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Title: Isoxazole analogues bind the system xc- transporter: structure-activity relationship and pharmacophore model.
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Title: The glutamate receptor GluR5 agonist (S)-2-amino-3-(3-hydroxy-7,8-dihydro-6H-cyclohepta[d]isoxazol-4-yl)propionic acid and the 8-methyl analogue: synthesis, molecular pharmacology, and biostructural characterization.
Journal: Journal of medicinal chemistry 20090813
Title: Hierarchical recruitment by AMPA but not staurosporine of pro-apoptotic mitochondrial signaling in cultured cortical neurons: evidence for caspase-dependent/independent cross-talk.
Journal: Journal of neurochemistry 20071201
Title: Synthesis and pharmacology of willardiine derivatives acting as antagonists of kainate receptors.
Journal: Journal of medicinal chemistry 20051201
Title: Convergent synthesis and pharmacology of substituted tetrazolyl-2-amino-3-(3-hydroxy-5-methyl-4-isoxazolyl)propionic acid analogues.
Journal: Journal of medicinal chemistry 20050505
Title: Isoxazole ionotropic glutamate neurotransmitters.
Journal: Current medicinal chemistry 20050101
Title: Synaptic activity augments muscarinic acetylcholine receptor-stimulated inositol 1,4,5-trisphosphate production to facilitate Ca2+ release in hippocampal neurons.
Journal: The Journal of biological chemistry 20041119
Title: (S)-2-Amino-3-(3-hydroxy-7,8-dihydro-6H-cyclohepta[d]isoxazol-4-yl)propionic acid, a potent and selective agonist at the GluR5 subtype of ionotropic glutamate receptors. Synthesis, modeling, and molecular pharmacology.
Journal: Journal of medicinal chemistry 20030410
Title: Effects of acute ethanol on the Ca2+ response to AMPA in cultured rat cortical GABAergic nonpyramidal neurons.
Journal: Alcohol and alcoholism (Oxford, Oxfordshire) 20030101
Title: A glutamate receptor subtype antagonist inhibits seizures in rat hippocampal slices.
Journal: Neuroreport 20020304
Title: Regional mapping of low-affinity kainate receptors in mouse brain using [(3)H](2S,4R)-4-methylglutamate autoradiography.
Journal: European journal of pharmacology 20011123
Title: Effect of FK960, a putative cognitive enhancer, on synaptic transmission in CA1 neurons of rat hippocampus.
Journal: The Journal of pharmacology and experimental therapeutics 20010501
Title: Quinazolone-alkyl-carboxylic acid derivatives inhibit transmembrane Ca(2+) ion flux to (+)-(S)-alpha-amino-3-hydroxy-5-methylisoxazole-4-propionic acid.
Journal: Molecular pharmacology 20010401
Title: A new highly selective metabotropic excitatory amino acid agonist: 2-amino-4-(3-hydroxy-5-methylisoxazol-4-yl)butyric acid.
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