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Title: Functional and molecular expression of the proton-coupled oligopeptide transporters in spleen and macrophages from mouse and human.
Journal: Molecular pharmaceutics 20130401
Title: Expression profile and functional activity of peptide transporters in prostate cancer cells.
Journal: Molecular pharmaceutics 20130204
Title: Mechanistic insights into PEPT1-mediated transport of a novel antiepileptic, NP-647.
Journal: Molecular pharmaceutics 20120904
Title: Intestinal drug transport via the proton-coupled amino acid transporter PAT1 (SLC36A1) is inhibited by Gly-X(aa) dipeptides.
Journal: Molecular pharmaceutics 20120904
Title: Role of the intestinal peptide transporter PEPT1 in oseltamivir absorption: in vitro and in vivo studies.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20120801
Title: Species-dependent uptake of glycylsarcosine but not oseltamivir in Pichia pastoris expressing the rat, mouse, and human intestinal peptide transporter PEPT1.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20120701
Title: Construction, identification and application of HeLa cells stably transfected with human PEPT1 and PEPT2.
Journal: Peptides 20120401
Title: Pharmacokinetics of memantine in rats and mice.
Journal: PLoS currents 20120215
Title: Influence of fed-fasted state on intestinal PEPT1 expression and in vivo pharmacokinetics of glycylsarcosine in wild-type and Pept1 knockout mice.
Journal: Pharmaceutical research 20120201
Title: Effect of dose escalation on the in vivo oral absorption and disposition of glycylsarcosine in wild-type and Pept1 knockout mice.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20111201
Title: Characterizing the intramolecular H-bond and secondary structure in methylated GlyGlyH+ with H2 predissociation spectroscopy.
Journal: Journal of the American Society for Mass Spectrometry 20111101
Title: 3H-L-leucine transport by the promiscuous crustacean dipeptide-like cotransporter.
Journal: Journal of experimental zoology. Part A, Ecological genetics and physiology 20111001
Title: Differentiating passive from transporter-mediated uptake by PepT1: a comparison and evaluation of four methods.
Journal: The Journal of surgical research 20110901
Title: Peptide absorption after massive proximal small bowel resection: mechanisms of ileal adaptation.
Journal: Journal of gastrointestinal surgery : official journal of the Society for Surgery of the Alimentary Tract 20110901
Title: Effects of JBP485 on the expression and function of PEPT1 in indomethacin-induced intestinal injury in rats and damage in Caco-2 cells.
Journal: Peptides 20110501
Title: Bifunctional peptidomimetic prodrugs of didanosine for improved intestinal permeability and enhanced acidic stability: synthesis, transepithelial transport, chemical stability and pharmacokinetics.
Journal: Molecular pharmaceutics 20110404
Title: Uptake, transport and regulation of JBP485 by PEPT1 in vitro and in vivo.
Journal: Peptides 20110401
Title: 1α,25-dihydroxyvitamin D3 on intestinal transporter function: studies with the rat everted intestinal sac.
Journal: Biopharmaceutics & drug disposition 20110301
Title: Peptide transporter 1 is responsible for intestinal uptake of the dipeptide glycylsarcosine: studies in everted jejunal rings from wild-type and Pept1 null mice.
Journal: Journal of pharmaceutical sciences 20110201
Title: Intestinal adaptation for oligopeptide absorption via PepT1 after massive (70%) mid-small bowel resection.
Journal: Journal of gastrointestinal surgery : official journal of the Society for Surgery of the Alimentary Tract 20110201
Title: Distribution of glycylsarcosine and cefadroxil among cerebrospinal fluid, choroid plexus, and brain parenchyma after intracerebroventricular injection is markedly different between wild-type and Pept2 null mice.
Journal: Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism 20110101
Title: Molecular biology of the blood-brain and the blood-cerebrospinal fluid barriers: similarities and differences.
Journal: Fluids and barriers of the CNS 20110101
Title: The quest for targeted delivery in colon cancer: mucoadhesive valdecoxib microspheres.
Journal: International journal of nanomedicine 20110101
Title: Choroid plexus transport: gene deletion studies.
Journal: Fluids and barriers of the CNS 20110101
Title: Serine side chain-linked peptidomimetic conjugates of cyclic HPMPC and HPMPA: synthesis and interaction with hPEPT1.
Journal: Molecular pharmaceutics 20101206
Title: Ibuprofen is a non-competitive inhibitor of the peptide transporter hPEPT1 (SLC15A1): possible interactions between hPEPT1 substrates and ibuprofen.
Journal: British journal of pharmacology 20101201
Title: Functional role of the intracellular loop linking transmembrane domains 6 and 7 of the human dipeptide transporter hPEPT1.
Journal: The Journal of membrane biology 20101201
Title: Significance and regional dependency of peptide transporter (PEPT) 1 in the intestinal permeability of glycylsarcosine: in situ single-pass perfusion studies in wild-type and Pept1 knockout mice.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20101001
Title: The proton-coupled amino acid transporter, SLC36A1 (hPAT1), transports Gly-Gly, Gly-Sar and other Gly-Gly mimetics.
Journal: British journal of pharmacology 20101001
Title: The apical (hPepT1) and basolateral peptide transport systems of Caco-2 cells are regulated by AMP-activated protein kinase.
Journal: American journal of physiology. Gastrointestinal and liver physiology 20100701
Title: Gene ablation for PEPT1 in mice abolishes the effects of dipeptides on small intestinal fluid absorption, short-circuit current, and intracellular pH.
Journal: American journal of physiology. Gastrointestinal and liver physiology 20100701
Title: Role of insulin on jejunal PepT1 expression and function regulation in diabetic male and female rats.
Journal: Canadian journal of physiology and pharmacology 20100701
Title: Putative anion transporter-1 (Pat-1, Slc26a6) contributes to intracellular pH regulation during H+-dipeptide transport in duodenal villous epithelium.
Journal: American journal of physiology. Gastrointestinal and liver physiology 20100501
Title: The intestinal absorption of a prodrug of the mGlu2/3 receptor agonist LY354740 is mediated by PEPT1: in situ rat intestinal perfusion studies.
Journal: Journal of pharmaceutical sciences 20100301
Title: The bioactive dipeptide anserine is transported by human proton-coupled peptide transporters.
Journal: The FEBS journal 20100201
Title: Absorption of lisdexamfetamine dimesylate and its enzymatic conversion to d-amphetamine.
Journal: Neuropsychiatric disease and treatment 20100101
Title: Evidence of D-phenylglycine as delivering tool for improving L-dopa absorption.
Journal: Journal of biomedical science 20100101
Title: Pharmacokinetics and mechanism of intestinal absorption of JBP485 in rats.
Journal: Drug metabolism and pharmacokinetics 20100101
Title: Diurnal expression and function of peptide transporter 1 (PEPT1).
Journal: The Journal of surgical research 20090901
Title: Oseltamivir (tamiflu) is a substrate of peptide transporter 1.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20090801
Title: Direct evidence for efficient transport and minimal metabolism of L-cephalexin by oligopeptide transporter 1 in budded baculovirus fraction.
Journal: Biological & pharmaceutical bulletin 20090801
Title: PEPT1 involved in the uptake and transepithelial transport of cefditoren in vivo and in vitro.
Journal: European journal of pharmacology 20090610
Title: Investigation of the role of oligopeptide transporter PEPT1 and sodium/glucose cotransporter SGLT1 in intestinal absorption of their substrates using small GTP-binding protein Rab8-null mice.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20090301
Title: Interferon-gamma increases expression of the di/tri-peptide transporter, h-PEPT1, and dipeptide transport in cultured human intestinal monolayers.
Journal: Pharmacological research 20090301
Title: Rapid and sensitive hydrophilic interaction chromatography/tandem mass spectrometry method for the determination of glycyl-sarcosine in cell homogenates.
Journal: Journal of chromatography. B, Analytical technologies in the biomedical and life sciences 20090301
Title: Inhibition of intracellular dipeptide hydrolysis uncovers large outward transport currents of the peptide transporter PEPT1 in Xenopus oocytes.
Journal: Pflugers Archiv : European journal of physiology 20090201
Title: Transepithelial transport of the group II metabotropic glutamate 2/3 receptor agonist (1S,2S,5R,6S)-2-aminobicyclo[3.1.0]hexane-2,6-dicarboxylate (LY354740) and its prodrug (1S,2S,5R,6S)-2-[(2'S)-(2'-amino)propionyl]aminobicyclo[3.1.0]hexane-2,6-dicarboxylate (LY544344).
Journal: Drug metabolism and disposition: the biological fate of chemicals 20090101
Title: Transport and signaling via the amino acid binding site of the yeast Gap1 amino acid transceptor.
Journal: Nature chemical biology 20090101
Title: Synthesis, transport and pharmacokinetics of 5'-amino acid ester prodrugs of 1-beta-D-arabinofuranosylcytosine.
Journal: Molecular pharmaceutics 20090101
Title: Intestinal dipeptide absorption is preserved during thermal injury and cytokine treatment.
Journal: JPEN. Journal of parenteral and enteral nutrition 20090101
Title: Escherichia coli, an Intestinal Microorganism, as a Biosensor for Quantification of Amino Acid Bioavailability.
Journal: Sensors (Basel, Switzerland) 20090101
Title: Transport of angiotensin-converting enzyme inhibitors by H+/peptide transporters revisited.
Journal: The Journal of pharmacology and experimental therapeutics 20081101
Title: Enhanced cancer cell growth inhibition by dipeptide prodrugs of floxuridine: increased transporter affinity and metabolic stability.
Journal: Molecular pharmaceutics 20081006
Title: DtpB (YhiP) and DtpA (TppB, YdgR) are prototypical proton-dependent peptide transporters of Escherichia coli.
Journal: The FEBS journal 20080701
Title: hPEPT1 is responsible for uptake and transport of Gly-Sar in the human bronchial airway epithelial cell-line Calu-3.
Journal: Pflugers Archiv : European journal of physiology 20080601
Title: Ethanol inhibits functional activity of the human intestinal dipeptide transporter hPepT1 expressed in Xenopus oocytes.
Journal: Alcoholism, clinical and experimental research 20080501
Title: Cloning of the pig PEPT2 (pPEPT2) and characterization of the effects of epidermal growth factor (EGF) on pPEPT2-mediated peptide uptake in the renal porcine cell line LLC-PK1.
Journal: European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences 20080423
Title: Quantitative prediction of oral absorption of PEPT1 substrates based on in vitro uptake into Caco-2 cells.
Journal: International journal of pharmaceutics 20080416
Title: Cancer detection using a PET tracer, 11C-glycylsarcosine, targeted to H+/peptide transporter.
Journal: Journal of nuclear medicine : official publication, Society of Nuclear Medicine 20080401
Title: Oral absorption of ampicillin: role of paracellular route vs. PepT1 transporter.
Journal: Fundamental & clinical pharmacology 20080401
Title: Evaluation of the effect of ethanol's toxic metabolite acetaldehyde on the gastrointestinal oligopeptide transporter, PEPT1: in vitro and in vivo studies.
Journal: Alcoholism, clinical and experimental research 20080101
Title: Role and relevance of PEPT2 in drug disposition, dynamics, and toxicity.
Journal: Drug metabolism and pharmacokinetics 20080101
Title: The apical uptake transporter of levofloxacin is distinct from the peptide transporter in human intestinal epithelial Caco-2 cells.
Journal: Drug metabolism and pharmacokinetics 20080101
Title: Inhibitory effect of zinc on the absorption of beta-lactam antibiotic ceftibuten via the peptide transporters in rats.
Journal: Drug metabolism and pharmacokinetics 20080101
Title: Targeted disruption of peptide transporter Pept1 gene in mice significantly reduces dipeptide absorption in intestine.
Journal: Molecular pharmaceutics 20080101
Title: Changes in small intestinal nutrient transport and barrier function after lipopolysaccharide exposure in two pig breeds.
Journal: Journal of animal science 20071001
Title: Long-term effect of leptin on H+-coupled peptide cotransporter 1 activity and expression in vivo: evidence in leptin-deficient mice.
Journal: The Journal of pharmacology and experimental therapeutics 20071001
Title: Recognition of 2-aminothiazole-4-acetic acid derivatives by the peptide transporters PEPT1 and PEPT2.
Journal: European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences 20070901
Title: In vivo effects of glycyl-glutamate and glycyl-sarcosine on gabapentin oral absorption in rat.
Journal: Pharmaceutical research 20070801
Title: Dipeptide monoester ganciclovir prodrugs for transscleral drug delivery: targeting the oligopeptide transporter on rabbit retina.
Journal: Journal of ocular pharmacology and therapeutics : the official journal of the Association for Ocular Pharmacology and Therapeutics 20070801
Title: Regulation of intestinal hPepT1 (SLC15A1) activity by phosphodiesterase inhibitors is via inhibition of NHE3 (SLC9A3).
Journal: Biochimica et biophysica acta 20070701
Title: Intestinal absorption of novel-dipeptide prodrugs of saquinavir in rats.
Journal: International journal of pharmaceutics 20070524
Title: Cysteine scanning of transmembrane domain three of the human dipeptide transporter: implications for substrate transport.
Journal: Journal of drug targeting 20070401
Title: Functional characterization of peptide transporters in MDCKII-MDR1 cell line as a model for oral absorption studies.
Journal: International journal of pharmaceutics 20070306
Title: Demonstration of functional dipeptide transport with expression of PEPT2 in guinea pig cardiomyocytes.
Journal: Pflugers Archiv : European journal of physiology 20070301
Title: Cryptosporidiosis induces a transient upregulation of the oligopeptides transporter (PepT1) activity in neonatal rats.
Journal: Experimental biology and medicine (Maywood, N.J.) 20070301
Title: Effects of capsaicin on intestinal cephalexin absorption in rats.
Journal: Biological & pharmaceutical bulletin 20070301
Title: PEPT1 enhances the uptake of gabapentin via trans-stimulation of b0,+ exchange.
Journal: Pharmaceutical research 20070201
Title: Membrane transport function in primary cultures of human proximal tubular cells.
Journal: Toxicology 20061207
Title: Induction of intestinal peptide transporter 1 expression during fasting is mediated via peroxisome proliferator-activated receptor alpha.
Journal: American journal of physiology. Gastrointestinal and liver physiology 20061101
Title: Expression and functional characteristics of tubular transporters: P-glycoprotein, PEPT1, and PEPT2 in renal mass reduction and diabetes.
Journal: American journal of physiology. Renal physiology 20061101
Title: Mutation in an adaptor protein PDZK1 affects transport activity of organic cation transporter OCTNs and oligopeptide transporter PEPT2.
Journal: Drug metabolism and pharmacokinetics 20061001
Title: Molecular interactions between dipeptides, drugs and the human intestinal H+ -oligopeptide cotransporter hPEPT1.
Journal: The Journal of physiology 20060701
Title: The PDZ domain protein PDZK1 interacts with human peptide transporter PEPT2 and enhances its transport activity.
Journal: Kidney international 20060701
Title: Human PEPT1 pharmacophore distinguishes between dipeptide transport and binding.
Journal: Journal of medicinal chemistry 20060615
Title: Transepithelial flux of early and advanced glycation compounds across Caco-2 cell monolayers and their interaction with intestinal amino acid and peptide transport systems.
Journal: The British journal of nutrition 20060601
Title: Role of PEPT2 in glycylsarcosine transport in astrocyte and glioma cultures.
Journal: Neuroscience letters 20060403
Title: Prediction of glycylsarcosine transport in Caco-2 cell lines expressing PEPT1 at different levels.
Journal: Pflugers Archiv : European journal of physiology 20060401
Title: The functional evaluation of human peptide/histidine transporter 1 (hPHT1) in transiently transfected COS-7 cells.
Journal: European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences 20060401
Title: Investigation of the route of absorption of lipid and sugar modified leu-enkephalin analogues and their enzymatic stability using the caco-2 cell monolayer system.
Journal: Medicinal chemistry (Shariqah (United Arab Emirates)) 20060301
Title: Na+/H+ exchanger 3 affects transport property of H+/oligopeptide transporter 1.
Journal: Drug metabolism and pharmacokinetics 20051201
Title: Role and relevance of peptide transporter 2 (PEPT2) in the kidney and choroid plexus: in vivo studies with glycylsarcosine in wild-type and PEPT2 knockout mice.
Journal: The Journal of pharmacology and experimental therapeutics 20051001
Title: Rapid elimination of cefaclor from the cerebrospinal fluid is mediated by a benzylpenicillin-sensitive mechanism distinct from organic anion transporter 3.
Journal: The Journal of pharmacology and experimental therapeutics 20050801
Title: Computational modelling of H+-coupled peptide transport via human PEPT1.
Journal: The Journal of physiology 20050601
Title: Functional linkage of H+/peptide transporter PEPT2 and Na+/H+ exchanger in primary cultures of astrocytes from mouse cerebral cortex.
Journal: Brain research 20050517
Title: Increased protein level of PEPT1 intestinal H+-peptide cotransporter upregulates absorption of glycylsarcosine and ceftibuten in 5/6 nephrectomized rats.
Journal: American journal of physiology. Gastrointestinal and liver physiology 20050401
Title: In vitro and pharmacophore-based discovery of novel hPEPT1 inhibitors.
Journal: Pharmaceutical research 20050401
Title: Amino acid ester prodrugs of the antiviral agent 2-bromo-5,6-dichloro-1-(beta-D-ribofuranosyl)benzimidazole as potential substrates of hPEPT1 transporter.
Journal: Journal of medicinal chemistry 20050224
Title: Exploring the role of different drug transport routes in permeability screening.
Journal: Journal of medicinal chemistry 20050127
Title: H+-dependent transport mechanism of nateglinide in the brush-border membrane of the rat intestine.
Journal: The Journal of pharmacology and experimental therapeutics 20050101
Title: Functional characterization of a cloned pig intestinal peptide transporter (pPepT1).
Journal: Journal of animal science 20050101
Title: Characterization of rPEPT2-mediated Gly-Sar transport parameters in the rat kidney proximal tubule cell line SKPT-0193 cl.2 cultured in basic growth media.
Journal: Molecular pharmaceutics 20050101
Title: Amino acid ester prodrugs of the anticancer agent gemcitabine: synthesis, bioconversion, metabolic bioevasion, and hPEPT1-mediated transport.
Journal: Molecular pharmaceutics 20050101
Title: hPEPT1 affinity and translocation of selected Gln-Sar and Glu-Sar dipeptide derivatives.
Journal: Molecular pharmaceutics 20050101
Title: Genetic variants of the human H+/dipeptide transporter PEPT2: analysis of haplotype functions.
Journal: The Journal of pharmacology and experimental therapeutics 20041201
Title: Efflux properties of basolateral peptide transporter in human intestinal cell line Caco-2.
Journal: Pflugers Archiv : European journal of physiology 20041101
Title: Stable transfection of MDCK cells with epitope-tagged human PepT1.
Journal: Pharmaceutical research 20041101
Title: Screening of the interaction between xenobiotic transporters and PDZ proteins.
Journal: Pharmaceutical research 20041001
Title: Role of PEPT2 in the choroid plexus uptake of glycylsarcosine and 5-aminolevulinic acid: studies in wild-type and null mice.
Journal: Pharmaceutical research 20040901
Title: Decreased activity and expression of intestinal oligopeptide transporter PEPT1 in rats with hyperthyroidism in vivo.
Journal: Pharmaceutical research 20040601
Title: Transport of the phosphonodipeptide alafosfalin by the H+/peptide cotransporters PEPT1 and PEPT2 in intestinal and renal epithelial cells.
Journal: European journal of biochemistry 20040501
Title: Genetic variant Arg57His in human H+/peptide cotransporter 2 causes a complete loss of transport function.
Journal: Biochemical and biophysical research communications 20040402
Title: Modulation of intestinal P-glycoprotein function by cremophor EL and other surfactants by an in vitro diffusion chamber method using the isolated rat intestinal membranes.
Journal: Journal of pharmaceutical sciences 20040401
Title: Mechanism of a model dipeptide transport across blood-ocular barriers following systemic administration.
Journal: Experimental eye research 20040401
Title: Epidermal growth factor decreases PEPT2 transport capacity and expression in the rat kidney proximal tubule cell line SKPT0193 cl.2.
Journal: American journal of physiology. Renal physiology 20040201
Title: A novel high-throughput pepT1 transporter assay differentiates between substrates and antagonists.
Journal: Molecular pharmaceutics 20040112
Title: In-depth evaluation of Gly-Sar transport parameters as a function of culture time in the Caco-2 cell model.
Journal: European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences 20040101
Title: Effect of diabetes mellitus and insulin on the regulation of the PepT 1 symporter in rat jejunum.
Journal: Molecular pharmaceutics 20040101
Title: Comparison of human and monkey peptide transporters: PEPT1 and PEPT2.
Journal: Molecular pharmaceutics 20040101
Title: Analysis of transmembrane segment 7 of the dipeptide transporter hPepT1 by cysteine-scanning mutagenesis.
Journal: The Journal of biological chemistry 20031219
Title: Changes of biological functions of dipeptide transporter (PepT1) and hormonal regulation in severe scald rats.
Journal: World journal of gastroenterology 20031215
Title: Concentration-dependent atypical intestinal absorption of cyclic phenylalanylserine: small intestine acts as an interface between the body and ingested compounds.
Journal: Biological & pharmaceutical bulletin 20031101
Title: Preliminary investigation into the expression of proton-coupled oligopeptide transporters in neural retina and retinal pigment epithelium (RPE): lack of functional activity in RPE plasma membranes.
Journal: Pharmaceutical research 20030901
Title: Inhibitory effect of zinc on PEPT1-mediated transport of glycylsarcosine and beta-lactam antibiotics in human intestinal cell line Caco-2.
Journal: Pharmaceutical research 20030901
Title: High glucose concentration in isotonic media alters caco-2 cell permeability.
Journal: AAPS pharmSci 20030901
Title: Transmembrane segment 5 of the dipeptide transporter hPepT1 forms a part of the substrate translocation pathway.
Journal: Biochemical and biophysical research communications 20030620
Title: Epidermal growth factor and insulin short-term increase hPepT1-mediated glycylsarcosine uptake in Caco-2 cells.
Journal: Acta physiologica Scandinavica 20030601
Title: Postnatal development of nutrient transport in the intestine of dogs.
Journal: American journal of veterinary research 20030501
Title: Delivery of peptide drugs to the brain by adenovirus-mediated heterologous expression of human oligopeptide transporter at the blood-brain barrier.
Journal: The Journal of pharmacology and experimental therapeutics 20030401
Title: Interactions of the dipeptide ester prodrugs of acyclovir with the intestinal oligopeptide transporter: competitive inhibition of glycylsarcosine transport in human intestinal cell line-Caco-2.
Journal: The Journal of pharmacology and experimental therapeutics 20030201
Title: Inhibition of intestinal dipeptide transport by the neuropeptide VIP is an anti-absorptive effect via the VPAC1 receptor in a human enterocyte-like cell line (Caco-2).
Journal: British journal of pharmacology 20030201
Title: Uptake of dipeptide and beta-lactam antibiotics by the basolateral membrane vesicles prepared from rat kidney.
Journal: Biochimica et biophysica acta 20030110
Title: Transcellular transport of a highly polar 3+ net charge opioid tetrapeptide.
Journal: The Journal of pharmacology and experimental therapeutics 20030101
Title: Novel dipeptide prodrugs of acyclovir for ocular herpes infections: Bioreversion, antiviral activity and transport across rabbit cornea.
Journal: Current eye research 20030101
Title: Optimal absorptive transport of the dipeptide glycylsarcosine is dependent on functional Na+/H+ exchange activity.
Journal: Pflugers Archiv : European journal of physiology 20021001
Title: Ocular penetration of acyclovir and its peptide prodrugs valacyclovir and val-valacyclovir following systemic administration in rabbits: An evaluation using ocular microdialysis and LC-MS.
Journal: Current eye research 20021001
Title: Effects of nonionic surfactants on membrane transporters in Caco-2 cell monolayers.
Journal: European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences 20020901
Title: Uptake of cyclic dipeptide by PEPT1 in Caco-2 cells: phenolic hydroxyl group of substrate enhances affinity for PEPT1.
Journal: The Journal of pharmacy and pharmacology 20020901
Title: Ionic strength has a greater effect than does transmembrane electric potential difference on permeation of tryptamine and indoleacetic acid across Caco-2 cells.
Journal: Biochimica et biophysica acta 20020819
Title: Diurnal rhythm of H+-peptide cotransporter in rat small intestine.
Journal: American journal of physiology. Gastrointestinal and liver physiology 20020701
Title: H+-peptide cotransport in the human bile duct epithelium cell line SK-ChA-1.
Journal: American journal of physiology. Gastrointestinal and liver physiology 20020701
Title: Studies on intestinal absorption of sulpiride (1): carrier-mediated uptake of sulpiride in the human intestinal cell line Caco-2.
Journal: Biological & pharmaceutical bulletin 20020701
Title: Enhanced delivery of drugs to the liver by adenovirus-mediated heterologous expression of the human oligopeptide transporter PEPT1.
Journal: The Journal of pharmacology and experimental therapeutics 20020601
Title: Role of PEPT2 in peptide/mimetic trafficking at the blood-cerebrospinal fluid barrier: studies in rat choroid plexus epithelial cells in primary culture.
Journal: The Journal of pharmacology and experimental therapeutics 20020601
Title: Thyroid hormone regulates the activity and expression of the peptide transporter PEPT1 in Caco-2 cells.
Journal: American journal of physiology. Gastrointestinal and liver physiology 20020401
Title: Comparison of bidirectional cephalexin transport across MDCK and caco-2 cell monolayers: interactions with peptide transporters.
Journal: Pharmaceutical research 20020101
Title: Inhibitory effect of supramolecular polyrotaxane-dipeptide conjugates on digested peptide uptake via intestinal human peptide transporter.
Journal: Bioconjugate chemistry 20020101
Title: Concentration-dependent preferences of absorptive and excretive transport cause atypical intestinal absorption of cyclic phenylalanylserine: small intestine acts as an interface between the body and ingested compounds.
Journal: Research communications in molecular pathology and pharmacology 20020101
Title: Upregulation of H(+)-peptide cotransporter PEPT2 in rat remnant kidney.
Journal: American journal of physiology. Renal physiology 20011201
Title: PepT1-mediated epithelial transport of dipeptides and cephalexin is enhanced by luminal leptin in the small intestine.
Journal: The Journal of clinical investigation 20011115
Title: Application of enzymatically stable dipeptides for enhancement of intestinal permeability. Synthesis and in vitro evaluation of dipeptide-coupled compounds.
Journal: Bioorganic & medicinal chemistry 20011001
Title: Distinct transport characteristics of basolateral peptide transporters between MDCK and Caco-2 cells.
Journal: Pflugers Archiv : European journal of physiology 20011001
Title: Conformational limitations of glycylsarcosine as a prototypic substrate for peptide transporters.
Journal: Biochimica et biophysica acta 20010903
Title: Epidermal growth factor inhibits glycylsarcosine transport and hPepT1 expression in a human intestinal cell line.
Journal: American journal of physiology. Gastrointestinal and liver physiology 20010701
Title: PEPT2-mediated uptake of neuropeptides in rat choroid plexus.
Journal: Pharmaceutical research 20010601
Title: Effects of tacrolimus and cyclosporin A on peptide transporter PEPT1 in Caco-2 cells.
Journal: Pharmaceutical research 20010501
Title: Drug inhibition of Gly-Sar uptake and hPepT1 localization using hPepT1-GFP fusion protein.
Journal: AAPS pharmSci 20010301
Title: Significance of substrate hydrophobicity for recognition by an oligopeptide transporter (PEPT1).
Journal: Bioconjugate chemistry 20010101
Title: Immunohistochemical and functional characterization of pH-dependent intestinal absorption of weak organic acids by the monocarboxylic acid transporter MCT1.
Journal: The Journal of pharmacy and pharmacology 19991001
Title: hPepT1-mediated epithelial transport of bacteria-derived chemotactic peptides enhances neutrophil-epithelial interactions.
Journal: The Journal of clinical investigation 19981201
Title: 5'-Amino acid esters of antiviral nucleosides, acyclovir, and AZT are absorbed by the intestinal PEPT1 peptide transporter.
Journal: Pharmaceutical research 19980801
Title: Recognition of beta-lactam antibiotics by rat peptide transporters, PEPT1 and PEPT2, in LLC-PK1 cells.
Journal: The American journal of physiology 19971101
Title: The predominant contribution of oligopeptide transporter PepT1 to intestinal absorption of beta-lactam antibiotics in the rat small intestine.
Journal: The Journal of pharmacy and pharmacology 19970801
Title: Interaction of anionic cephalosporins with the intestinal and renal peptide transporters PEPT 1 and PEPT 2.
Journal: Biochimica et biophysica acta 19970313
Title: Human dipeptide transporter, hPEPT1, stably transfected into Chinese hamster ovary cells.
Journal: Pharmaceutical research 19961101
Title: Identification of the histidine residues involved in substrate recognition by a rat H+/peptide cotransporter, PEPT1.
Journal: FEBS letters 19960930
