Title: Zhou B, et al. Discovery of a Small-Molecule Degrader of Bromodomain and Extra-Terminal (BET) Proteins withPicomolar Cellular Potencies and Capable of Achieving Tumor Regression. J Med Chem. 2017 Mar 24.
Title: James Bradner, et al. Methods to induce targeted protein degradation through bifunctional molecules. WO 2017024317 A2.