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87051-43-2,MFCD00069341
Catalog No.:AA008DMV

87051-43-2 | RITANSERIN

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5mg
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$52.00   $36.00
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10mg
≥95%
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25mg
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  • Technical Information
  • Properties
  • Literature
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  • Technical Information
  • Properties
  • Literature
Technical Information
Catalog Number:
AA008DMV
Chemical Name:
RITANSERIN
CAS Number:
87051-43-2
Molecular Formula:
C27H25F2N3OS
Molecular Weight:
477.5687
MDL Number:
MFCD00069341
SMILES:
Fc1ccc(cc1)C(=C1CCN(CC1)CCc1c(C)nc2n(c1=O)ccs2)c1ccc(cc1)F
NSC Number:
758470
Properties
Computed Properties
 
Complexity:
877  
Covalently-Bonded Unit Count:
1  
Heavy Atom Count:
34  
Hydrogen Bond Acceptor Count:
6  
Rotatable Bond Count:
5  
XLogP3:
5.2  

Literature

Title: A high-throughput screen for teratogens using human pluripotent stem cells.

Journal: Toxicological sciences : an official journal of the Society of Toxicology 20140101

Title: Vasoconstrictor 5-HT receptors in the smooth muscle of the rat middle cerebral artery.

Journal: European journal of pharmacology 20120815

Title: Modulation of antipsychotic-induced extrapyramidal side effects by medications for mood disorders.

Journal: Progress in neuro-psychopharmacology & biological psychiatry 20120807

Title: Effects of diphenyl diselenide on depressive-like behavior in ovariectomized mice submitted to subchronic stress: involvement of the serotonergic system.

Journal: Psychopharmacology 20120801

Title: Long-term depression of nociceptive synapses by non-nociceptive afferent activity: role of endocannabinoids, Ca²+, and calcineurin.

Journal: Brain research 20120615

Title: p-Chloro-diphenyl diselenide, an organoselenium compound, with antidepressant-like and memory enhancer actions in aging male rats.

Journal: Biogerontology 20120601

Title: Opposing effects of 5,7-DHT lesions to the core and shell of the nucleus accumbens on the processing of irrelevant stimuli.

Journal: The international journal of neuropsychopharmacology 20120501

Title: Influence of Withania somnifera on obsessive compulsive disorder in mice.

Journal: Asian Pacific journal of tropical medicine 20120501

Title: Italian guidelines for primary headaches: 2012 revised version.

Journal: The journal of headache and pain 20120501

Title: Mutual independence of 5-HT(2) and α1 noradrenergic receptors in mediating deficits in sensorimotor gating.

Journal: Psychopharmacology 20120401

Title: Vasoconstrictor and vasodilator responses to tryptamine of rat-isolated perfused mesentery: comparison with tyramine and β-phenylethylamine.

Journal: British journal of pharmacology 20120401

Title: Serotonergic and dopaminergic distinctions in the behavioral pharmacology of (±)-1-(2,5-dimethoxy-4-iodophenyl)-2-aminopropane (DOI) and lysergic acid diethylamide (LSD).

Journal: Pharmacology, biochemistry, and behavior 20120301

Title: Arousal effects of orexin A on acute alcohol intoxication-induced coma in rats.

Journal: Neuropharmacology 20120201

Title: 5-HT2A/C receptors mediate the antipsychotic-like effects of alstonine.

Journal: Progress in neuro-psychopharmacology & biological psychiatry 20120110

Title: On the mechanism of anti-hyperthermic effects of LY379268 and LY487379, group II mGlu receptors activators, in the stress-induced hyperthermia in singly housed mice.

Journal: Neuropharmacology 20120101

Title: The effects of acute tryptophan depletion on costly information sampling: impulsivity or aversive processing?

Journal: Psychopharmacology 20120101

Title: Treatment-resistant Schizophrenia: Evidence-based Strategies.

Journal: Mens sana monographs 20120101

Title: A hidden Markov model to assess drug-induced sleep fragmentation in the telemetered rat.

Journal: Journal of pharmacokinetics and pharmacodynamics 20111201

Title: Postnatal serotonin type 2 receptor blockade prevents the emergence of anxiety behavior, dysregulated stress-induced immediate early gene responses, and specific transcriptional changes that arise following early life stress.

Journal: Biological psychiatry 20111201

Title: Myenteric neural network activated by motilin in the stomach of Suncus murinus (house musk shrew).

Journal: Neurogastroenterology and motility : the official journal of the European Gastrointestinal Motility Society 20111201

Title: Decoding the signaling of a GPCR heteromeric complex reveals a unifying mechanism of action of antipsychotic drugs.

Journal: Cell 20111123

Title: Antinociceptive and antihyperalgesic effects of tapentadol in animal models of inflammatory pain.

Journal: The Journal of pharmacology and experimental therapeutics 20111101

Title: Role of growth hormone-releasing hormone in sleep and growth impairments induced by upper airway obstruction in rats.

Journal: The European respiratory journal 20111001

Title: Diltiazem potentiates pentobarbital-induced hypnosis via 5-HT1A and 5-HT2A/2C receptors: role for dorsal raphe nucleus.

Journal: Pharmacology, biochemistry, and behavior 20111001

Title: Clozapine increases reward evaluation but not overall ingestive behaviour in rats licking for sucrose.

Journal: Psychopharmacology 20110801

Title: Identification of antidepressant-like ingredients in ginseng root (Panax ginseng C.A. Meyer) using a menopausal depressive-like state in female mice: participation of 5-HT2A receptors.

Journal: Psychopharmacology 20110801

Title: Serotonin control of sleep-wake behavior.

Journal: Sleep medicine reviews 20110801

Title: Pharmacological stimulation of locus coeruleus reveals a new antipsychotic-responsive pathway for deficient sensorimotor gating.

Journal: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20110701

Title: Serotonergic mechanism underlying tranylcypromine enhancement of nicotine self-administration.

Journal: Synapse (New York, N.Y.) 20110601

Title: Antidepressant-like effect of m-trifluoromethyl-diphenyl diselenide in the mouse forced swimming test involves opioid and serotonergic systems.

Journal: European journal of pharmacology 20110511

Title: Interactive effects of mGlu5 and 5-HT2A receptors on locomotor activity in mice.

Journal: Psychopharmacology 20110501

Title: Residual effects of esmirtazapine on actual driving performance: overall findings and an exploratory analysis into the role of CYP2D6 phenotype.

Journal: Psychopharmacology 20110501

Title: Efficacy of antidepressants for dysthymia: a meta-analysis of placebo-controlled randomized trials.

Journal: The Journal of clinical psychiatry 20110401

Title: A pronociceptive role for the 5-HT2 receptor on spinal nociceptive transmission: an in vivo electrophysiological study in the rat.

Journal: Brain research 20110325

Title: Effect of alpha-melanocyte stimulating hormone on locomotor recovery following spinal cord injury in mice: Role of serotonergic system.

Journal: Neuropeptides 20110201

Title: Fluoxetine, trazodone and ritanserin are more effective than placebo when used as add-on therapies for negative symptoms of schizophrenia.

Journal: Evidence-based mental health 20110201

Title: Early postnatal protein-calorie malnutrition and cognition: a review of human and animal studies.

Journal: International journal of environmental research and public health 20110201

Title: [The relationships among raphe magnus nucleus, locus coeruleus and dorsal motor nucleus of vagus in the descending regulation of gastric motility].

Journal: Zhongguo ying yong sheng li xue za zhi = Zhongguo yingyong shenglixue zazhi = Chinese journal of applied physiology 20110201

Title: Switching-on of serotonergic calcium signaling in activated hepatic stellate cells.

Journal: World journal of gastroenterology 20110114

Title: Serotonergic modulation of extrapyramidal motor disorders in mice and rats: role of striatal 5-HT3 and 5-HT6 receptors.

Journal: Neuropharmacology 20110101

Title: Evaluation of the Anxiolytic Activity of NR-ANX-C (a Polyherbal Formulation) in Ethanol Withdrawal-Induced Anxiety Behavior in Rats.

Journal: Evidence-based complementary and alternative medicine : eCAM 20110101

Title: Bacopa monniera Attenuates Scopolamine-Induced Impairment of Spatial Memory in Mice.

Journal: Evidence-based complementary and alternative medicine : eCAM 20110101

Title: Standard operation procedures for conducting the on-the-road driving test, and measurement of the standard deviation of lateral position (SDLP).

Journal: International journal of general medicine 20110101

Title: Evidence of a pharmacodynamic EEG profile in rats following clonidine administration using a nonlinear analysis.

Journal: Nonlinear biomedical physics 20110101

Title: Pharmacological treatment of insomnia in alcohol recovery: a systematic review.

Journal: Alcohol and alcoholism (Oxford, Oxfordshire) 20110101

Title: The 5-HT(2A) Receptor Antagonist M100907 Produces Antiparkinsonian Effects and Decreases Striatal Glutamate.

Journal: Frontiers in systems neuroscience 20110101

Title: Narcolepsy: a review.

Journal: Neuropsychiatric disease and treatment 20110101

Title: The involvement of the serotonergic transmission system in neonatal and adult rat ileum contractility varies with age.

Journal: Pharmacology 20110101

Title: Anxiolytic-like activity of MGS0039, a selective group II mGlu receptor antagonist, is serotonin- and GABA-dependent.

Journal: Pharmacological reports : PR 20110101

Title: Adolescent oxytocin exposure causes persistent reductions in anxiety and alcohol consumption and enhances sociability in rats.

Journal: PloS one 20110101

Title: Differential effects of HIF-1 inhibition by YC-1 on the overall outcome and blood-brain barrier damage in a rat model of ischemic stroke.

Journal: PloS one 20110101

Title: On the mechanism of the antidepressant-like action of group II mGlu receptor antagonist, MGS0039.

Journal: Psychopharmacology 20101201

Title: Metabotropic glutamate receptor 4 novel agonist LSP1-2111 with anxiolytic, but not antidepressant-like activity, mediated by serotonergic and GABAergic systems.

Journal: Neuropharmacology 20101201

Title: Neuro-psychopharmacogenetics and Neurological Antecedents of Posttraumatic Stress Disorder: Unlocking the Mysteries of Resilience and Vulnerability.

Journal: Current neuropharmacology 20101201

Title: Dopamine release induced by atypical antipsychotics in prefrontal cortex requires 5-HT(1A) receptors but not 5-HT(2A) receptors.

Journal: The international journal of neuropsychopharmacology 20101101

Title: Antinociceptive effect of butyl (2-phenylethynyl) selenide on formalin test in mice: Evidences for the involvement of serotonergic and adenosinergic systems.

Journal: European journal of pharmacology 20101010

Title: Mirtazapine abolishes hyperthermia in an animal model of serotonin syndrome.

Journal: Neuroscience letters 20101004

Title: Antidepressant-like pharmacological profile of 3-(4-fluorophenylselenyl)-2,5-diphenylselenophene: Involvement of serotonergic system.

Journal: Neuropharmacology 20100901

Title: Differential contribution of opioid and noradrenergic mechanisms of tapentadol in rat models of nociceptive and neuropathic pain.

Journal: European journal of pain (London, England) 20100901

Title: The antidepressant-like action of metabotropic glutamate 7 receptor agonist N,N'-bis(diphenylmethyl)-1,2-ethanediamine (AMN082) is serotonin-dependent.

Journal: The Journal of pharmacology and experimental therapeutics 20100901

Title: Cardiovascular effects of a novel synthetic analogue of naturally occurring piperamides.

Journal: Journal of cardiovascular pharmacology 20100901

Title: Efficacy of antidepressants in treating the negative symptoms of chronic schizophrenia: meta-analysis.

Journal: The British journal of psychiatry : the journal of mental science 20100901

Title: Dopamine receptor alterations in female rats with diet-induced decreased brain docosahexaenoic acid (DHA): interactions with reproductive status.

Journal: Nutritional neuroscience 20100801

Title: Obsessive-compulsive disorder and its related disorders: a reappraisal of obsessive-compulsive spectrum concepts.

Journal: Dialogues in clinical neuroscience 20100601

Title: Escitalopram prolonged fear induced by simulated public speaking and released hypothalamic-pituitary-adrenal axis activation.

Journal: Journal of psychopharmacology (Oxford, England) 20100501

Title: Serotonin-induced region-specific responses of the arcuate and ventromedial hypothalamic nuclei.

Journal: The International journal of neuroscience 20100501

Title: Serotonin 5-HT(2A) receptor antagonists in the treatment of insomnia: present status and future prospects.

Journal: Drugs of today (Barcelona, Spain : 1998) 20100301

Title: A cell protection screen reveals potent inhibitors of multiple stages of the hepatitis C virus life cycle.

Journal: Proceedings of the National Academy of Sciences of the United States of America 20100223

Title: Unilateral lesion of the nigrostriatal pathway decreases the response of interneurons in medial prefrontal cortex to 5-HT 2A/2C receptor stimulation in the rat.

Journal: Brain research 20100202

Title: [Pharmacological hypotheses and therapeutic strategies for gait disorders in Parkinson's disease].

Journal: Revue neurologique 20100201

Title: Identification of molecular targets associated with ethanol toxicity and implications in drug development.

Journal: Current pharmaceutical design 20100101

Title: 5-HT2A receptor antagonists improve motor impairments in the MPTP mouse model of Parkinson's disease.

Journal: Neuropharmacology 20100101

Title: Medications acting on the serotonergic system for the treatment of alcohol dependent patients.

Journal: Current pharmaceutical design 20100101

Title: Serotonergic modulation of absence-like seizures in groggy rats: a novel rat model of absence epilepsy.

Journal: Journal of pharmacological sciences 20100101

Title: Hypertension in Cushing's syndrome: from pathogenesis to treatment.

Journal: Neuroendocrinology 20100101

Title: [Selective involvement of cerebellar neurotransmitter systems in mechanisms of various types of defensive behavior].

Journal: Zhurnal vysshei nervnoi deiatelnosti imeni I P Pavlova 20100101

Title: Effect of ritanserin and leuprolide alone and combined on marble-burying behavior of mice.

Journal: Acta poloniae pharmaceutica 20100101

Title: Tricyclic antidepressants and headaches: systematic review and meta-analysis.

Journal: BMJ (Clinical research ed.) 20100101

Title: Classification of drugs based on properties of sodium channel inhibition: a comparative automated patch-clamp study.

Journal: PloS one 20100101

Title: Formalin pain increases the concentration of serotonin and its 5-hydroxyindoleacetic acid metabolite in the CA1 region of hippocampus.

Journal: Daru : journal of Faculty of Pharmacy, Tehran University of Medical Sciences 20100101

Title: Buspirone improves haloperidol-induced Parkinson disease in mice through 5-HT(1A) recaptors.

Journal: Daru : journal of Faculty of Pharmacy, Tehran University of Medical Sciences 20100101

Title: Involvement of the serotonergic system in the anxiolytic-like effect caused by m-trifluoromethyl-diphenyl diselenide in mice.

Journal: Behavioural brain research 20091228

Title: [Role of serotonin receptors in vascular tone in the pithed rat].

Journal: Archivos de cardiologia de Mexico 20091201

Title: Asenapine effects in animal models of psychosis and cognitive function.

Journal: Psychopharmacology 20091101

Title: A new homogeneous high-throughput screening assay for profiling compound activity on the human ether-a-go-go-related gene channel.

Journal: Analytical biochemistry 20091101

Title: Discriminative stimulus effects of 1-(2,5-dimethoxy-4-methylphenyl)-2-aminopropane (DOM), ketanserin, and (R)-(+)-{alpha}-(2,3-dimethoxyphenyl)-1-[2-(4-fluorophenyl)ethyl]-4-pipidinemethanol (MDL100907) in rats.

Journal: The Journal of pharmacology and experimental therapeutics 20091101

Title: Potentiation of excitatory serotonergic responses by MK-801 in the medial prefrontal cortex.

Journal: Naunyn-Schmiedeberg's archives of pharmacology 20091101

Title: Further pharmacological characterization of 5-HT(2C) receptor agonist-induced inhibition of 5-HT neuronal activity in the dorsal raphe nucleus in vivo.

Journal: British journal of pharmacology 20091101

Title: Characterization of the contractile 5-hydroxytryptamine receptor in the autoperfused kidney of L-NAME hypertensive rats.

Journal: European journal of pharmacology 20091012

Title: Physical binding pocket induction for affinity prediction.

Journal: Journal of medicinal chemistry 20091008

Title: The bovine mammary gland expresses multiple functional isoforms of serotonin receptors.

Journal: The Journal of endocrinology 20091001

Title: Genetic mapping of targets mediating differential chemical phenotypes in Plasmodium falciparum.

Journal: Nature chemical biology 20091001

Title: In vivo effects of activation and blockade of 5-HT(2A/2C) receptors in the firing activity of pyramidal neurons of medial prefrontal cortex in a rodent model of Parkinson's disease.

Journal: Experimental neurology 20090901

Title: The group III mGlu receptor agonist ACPT-I exerts anxiolytic-like but not antidepressant-like effects, mediated by the serotonergic and GABA-ergic systems.

Journal: Neuropharmacology 20090901

Title: Inhibitory effect of serotonin antagonists on JC virus propagation in a carrier culture of human neuroblastoma cells.

Journal: Microbiology and immunology 20090901

Title: Activity of sap from Croton lechleri on rat vascular and gastric smooth muscles.

Journal: Phytomedicine : international journal of phytotherapy and phytopharmacology 20090801

Title: Individual differences in the sensitivity to serotonergic drugs: a pharmacobehavioural approach using rats selected on the basis of their response to novelty.

Journal: Psychopharmacology 20090801

Title: Sedative and hypothermic effects of gamma-hydroxybutyrate (GHB) in rats alone and in combination with other drugs: assessment using biotelemetry.

Journal: Drug and alcohol dependence 20090801

Title: Depression-like behavior in the forced swimming test in PACAP-deficient mice: amelioration by the atypical antipsychotic risperidone.

Journal: Journal of neurochemistry 20090701

Title: Decrease in the kainate-induced wet dog shake behavior in genetically epilepsy-prone rats: possible involvement of an impaired synaptic transmission to the 5-HT(2A) receptor.

Journal: Journal of pharmacological sciences 20090701

Title: 5-Hydroxytryptamine Receptor Subtypes and their Modulators with Therapeutic Potentials.

Journal: Journal of clinical medicine research 20090601

Title: Guinea pig hippocampal 5-HT(1E) receptors: a tool for selective drug development.

Journal: Journal of neurochemistry 20090401

Title: Evidence for the involvement of the monoaminergic system in the antidepressant-like effect of magnesium.

Journal: Progress in neuro-psychopharmacology & biological psychiatry 20090317

Title: The involvement of serotonergic system in the antidepressant effect of zinc in the forced swim test.

Journal: Progress in neuro-psychopharmacology & biological psychiatry 20090317

Title: Discriminative stimulus effects of 1-(2,5-dimethoxy-4-methylphenyl)-2-aminopropane in rhesus monkeys: antagonism and apparent pA2 analyses.

Journal: The Journal of pharmacology and experimental therapeutics 20090301

Title: Evidence that oxytocin exerts anxiolytic effects via oxytocin receptor expressed in serotonergic neurons in mice.

Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience 20090218

Title: Cell surface delivery and structural re-organization by pharmacological chaperones of an oligomerization-defective alpha(1b)-adrenoceptor mutant demonstrates membrane targeting of GPCR oligomers.

Journal: The Biochemical journal 20090101

Title: Panic disorder: is the PAG involved?

Journal: Neural plasticity 20090101

Title: Nociception-induced spatial and temporal plasticity of synaptic connection and function in the hippocampal formation of rats: a multi-electrode array recording.

Journal: Molecular pain 20090101

Title: Synthesis, Structure Activity Relationship Studies and Pharmacological Evaluation of 2-Phenyl-3-(Substituted Phenyl)-3H-Quinazolin-4-ones as Serotonin 5-HT(2) Antagonists.

Journal: Indian journal of pharmaceutical sciences 20090101

Title: Effect of ritanserin, a 5HT2A/2C antagonist, on negative symptoms of schizophrenia: a double-blind randomized placebo-controlled study.

Journal: Progress in neuro-psychopharmacology & biological psychiatry 20081212

Title: Risperidone attenuates and reverses hyperthermia induced by 3,4-methylenedioxymethamphetamine (MDMA) in rats.

Journal: Neurotoxicology 20081101

Title: Upper airway loading induces growth retardation and change in local chondrocyte IGF-I expression is reversed by stimulation of GH release in juvenile rats.

Journal: Journal of applied physiology (Bethesda, Md. : 1985) 20081101

Title: Miscellaneous.

Journal: Indian journal of pharmacology 20081001

Title: Characterization of contractile 5-hydroxytryptamine receptor subtypes in the in situ autoperfused kidney in the anaesthetized rat.

Journal: European journal of pharmacology 20080911

Title: Fluoxetine potentiates GABAergic IPSCs in rat hippocampal neurons.

Journal: Neuroscience letters 20080905

Title: Hypersensitivity of 5-HT2 receptors in OCD patients. An increased prolactin response after a challenge with meta-chlorophenylpiperazine and pre-treatment with ritanserin and placebo.

Journal: Journal of psychiatric research 20080901

Title: A comparison of the discriminative stimulus properties of the atypical antipsychotic drug clozapine in DBA/2 and C57BL/6 inbred mice.

Journal: Behavioural pharmacology 20080901

Title: The structure of human serotonin 2c G-protein-coupled receptor bound to agonists and antagonists.

Journal: Journal of molecular graphics & modelling 20080801

Title: Diphenyl diselenide exerts anxiolytic-like effect in Wistar rats: putative roles of GABAA and 5HT receptors.

Journal: Progress in neuro-psychopharmacology & biological psychiatry 20080801

Title: Off-target effects of psychoactive drugs revealed by genome-wide assays in yeast.

Journal: PLoS genetics 20080801

Title: Prediction and identification of drug interactions with the human ATP-binding cassette transporter multidrug-resistance associated protein 2 (MRP2; ABCC2).

Journal: Journal of medicinal chemistry 20080612

Title: Behavioral and biochemical effects of amperozide and serotonin agents on nigrostriatal and mesolimbic dopamine systems.

Journal: The Chinese journal of physiology 20080430

Title: The role of lipophilicity in determining binding affinity and functional activity for 5-HT2A receptor ligands.

Journal: Bioorganic & medicinal chemistry 20080415

Title: 2-Alkyl-4-aryl-pyrimidine fused heterocycles as selective 5-HT2A antagonists.

Journal: Bioorganic & medicinal chemistry letters 20080315

Title: Effects of antipsychotics and reference monoaminergic ligands on marble burying behavior in mice.

Journal: Behavioural pharmacology 20080301

Title: 5-HT 1B receptor-mediated serotoninergic modulation of methylphenidate-induced locomotor activation in rats.

Journal: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20080201

Title: Discriminative stimulus effects of 1-(2,5-dimethoxy-4-methylphenyl)-2-aminopropane in rhesus monkeys.

Journal: The Journal of pharmacology and experimental therapeutics 20080201

Title: Serotonin, inhibition, and negative mood.

Journal: PLoS computational biology 20080201

Title: Identification of new functional inhibitors of acid sphingomyelinase using a structure-property-activity relation model.

Journal: Journal of medicinal chemistry 20080124

Title: Antidepressant drugs for narcolepsy.

Journal: The Cochrane database of systematic reviews 20080123

Title: The antidepressant effects of curcumin in the forced swimming test involve 5-HT1 and 5-HT2 receptors.

Journal: European journal of pharmacology 20080106

Title: Differential effects of dialysis and ultrafiltrate from individuals with CKD, with or without diabetes, on platelet phosphatidylserine externalization.

Journal: American journal of physiology. Renal physiology 20080101

Title: Update on neuropharmacological treatments for alcoholism: scientific basis and clinical findings.

Journal: Biochemical pharmacology 20080101

Title: 5-HT1B receptor subtype and aging in rat resistance vessels.

Journal: Pharmacology 20080101

Title: Comparison of the effects of deramciclane, ritanserin and buspirone on extracellular dopamine and its metabolites in striatum and nucleus accumbens of freely moving rats.

Journal: Basic & clinical pharmacology & toxicology 20080101

Title: Heterogeneity in 5-HT-induced contractile and proliferative responses in rat pulmonary arterial bed.

Journal: Journal of vascular research 20080101

Title: Neuropsychotoxicity of abused drugs: effects of serotonin receptor ligands on methamphetamine- and cocaine-induced behavioral sensitization in mice.

Journal: Journal of pharmacological sciences 20080101

Title: Antidepressant-like effect of chromium chloride in the mouse forced swim test: involvement of glutamatergic and serotonergic receptors.

Journal: Pharmacological reports : PR 20080101

Title: Tryptophan research in panic disorder.

Journal: International journal of tryptophan research : IJTR 20080101

Title: Role of endocannabinoids in regulating drug dependence.

Journal: Neuropsychiatric disease and treatment 20071201

Title: Endocannabinoid signaling in midbrain dopamine neurons: more than physiology?

Journal: Current neuropharmacology 20071201

Title: Anxiolytic-like action of MTEP expressed in the conflict drinking Vogel test in rats is serotonin dependent.

Journal: Neuropharmacology 20071101

Title: Possible involvement of endogenous 5-HT in aggravation of cerulein-induced acute pancreatitis in mice.

Journal: Journal of pharmacological sciences 20071101

Title: Potential cognitive enhancing and disease modification effects of SSRIs for Alzheimer's disease.

Journal: Neuropsychiatric disease and treatment 20071001

Title: Effect of 5-HT(2) receptor blockade on cadmium-induced acute toxicity.

Journal: Digestive diseases and sciences 20070901

Title: Ritanserin reverses repeated methamphetamine-induced behavioral and neurochemical sensitization in mice.

Journal: Synapse (New York, N.Y.) 20070901

Title: Exogenous serotonin regulates proliferation of interstitial cells of Cajal in mouse jejunum through 5-HT2B receptors.

Journal: Gastroenterology 20070901

Title: Ameliorating effect of emodin, a constitute of Polygonatum multiflorum, on cycloheximide-induced impairment of memory consolidation in rats.

Journal: Journal of ethnopharmacology 20070725

Title: Advanced glycation end products elicit externalization of phosphatidylserine in a subpopulation of platelets via 5-HT2A/2C receptors.

Journal: American journal of physiology. Cell physiology 20070701

Title: Risperidone attenuates MK-801-induced hyperlocomotion in mice via the blockade of serotonin 5-HT 2A/2C receptors.

Journal: European journal of pharmacology 20070614

Title: Serotonergic modulation of plasticity of the auditory cortex elicited by fear conditioning.

Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience 20070502

Title: The role of 5-HT(7) receptors in the control of seizures.

Journal: Brain research 20070413

Title: A61603-induced contractions of the porcine meningeal artery are mediated by alpha1- and alpha2-adrenoceptors.

Journal: Basic & clinical pharmacology & toxicology 20070401

Title: Anxiolytic-like effect of group III mGlu receptor antagonist is serotonin-dependent.

Journal: Neuropharmacology 20070201

Title: Neurotransmitter mechanisms mediating low-glucose signalling in cocultures and fresh tissue slices of rat carotid body.

Journal: The Journal of physiology 20070201

Title: Serotonin decreases generation of dopaminergic neurons from mesencephalic precursors via serotonin type 7 and type 4 receptors.

Journal: Developmental neurobiology 20070101

Title: In vivo evidence that 5-HT(2C) receptors inhibit 5-HT neuronal activity via a GABAergic mechanism.

Journal: British journal of pharmacology 20061201

Title: Clozapine and olanzapine, but not haloperidol, suppress serotonin efflux in the medial prefrontal cortex elicited by phencyclidine and ketamine.

Journal: The international journal of neuropsychopharmacology 20061001

Title: Differential attenuation of d-amphetamine-induced disruption of conditional discrimination performance by dopamine and serotonin antagonists.

Journal: Psychopharmacology 20061001

Title: Inverse agonist activity of sarpogrelate, a selective 5-HT2A-receptor antagonist, at the constitutively active human 5-HT2A receptor.

Journal: Journal of pharmacological sciences 20061001

Title: Involvement of 5-HT(2) serotonergic receptors of the nucleus raphe magnus and nucleus reticularis gigantocellularis/paragigantocellularis complex neural networks in the antinociceptive phenomenon that follows the post-ictal immobility syndrome.

Journal: Experimental neurology 20060901

Title: Increased hippocampal nitric oxide synthase activity and stress responsiveness after imipramine discontinuation: role of 5HT 2A/C-receptors.

Journal: Metabolic brain disease 20060901

Title: Effects of osemozotan, ritanserin and azasetron on cocaine-induced behavioral sensitization in mice.

Journal: Pharmacology, biochemistry, and behavior 20060901

Title: Obstructive sleep apnea - management update.

Journal: Neuropsychiatric disease and treatment 20060901

Title: Serotonergic mediation of constant light-potentiated nonphotic phase shifting of the circadian locomotor activity rhythm in Syrian hamsters.

Journal: American journal of physiology. Regulatory, integrative and comparative physiology 20060701

Title: Microsphere-based protease assays and screening application for lethal factor and factor Xa.

Journal: Cytometry. Part A : the journal of the International Society for Analytical Cytology 20060501

Title: Pharmacotherapy for alcohol dependence: anticraving medications for relapse prevention.

Journal: Yonsei medical journal 20060430

Title: Microinjection of ritanserin into the CA1 region of hippocampus improves scopolamine-induced amnesia in adult male rats.

Journal: Behavioural brain research 20060403

Title: Microinjection of ritanserin into the dorsal hippocampal CA1 and dentate gyrus decrease nociceptive behavior in adult male rat.

Journal: Behavioural brain research 20060403

Title: Mirtazapine in bupropion-induced dyskinesias: a case report.

Journal: Movement disorders : official journal of the Movement Disorder Society 20060401

Title: Potential vascular alpha1-adrenoceptor blocking properties of an array of 5-HT receptor ligands in the rat.

Journal: European journal of pharmacology 20060327

Title: Discriminative stimulus properties of the atypical antipsychotic drug clozapine in rats trained to discriminate 1.25 mg/kg clozapine vs. 5.0 mg/kg clozapine vs. vehicle.

Journal: Behavioural pharmacology 20060301

Title: The alkaloid alstonine: a review of its pharmacological properties.

Journal: Evidence-based complementary and alternative medicine : eCAM 20060301

Title: The activation of 5-HT receptors in prefrontal cortex enhances dopaminergic activity.

Journal: Journal of neurochemistry 20051201

Title: Fluvoxamine in the treatment of anxiety disorders.

Journal: Neuropsychiatric disease and treatment 20051201

Title: Adjunctive treatment with mianserin enhances effects of raclopride on cortical dopamine output and, in parallel, its antipsychotic-like effect.

Journal: Neuropsychiatric disease and treatment 20051201

Title: 5-HT1B receptors modulate the feeding inhibitory effects of enterostatin.

Journal: Brain research 20051116

Title: Behavioral effects of systemically administered MK-212 are prevented by ritanserin microinfusion into the basolateral amygdala of rats exposed to the elevated plus-maze.

Journal: Psychopharmacology 20051101

Title: Short-term constant light potentiation of large-magnitude circadian phase shifts induced by 8-OH-DPAT: effects on serotonin receptors and gene expression in the hamster suprachiasmatic nucleus.

Journal: The European journal of neuroscience 20051101

Title: Effect of 5-hydroxytryptamine on neurogenic vasoconstriction in the isolated, autoperfused hindquarters of the rat.

Journal: Clinical and experimental pharmacology & physiology 20051001

Title: Adjunctive treatment with mianserin enhances effects of raclopride on cortical dopamine output and, in parallel, its antipsychotic-like effect.

Journal: Neuropsychiatric disease and treatment 20050901

Title: Lack of involvement of dopamine and serotonin during the orphanin FQ/Nociceptin (OFQ/N)-induced prolactin secretory response.

Journal: Life sciences 20050812

Title: Diabetes-induced changes in the 5-hydroxytryptamine inhibitory receptors involved in the pressor effect elicited by sympathetic stimulation in the pithed rat.

Journal: British journal of pharmacology 20050701

Title: A role for midbrain raphe gamma aminobutyric acid neurons in 5-hydroxytryptamine feedback control.

Journal: Neuroreport 20050621

Title: Attenuation of benzodiazepine withdrawal anxiety in the rat by serotonin antagonists.

Journal: Behavioural brain research 20050620

Title: Serotonin receptor mechanisms mediate the discriminative stimulus properties of the atypical antipsychotic clozapine in C57BL/6 mice.

Journal: Psychopharmacology 20050601

Title: Effects of serotonin and serotonergic agonists and antagonists on the production of tumor necrosis factor alpha and interleukin-6.

Journal: Psychiatry research 20050430

Title: A pharmacophore hypothesis for P-glycoprotein substrate recognition using GRIND-based 3D-QSAR.

Journal: Journal of medicinal chemistry 20050421

Title: Evidence for a spinal serotonergic control of the peripheral inflammation in the rat.

Journal: Life sciences 20050401

Title: Circadian rhythm phenotype of 5-HT7 receptor knockout mice: 5-HT and 8-OH-DPAT-induced phase advances of SCN neuronal firing.

Journal: Journal of biological rhythms 20050401

Title: A serotonin receptor antagonist induces oocyte maturation in both frogs and mice: evidence that the same G protein-coupled receptor is responsible for maintaining meiosis arrest in both species.

Journal: Journal of cellular physiology 20050301

Title: Serotonergic modulation of carbachol-induced rhythmic activity in hippocampal slices.

Journal: Neuropharmacology 20050301

Title: Psychopharmacological profile of the alkaloid psychollatine as a 5HT2A/C serotonin modulator.

Journal: Journal of natural products 20050301

Title: Role of nitric oxide on motor behavior.

Journal: Cellular and molecular neurobiology 20050301

Title: The effect of intrahippocampal injections of ritanserin (5HT2A/2C antagonist) and granisetron (5HT3 antagonist) on learning as assessed in the spatial version of the water maze.

Journal: Behavioural brain research 20050227

Title: Discriminative stimulus properties of the atypical antipsychotic clozapine and the typical antipsychotic chlorpromazine in a three-choice drug discrimination procedure in rats.

Journal: Psychopharmacology 20050201

Title: m-CPP, a 5-HT2C receptor agonist that modifies the perfusion pressure of the hindquarter vascular bed of anesthetized rat.

Journal: Pharmacology 20050201

Title: In-vivo effects of the 1,2,4-piperazine derivatives MM5 and MC1, putative 5-HT agonists, on dopamine and serotonin release in rat prefrontal cortex.

Journal: The Journal of pharmacy and pharmacology 20050201

Title: Pharmacologic management of Cushing syndrome : new targets for therapy.

Journal: Treatments in endocrinology 20050101

Title: Phobic memory and somatic vulnerabilities in anorexia nervosa: a necessary unity?

Journal: Annals of general psychiatry 20050101

Title: Serotonin-induced phase advances of SCN neuronal firing in vitro: a possible role for 5-HT5A receptors?

Journal: Synapse (New York, N.Y.) 20041101

Title: Evidence for serotonin receptor subtypes involvement in agmatine antidepressant like-effect in the mouse forced swimming test.

Journal: Brain research 20041015

Title: 5-HT1A, 5-HT2, and GABAB receptors interact to modulate neurotransmitter release probability in layer 2/3 somatosensory rat cortex as evaluated by the paired pulse protocol.

Journal: Journal of neuroscience research 20041015

Title: Regulation of serotonin 5-HT2C receptors by chronic ligand exposure.

Journal: European journal of pharmacology 20040913

Title: Fluoxetine attenuates thermal hyperalgesia through 5-HT1/2 receptors in streptozotocin-induced diabetic mice.

Journal: European journal of pharmacology 20040830

Title: Increased wakefulness, motor activity and decreased theta activity after blockade of the 5-HT2B receptor by the subtype-selective antagonist SB-215505.

Journal: British journal of pharmacology 20040801

Title: Pharmacological characterisation of the agonist radioligand binding site of 5-HT(2A), 5-HT(2B) and 5-HT(2C) receptors.

Journal: Naunyn-Schmiedeberg's archives of pharmacology 20040801

Title: Differential inverse agonist efficacies of SB-258719, SB-258741 and SB-269970 at human recombinant serotonin 5-HT7 receptors.

Journal: European journal of pharmacology 20040714

Title: Cloning and pharmacological characterisation of the guinea pig 5-ht5A receptor.

Journal: European journal of pharmacology 20040628

Title: Serotonin-mediated phosphorylation of extracellular regulated kinases in platelets of patients with panic disorder versus controls.

Journal: Neurochemistry international 20040601

Title: Vasoconstrictor responses to 5-hydroxytryptamine in the autoperfused hindquarters of spontaneously hypertensive rats.

Journal: Pharmacology 20040601

Title: Restoration of baroreflex function by ketanserin is not blood pressure dependent in conscious freely moving rats.

Journal: Journal of hypertension 20040601

Title: Gateways to clinical trials.

Journal: Methods and findings in experimental and clinical pharmacology 20040601

Title: Pharmacological analysis of the mechanisms involved in the tachycardic and vasopressor responses to the antimigraine agent, isometheptene, in pithed rats.

Journal: Life sciences 20040514

Title: Opposing regulation of cell proliferation by retinoic acid and the serotonin2B receptor in the mouse frontonasal mass.

Journal: Anatomy and embryology 20040501

Title: 5-HT7 receptor subtype as a mediator of the serotonergic regulation of luteinizing hormone release in the zona incerta.

Journal: European journal of pharmacology 20040426

Title: Study of the behavioural responses related to the potential addictive properties of MDMA in mice.

Journal: Naunyn-Schmiedeberg's archives of pharmacology 20040301

Title: Anxiolytic properties of the antipsychotic alkaloid alstonine.

Journal: Pharmacology, biochemistry, and behavior 20040301

Title: Hormonal and temperature responses to flesinoxan in normal volunteers: an antagonist study.

Journal: European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology 20040301

Title: Antidepressant-like activity of S 20098 (agomelatine) in the forced swimming test in rodents: involvement of melatonin and serotonin receptors.

Journal: Journal of psychiatry & neuroscience : JPN 20040301

Title: Serotonin blockade protects against early microvascular constriction following atherosclerotic plaque rupture.

Journal: European journal of pharmacology 20040213

Title: 8-OH-DPAT as a 5-HT7 agonist: phase shifts of the circadian biological clock through increases in cAMP production.

Journal: Neuropharmacology 20040101

Title: Ritanserin counteracts both rat vacuous chewing movements and nigro-striatal tyrosine hydroxylase-immunostaining alterations induced by haloperidol.

Journal: European journal of pharmacology 20040101

Title: A new class of arylpiperazine derivatives: the library synthesis on SynPhase lanterns and biological evaluation on serotonin 5-HT(1A) and 5-HT(2A) receptors.

Journal: Journal of combinatorial chemistry 20040101

Title: Role of the serotonergic system in the neurobiology of alcoholism: implications for treatment.

Journal: CNS drugs 20040101

Title: Optimization of the pharmacophore model for 5-HT7R antagonism. Design and synthesis of new naphtholactam and naphthosultam derivatives.

Journal: Journal of medicinal chemistry 20031218

Title: The modulation by 5-HT of glutamatergic inputs from the raphe pallidus to rat hypoglossal motoneurones, in vitro.

Journal: The Journal of physiology 20031215

Title: Intrastriatal serotonin 5-HT2 receptors mediate dopamine D1-induced hyperlocomotion in 6-hydroxydopamine-lesioned rats.

Journal: Synapse (New York, N.Y.) 20031101

Title: Pharmacological characterization of a serotonin receptor (5-HT7) stimulating cAMP production in human corneal epithelial cells.

Journal: Investigative ophthalmology & visual science 20031101

Title: [Molecular pharmacology of sarpogrelate].

Journal: Nihon yakurigaku zasshi. Folia pharmacologica Japonica 20031101

Title: Group II metabotropic glutamate receptor antagonists LY341495 and LY366457 increase locomotor activity in mice.

Journal: Neuropharmacology 20031001

Title: Haloperidol, but not clozapine, produces dramatic catalepsy in delta9-THC-treated rats: possible clinical implications.

Journal: British journal of pharmacology 20031001

Title: Pharmacological profile of the 5-HT-induced inhibition of cardioaccelerator sympathetic outflow in pithed rats: correlation with 5-HT1 and putative 5-ht5A/5B receptors.

Journal: British journal of pharmacology 20031001

Title: Presynaptic modulation of rat arterial chemoreceptor function by 5-HT: role of K+ channel inhibition via protein kinase C.

Journal: The Journal of physiology 20030915

Title: Role of the serotonin 5-HT(2A) receptor in learning.

Journal: Learning & memory (Cold Spring Harbor, N.Y.) 20030901

Title: The role of serotonergic agents as treatments for alcoholism.

Journal: Drugs of today (Barcelona, Spain : 1998) 20030901

Title: Role of 5-HT1B receptors in the regulation of extracellular serotonin and dopamine in the dorsal striatum of mice.

Journal: European journal of pharmacology 20030822

Title: Higher-end serotonin receptors: 5-HT(5), 5-HT(6), and 5-HT(7).

Journal: Journal of medicinal chemistry 20030703

Title: Risperidone attenuates the discriminative-stimulus effects of d-amphetamine in humans.

Journal: The Journal of pharmacology and experimental therapeutics 20030701

Title: Evidence that central 5-HT2A and 5-HT2B/C receptors regulate 5-HT cell firing in the dorsal raphe nucleus of the anaesthetised rat.

Journal: British journal of pharmacology 20030701

Title: Ritanserin improves sleep quality in narcolepsy.

Journal: Pharmacopsychiatry 20030701

Title: A 5-HT1A agonist and a 5-HT2c antagonist reduce social interaction deficit induced by multiple ethanol withdrawals in rats.

Journal: Psychopharmacology 20030601

Title: Functional study of rat 5-HT2A receptors using antisense oligonucleotides.

Journal: Journal of neurochemistry 20030601

Title: Efficacy of low-dose mirtazapine in neuroleptic-induced akathisia: a double-blind randomized placebo-controlled pilot study.

Journal: Journal of clinical psychopharmacology 20030601

Title: Insurmountable antagonism of AT-1015, a 5-HT2 antagonist, on serotonin-induced endothelium-dependent relaxation in porcine coronary artery.

Journal: The Journal of pharmacy and pharmacology 20030601

Title: 5-HT2 and 3 receptor antagonists suppress the response of rat type I slowly adapting mechanoreceptor: an in vitro study.

Journal: Brain research 20030418

Title: Ketanserin stabilizes blood pressure in conscious spontaneously hypertensive rats.

Journal: Clinical and experimental pharmacology & physiology 20030301

Title: Pharmacological characterization of an adenylyl cyclase-coupled 5-HT receptor in aplysia: comparison with mammalian 5-HT receptors.

Journal: Journal of neurophysiology 20030301

Title: Localization of serotonin and its possible role in early embryos of Tritonia diomedea(Mollusca: Nudibranchia).

Journal: Cell and tissue research 20030201

Title: Further evidence that the discriminative stimulus properties of indorenate are mediated by 5-HT 1A/1B/2C receptors.

Journal: Pharmacology, biochemistry, and behavior 20030101

Title: Evidence that the anorexia induced by lipopolysaccharide is mediated by the 5-HT2C receptor.

Journal: Pharmacology, biochemistry, and behavior 20030101

Title: Benefits and risks of pharmacotherapy for dysthymia: a systematic appraisal of the evidence.

Journal: Drug safety 20030101

Title: Characterization of the 5-hydroxytryptamine receptors mediating contraction in the pig isolated intravesical ureter.

Journal: British journal of pharmacology 20030101

Title: Excitation by dopamine of rat subthalamic nucleus neurones in vitro-a direct action with unconventional pharmacology.

Journal: Neuroscience 20030101

Title: Dopamine and serotonin receptors mediating contractions of the snail, Helix pomatia, salivary duct.

Journal: Neuroscience 20030101

Title: Anxiolytic effect of ting-chih-wan in mouse behavior models of anxiety.

Journal: The American journal of Chinese medicine 20030101

Title: Ritanserin as an adjunct to lithium and haloperidol for the treatment of medication-naive patients with acute mania: a double blind and placebo controlled trial.

Journal: BMC psychiatry 20030101

Title: Mirtazapine in L-dopa-induced dyskinesias.

Journal: Clinical neuropharmacology 20030101

Title: Combined intrastriatal dopamine D1 and serotonin 5-HT2 receptor stimulation reveals a mechanism for hyperlocomotion in 6-hydroxydopamine-lesioned rats.

Journal: Neuroscience 20030101

Title: Sea urchin embryos and larvae as biosensors for neurotoxicants.

Journal: Current protocols in toxicology 20030101

Title: Smooth muscle 5-HT2A receptors mediating contraction of porcine isolated proximal stomach strips.

Journal: British journal of pharmacology 20021201

Title: Functional cooperation between neurosteroids and D2 dopamine antagonists on KCl-evoked [3H]noradrenaline release: modulation by calcium channel blockers.

Journal: Journal of neuroendocrinology 20021201

Title: Sleep-wake mechanisms and drug discovery: sleep EEG as a tool for the development of CNS-acting drugs.

Journal: Dialogues in clinical neuroscience 20021201

Title: Hypotension caused by extracorporeal circulation: serotonin from pump-activated platelets triggers nitric oxide release.

Journal: Circulation 20021112

Title: Involvement of 5-HT7 receptors in serotonergic effects on spike afterpotentials in presumed jaw-closing motoneurons of rats.

Journal: Brain research 20021108

Title: Differential regulation of hippocampal BDNF mRNA by typical and atypical antipsychotic administration.

Journal: Brain research 20021101

Title: Prenatal opiate withdrawal activates the chick embryo hypothalamic pituitary-adrenal axis and dilates vitelline blood vessels via serotonin(2) receptors.

Journal: The Journal of pharmacology and experimental therapeutics 20021001

Title: Effect of a 5-HT(2C) serotonin agonist, dexnorfenfluramine, on amyloid precursor protein metabolism in guinea pigs.

Journal: Brain research 20020927

Title: Vasodilator and vasoconstrictor responses induced by 5-hydroxytryptamine in the in situ blood autoperfused hindquarters of the anaesthetized rat.

Journal: Naunyn-Schmiedeberg's archives of pharmacology 20020801

Title: Effects of sarpogrelate, a novel 5-HT2 antagonist, on 5-HT-induced endothelium-dependent relaxations in porcine coronary artery.

Journal: Japanese journal of pharmacology 20020801

Title: Acute and long-term effects of the 5-HT2 receptor antagonist ritanserin on EEG power spectra, motor activity, and sleep: changes at the light-dark phase shift.

Journal: Brain research 20020705

Title: 5-HT2A and 5-HT2C serotonin receptors differentially modulate mouse sexual arousal and the hypothalamo-pituitary-testicular response to the presence of a female.

Journal: Neuroendocrinology 20020701

Title: Decrease of core body temperature in mice by dehydroepiandrosterone.

Journal: Experimental biology and medicine (Maywood, N.J.) 20020601

Title: Recent advances in 5-HT1B/1D receptor antagonists and agonists and their potential therapeutic applications.

Journal: Current topics in medicinal chemistry 20020601

Title: Ritanserin antagonism of m-chlorophenylpiperazine effects in neuroleptic-free schizophrenics patients: support for serotonin-2 receptor modulation of schizophrenia symptoms.

Journal: Psychopharmacology 20020601

Title: Erratum to 'CNS drugs in Cushing's disease: pathophysiological and therapeutic implications for mood disorders' [Prog. Neuro-Psycol. Biol. Psychiatry, 26, 763 (2002)].

Journal: Progress in neuro-psychopharmacology & biological psychiatry 20020601

Title: Modulation by 5-hT2A receptors of aggressive behavior in isolated mice.

Journal: Japanese journal of pharmacology 20020501

Title: Nefazodone treatment of dysthymic disorder an open, long-term, prospective pilot study.

Journal: Progress in neuro-psychopharmacology & biological psychiatry 20020501

Title: Residual symptoms in depression an emerging therapeutic concept.

Journal: Progress in neuro-psychopharmacology & biological psychiatry 20020501

Title: Sustained ER Ca2+ depletion suppresses protein synthesis and induces activation-enhanced cell death in mast cells.

Journal: The Journal of biological chemistry 20020419

Title: Peripheral 5-HT(2A)-receptor-mediated formation of an inhibitor of atrial natriuretic peptide binding involves inflammation.

Journal: European journal of pharmacology 20020405

Title: Specific labelling of serotonin 5-HT(1B) receptors in rat frontal cortex with the novel, phenylpiperazine derivative, [3H]GR125,743. A pharmacological characterization.

Journal: Pharmacology, biochemistry, and behavior 20020401

Title: Effect of SB-243213, a selective 5-HT(2C) receptor antagonist, on the rat sleep profile: a comparison to paroxetine.

Journal: Pharmacology, biochemistry, and behavior 20020401

Title: Role of central 5-HT(2) receptors in fluoxetine-induced decreases in T lymphocyte activity.

Journal: Brain, behavior, and immunity 20020401

Title: Involvement of the serotonergic system in orexin-induced behavioral alterations in rats.

Journal: Regulatory peptides 20020315

Title: Ritanserin, a serotonin-2 receptor antagonist, improves ultradian sleep rhythmicity in young poor sleepers.

Journal: Clinical neurophysiology : official journal of the International Federation of Clinical Neurophysiology 20020301

Title: The atypical 5-HT2 receptor mediating tachycardia in pithed rats: pharmacological correlation with the 5-HT2A receptor subtype.

Journal: British journal of pharmacology 20020301

Title: The human 5-HT7 serotonin receptor splice variants: constitutive activity and inverse agonist effects.

Journal: British journal of pharmacology 20020301

Title: Modulation of cannabinoid agonist binding by 5-HT in the rat cerebellum.

Journal: Journal of neurochemistry 20020301

Title: Methiothepin attenuates gastric secretion and motility effects of vagal stimulants at the dorsal vagal complex.

Journal: European journal of pharmacology 20020201

Title: 5-HT(1B) but not 5-HT(6) or 5-HT(7) receptors mediate depression of spinal nociceptive reflexes in vitro.

Journal: British journal of pharmacology 20020201

Title: Calcium-antagonistic activity of sumatriptan in the rat anococcygeus muscle.

Journal: Pharmacology 20020101

Title: The pharmacology of the acute hyperthermic response that follows administration of 3,4-methylenedioxymethamphetamine (MDMA, 'ecstasy') to rats.

Journal: British journal of pharmacology 20020101

Title: Serotonin localization in Phallusia mammillata larvae and effects of 5-HT antagonists during larval development.

Journal: Development, growth & differentiation 20011201

Title: The 5-HT2C/2B receptor agonist m-chlorophenylpiperazine (mCPP) inhibits 2-deoxy-D-glucose (2-DG)-induced hyperphagia in rats.

Journal: Biological & pharmaceutical bulletin 20011201

Title: Serotonergic regulation of inhibitory avoidance and one-way escape in the rat elevated T-maze.

Journal: Neuroscience and biobehavioral reviews 20011201

Title: m-CPP hypolocomotion is selectively antagonized by compounds with high affinity for 5-HT(2C) receptors but not 5-HT(2A) or 5-HT(2B) receptors.

Journal: Behavioural pharmacology 20011201

Title: RNA editing of the human serotonin 5-HT2C receptor alters receptor-mediated activation of G13 protein.

Journal: The Journal of biological chemistry 20011130

Title: 5-HT(2A/2C) receptor-mediated hypopnea in the newborn rat: relationship to Fos immunoreactivity.

Journal: Pediatric research 20011101

Title: Assessment of affinity and dissociation ability of a newly synthesized 5-HT2 antagonist, AT-1015: comparison with other 5-HT2 antagonists.

Journal: Japanese journal of pharmacology 20011101

Title: Inverse agonist actions of typical and atypical antipsychotic drugs at the human 5-hydroxytryptamine(2C) receptor.

Journal: The Journal of pharmacology and experimental therapeutics 20011001

Title: Binding affinity of a newly synthesized 5-HT2 antagonist, AT-1015 (N-[2-[4-(5H-Dibenzo[a,d]cyclohepten-5-ylidene)-piperidino]ethyl]-1-formyl-4-piperidinecarboxamide monohydrochloride monohydrate), in the rabbit platelet membrane.

Journal: Biological & pharmaceutical bulletin 20011001

Title: Effects of the 5-HT2 receptor antagonist, ritanserin on hyperthermia and depletion of 5-HT in frontal cortex induced by a 5-HT releasing drug, p-chloroamphetamine (PCA) in mice.

Journal: Biological & pharmaceutical bulletin 20011001

Title: Effect of 5-HT1A and 5-HT2A/2C receptor modulation on neuroleptic-induced vacuous chewing movements.

Journal: European journal of pharmacology 20010928

Title: Embryonic 'binge' cocaine exposure alters neural-immune and neural-endocrine interactions in young chickens: involvement of serotonin(2) receptors.

Journal: Brain research. Developmental brain research 20010923

Title: Serotonin 2A receptor regulation of striatal neuropeptide gene expression is selective for tachykinin, but not enkephalin neurons following dopamine depletion.

Journal: Brain research. Molecular brain research 20010815

Title: Fenfluramine-induced pulmonary vasoconstriction: role of serotonin receptors and potassium channels.

Journal: Journal of applied physiology (Bethesda, Md. : 1985) 20010801

Title: In vivo resetting of the hamster circadian clock by 5-HT7 receptors in the suprachiasmatic nucleus.

Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience 20010715

Title: Serotonin-based pharmacotherapy for acute neuroleptic-induced akathisia: a new approach to an old problem.

Journal: The British journal of psychiatry : the journal of mental science 20010701

Title: Role of 5-HT(1A) and 5-HT(7) receptors in the facilitatory response induced by 8-OH-DPAT on learning consolidation.

Journal: Behavioural brain research 20010601

Title: Vascular actions of MDMA involve alpha1 and alpha2-adrenoceptors in the anaesthetized rat.

Journal: British journal of pharmacology 20010601

Title: The cloned human 5-HT7 receptor splice variants: a comparative characterization of their pharmacology, function and distribution.

Journal: Naunyn-Schmiedeberg's archives of pharmacology 20010601

Title: Affinity of serotonin receptor antagonists and agonists to recombinant and native alpha1-adrenoceptor subtypes.

Journal: Japanese journal of pharmacology 20010601

Title: An investigation of the mechanisms responsible for acute fluoxetine-induced anxiogenic-like effects in mice.

Journal: Behavioural pharmacology 20010601

Title: Human 5-HT(5) receptors: the 5-HT(5A) receptor is functional but the 5-HT(5B) receptor was lost during mammalian evolution.

Journal: European journal of pharmacology 20010427

Title: Cataleptic effect of neurosteroid 3alpha-hydroxy-5alpha-pregnan-20-one in mice: modulation by serotonergic agents.

Journal: Brain research 20010413

Title: A 5-HT(7) receptor-mediated depolarization in the anterodorsal thalamus. I. Pharmacological characterization.

Journal: The Journal of pharmacology and experimental therapeutics 20010401

Title: Serotonergic modulation of ventilation and upper airway stability in obese Zucker rats.

Journal: American journal of respiratory and critical care medicine 20010401

Title: Evidence for 5-HT(1B/1D) and 5-HT(2A) receptors mediating constriction of the canine internal carotid circulation.

Journal: British journal of pharmacology 20010301

Title: The GR127935-sensitive 5-HT(1) receptors mediating canine internal carotid vasoconstriction: resemblance to the 5-HT(1B), but not to the 5-HT(1D) or 5-ht(1F), receptor subtype.

Journal: British journal of pharmacology 20010301

Title: Discriminative stimulus properties of indorenate, a 5-HT1A, 5-HT1B and 5-HT2C agonist: a study in rats.

Journal: Journal of psychopharmacology (Oxford, England) 20010301

Title: The inhibitory effect of serotonin on the spontaneous discharge of suprachiasmatic neurons in hypothalamic slice is mediated by 5-HT(7) receptor.

Journal: Brain research bulletin 20010301

Title: Subchronic effects of the GABA-agonist lorazepam and the 5-HT2A/2C antagonist ritanserin on driving performance, slow wave sleep and daytime sleepiness in healthy volunteers.

Journal: Psychopharmacology 20010301

Title: Endogenous 5-HT tonically inhibits spontaneous firing activity of dorsal hippocampus CA1 pyramidal neurons through stimulation of 5-HT(1A) receptors in quiet awake rats: in vivo electrophysiological evidence.

Journal: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20010201

Title: Serotonergic modulation of retinal input to the mouse suprachiasmatic nucleus mediated by 5-HT1B and 5-HT7 receptors.

Journal: Journal of biological rhythms 20010201

Title: Potent serotonin (5-HT)(2A) receptor antagonists completely prevent the development of hyperthermia in an animal model of the 5-HT syndrome.

Journal: Brain research 20010126

Title: The antidepressant activity of inositol in the forced swim test involves 5-HT(2) receptors.

Journal: Behavioural brain research 20010108

Title: Effects of the 5-HT(6) receptor antagonist Ro 04-6790 on learning consolidation.

Journal: Behavioural brain research 20010108

Title: A randomized, double-blind, placebo-controlled study of ritanserin pharmacotherapy for cocaine dependence.

Journal: Drug and alcohol dependence 20010101

Title: The ameliorating effect of the water layer of Fructus Schisandrae on cycloheximide-induced amnesia in rats: interaction with drugs acting at neurotransmitter receptors.

Journal: Pharmacological research 20010101

Title: New developments in the pharmacotherapy of alcohol dependence.

Journal: The American journal on addictions 20010101

Title: Embryonic cocaine exposure and corticosterone: serotonin(2) receptor mediation.

Journal: Pharmacology, biochemistry, and behavior 20010101

Title: On the mechanism of tolerance to morphine-induced Straub tail reaction in mice.

Journal: Pharmacology, biochemistry, and behavior 20010101

Title: Neonatal dopamine depletion reveals a synergistic mechanism of mRNA regulation that is mediated by dopamine(D1) and serotonin(2) receptors and is targeted to tachykinin neurons of the dorsomedial striatum.

Journal: Neuroscience 20010101

Title: The neuropharmacology of upper airway motor control in the awake and asleep states: implications for obstructive sleep apnoea.

Journal: Respiratory research 20010101

Title: The effect of Psilocybe cubensis extract on hippocampal neurons in vitro.

Journal: Fiziolohichnyi zhurnal (Kiev, Ukraine : 1994) 20010101

Title: Expression of 5-HT(2A), 5-HT(2B) and 5-HT(2C) receptors in the mouse embryo.

Journal: International journal of developmental neuroscience : the official journal of the International Society for Developmental Neuroscience 20001101

Title: Differential modes of agonist binding to 5-hydroxytryptamine(2A) serotonin receptors revealed by mutation and molecular modeling of conserved residues in transmembrane region 5.

Journal: Molecular pharmacology 20001101

Title: The serotonin 5-HT(2A) receptor subtype does not mediate apomorphine-induced aggressive behaviour in male Wistar rats.

Journal: Pharmacology, biochemistry, and behavior 20001001

Title: Effects of the serotonin 5-HT(2) antagonist, ritanserin, and the serotonin 5-HT(1A) antagonist, WAY 100635, on cocaine-seeking in rats.

Journal: Pharmacology, biochemistry, and behavior 20001001

Title: Effects of serotoninergic drugs on tremor induced by physostigmine in rats.

Journal: Behavioural brain research 20000501

Title: RS-127445: a selective, high affinity, orally bioavailable 5-HT2B receptor antagonist.

Journal: British journal of pharmacology 19990701

Title: 5-HT2 receptor antagonism reduces hyperactivity induced by amphetamine, cocaine, and MK-801 but not D1 agonist C-APB.

Journal: Pharmacology, biochemistry, and behavior 19990601

Title: Attenuation of haloperidol-induced catalepsy by a 5-HT2C receptor antagonist.

Journal: British journal of pharmacology 19990201

Title: Chimeric receptor analysis of the ketanserin binding site in the human 5-Hydroxytryptamine1D receptor: importance of the second extracellular loop and fifth transmembrane domain in antagonist binding.

Journal: Molecular pharmacology 19981201

Title: Identification of residues in transmembrane regions III and VI that contribute to the ligand binding site of the serotonin 5-HT6 receptor.

Journal: Journal of neurochemistry 19981101

Title: The 5-hydroxytryptamine6 receptor-selective radioligand [3H]Ro 63-0563 labels 5-hydroxytryptamine receptor binding sites in rat and porcine striatum.

Journal: Molecular pharmacology 19980901

Title: Agonistic properties of alniditan, sumatriptan and dihydroergotamine on human 5-HT1B and 5-HT1D receptors expressed in various mammalian cell lines.

Journal: British journal of pharmacology 19980401

Title: Serotonergic regulation of neuropeptide and glutamic acid decarboxylase mRNA levels in the rat striatum and globus pallidus: studies with fluoxetine and DOI.

Journal: Brain research. Molecular brain research 19980201

Title: [3H]Rauwolscine: an antagonist radioligand for the cloned human 5-hydroxytryptamine2b (5-HT2B) receptor.

Journal: Naunyn-Schmiedeberg's archives of pharmacology 19980101

Title: Interaction of tryptamine and ergoline compounds with threonine 196 in the ligand binding site of the 5-hydroxytryptamine6 receptor.

Journal: Molecular pharmacology 19970901

Title: Characterization of human serotonin 1D and 1B receptors using [3H]-GR-125743, a novel radiolabelled serotonin 5HT1D/1B receptor antagonist.

Journal: Naunyn-Schmiedeberg's archives of pharmacology 19970901

Title: 8-OH-DPAT, a 5-HT1A agonist and ritanserin, a 5-HT2A/C antagonist, reverse haloperidol-induced catalepsy in rats independently of striatal dopamine release.

Journal: Psychopharmacology 19970501

Title: Mechanism of action of clozapine-induced modification of motor behavior in an animal model of the 'super-off' phenomenon.

Journal: Movement disorders : official journal of the Movement Disorder Society 19970301

Title: Pharmacological characterization of recombinant human 5-hydroxytryptamine1A receptors using a novel antagonist radioligand, [3H]WAY-100635.

Journal: Life sciences 19970101

Title: Functional and radioligand binding characterization of rat 5-HT6 receptors stably expressed in HEK293 cells.

Journal: Neuropharmacology 19970101

Title: Alniditan, a new 5-hydroxytryptamine1D agonist and migraine-abortive agent: ligand-binding properties of human 5-hydroxytryptamine1D alpha, human 5-hydroxytryptamine1D beta, and calf 5-hydroxytryptamine1D receptors investigated with [3H]5-hydroxytryptamine and [3H]alniditan.

Journal: Molecular pharmacology 19961201

Title: 5-HT3-like receptors in the rat medial prefrontal cortex: further pharmacological characterization.

Journal: Brain research 19960909

Title: Cloning, characterization, and chromosomal localization of a human 5-HT6 serotonin receptor.

Journal: Journal of neurochemistry 19960101

Title: Binding affinity of sarpogrelate, a new antiplatelet agent, and its metabolite for serotonin receptor subtypes.

Journal: Archives internationales de pharmacodynamie et de therapie 19960101

Title: Differential effects of classical and newer antipsychotics on the hypermotility induced by two dose levels of D-amphetamine.

Journal: European journal of pharmacology 19950905

Title: In-vitro pharmacology of sarpogrelate and the enantiomers of its major metabolite: 5-HT2A receptor specificity, stereoselectivity and modulation of ritanserin-induced depression of 5-HT contractions in rat tail artery.

Journal: The Journal of pharmacy and pharmacology 19950401

Title: Penile erection and yawning induced by 5-HT1C receptor agonists in male rats: relationship with dopaminergic and oxytocinergic transmission.

Journal: European journal of pharmacology 19940811

Title: Cloning of a novel human serotonin receptor (5-HT7) positively linked to adenylate cyclase.

Journal: The Journal of biological chemistry 19931105

Title: Molecular cloning and expression of a 5-hydroxytryptamine7 serotonin receptor subtype.

Journal: The Journal of biological chemistry 19930825

Title: Cloning and expression of a novel serotonin receptor with high affinity for tricyclic psychotropic drugs.

Journal: Molecular pharmacology 19930301

Title: Pharmacological characteristics of the newly cloned rat 5-hydroxytryptamine2F receptor.

Journal: Molecular pharmacology 19930301

Title: Effect of amperozide on rat cortical 5-HT2 and striatal and limbic dopamine D2 receptor occupancy: implications for antipsychotic action.

Journal: European journal of pharmacology 19920527

Title: Opioid and nonopioid components independently contribute to the mechanism of action of tramadol, an 'atypical' opioid analgesic.

Journal: The Journal of pharmacology and experimental therapeutics 19920101

Title: Effects of 5-HT1A agonists and 5-HT2 antagonists on haloperidol-induced dyskinesias in squirrel monkeys: no evidence for reciprocal 5-HT-dopamine interaction.

Journal: Psychopharmacology 19890101

Title: Interference of ketanserin with baroreflex control of the circulation in the conscious spontaneously hypertensive rat.

Journal: Drugs 19880101

Title: Leysen JE, et al. Receptor-binding properties in vitro and in vivo of ritanserin: A very potent and long acting serotonin-S2 antagonist. Mol Pharmacol. 1985 Jun;27(6):600-11.

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