Title: Vitamin D inhibits CEACAM1 to promote insulin/IGF-I receptor signaling without compromising anti-proliferative action.
Journal: Laboratory investigation; a journal of technical methods and pathology 20110101
Title: Synergistic induction of gene expression during the differentiation into mature macrophage in human myeloblastic leukemia cells treated with TPA and KH1060.
Journal: Leukemia research 20090601
Title: Vitamin D-binding protein influences total circulating levels of 1,25-dihydroxyvitamin D3 but does not directly modulate the bioactive levels of the hormone in vivo.
Journal: Endocrinology 20080701
Title: Interaction among vitamin D(3) analogue KH 1060, TNF-alpha, and vitamin D receptor protein in peripheral blood mononuclear cells of inflammatory bowel disease patients.
Journal: International immunopharmacology 20060701
Title: Vitamin D receptor: ligand recognition and allosteric network.
Journal: Journal of medicinal chemistry 20060223
Title: Human cathelicidin antimicrobial peptide (CAMP) gene is a direct target of the vitamin D receptor and is strongly up-regulated in myeloid cells by 1,25-dihydroxyvitamin D3.
Journal: FASEB journal : official publication of the Federation of American Societies for Experimental Biology 20050701
Title: Biochemical effects of KH 1060 and anti-TNF monoclonal antibody on human peripheral blood mononuclear cells.
Journal: International immunopharmacology 20050401
Title: Targacept active conformation search: a new method for predicting the conformation of a ligand bound to its protein target.
Journal: Journal of medicinal chemistry 20041230
Title: 9-cis retinoic acid accelerates calcitriol-induced osteocalcin production and promotes degradation of both vitamin D receptor and retinoid X receptor in human osteoblastic cells.
Journal: Journal of cellular biochemistry 20030815
Title: Inhibition of MG-63 cell cycle progression by synthetic vitamin D3 analogs mediated by p27, Cdk2, cyclin E, and the retinoblastoma protein.
Journal: Biochemical pharmacology 20030801
Title: 1,25-dihydroxyvitamin D3-induced apoptosis of retinoblastoma cells is associated with reciprocal changes of Bcl-2 and bax.
Journal: Experimental eye research 20030701
Title: Anti-proliferative effects of 20-epi-vitamin-D3 analogue, KH1060 in human neuroblastoma: induction of RAR-beta and p21(Cip1).
Journal: Cancer letters 20030210
Title: Involvement of diverse protein kinase C isoforms in the differentiation of ML-1 human myeloblastic leukemia cells induced by the vitamin D3 analogue KH1060 and the phorbol ester TPA.
Journal: Cancer letters 20021201
Title: Synergistic inhibitory effect of cyclosporin A and vitamin D derivatives on T-lymphocyte proliferation in active ulcerative colitis.
Journal: The American journal of gastroenterology 20020301
Title: Synergistic effect of vitamin D derivatives and retinoids on C2C12 skeletal muscle cells.
Journal: IUBMB life 20020301
Title: A combination of KH1060, a vitamin D(3) analogue, and cyclosporin prevents early graft failure and prolongs graft survival of xenogeneic islets in nonobese diabetic mice.
Journal: Transplantation proceedings 20010501
Title: Vitamin D(3) and its synthetic analogs inhibit the spontaneous in vitro immunoglobulin production by SLE-derived PBMC.
Journal: Clinical immunology (Orlando, Fla.) 20010401
Title: Suppressive effect of 1,25-dihydroxyvitamin D3 and its analogues EB 1089 and KH 1060 on T lymphocyte proliferation in active ulcerative colitis.
Journal: Biochemical pharmacology 20010201
Title: Cytotoxic effects of 1 alpha,25-dihydroxyvitamin D3 and synthetic vitamin D3 analogues on a glioma cell line.
Journal: Cancer letters 19960227
Title: Studies on two new vitamin D analogs, EB 1089 and KH 1060: effects on bone resorption and osteoclast recruitment in vitro.
Journal: Bone 19951001
Title: L Binderup, et al. 20-epi-vitamin D3 analogues: a novel class of potent regulators of cell growth and immune responses. Biochem Pharmacol. 1991 Sep 27;42(8):1569-75.
Title: C Gysemans, et al. A combination of KH1060, a vitamin D(3) analogue, and cyclosporin prevents early graft failure and prolongs graft survival of xenogeneic islets in nonobese diabetic mice. Transplant Proc. 2001 May;33(3):2365.
