Home Boronic Acids 957060-88-7
957060-88-7,MFCD06798255
Catalog No.:AA003BOX

957060-88-7 | 3-Chloro-2-methoxypyridine-4-boronic acid

Pack Size
Purity
Availability
Price(USD)
Quantity
  
100mg
98%
in stock  
$21.00   $15.00
- +
1g
95%
in stock  
$47.00   $33.00
- +
5g
98%
in stock  
$162.00   $114.00
- +
10g
97%
in stock  
$311.00   $218.00
- +
25g
97%
in stock  
$610.00   $427.00
- +
100g
97%
in stock  
$1,640.00   $1,148.00
- +
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Technical Information
Catalog Number:
AA003BOX
Chemical Name:
3-Chloro-2-methoxypyridine-4-boronic acid
CAS Number:
957060-88-7
Molecular Formula:
C6H7BClNO3
Molecular Weight:
187.3887
MDL Number:
MFCD06798255
SMILES:
COc1nccc(c1Cl)B(O)O
Properties
Properties
 
BP:
344.3°C at 760 mmHg  
Form:
Solid  
MP:
140 °C  
Storage:
Keep in dry area;2-8℃;  


Downstream Synthesis Route

[1]CurrentPatentAssignee:VERTEXPHARMACEUTICALS(OLD)-WO2008/141119,2008,A2Locationinpatent:Page/Pagecolumn157

[1]CurrentPatentAssignee:ROCHEHOLDINGAG-US2011/71150,2011,A1Locationinpatent:Page/Pagecolumn64

[1]Li,Zhihong;Wang,Xianghong;Eksterowicz,John;Gribble,MichaelW.;Alba,GraceQ.;Ayres,Merrill;Carlson,TimothyJ.;Chen,Ada;Chen,Xiaoqi;Cho,Robert;Connors,RichardV.;Degraffenreid,Michael;Deignan,JeffreyT.;Duquette,Jason;Fan,Pingchen;Fisher,Benjamin;Fu,Jiasheng;Huard,JustinN.;Kaizerman,Jacob;Keegan,KathleenS.;Li,Cong;Li,Kexue;Li,Yunxiao;Liang,Lingming;Liu,Wen;Lively,SarahE.;Lo,Mei-Chu;Ma,Ji;McMinn,DustinL.;Mihalic,JeffreyT.;Modi,Kriti;Ngo,Rachel;Pattabiraman,Kanaka;Piper,DerekE.;Queva,Christophe;Ragains,MarkL.;Suchomel,Julia;Thibault,Steve;Walker,Nigel;Wang,Xiaodong;Wang,Zhulun;Wanska,Malgorzata;Wehn,PaulM.;Weidner,MargaretF.;Zhang,AlexJ.;Zhao,Xiaoning;Kamb,Alexander;Wickramasinghe,Dineli;Dai,Kang;McGee,LawrenceR.;Medina,JulioC.[JournalofMedicinalChemistry,2014,vol.57,#8,p.3430-3449]

[2]Li,Zhihong;Wang,Xianghong;Eksterowicz,John;Gribble,MichaelW.;Alba,GraceQ.;Ayres,Merrill;Carlson,TimothyJ.;Chen,Ada;Chen,Xiaoqi;Cho,Robert;Connors,RichardV.;Degraffenreid,Michael;Deignan,JeffreyT.;Duquette,Jason;Fan,Pingchen;Fisher,Benjamin;Fu,Jiasheng;Huard,JustinN.;Kaizerman,Jacob;Keegan,KathleenS.;Li,Cong;Li,Kexue;Li,Yunxiao;Liang,Lingming;Liu,Wen;Lively,SarahE.;Lo,Mei-Chu;Ma,Ji;McMinn,DustinL.;Mihalic,JeffreyT.;Modi,Kriti;Ngo,Rachel;Pattabiraman,Kanaka;Piper,DerekE.;Queva,Christophe;Ragains,MarkL.;Suchomel,Julia;Thibault,Steve;Walker,Nigel;Wang,Xiaodong;Wang,Zhulun;Wanska,Malgorzata;Wehn,PaulM.;Weidner,MargaretF.;Zhang,AlexJ.;Zhao,Xiaoning;Kamb,Alexander;Wickramasinghe,Dineli;Dai,Kang;McGee,LawrenceR.;Medina,JulioC.[JournalofMedicinalChemistry,2014,vol.57,#8,p.3430-3449]

957060-88-7   
2-(3R)-3-methylmorpholin-4-yl-8-1-(tetrahydro-2H-pyran-2-yl)-1H-pyrazol-5-yl-1,7-naphthyridin-4-yltrifluoromethanesulfonate 
 
4-(3-chloro-2-methoxypyridin-4-yl)-2-(3R)-3-methylmorpholin-4-yl-8-(1H-pyrazol-5-yl)-1,7-naphthyridine 

[1]CurrentPatentAssignee:POLINUTRIALIMENTOSSA;BAYERAG-WO2016/20320,2016,A1Locationinpatent:Page/Pagecolumn254;255

957060-88-7   
4,5,6,7-tetrachloro-1,3-dioxoisoindolin-2-yl1-benzoylpiperidine-4-carboxylate 
 
(4-(3-chloro-2-methoxypyridin-4-yl)piperidin-1-yl)(phenyl)methanone 

[1]Sandfort,Frederik;O'Neill,MatthewJ.;Cornella,Josep;Wimmer,Laurin;Baran,PhilS.[AngewandteChemie-InternationalEdition,2017,vol.56,#12,p.3319-3323][Angew.Chem.,2017,vol.129,p.3367-3371,5]

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Tags:957060-88-7 Molecular Formula|957060-88-7 MDL|957060-88-7 SMILES|957060-88-7 3-Chloro-2-methoxypyridine-4-boronic acid