, Rana pipiens.

Journal: Brain, behavior and evolution 20010601

Title: Differential effects of 5-HT1A receptor deletion upon basal and fluoxetine-evoked 5-HT concentrations as revealed by in vivo microdialysis.

Journal: Brain research 20010525

Title: Reversible decrease of dopamine D2 receptor density in the striatum of rats with acute hepatic failure.

Journal: Brain research 20010504

Title: D2 but not D3 receptors are elevated after 9 or 11 months chronic haloperidol treatment: influence of withdrawal period.

Journal: Synapse (New York, N.Y.) 20010501

Title: D(3) dopamine receptors in rat spinal cord: implications for sensory and motor function.

Journal: Neuroscience letters 20010427

Title: Effects of dopaminergic agents on carrageenan hyperalgesia after intrathecal administration to rats.

Journal: European journal of pharmacology 20010420

Title: Cis- and trans-N-benzyl-octahydrobenzo[g]quinolines. Adrenergic and dopaminergic activity studies.

Journal: Bioorganic & medicinal chemistry letters 20010409

Title: Characterization of the serotonin receptor mediating contraction in the mouse thoracic aorta and signal pathway coupling.

Journal: The Journal of pharmacology and experimental therapeutics 20010401

Title: Mechanisms of inverse agonism of antipsychotic drugs at the D(2) dopamine receptor: use of a mutant D(2) dopamine receptor that adopts the activated conformation.

Journal: Journal of neurochemistry 20010401

Title: The role of D2-like dopamine receptors in the locomotor stimulant effects of cocaine in mice.

Journal: Psychopharmacology 20010401

Title: Alteration of dopamine transport in the striatum and nucleus accumbens of ovariectomized and estrogen-primed rats following N-(p-isothiocyanatophenethyl) spiperone (NIPS) treatment.

Journal: Brain research bulletin 20010401

Title: S 14506: novel receptor coupling at 5-HT(1A) receptors.

Journal: Neuropharmacology 20010301

Title: Failure of AH11110A to functionally discriminate between alpha(1)-adrenoceptor subtypes A, B and D or between alpha(1)- and alpha(2)-adrenoceptors.

Journal: European journal of pharmacology 20010301

Title: Stimulus properties of 7-OH-DPAT versus auto- and postsynaptic receptor-specific doses of quinpirole.

Journal: Pharmacology, biochemistry, and behavior 20010301

Title: Effects of intrastriatal infusion of D2 and D3 dopamine receptor preferring antagonists on dopamine release in rat dorsal striatum (in vivo microdialysis study).

Journal: Pharmacological research 20010301

Title: Increased 5-hydroxytryptamine-2 receptor binding in the frontal cortex of depressed patients responding to paroxetine treatment: a positron emission tomography scan study.

Journal: Journal of clinical psychopharmacology 20010201

Title: The effect of nicotine and haloperidol co-treatment on nicotinic receptor levels in the rat brain.

Journal: Brain research. Molecular brain research 20010131

Title: Modulation of 5-HT(1A) receptor activation by its interaction with wild-type and mutant g(alphai3) proteins.

Journal: Neuropharmacology 20010101

Title: Differential modulation by GTPgammaS of agonist and inverse agonist binding to h5-HT(1A) receptors revealed by [3H]-WAY100,635.

Journal: British journal of pharmacology 20010101

Title: Dopaminergic activity in transgenic mice underexpressing glucocorticoid receptors: effect of antidepressants.

Journal: Neuroscience 20010101

Title: Recent advances in imaging endogenous or transferred gene expression utilizing radionuclide technologies in living subjects: applications to breast cancer.

Journal: Breast cancer research : BCR 20010101

Title: A consideration of the dopamine D2 receptor monomer-dimer equilibrium and the anomalous binding properties of the dopamine D2 receptor ligand, N-methyl spiperone.

Journal: Journal of neural transmission (Vienna, Austria : 1996) 20010101

Title: Effects of lithium on dopamine D2 receptor expression in the rat brain striatum.

Journal: Journal of neural transmission (Vienna, Austria : 1996) 20010101

Title: Dopamine depletion with 6-OHDA enhances dopamine D1-receptor modulation of potassium currents in retinal bipolar cells.

Journal: Visual neuroscience 20010101

Title: Patterns of cyclic AMP formation by coexpressed D1 and D2L dopamine receptors in HEK 293 cells.

Journal: Receptors & channels 20010101

Title: Differential modes of agonist binding to 5-hydroxytryptamine(2A) serotonin receptors revealed by mutation and molecular modeling of conserved residues in transmembrane region 5.

Journal: Molecular pharmacology 20001101

Title: Inverse agonist activity of atypical antipsychotic drugs at human 5-hydroxytryptamine2C receptors.

Journal: The Journal of pharmacology and experimental therapeutics 20001001

Title: Regulation of human D(1), d(2(long)), d(2(short)), D(3) and D(4) dopamine receptors by amiloride and amiloride analogues.

Journal: British journal of pharmacology 20000701

Title: The effects of benzamide analogues on cocaine self-administration in rhesus monkeys.

Journal: Psychopharmacology 19991101

Title: Enhanced striatal dopamine D(2) receptor-induced [35S]GTPgammaS binding after haloperidol treatment.

Journal: European journal of pharmacology 19991008

Title: Synthesis and preliminary pharmacological investigations of 1-(1,2-dihydro-2-acenaphthylenyl)piperazine derivatives as potential atypical antipsychotic agents in mice.

Journal: Farmaco (Societa chimica italiana : 1989) 19990830

Title: Zinc modulates antagonist interactions with D2-like dopamine receptors through distinct molecular mechanisms.

Journal: The Journal of pharmacology and experimental therapeutics 19990501

Title: High-affinity agonist binding correlates with efficacy (intrinsic activity) at the human serotonin 5-HT2A and 5-HT2C receptors: evidence favoring the ternary complex and two-state models of agonist action.

Journal: Journal of neurochemistry 19990501

Title: Characterization of alpha1-adrenoceptor subtypes mediating noradrenaline-induced contraction of rat epididymal vas deferens in calcium-free medium.

Journal: Life sciences 19990101

Title: Agonist and antagonist actions of antipsychotic agents at 5-HT1A receptors: a [35S]GTPgammaS binding study.

Journal: European journal of pharmacology 19980821

Title: Creation of a constitutively activated state of the 5-hydroxytryptamine2A receptor by site-directed mutagenesis: inverse agonist activity of antipsychotic drugs.

Journal: The Journal of pharmacology and experimental therapeutics 19980701

Title: Labelling of recombinant human and native rat serotonin 5-HT1A receptors by a novel, selective radioligand, [3H]-S 15535: definition of its binding profile using agonists, antagonists and inverse agonists.

Journal: Naunyn-Schmiedeberg's archives of pharmacology 19980301

Title: [3H]Rauwolscine: an antagonist radioligand for the cloned human 5-hydroxytryptamine2b (5-HT2B) receptor.

Journal: Naunyn-Schmiedeberg's archives of pharmacology 19980101

Title: Cloning, expression and pharmacology of a truncated splice variant of the human 5-HT7 receptor (h5-HT7b).

Journal: British journal of pharmacology 19970901

Title: Zinc allosterically modulates antagonist binding to cloned D1 and D2 dopamine receptors.

Journal: Journal of neurochemistry 19970501

Title: Bromocriptine transcriptionally activates the multidrug resistance gene (pgp2/mdr1b) by a novel pathway.

Journal: The Journal of biological chemistry 19970425

Title: The behavioural effects of pramipexole, a novel dopamine receptor agonist.

Journal: European journal of pharmacology 19970411

Title: Synthesis and biological profile of the enantiomers of [4-(4-amino-6,7-dimethoxyquinazolin-2-yl)-cis-octahydroquinoxalin- 1-yl]furan-2-ylmethanone (cyclazosin), a potent competitive alpha 1B- adrenoceptor antagonist.

Journal: Journal of medicinal chemistry 19961108

Title: Nefiracetam (DM-9384) reverses apomorphine-induced amnesia of a passive avoidance response: delayed emergence of the memory retention effects.

Journal: Neurochemical research 19960601

Title: Critical reevaluation of spiperone and benzamide binding to dopamine D2 receptors: evidence for identical binding sites.

Journal: European journal of pharmacology 19960506

Title: Radiolabelling of the human 5-HT2A receptor with an agonist, a partial agonist and an antagonist: effects on apparent agonist affinities.

Journal: Biochemical pharmacology 19960112

Title: ABT-431: the diacetyl prodrug of A-86929, a potent and selective dopamine D1 receptor agonist: in vitro characterization and effects in animal models of Parkinson's disease.

Journal: The Journal of pharmacology and experimental therapeutics 19960101

Title: Roxindole, a potential antidepressant. I. Effect on the dopamine system.

Journal: Journal of neural transmission (Vienna, Austria : 1996) 19960101

Title: Neurochemical and functional characterization of the preferentially selective dopamine D3 agonist PD 128907.

Journal: The Journal of pharmacology and experimental therapeutics 19951201

Title: Functional correlates of dopamine D3 receptor activation in the rat in vivo and their modulation by the selective antagonist, (+)-S 14297: 1. Activation of postsynaptic D3 receptors mediates hypothermia, whereas blockade of D2 receptors elicits prolactin secretion and catalepsy.

Journal: The Journal of pharmacology and experimental therapeutics 19951101

Title: Alpha- and beta-adrenoceptors: from the gene to the clinic. 1. Molecular biology and adrenoceptor subclassification.

Journal: Journal of medicinal chemistry 19950901

Title: Pramipexole binding and activation of cloned and expressed dopamine D2, D3 and D4 receptors.

Journal: European journal of pharmacology 19950623

Title: Behavioral and biochemical changes after bilateral electrolytic lesions of the red nucleus of rat.

Journal: Pharmacology, biochemistry, and behavior 19950501

Title: Differential effects of [3H]nemonapride and [3H]spiperone binding on human dopamine D4 receptors.

Journal: Neuroscience letters 19950217

Title: Is clozapine selective for the dopamine D4 receptor?

Journal: Life sciences 19950101

Title: Some behavioral effects of CNQX AND NBQX, AMPA receptor antagonists.

Journal: Polish journal of pharmacology 19950101

Title: Elimination of cocaine-induced hyperactivity and dopamine-mediated neurophysiological effects in dopamine D1 receptor mutant mice.

Journal: Cell 19941216

Title: Molecular cloning, functional expression, and mRNA tissue distribution of the human 5-hydroxytryptamine2B receptor.

Journal: Molecular pharmacology 19940801

Title: Binding of typical and atypical antipsychotic agents to 5-hydroxytryptamine-6 and 5-hydroxytryptamine-7 receptors.

Journal: The Journal of pharmacology and experimental therapeutics 19940301

Title: Characterization of the human dopamine D3 receptor expressed in transfected cell lines.

Journal: European journal of pharmacology 19940101

Title: Some central effects of kynurenic acid, 7-chlorokynurenic acid and 5,7- dichloro-kynurenic acid, glycine site antagonists.

Journal: Polish journal of pharmacology 19940101

Title: Pharmacological and functional characterization of D2, D3 and D4 dopamine receptors in fibroblast and dopaminergic cell lines.

Journal: The Journal of pharmacology and experimental therapeutics 19940101

Title: Dopamine D2 and serotonin S2 receptors in susceptibility to methamphetamine psychosis detected by positron emission tomography.

Journal: Psychiatry research 19931201

Title: Cloning of a novel human serotonin receptor (5-HT7) positively linked to adenylate cyclase.

Journal: The Journal of biological chemistry 19931105

Title: Molecular cloning, characterization, and localization of a high-affinity serotonin receptor (5-HT7) activating cAMP formation.

Journal: Proceedings of the National Academy of Sciences of the United States of America 19930915

Title: Low density of dopamine D4 receptors in Parkinson's, schizophrenia, and control brain striata.

Journal: Synapse (New York, N.Y.) 19930801

Title: Molecular cloning of a mammalian serotonin receptor that activates adenylate cyclase.

Journal: Molecular pharmacology 19930801

Title: Strain differences in clonidine-induced aggressiveness in mice and its interaction with the dopamine system.

Journal: Pharmacology, biochemistry, and behavior 19930401

Title: The role of receptor binding in drug discovery.

Journal: Journal of natural products 19930401

Title: Pharmacological characteristics of the newly cloned rat 5-hydroxytryptamine2F receptor.

Journal: Molecular pharmacology 19930301

Title: Cloning of another human serotonin receptor (5-HT1F): a fifth 5-HT1 receptor subtype coupled to the inhibition of adenylate cyclase.

Journal: Proceedings of the National Academy of Sciences of the United States of America 19930115

Title: Pharmacological profile of AD-5423, a novel antipsychotic with both potent dopamine-D2 and serotonin-S2 antagonist properties.

Journal: The Journal of pharmacology and experimental therapeutics 19930101

Title: High-level stable expression of recombinant 5-HT1A 5-hydroxytryptamine receptors in Chinese hamster ovary cells.

Journal: The Biochemical journal 19920801

Title: Upregulation of postsynaptic dopamine receptors in the striatum does not influence haloperidol-induced catalepsy in mice.

Journal: Pharmacology, biochemistry, and behavior 19920801

Title: Human serotonin 1D receptor is encoded by a subfamily of two distinct genes: 5-HT1D alpha and 5-HT1D beta.

Journal: Proceedings of the National Academy of Sciences of the United States of America 19920415

Title: Mouse 5HT1B serotonin receptor: cloning, functional expression, and localization in motor control centers.

Journal: Proceedings of the National Academy of Sciences of the United States of America 19920401

Title: Effect of mesulergine on prolactin secretion and dopamine D2 receptors-adaptive changes in diethylstilbestrol-induced hyperplasia of the rat anterior pituitary.

Journal: Endocrine regulations 19920301

Title: Fluorescent probes for dopamine receptors: synthesis and characterization of fluorescein and 7-nitrobenz-2-oxa-1,3-diazol-4-yl conjugates of D-1 and D-2 receptor ligands.

Journal: Journal of medicinal chemistry 19911101

Title: Primary structure and functional characterization of a human 5-HT1D-type serotonin receptor.

Journal: Molecular pharmacology 19910801

Title: Reduced D2 dopamine and muscarinic cholinergic receptor densities in caudate specimens from fluctuating parkinsonian patients.

Journal: Annals of neurology 19910801

Title: Cloning of the gene for a human dopamine D5 receptor with higher affinity for dopamine than D1.

Journal: Nature 19910418

Title: Cloning of the gene for a human dopamine D4 receptor with high affinity for the antipsychotic clozapine.

Journal: Nature 19910418

Title: Simultaneous quantitation of loxapine, amoxapine and their 7- and 8-hydroxy metabolites in plasma by high-performance liquid chromatography.

Journal: Journal of chromatography 19910308

Title: Behavioural and electoencephalographic interactions between haloperidol and PCP/sigma ligands in the rat.

Journal: Psychopharmacology 19910101

Title: Antidopaminergic effects of the stereoisomers of N-[(1-alkyl-2- pyrrolidinyl)methyl]-5-sulfamoylbenzamides and -2,3-dihydrobenzofuran-7-carboxamides.

Journal: Journal of medicinal chemistry 19910101

Title: On the selection of mice for haloperidol response and non-response.

Journal: Psychopharmacology 19910101

Title: Effects of subchronic amphetamine or amfonelic acid on rat brain dopaminergic and serotonergic function.

Journal: Journal of neural transmission. General section 19910101

Title: [3H]-DOB(4-bromo-2,5-dimethoxyphenylisopropylamine) and [3H] ketanserin label two affinity states of the cloned human 5-hydroxytryptamine2 receptor.

Journal: Molecular pharmacology 19901101

Title: Modulation of dopamine receptors by cations in 7315a, MtTW15 and estradiol-induced pituitary tumors.

Journal: Biochemical pharmacology 19900915

Title: Molecular cloning and characterization of a novel dopamine receptor (D3) as a target for neuroleptics.

Journal: Nature 19900913

Title: Evidence that central 5-HT1A-receptors play a role in the von Bezold-Jarisch reflex in the rat.

Journal: British journal of pharmacology 19900801

Title: Pharmacological actions of SM-9018, a new neuroleptic drug with both potent 5-hydroxytryptamine2 and dopamine2 antagonistic actions.

Journal: Japanese journal of pharmacology 19900701

Title: Dopamine receptor agonists: selectivity and dopamine D1 receptor efficacy.

Journal: European journal of pharmacology 19900612

Title: Dihydrexidine, a novel selective high potency full dopamine D-1 receptor agonist.

Journal: European journal of pharmacology 19890704

Title: Dopamine blockade and clinical response: evidence for two biological subgroups of schizophrenia.

Journal: The American journal of psychiatry 19890701

Title: Cloning and expression of a rat D2 dopamine receptor cDNA.

Journal: Nature 19881201

Title: In vitro estrogen-like effects of 7,12-dimethylbenz(a)anthracene on anterior pituitary dopamine receptors of rats.

Journal: Cancer research 19881115

Title: Receptor mechanisms of nicotine-induced locomotor hyperactivity in chronic nicotine-treated rats.

Journal: European journal of pharmacology 19880802

Title: Alpha 2-adrenoceptors as a target for formamidine pesticides: in vitro and in vivo studies in mice.

Journal: Toxicology and applied pharmacology 19880401

Title: High doses of morphine do not change characteristics of the cerebral catecholamine receptors in the rat.

Journal: Polish journal of pharmacology and pharmacy 19880101

Title: Antagonism by neuroleptics of serotonin 5-HT1A and 5-HT2 receptors of normal human brain in vitro.

Journal: European journal of pharmacology 19871110

Title: MPTP-induced parkinsonism in the monkey: neurochemical pathology, complications of treatment and pathophysiological mechanisms.

Journal: The Canadian journal of neurological sciences. Le journal canadien des sciences neurologiques 19870801

Title: Experimental study on resting tremor and L-dopa-induced dyskinesia.

Journal: European neurology 19870101

Title: The selective dopamine D2 receptor antagonist raclopride discriminates between dopamine-mediated motor functions.

Journal: Psychopharmacology 19860101

Title: Simultaneous catalepsy and apomorphine-induced stereotypic behavior in mice.

Journal: Life sciences 19851104

Title: Prenatal exposure of rats to antidepressants enhances agonist affinity of brain dopamine receptors and dopamine-mediated behaviour.

Journal: European journal of pharmacology 19851022

Title: Repeated treatment with imipramine or amitriptyline increases the locomotor response of rats to (+)-amphetamine given into the nucleus accumbens.

Journal: The Journal of pharmacy and pharmacology 19850501

Title: The role of the GABA mechanisms of the globus pallidus in mediating catalepsy, stereotypy and locomotor activity.

Journal: Pharmacology, biochemistry, and behavior 19841201

Title: [Effect of repeated haloperidol and apomorphine administration on the development of tolerance for catalepsy and dopamine receptor hypersensitivity in mice].

Journal: Biulleten' eksperimental'noi biologii i meditsiny 19841001

Title: Sigma opiates and certain antipsychotic drugs mutually inhibit (+)-[3H] SKF 10,047 and [3H]haloperidol binding in guinea pig brain membranes.

Journal: Proceedings of the National Academy of Sciences of the United States of America 19840901

Title: Dopamine receptors in rat pituitary and estradiol-induced pituitary tumor: effect of chronic treatment with bromocriptine.

Journal: Biochemical and biophysical research communications 19840830

Title: Remoxipride, a new potential antipsychotic compound with selective antidopaminergic actions in the rat brain.

Journal: European journal of pharmacology 19840720

Title: Interactions of neurotensin with brain dopamine systems: biochemical and behavioral studies.

Journal: The Journal of pharmacology and experimental therapeutics 19830501

Title: CGS 7525A, a new, centrally active alpha 2 adrenoceptor antagonist.

Journal: Life sciences 19830124

Title: Assessment of the antidepressant activity of dothiepin and its metabolites by preclinical tests.

Journal: Journal of affective disorders 19820901

Title: Possible involvement of serotonergic neurons in the reduction of locomotor hyperactivity caused by amphetamine in neonatal rats depleted of brain dopamine.

Journal: Brain research 19820722

Title: Cataleptogenic doses of morphine suppress 3H-spiroperidol binding to striatal membranes.

Journal: Naunyn-Schmiedeberg's archives of pharmacology 19820501

Title: Septo-hippocampal system: target for substituted benzamides.

Journal: European journal of pharmacology 19820423

Title: Central neurotropic activity of homovanillic acid.

Journal: Acta physiologica Polonica 19810101

Title: Chronic treatment with antidepressant drugs: potentiation of apomorphine-induced aggressive behaviour in rats.

Journal: Neuroscience letters 19790801

Title: On the anticataleptic action of cyproheptadine.

Journal: Pharmacology, biochemistry, and behavior 19760801

Title: Influence of WA-335, a factor which blocks serotonin receptors, on neuroleptic-induced catalepsy.

Journal: Archivum immunologiae et therapiae experimentalis 19760101

Title: Antagonistic effect of cyproheptadine on neuroleptic-induced catalepsy.

Journal: Pharmacology, biochemistry, and behavior 19750101

Title: The effect of 5-hydroxytrytamine synthesis inhibitors on neuroleptic-induced catalepsy in rats.

Journal: Archivum immunologiae et therapiae experimentalis 19750101

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Tags:749-02-0 Molecular Formula|749-02-0 MDL|749-02-0 SMILES|749-02-0 Spiperone