Title: Discovery of new quinoline ether inhibitors with high affinity and selectivity for PDGFR tyrosine kinases.
Journal: Bioorganic & medicinal chemistry letters 20120501
Title: Discovery of AZD2932, a new Quinazoline Ether Inhibitor with high affinity for VEGFR-2 and PDGFR tyrosine kinases.
Journal: Bioorganic & medicinal chemistry letters 20120101
Title: Plé PA, et al. Discovery of AZD2932, a new Quinazoline Ether Inhibitor with high affinity for VEGFR-2 and PDGFR tyrosine kinases. Bioorg Med Chem Lett. 2012 Jan 1;22(1):262-6.