Title: Identification of potent Yes1 kinase inhibitors using a library screening approach.
Journal: Bioorganic & medicinal chemistry letters 20130801
Title: The role of neurotensin in passive avoidance learning in the rat central nucleus of amygdala.
Journal: Behavioural brain research 20120115
Title: Neurotensin decreases high affinity [3H]-ouabain binding to cerebral cortex membranes.
Journal: Regulatory peptides 20111210
Title: Inhibition of neurotensin receptor 1 selectively sensitizes prostate cancer to ionizing radiation.
Journal: Cancer research 20111101
Title: Neurotensin inhibits background K+ channels and facilitates glutamatergic transmission in rat spinal cord dorsal horn.
Journal: The European journal of neuroscience 20111001
Title: The many faces of the adamantyl group in drug design.
Journal: European journal of medicinal chemistry 20110601
Title: Pancreatic cancer bears overexpression of neurotensin and neurotensin receptor subtype-1 and SR 48692 counteracts neurotensin induced cell proliferation in human pancreatic ductal carcinoma cell line PANC-1.
Journal: Neuropeptides 20110401
Title: In vivo investigations of neurotensin receptors in adipocytes, hepatocytes and enterocytes of rat.
Journal: Annals of agricultural and environmental medicine : AAEM 20110101
Title: Neurotensin is a regulator of insulin secretion in pancreatic beta-cells.
Journal: The international journal of biochemistry & cell biology 20101001
Title: Effects of neurotensin in amygdaloid spatial learning mechanisms.
Journal: Behavioural brain research 20100711
Title: The role of neurotensin in positive reinforcement in the rat central nucleus of amygdala.
Journal: Behavioural brain research 20100402
Title: Intra-accumbens shell injections of SR48692 enhanced cocaine self-administration intake in rats exposed to an environmentally-elicited reinstatement paradigm.
Journal: Brain research 20090714
Title: Neurotensin inhibition of GABAergic transmission via mGluR-induced endocannabinoid signalling in rat periaqueductal grey.
Journal: The Journal of physiology 20090601
Title: Comparison of N-terminal modifications on neurotensin(8-13) analogues correlates peptide stability but not binding affinity with in vivo efficacy.
Journal: Journal of medicinal chemistry 20090409
Title: The identification of nonpeptide neurotensin receptor partial agonists from the potent antagonist SR48692 using a calcium mobilization assay.
Journal: Bioorganic & medicinal chemistry letters 20090301
Title: Neurotensin inversely modulates maternal aggression.
Journal: Neuroscience 20090218
Title: Electrophysiological effects of neurotensin on globus pallidus neurons of 6-hydroxydopamine-lesioned rats.
Journal: Neuro-Signals 20090101
Title: Heightened amygdala long-term potentiation in neurotensin receptor type-1 knockout mice.
Journal: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20081201
Title: Stimulation by neurotensin of dopamine and 5-hydroxytryptamine (5-HT) release from rat prefrontal cortex: possible role of NTR1 receptors in neuropsychiatric disorders.
Journal: Neurochemistry international 20081201
Title: High-affinity neurotensin receptor is involved in phosphoinositide turnover increase by inhibition of sodium pump in neonatal rat brain.
Journal: Neurochemical research 20081101
Title: Novel insights into GPCR-peptide interactions: mutations in extracellular loop 1, ligand backbone methylations and molecular modeling of neurotensin receptor 1.
Journal: Bioorganic & medicinal chemistry 20081015
Title: Neurotensin modulation of acetylcholine, GABA, and aspartate release from rat prefrontal cortex studied in vivo with microdialysis.
Journal: Brain research bulletin 20080930
Title: Neurotensin in the ventral pallidum increases extracellular gamma-aminobutyric acid and differentially affects cue- and cocaine-primed reinstatement.
Journal: The Journal of pharmacology and experimental therapeutics 20080501
Title: Neurotensin receptor antagonist administered during cocaine withdrawal decreases locomotor sensitization and conditioned place preference.
Journal: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20071201
Title: Blockade of neurotensin receptors during amphetamine discontinuation indicates individual variability.
Journal: Neuropeptides 20070401
Title: Impact of chronic beta-adrenoceptor activation on neurotensin-induced myocardial effects in rats.
Journal: European journal of pharmacology 20061228
Title: Interactions between NTS2 neurotensin and opioid receptors on two nociceptive responses assessed on the hot plate test in mice.
Journal: Behavioural brain research 20061215
Title: Bidirectional regulation of dopamine D2 and neurotensin NTS1 receptors in dopamine neurons.
Journal: The European journal of neuroscience 20061101
Title: Microinfusions of neurotensin antagonist SR 48692 within the nucleus accumbens core impair spatial learning in rats.
Journal: Behavioral neuroscience 20061001
Title: Neurotensin selectively facilitates glutamatergic transmission in globus pallidus.
Journal: Neuroscience 20060915
Title: Amphetamine-elicited striatal Fos expression is attenuated in neurotensin null mutant mice.
Journal: Neuroscience letters 20060710
Title: Biophysical characteristics of neurotensin polyplex for in vitro and in vivo gene transfection.
Journal: Biochimica et biophysica acta 20060701
Title: Neurotensin enhances nitric oxide generation via the JAK2-STAT1 pathway in murine macrophage Raw264.7 cells during costimulation with LPS and IFNgamma.
Journal: Neuropeptides 20060601
Title: Neurotensin-induced myocardial noradrenergic effects in spontaneously hypertensive rats.
Journal: Journal of cardiovascular pharmacology 20060201
Title: Impact and mechanisms of action of neurotensin on cardiac contractility in the rat left ventricle.
Journal: European journal of pharmacology 20050927
Title: Neuropeptide neurotensin stimulates intestinal wound healing following chronic intestinal inflammation.
Journal: American journal of physiology. Gastrointestinal and liver physiology 20050401
Title: Neurotensin receptor agonists and antagonists for schizophrenia.
Journal: The American journal of psychiatry 20050301
Title: Neurotensin receptor agonists and antagonists for schizophrenia.
Journal: The American journal of psychiatry 20050301
Title: Neurotensin activates GABAergic interneurons in the prefrontal cortex.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience 20050216
Title: High-affinity neurotensin receptor is involved in phosphoinositide hydrolysis stimulation by carbachol in neonatal rat brain.
Journal: Brain research. Developmental brain research 20050208
Title: Participation of ATP in nonadrenergic, noncholinergic relaxation of longitudinal muscle of wistar rat jejunum.
Journal: Journal of pharmacological sciences 20050101
Title: Neurotensin modulates synaptic transmission in the nucleus of the solitary tract of the rat.
Journal: Neuroscience 20050101
Title: The neurotensin agonist PD149163 increases Fos expression in the prefrontal cortex of the rat.
Journal: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20041001
Title: Endogenous neurotensin attenuates dopamine-dependent locomotion and stereotypy.
Journal: Brain research 20041001
Title: Blockade of neurotensin receptors affects differently hypo-locomotion and catalepsy induced by haloperidol in mice.
Journal: Neuropharmacology 20040701
Title: Characterization of neurotensin receptors.
Journal: Current protocols in pharmacology 20040501
Title: SR 48692, a specific neurotensin receptor antagonist, has no effect on oesophageal motility in humans.
Journal: Alimentary pharmacology & therapeutics 20040415
Title: Neurotensin enhances endogenous extracellular glutamate levels in primary cultures of rat cortical neurons: involvement of neurotensin receptor in NMDA induced excitotoxicity.
Journal: Cerebral cortex (New York, N.Y. : 1991) 20040401
Title: Role of calcium in neurotensin-evoked enhancement in firing in mesencephalic dopamine neurons.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience 20040310
Title: Sezary syndrome cells unlike normal circulating T lymphocytes fail to migrate following engagement of NT1 receptor.
Journal: The Journal of investigative dermatology 20040101
Title: Neurotensin depolarizes globus pallidus neurons in rats via neurotensin type-1 receptor.
Journal: Neuroscience 20040101
Title: Neurokinin B, neurotensin, and cannabinoid receptor antagonists and Parkinson disease.
Journal: Clinical neuropharmacology 20040101
Title: Endogenous neurotensin facilitates visceral nociception and is required for stress-induced antinociception in mice and rats.
Journal: Neuroscience 20040101
Title: Regulation of DARPP-32 Thr75 phosphorylation by neurotensin in neostriatal neurons: involvement of glutamate signalling.
Journal: The European journal of neuroscience 20030901
Title: Central administration of the neurotensin receptor antagonist SR48692 attenuates vacuous chewing movements in a rodent model of tardive dyskinesia.
Journal: Neuroscience 20030101
Title: Neurotensin enhances glutamate excitotoxicity in mesencephalic neurons in primary culture.
Journal: Journal of neuroscience research 20021215
Title: Pharmacology and functional properties of NTS2 neurotensin receptors in cerebellar granule cells.
Journal: The Journal of biological chemistry 20020927
Title: Neurotensin phase-shifts the firing rate rhythm of neurons in the rat suprachiasmatic nuclei in vitro.
Journal: The European journal of neuroscience 20020701
Title: Neurotensin causes tyrosine phosphorylation of focal adhesion kinase in lung cancer cells.
Journal: European journal of pharmacology 20020510
Title: Neurotensin-induced modulation of dopamine D2 receptors and their function in rat striatum: counteraction by a NTR1-like receptor antagonist.
Journal: Neuroreport 20020507
Title: Effects of neurotensin receptor antagonism on latent inhibition in Sprague-Dawley rats.
Journal: Psychopharmacology 20020501
Title: Neurotensin regulates DARPP-32 thr34 phosphorylation in neostriatal neurons by activation of dopamine D1-type receptors.
Journal: Journal of neurochemistry 20020401
Title: Stress-induced activation of median raphe serotonergic neurons in rats is potentiated by the neurotensin antagonist, SR 48692.
Journal: Neuroscience letters 20020208
Title: Constitutive activation of the neurotensin receptor 1 by mutation of Phe(358) in Helix seven.
Journal: British journal of pharmacology 20020201
Title: Chronic blockade of neurotensin receptors strongly reduces sensitized, but not acute, behavioral response to D-amphetamine.
Journal: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20020101
Title: Agonism, inverse agonism, and neutral antagonism at the constitutively active human neurotensin receptor 2.
Journal: Molecular pharmacology 20011201
Title: Characterization of the profile of neurokinin-2 and neurotensin receptor antagonists in the mouse defense test battery.
Journal: Neuroscience and biobehavioral reviews 20011201
Title: The neurotensin receptor antagonist, SR48692, attenuates the expression of amphetamine-induced behavioural sensitisation in mice.
Journal: European journal of pharmacology 20010928
Title: K(+)-p-nitrophenylphosphatase inhibition by neurotensin involves high affinity neurotensin receptor: influence of potassium concentration and enzyme phosphorylation.
Journal: Regulatory peptides 20010915
Title: Neurotensin induces mating in Saccharomyces cerevisiae cells that express human neurotensin receptor type 1 in place of the endogenous pheromone receptor.
Journal: European journal of biochemistry 20010901
Title: Neurotensin excitation of serotonergic neurons in the rat nucleus raphe magnus: ionic and molecular mechanisms.
Journal: Neuropharmacology 20010601
Title: Endogenous neurotensin down-regulates dopamine efflux in the nucleus accumbens as revealed by SR-142948A, a selective neurotensin receptor antagonist.
Journal: Journal of neurochemistry 20010601
Title: The neurotensin antagonist SR 48692 attenuates haloperidol-induced striatal Fos expression in the rat.
Journal: Neuroscience letters 20010427
Title: In vivo gene transfer to dopamine neurons of rat substantia nigra via the high-affinity neurotensin receptor.
Journal: Molecular medicine (Cambridge, Mass.) 20010301
Title: Evidence that neurotensin mediates the central effect of leptin on food intake in rat.
Journal: Brain research 20010112
Title: SR48692 is a neurotensin receptor antagonist which inhibits the growth of small cell lung cancer cells.
Journal: Peptides 20010101
Title: Nigral neurotensin receptor regulation of nigral glutamate and nigroventral thalamic GABA transmission: a dual-probe microdialysis study in intact conscious rat brain.
Journal: Neuroscience 20010101
Title: Neurotensin modulates the electrical activity of frog pituitary melanotropes via activation of a G-protein-coupled receptor pharmacologically related to both the NTS1 and nts2 receptors of mammals.
Journal: Neuroendocrinology 20001201
Title: Mutagenesis and modeling of the neurotensin receptor NTR1. Identification of residues that are critical for binding SR 48692, a nonpeptide neurotensin antagonist.
Journal: The Journal of biological chemistry 19980626
Title: Stable expression of the mouse levocabastine-sensitive neurotensin receptor in HEK 293 cell line: binding properties, photoaffinity labeling, and internalization mechanism.
Journal: Biochemical and biophysical research communications 19980213
Title: Biochemical and pharmacological activities of SR 142948A, a new potent neurotensin receptor antagonist.
Journal: The Journal of pharmacology and experimental therapeutics 19970201
Title: [3H]SR 48692, the first nonpeptide neurotensin antagonist radioligand: characterization of binding properties and evidence for distinct agonist and antagonist binding domains on the rat neurotensin receptor.
Journal: Molecular pharmacology 19950501
