[1]CurrentPatentAssignee:IVASHCHENKO;ALLACHEMLLC-US2011/178078,2011,A1Locationinpatent:Page/Pagecolumn23;85;94
[1]Locationinpatent:experimentalpartIvachtchenko,AlexandreV.;Golovina,ElenaS.;Kadieva,MadinaG.;Kysil,VolodymyrM.;Mitkin,OlegD.;Tkachenko,SergeyE.;Okun,IlyaM.[JournalofMedicinalChemistry,2011,vol.54,#23,p.8161-8173]
Title: Synthesis and structure-activity relationship (SAR) of (5,7-disubstituted 3-phenylsulfonyl-pyrazolo[1,5-a]pyrimidin-2-yl)-methylamines as potent serotonin 5-HT(6) receptor (5-HT(6)R) antagonists.
Journal: Journal of medicinal chemistry 20111208
Title: Ivachtchenko AV, et al. AVN-492, A Novel Highly Selective 5-HT6R Antagonist: Preclinical Evaluation. J Alzheimers Dis. 2017;58(4):1043-1063.