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923565-22-4,MFCD18251560
Catalog No.:AA00GU0S

923565-22-4 | GSK962040 (HCl salt)

Pack Size
Purity
Availability
Price(USD)
Quantity
  
1mg
95%
1 week  
$244.00   $171.00
- +
5mg
95%
1 week  
$454.00   $318.00
- +
10mg
95%
1 week  
$626.00   $438.00
- +
25mg
95%
1 week  
$964.00   $675.00
- +
50mg
95%
1 week  
$1,349.00   $944.00
- +
100mg
95%
1 week  
$1,795.00   $1,256.00
- +
500mg
95%
1 week  
$3,452.00   $2,416.00
- +
  • Technical Information
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  • Technical Information
  • Properties
  • Literature
Technical Information
Catalog Number:
AA00GU0S
Chemical Name:
GSK962040 (HCl salt)
CAS Number:
923565-22-4
Molecular Formula:
C25H34ClFN4O
Molecular Weight:
461.0151
MDL Number:
MFCD18251560
SMILES:
C[C@@H]1NCCN(C1)Cc1ccc(cc1)CC(=O)N1CCC(CC1)Nc1cccc(c1)F.Cl
Properties

Literature

Title: Sanger, G.J., et al., GSK962040: a small molecule, selective motilin receptor agonist, effective as a stimulant of human and rabbit gastrointestinal motility. Neurogastroenterol Motil, 2009. 21(6): p. 657-64, e30-1.

Title: Leming, S., et al., GSK962040: a small molecule motilin receptor agonist which increases gastrointestinal motility in conscious dogs. Neurogastroenterol Motil, 2011. 23(10): p. 958-e410.

Title: Westaway, S.M., et al., Discovery of N-(3-fluorophenyl)-1-[(4-([(3S)-3-methyl-1-piperazinylmethyl)phenyl)acetyl-4-pi peridinamine (GSK962040), the first small molecule motilin receptor agonist clinical candidate. J Med Chem, 2009. 52(4): p. 1180-9.

Title: Broad, J., et al., Regional- and agonist-dependent facilitation of human neurogastrointestinal functions by motilin receptor agonists. Br J Pharmacol, 2012. 167(4): p. 763-74.

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