Title: Profiling 976 ToxCast chemicals across 331 enzymatic and receptor signaling assays.
Journal: Chemical research in toxicology 20130617
Title: 5-HT(2A) receptor blockade and 5-HT(2C) receptor activation interact to reduce cocaine hyperlocomotion and Fos protein expression in the caudate-putamen.
Journal: Synapse (New York, N.Y.) 20121201
Title: 5-HT2A receptors in the orbitofrontal cortex facilitate reversal learning and contribute to the beneficial cognitive effects of chronic citalopram treatment in rats.
Journal: The international journal of neuropsychopharmacology 20121001
Title: Involvement of 5-HT2A receptor and α2-adrenoceptor blockade in the asenapine-induced elevation of prefrontal cortical monoamine outflow.
Journal: Synapse (New York, N.Y.) 20120701
Title: Effects of the 5-HT2C receptor agonist Ro60-0175 and the 5-HT2A receptor antagonist M100907 on nicotine self-administration and reinstatement.
Journal: Neuropharmacology 20120601
Title: Sustained recreational use of ecstasy is associated with altered pre and postsynaptic markers of serotonin transmission in neocortical areas: a PET study with [¹¹C]DASB and [¹¹C]MDL 100907.
Journal: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20120501
Title: Effects of the selective 5-HT(7) receptor antagonist SB-269970 in animal models of psychosis and cognition.
Journal: Behavioural brain research 20120301
Title: The neuropharmacology of prolactin secretion elicited by 3,4-methylenedioxymethamphetamine ('ecstasy'): a concurrent microdialysis and plasma analysis study.
Journal: Hormones and behavior 20120201
Title: 5-HT2A receptor antagonist M100907 reduces serotonin synthesis: an autoradiographic study.
Journal: Brain research bulletin 20120104
Title: Extended characterisation of the serotonin 2A (5-HT2A) receptor-selective PET radiotracer 11C-MDL100907 in humans: quantitative analysis, test-retest reproducibility, and vulnerability to endogenous 5-HT tone.
Journal: NeuroImage 20120102
Title: Dorsal-striatal 5-HT₂A and 5-HT₂C receptors control impulsivity and perseverative responding in the 5-choice serial reaction time task.
Journal: Psychopharmacology 20120101
Title: The 5-HT(2A) receptor and serotonin transporter in Asperger's disorder: A PET study with [¹¹C]MDL 100907 and [¹¹C]DASB.
Journal: Psychiatry research 20111230
Title: Serotonin 2A receptors in obsessive-compulsive disorder: a positron emission tomography study with [11C]MDL 100907.
Journal: Biological psychiatry 20111101
Title: p-Hydroxyamphetamine causes prepulse inhibition disruption in mice: contribution of serotonin neurotransmission.
Journal: Behavioural brain research 20111010
Title: Pimavanserin, a 5-HT2A inverse agonist, reverses psychosis-like behaviors in a rodent model of Parkinson's disease.
Journal: Behavioural pharmacology 20111001
Title: Impulsive action induced by amphetamine, cocaine and MK801 is reduced by 5-HT(2C) receptor stimulation and 5-HT(2A) receptor blockade.
Journal: Neuropharmacology 20110901
Title: Serotonin 2A receptor antagonists for treatment of schizophrenia.
Journal: Expert opinion on investigational drugs 20110901
Title: Serotonin control of sleep-wake behavior.
Journal: Sleep medicine reviews 20110801
Title: Effects of 5-HT(2A) and 5-HT(2C) receptor antagonists on acute and chronic dyskinetic effects induced by haloperidol in rats.
Journal: Behavioural brain research 20110601
Title: Serotonin (5-hydroxytryptamine) 5-HT(2A) receptor: association with inherent and cocaine-evoked behavioral disinhibition in rats.
Journal: Behavioural pharmacology 20110601
Title: Effects of direct- and indirect-acting serotonin receptor agonists on the antinociceptive and discriminative stimulus effects of morphine in rhesus monkeys.
Journal: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20110401
Title: Blockade of nucleus accumbens 5-HT2A and 5-HT2C receptors prevents the expression of cocaine-induced behavioral and neurochemical sensitization in rats.
Journal: Psychopharmacology 20110201
Title: Blockade of 5-HT2A receptors in the medial prefrontal cortex attenuates reinstatement of cue-elicited cocaine-seeking behavior in rats.
Journal: Psychopharmacology 20110201
Title: P-glycoprotein influence on the brain uptake of a 5-HT(2A) ligand: [(18)F]MH.MZ.
Journal: Neuropsychobiology 20110101
Title: Possible involvement of serotonin 5-HT2 receptor in the regulation of feeding behavior through the histaminergic system.
Journal: Neuropharmacology 20110101
Title: Interaction of 5-HT2A and 5-HT2C receptors in R(-)-2,5-dimethoxy-4-iodoamphetamine-elicited head twitch behavior in mice.
Journal: The Journal of pharmacology and experimental therapeutics 20101201
Title: Novel spirotetracyclic zwitterionic dual H(1)/5-HT(2A) receptor antagonists for the treatment of sleep disorders.
Journal: Journal of medicinal chemistry 20101111
Title: The alpha2 adrenergic receptor antagonist idazoxan, but not the serotonin-2A receptor antagonist M100907, partially attenuated reward deficits associated with nicotine, but not amphetamine, withdrawal in rats.
Journal: European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology 20101001
Title: Structural combination of established 5-HT(2A) receptor ligands: new aspects of the binding mode.
Journal: Chemical biology & drug design 20101001
Title: Differential effects of serotonin (5-HT)2 receptor-targeting ligands on locomotor responses to nicotine-repeated treatment.
Journal: Synapse (New York, N.Y.) 20100701
Title: Synergistic effect of decreased opioid activity and sleep deprivation on head-twitch response in mice.
Journal: Pharmacology, biochemistry, and behavior 20100701
Title: Increased serotonin 2A receptor availability in the orbitofrontal cortex of physically aggressive personality disordered patients.
Journal: Biological psychiatry 20100615
Title: Non-basic ligands for aminergic GPCRs: the discovery and development diaryl sulfones as selective, orally bioavailable 5-HT2A receptor antagonists for the treatment of sleep disorders.
Journal: Bioorganic & medicinal chemistry letters 20100615
Title: CRF receptor 1 regulates anxiety behavior via sensitization of 5-HT2 receptor signaling.
Journal: Nature neuroscience 20100501
Title: 18F-labeling and evaluation of novel MDL 100907 derivatives as potential 5-HT2A antagonists for molecular imaging.
Journal: Nuclear medicine and biology 20100501
Title: Simplified quantification of 5-HT2A receptors in the human brain with [11C]MDL 100,907 PET and non-invasive kinetic analyses.
Journal: NeuroImage 20100415
Title: Antagonism at serotonin 5-HT(2A) receptors modulates functional activity of frontohippocampal circuit.
Journal: Psychopharmacology 20100301
Title: Attenuation of phencyclidine-induced object recognition deficits by the combination of atypical antipsychotic drugs and pimavanserin (ACP 103), a 5-hydroxytryptamine(2A) receptor inverse agonist.
Journal: The Journal of pharmacology and experimental therapeutics 20100201
Title: Blockade of serotonin 2A receptors prevents PCP-induced attentional performance deficit and CREB phosphorylation in the dorsal striatum of DBA/2 mice.
Journal: Psychopharmacology 20100201
Title: Enhancement of spatial reversal learning by 5-HT2C receptor antagonism is neuroanatomically specific.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience 20100120
Title: Sertindole improves sub-chronic PCP-induced reversal learning and episodic memory deficits in rodents: involvement of 5-HT(6) and 5-HT (2A) receptor mechanisms.
Journal: Psychopharmacology 20100101
Title: 5-HT2A receptor antagonists improve motor impairments in the MPTP mouse model of Parkinson's disease.
Journal: Neuropharmacology 20100101
Title: Plaque deposition dependent decrease in 5-HT2A serotonin receptor in AbetaPPswe/PS1dE9 amyloid overexpressing mice.
Journal: Journal of Alzheimer's disease : JAD 20100101
Title: Discriminative stimulus effects of 1-(2,5-dimethoxy-4-methylphenyl)-2-aminopropane (DOM), ketanserin, and (R)-(+)-{alpha}-(2,3-dimethoxyphenyl)-1-[2-(4-fluorophenyl)ethyl]-4-pipidinemethanol (MDL100907) in rats.
Journal: The Journal of pharmacology and experimental therapeutics 20091101
Title: Combined administration of an mGlu2/3 receptor agonist and a 5-HT 2A receptor antagonist markedly attenuate the psychomotor-activating and neurochemical effects of psychostimulants.
Journal: Psychopharmacology 20091101
Title: Enhanced 5-HT(2A) receptors in brain stem and ALDH activity in brain stem and liver: 5-HT(2A) regulation on ALDH in primary hepatocytes cultures in vitro.
Journal: Neurochemical research 20090901
Title: Effect of sertindole on extracellular dopamine, acetylcholine, and glutamate in the medial prefrontal cortex of conscious rats: a comparison with risperidone and exploration of mechanisms involved.
Journal: Psychopharmacology 20090901
Title: Serotonergic hyperinnervation and effective serotonin blockade in an FGF receptor developmental model of psychosis.
Journal: Schizophrenia research 20090901
Title: Interactions of serotonin (5-HT)2 receptor-targeting ligands and nicotine: locomotor activity studies in rats.
Journal: Synapse (New York, N.Y.) 20090801
Title: Role of dopamine transporters in the behavioral effects of 3,4-methylenedioxymethamphetamine (MDMA) in nonhuman primates.
Journal: Psychopharmacology 20090801
Title: Side chain flexibilities in the human ether-a-go-go related gene potassium channel (hERG) together with matched-pair binding studies suggest a new binding mode for channel blockers.
Journal: Journal of medicinal chemistry 20090723
Title: Relevance of dorsal raphe nucleus firing in serotonin 5-HT(2C) receptor blockade-induced augmentation of SSRIs effects.
Journal: Neuropharmacology 20090701
Title: Activation of glucocorticoid receptors increases 5-HT2A receptor levels.
Journal: Experimental neurology 20090701
Title: Activation of the JAK-STAT pathway is necessary for desensitization of 5-HT2A receptor-stimulated phospholipase C signalling by olanzapine, clozapine and MDL 100907.
Journal: The international journal of neuropsychopharmacology 20090601
Title: The brain 5-HT4 receptor binding is down-regulated in the Flinders Sensitive Line depression model and in response to paroxetine administration.
Journal: Journal of neurochemistry 20090601
Title: Simultaneous telemetric monitoring of tail-skin and core body temperature in a rat model of thermoregulatory dysfunction.
Journal: Journal of neuroscience methods 20090415
Title: Synthesis and in vitro affinities of various MDL 100907 derivatives as potential 18F-radioligands for 5-HT2A receptor imaging with PET.
Journal: Bioorganic & medicinal chemistry 20090415
Title: Genetic deletion of MAO-A promotes serotonin-dependent ventricular hypertrophy by pressure overload.
Journal: Journal of molecular and cellular cardiology 20090401
Title: Blockade of the serotonin 5-HT2A receptor suppresses cue-evoked reinstatement of cocaine-seeking behavior in a rat self-administration model.
Journal: Behavioral neuroscience 20090401
Title: Discriminative stimulus effects of 1-(2,5-dimethoxy-4-methylphenyl)-2-aminopropane in rhesus monkeys: antagonism and apparent pA2 analyses.
Journal: The Journal of pharmacology and experimental therapeutics 20090301
Title: Pharmacological properties and discriminative stimulus effects of a novel and selective 5-HT2 receptor agonist AL-38022A [(S)-2-(8,9-dihydro-7H-pyrano[2,3-g]indazol-1-yl)-1-methylethylamine].
Journal: Pharmacology, biochemistry, and behavior 20090101
Title: Endogenous serotonin and serotonin2C receptors are involved in the ability of M100907 to suppress cortical glutamate release induced by NMDA receptor blockade.
Journal: Journal of neurochemistry 20090101
Title: Fluoxetine-mediated 5-HT2B receptor stimulation in astrocytes causes EGF receptor transactivation and ERK phosphorylation.
Journal: Psychopharmacology 20081201
Title: The 5-hydroxytryptamine2A receptor antagonist R-(+)-alpha-(2,3-dimethoxyphenyl)-1-[2-(4-fluorophenyl)ethyl-4-piperidinemethanol (M100907) attenuates impulsivity after both drug-induced disruption (dizocilpine) and enhancement (antidepressant drugs) of differential-reinforcement-of-low-rate 72-s behavior in the rat.
Journal: The Journal of pharmacology and experimental therapeutics 20081201
Title: Validation of a rat in vivo [(3)H]M100907 binding assay to determine a translatable measure of 5-HT(2A) receptor occupancy.
Journal: European journal of pharmacology 20080904
Title: Opposing roles for 5-HT2A and 5-HT2C receptors in the nucleus accumbens on inhibitory response control in the 5-choice serial reaction time task.
Journal: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20080901
Title: The hallucinogen DOI reduces low-frequency oscillations in rat prefrontal cortex: reversal by antipsychotic drugs.
Journal: Biological psychiatry 20080901
Title: Chronic phenethylamine hallucinogen treatment alters behavioral sensitivity to a metabotropic glutamate 2/3 receptor agonist.
Journal: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20080801
Title: Dissociable effects of selective 5-HT2A and 5-HT2C receptor antagonists on serial spatial reversal learning in rats.
Journal: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20080701
Title: Lorcaserin, a novel selective human 5-hydroxytryptamine2C agonist: in vitro and in vivo pharmacological characterization.
Journal: The Journal of pharmacology and experimental therapeutics 20080501
Title: Evidence that genetic variation in 5-HT transporter expression is linked to changes in 5-HT2A receptor function.
Journal: Neuropharmacology 20080401
Title: 2-Alkyl-4-aryl-pyrimidine fused heterocycles as selective 5-HT2A antagonists.
Journal: Bioorganic & medicinal chemistry letters 20080315
Title: Total synthesis and evaluation of [18F]MHMZ.
Journal: Bioorganic & medicinal chemistry letters 20080215
Title: Abnormally persistent latent inhibition induced by MK801 is reversed by risperidone and by positive modulators of NMDA receptor function: differential efficacy depending on the stage of the task at which they are administered.
Journal: Psychopharmacology 20080201
Title: In vivo pharmacology of MDMA and its enantiomers in rhesus monkeys.
Journal: Experimental and clinical psychopharmacology 20080201
Title: Hallucinogen-like effects of N,N-dipropyltryptamine (DPT): possible mediation by serotonin 5-HT1A and 5-HT2A receptors in rodents.
Journal: Pharmacology, biochemistry, and behavior 20080101
Title: The stimulus effects of 8-OH-DPAT: evidence for a 5-HT2A receptor-mediated component.
Journal: Pharmacology, biochemistry, and behavior 20080101
Title: Selective 5HT2A and 5HT6 receptor antagonists promote sleep in rats.
Journal: Sleep 20080101
Title: Effects of 5-HT drugs in prefrontal cortex during memory formation and the ketamine amnesia-model.
Journal: Hippocampus 20080101
Title: 5-HT(2A) inverse-agonists for the treatment of insomnia.
Journal: Current topics in medicinal chemistry 20080101
Title: Opposing effects of 5-HT(2A) and 5-HT(2C) receptor antagonists in the rat and mouse on premature responding in the five-choice serial reaction time test.
Journal: Psychopharmacology 20071201
Title: Behavioral response to emotional stress in rabbits: role of serotonin and serotonin2A receptors.
Journal: Behavioural pharmacology 20071101
Title: Effects of the serotonin 5-HT2A and 5-HT2C receptor ligands on the discriminative stimulus effects of nicotine in rats.
Journal: European journal of pharmacology 20071001
Title: Hippocampal Bcl-2 expression is selectively increased following chronic but not acute treatment with antidepressants, 5-HT(1A) or 5-HT(2C/2B) receptor antagonists.
Journal: European journal of pharmacology 20070813
Title: Mechanical, thermal and formalin-induced nociception is differentially altered in 5-HT1A-/-, 5-HT1B-/-, 5-HT2A-/-, 5-HT3A-/- and 5-HTT-/- knock-out male mice.
Journal: Pain 20070801
Title: Behavioral effects of dipropyltryptamine in rats: evidence for 5-HT1A and 5-HT2A agonist activity.
Journal: Behavioural pharmacology 20070701
Title: Blockade of 5-HT2a receptors reduces haloperidol-induced attenuation of reward.
Journal: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20070301
Title: 5-Hydroxytryptamine (serotonin)2A receptors in rat anterior cingulate cortex mediate the discriminative stimulus properties of d-lysergic acid diethylamide.
Journal: The Journal of pharmacology and experimental therapeutics 20070201
Title: Validation of a tracer kinetic model for the quantification of 5-HT(2A) receptors in human brain with [(11)C]MDL 100,907.
Journal: Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism 20070101
Title: Effects of d-amphetamine and DOI (2,5-dimethoxy-4-iodoamphetamine) on timing behavior: interaction between D1 and 5-HT2A receptors.
Journal: Psychopharmacology 20061201
Title: Cardiac baroreflex facilitation evoked by hypothalamus and prefrontal cortex stimulation: role of the nucleus tractus solitarius 5-HT2A receptors.
Journal: American journal of physiology. Regulatory, integrative and comparative physiology 20061001
Title: Increased 5-HT(2A) receptor binding in euthymic, medication-free patients recovered from depression: a positron emission study with [(11)C]MDL 100,907.
Journal: The American journal of psychiatry 20060901
Title: Serotonin 2A receptor antagonist treatment reduces dopamine D1 receptor-mediated rotational behavior but not L-DOPA-induced abnormal involuntary movements in the unilateral dopamine-depleted rat.
Journal: Neuropharmacology 20060501
Title: Dissociable contribution of 5-HT1A and 5-HT2A receptors in the medial prefrontal cortex to different aspects of executive control such as impulsivity and compulsive perseveration in rats.
Journal: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20060401
Title: Effects of 5-HT2A receptor stimulation on the discrimination of durations by rats.
Journal: Behavioural pharmacology 20060201
Title: Hallucinogen-like actions of 5-methoxy-N,N-diisopropyltryptamine in mice and rats.
Journal: Pharmacology, biochemistry, and behavior 20060101
Title: Binding characteristics of the 5-HT2A receptor antagonists altanserin and MDL 100907.
Journal: Synapse (New York, N.Y.) 20051215
Title: Use of LC/MS to assess brain tracer distribution in preclinical, in vivo receptor occupancy studies: dopamine D2, serotonin 2A and NK-1 receptors as examples.
Journal: Life sciences 20051212
Title: The selective 5-HT2A receptor antagonist M100907 enhances antidepressant-like behavioral effects of the SSRI fluoxetine.
Journal: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20051201
Title: Relationship of cocaine-induced c-Fos expression to behaviors and the role of serotonin 5-HT2A receptors in cocaine-induced c-Fos expression.
Journal: Behavioral neuroscience 20051001
Title: The role of 5-HT(2A) receptor antagonism in amphetamine-induced inhibition of A10 dopamine neurons in vitro.
Journal: European journal of pharmacology 20050927
Title: Behavioral tolerance to lysergic acid diethylamide is associated with reduced serotonin-2A receptor signaling in rat cortex.
Journal: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20050901
Title: Serotonin 5-HT2A but not 5-HT2C receptor antagonism reduces hyperlocomotor activity induced in dopamine-depleted rats by striatal administration of the D1 agonist SKF 82958.
Journal: Neuropharmacology 20050901
Title: Serotonergic regulation of calcium-activated potassium currents in rodent prefrontal cortex.
Journal: The European journal of neuroscience 20050901
Title: 4-Fluorosulfonylpiperidines: selective 5-HT2A ligands for the treatment of insomnia.
Journal: Bioorganic & medicinal chemistry letters 20050815
Title: The stimulus properties of LSD in C57BL/6 mice.
Journal: Pharmacology, biochemistry, and behavior 20050801
Title: Lithium differs from anticonvulsant mood stabilizers in prefrontal cortical and accumbal dopamine release: role of 5-HT(1A) receptor agonism.
Journal: Brain research 20050712
Title: Distinct temporal phases in the behavioral pharmacology of LSD: dopamine D2 receptor-mediated effects in the rat and implications for psychosis.
Journal: Psychopharmacology 20050701
Title: A role for midbrain raphe gamma aminobutyric acid neurons in 5-hydroxytryptamine feedback control.
Journal: Neuroreport 20050621
Title: Complex discriminative stimulus properties of (+)lysergic acid diethylamide (LSD) in C57Bl/6J mice.
Journal: Psychopharmacology 20050601
Title: Role of the serotonin 5-HT2A receptor in the hyperlocomotive and hyperthermic effects of (+)-3,4-methylenedioxymethamphetamine.
Journal: Psychopharmacology 20050401
Title: Serotonin 2A receptors modulate tail-skin temperature in two rodent models of estrogen deficiency-related thermoregulatory dysfunction.
Journal: Brain research 20041203
Title: 5-HT2A and 5-HT2C receptor antagonists have opposing effects on a measure of impulsivity: interactions with global 5-HT depletion.
Journal: Psychopharmacology 20041101
Title: The 5-HT receptor antagonist M100,907 prevents extracellular glutamate rising in response to NMDA receptor blockade in the mPFC.
Journal: Journal of neurochemistry 20041001
Title: Cutting edge: serotonin is a chemotactic factor for eosinophils and functions additively with eotaxin.
Journal: Journal of immunology (Baltimore, Md. : 1950) 20040915
Title: The serotonin 5-HT2A receptors antagonist M100907 prevents impairment in attentional performance by NMDA receptor blockade in the rat prefrontal cortex.
Journal: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20040901
Title: Pharmacological characterisation of the agonist radioligand binding site of 5-HT(2A), 5-HT(2B) and 5-HT(2C) receptors.
Journal: Naunyn-Schmiedeberg's archives of pharmacology 20040801
Title: Desensitization of 5-HT1A receptors by 5-HT2A receptors in neuroendocrine neurons in vivo.
Journal: The Journal of pharmacology and experimental therapeutics 20040701
Title: Nantenine: an antagonist of the behavioral and physiological effects of MDMA in mice.
Journal: Psychopharmacology 20040501
Title: Serotonergic facilitation of synaptic activity in the developing rat prefrontal cortex.
Journal: The Journal of physiology 20040501
Title: The selective serotonin-2A receptor antagonist M100907 reverses behavioral deficits in dopamine transporter knockout mice.
Journal: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20040201
Title: Discriminative stimulus properties of 1.25 and 5.0 mg/kg doses of clozapine in rats: examination of the role of dopamine, serotonin, and muscarinic receptor mechanisms.
Journal: Pharmacology, biochemistry, and behavior 20040201
Title: Fenfluramine evokes 5-HT2A receptor-mediated responses but does not displace [11C]MDL 100907: small animal PET and gene expression studies.
Journal: Synapse (New York, N.Y.) 20031201
Title: The 5-HT2A receptor antagonist M100,907 attenuates motor and 'impulsive-type' behaviours produced by NMDA receptor antagonism.
Journal: Psychopharmacology 20031101
Title: Pharmacological characterization of a serotonin receptor (5-HT7) stimulating cAMP production in human corneal epithelial cells.
Journal: Investigative ophthalmology & visual science 20031101
Title: Group II metabotropic glutamate receptor antagonists LY341495 and LY366457 increase locomotor activity in mice.
Journal: Neuropharmacology 20031001
Title: Latent inhibition in 35-day-old rats is not an 'adult' latent inhibition: implications for neurodevelopmental models of schizophrenia.
Journal: Psychopharmacology 20030901
Title: In vivo modulation of 5-hydroxytryptamine release in mouse prefrontal cortex by local 5-HT(2A) receptors: effect of antipsychotic drugs.
Journal: The European journal of neuroscience 20030901
Title: The hallucinogen 1-[2,5-dimethoxy-4-iodophenyl]-2-aminopropane (DOI) increases cortical extracellular glutamate levels in rats.
Journal: Neuroscience letters 20030807
Title: Regulation of septo-hippocampal activity by 5-hydroxytryptamine(2C) receptors.
Journal: The Journal of pharmacology and experimental therapeutics 20030801
Title: Evaluation of the ocular hypotensive response of serotonin 5-HT1A and 5-HT2 receptor ligands in conscious ocular hypertensive cynomolgus monkeys.
Journal: The Journal of pharmacology and experimental therapeutics 20030701
Title: 5-HT 2A receptor stimulation by DOI, a 5-HT 2A/2C receptor agonist, potentiates amphetamine-induced dopamine release in rat medial prefrontal cortex and nucleus accumbens.
Journal: Brain research 20030516
Title: Intra-prefrontal 8-OH-DPAT and M100907 improve visuospatial attention and decrease impulsivity on the five-choice serial reaction time task in rats.
Journal: Psychopharmacology 20030501
Title: Generalization of clozapine as compared to other antipsychotic agents to a discriminative stimulus elicited by the serotonin (5-HT)2A antagonist, MDL100,907.
Journal: Neuropharmacology 20030401
Title: Discriminative stimulus properties of (+/-)-fenfluramine: the role of 5-HT2 receptor subtypes.
Journal: Behavioral neuroscience 20030401
Title: Pharmacological characterization of the effects of 3,4-methylenedioxymethamphetamine ('ecstasy') and its enantiomers on lethality, core temperature, and locomotor activity in singly housed and crowded mice.
Journal: Psychopharmacology 20030301
Title: Neuroendocrine evidence that (S)-2-(chloro-5-fluoro-indol- l-yl)-1-methylethylamine fumarate (Ro 60-0175) is not a selective 5-hydroxytryptamine(2C) receptor agonist.
Journal: The Journal of pharmacology and experimental therapeutics 20030301
Title: Discriminative stimulus properties of 1-(2,5-dimethoxy-4-iodophenyl)-2-aminopropane [(+/-)DOI] in C57BL/6J mice.
Journal: Psychopharmacology 20030201
Title: Protein kinase C is involved in clozapine's facilitation of N-methyl-D-aspartate- and electrically evoked responses in pyramidal cells of the medial prefrontal cortex.
Journal: Neuroscience 20030101
Title: Serotonin mechanisms in heart valve disease II: the 5-HT2 receptor and its signaling pathway in aortic valve interstitial cells.
Journal: The American journal of pathology 20021201
Title: Evidence that 5-HT2A receptors in the hypothalamic paraventricular nucleus mediate neuroendocrine responses to (-)DOI.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience 20021101
Title: Differential effects of the 5-HT(2A) receptor antagonist M100907 and the 5-HT(2C) receptor antagonist SB242084 on cocaine-induced locomotor activity, cocaine self-administration and cocaine-induced reinstatement of responding.
Journal: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20021001
Title: SR46349-B, a 5-HT(2A/2C) receptor antagonist, potentiates haloperidol-induced dopamine release in rat medial prefrontal cortex and nucleus accumbens.
Journal: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20020901
Title: 5-HT(2A) receptor antagonism potentiates haloperidol-induced dopamine release in rat medial prefrontal cortex and inhibits that in the nucleus accumbens in a dose-dependent manner.
Journal: Brain research 20020830
Title: 5-HT(1A) and 5-HT(2A) receptors minimally contribute to clozapine-induced acetylcholine release in rat medial prefrontal cortex.
Journal: Brain research 20020607
Title: Synthesis, receptor potency, and selectivity of halogenated diphenylpiperidines as serotonin 5-HT2A ligands for PET or SPECT brain imaging.
Journal: Journal of medicinal chemistry 20020523
Title: The selective serotonin(2A) receptor antagonist, MDL100,907, elicits a specific interoceptive cue in rats.
Journal: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20020401
Title: Attenuation of ischemic efflux of endogenous amino acids by the novel 5-HT(1A)/5-HT(2) receptor ligand adatanserin.
Journal: Neurochemistry international 20020301
Title: Comparison of the potency of MDL 100,907 and SB 242084 in blocking the serotonin (5-HT)(2) receptor agonist-induced increases in rat serum corticosterone concentrations: evidence for 5-HT(2A) receptor mediation of the HPA axis.
Journal: Neuropharmacology 20020201
Title: 4-(Phenylsulfonyl)piperidines: novel, selective, and bioavailable 5-HT(2A) receptor antagonists.
Journal: Journal of medicinal chemistry 20020117
Title: Pharmacological studies of the acute effects of (+)-3,4-methylenedioxymethamphetamine on locomotor activity: role of 5-HT(1B/1D) and 5-HT(2) receptors.
Journal: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20020101
Title: Effects of phencyclidine (PCP) and MK 801 on the EEGq in the prefrontal cortex of conscious rats; antagonism by clozapine, and antagonists of AMPA-, alpha(1)- and 5-HT(2A)-receptors.
Journal: British journal of pharmacology 20020101
Title: Control of serotonergic function in medial prefrontal cortex by serotonin-2A receptors through a glutamate-dependent mechanism.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience 20011215
Title: Functional and pharmacological characterization of the modulatory role of serotonin on the firing activity of locus coeruleus norepinephrine neurons.
Journal: Brain research 20011213
Title: m-CPP hypolocomotion is selectively antagonized by compounds with high affinity for 5-HT(2C) receptors but not 5-HT(2A) or 5-HT(2B) receptors.
Journal: Behavioural pharmacology 20011201
Title: Effect of clozapine, haloperidol, or M100907 on phencyclidine-activated glutamate efflux in the prefrontal cortex.
Journal: Biological psychiatry 20011115
Title: Characterization of the functional heterologous desensitization of hypothalamic 5-HT(1A) receptors after 5-HT(2A) receptor activation.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience 20011015
Title: Multiple conformations of native and recombinant human 5-hydroxytryptamine(2a) receptors are labeled by agonists and discriminated by antagonists.
Journal: Molecular pharmacology 20011001
Title: Differential regulation of the mesoaccumbens circuit by serotonin 5-hydroxytryptamine (5-HT)2A and 5-HT2C receptors.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience 20011001
Title: DOI, a 5-HT2A/2C receptor agonist, attenuates clozapine-induced cortical dopamine release.
Journal: Brain research 20010713
Title: 5-HT2A receptors stimulate ACTH, corticosterone, oxytocin, renin, and prolactin release and activate hypothalamic CRF and oxytocin-expressing cells.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience 20010515
Title: Acute and repeated administration of the selective 5-HT(2A) receptor antagonist M100907 significantly alters the activity of midbrain dopamine neurons: an in vivo electrophysiological study.
Journal: Synapse (New York, N.Y.) 20010501
Title: M100907, a selective 5-HT(2A) receptor antagonist, attenuates phencyclidine-induced Fos expression in discrete regions of rat brain.
Journal: European journal of pharmacology 20010413
Title: Antagonism of 5-hydroxytryptamine(2a) receptors attenuates the behavioral effects of cocaine in rats.
Journal: The Journal of pharmacology and experimental therapeutics 20010401
Title: [Synthesis and biological activities of new 5-HT2A selective ligands--N-substituted-piperidinyl-4-phenylthioether and sulfone derivatives].
Journal: Yao xue xue bao = Acta pharmaceutica Sinica 20010401
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