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Title: Impaired complement-mediated phagocytosis by HIV type-1-infected human monocyte-derived macrophages involves a cAMP-dependent mechanism.
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Title: Microsphere-based protease assays and screening application for lethal factor and factor Xa.
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Title: Phosphorylation of paracellin-1 at Ser217 by protein kinase A is essential for localization in tight junctions.
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Title: 2'-deoxy-4'-C-ethynyl-2-fluoroadenosine, a nucleoside reverse transcriptase inhibitor, is highly potent against all human immunodeficiency viruses type 1 and has low toxicity.
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Title: Influence of dipeptidyl peptidase IV on enzymatic properties of adenosine deaminase.
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Title: Enhancement of cellular adenosine triphosphate levels in PC12 cells by 2,5-dideoxyadenosine, a P-site inhibitor of adenylate cyclase.
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Title: Mechanisms of action of angiotensin II on mammalian sperm function.
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Title: Nicotine and epibatidine triggered prolonged rise in calcium and TH gene transcription in PC12 cells.
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Title: Effects of primer-template sequence on ATP-dependent removal of chain-terminating nucleotide analogues by HIV-1 reverse transcriptase.
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Title: Glucagon-like peptide-2: divergent signaling pathways.
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Title: Human chorionic gonadotropin decreases proliferation and invasion of breast cancer MCF-7 cells by inhibiting NF-kappaB and AP-1 activation.
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Title: PGE2 induces IL-1beta gene expression in mouse osteoblasts through a cAMP-PKA signaling pathway.
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Title: Enhanced inhibition of the EDHF phenomenon by a phenyl methoxyalaninyl phosphoramidate derivative of dideoxyadenosine.
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Title: Atrial natriuretic peptide-C receptor-induced attenuation of adenylyl cyclase signaling activates phosphatidylinositol turnover in A10 vascular smooth muscle cells.
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Title: Synthesis of 2',5'-dideoxy-2-fluoroadenosine and 2',5'-dideoxy-2,5'-difluoroadenosine: potent P-site inhibitors of adenylyl cyclase.
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Title: Determination of carrier-mediated transport of 2',3'-dideoxypurine nucleosides in the rat ileum using a bidirectional perfusion technique.
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Title: Structure of the N-terminal domain of GRP94. Basis for ligand specificity and regulation.
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Title: Evidence for multiple distinctly localized adenylyl cyclase isoforms in mammalian spermatozoa.
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Title: Phosphoramidate protides of 2',3'-dideoxy-3'-fluoroadenosine and related nucleosides with potent activity against HIV and HBV.
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Title: Anti-HIV-1 activity of 3-deaza-adenosine analogs. Inhibition of S-adenosylhomocysteine hydrolase and nucleotide congeners.
Journal: European journal of biochemistry 20030901
Title: Decreased adenylyl cyclase and cAMP-dependent protein kinase activities inhibit the cytotoxic function of human natural killer cells.
Journal: Human immunology 20030901
Title: Inhibition of hepatitis B virus by a novel L-nucleoside, beta-L-D4A and related analogues.
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Title: A strategy for liquid chromatography/tandem mass spectrometric assays of intracellular drugs: application to the validation of the triphosphorylated anabolite of antiretrovirals in peripheral blood mononuclear cells.
Journal: Journal of mass spectrometry : JMS 20030801
Title: [Inhibition of the replication of hepatitis B virus in vitro by a novel nucleoside analogue (beta-L-D4A)].
Journal: Zhonghua gan zang bing za zhi = Zhonghua ganzangbing zazhi = Chinese journal of hepatology 20030701
Title: HPLC and mass spectrometry analysis of the enzymatic hydrolysis of anti-HIV pronucleotide diastereomers.
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Title: [Effect and mechanism of beta-L-D4A (a novel nucleoside analog) against hepatitis B virus].
Journal: Zhonghua gan zang bing za zhi = Zhonghua ganzangbing zazhi = Chinese journal of hepatology 20030501
Title: Cyclopropyl and related analogs of the anti-HIV compound, isodideoxyadenosine.
Journal: Nucleosides, nucleotides & nucleic acids 20030301
Title: Exposure-disease continuum for 2-chloro-2'-deoxyadenosine, a prototype ocular teratogen. 3. Intervention with PK11195.
Journal: Birth defects research. Part A, Clinical and molecular teratology 20030201
Title: A selective role for phosphatidylinositol 3,4,5-trisphosphate in the Gi-dependent activation of platelet Rap1B.
Journal: The Journal of biological chemistry 20030103
Title: Components of the intracellular cAMP system supporting the olfactory reception of amyl alcohol.
Journal: Neuroscience and behavioral physiology 20030101
Title: An industrial process for synthesizing Lodenosine (FddA).
Journal: Nucleosides, nucleotides & nucleic acids 20030101
Title: A facile synthetic method for 3'-alpha-fluoro-2',3'-dideoxyadenosine.
Journal: Nucleosides, nucleotides & nucleic acids 20030101
Title: Synthesis and studies of 3'-C-trifluoromethyl nucleoside analogues bearing adenine or cytosine as the base.
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Title: Synthesis and biological evaluation of endocyclic 2',3'-didehydro-2',3'-dideoxymethanocarba adenosine.
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Title: Adenine and deazaadenine nucleoside and deoxynucleoside analogues: inhibition of viral replication of sheep MVV (in vitro model for HIV) and bovine BHV-1.
Journal: Bioorganic & medicinal chemistry 20020901
Title: Synthesis, conformational analysis and antiviral and antitumoral activity of new 1,2-disubstituted carbocyclic nucleosides.
Journal: European journal of medicinal chemistry 20020901
Title: Specificity of human and rat orthologs of the concentrative nucleoside transporter, SPNT.
Journal: American journal of physiology. Renal physiology 20020801
Title: PGE(2) increases release of substance P from renal sensory nerves by activating the cAMP-PKA transduction cascade.
Journal: American journal of physiology. Regulatory, integrative and comparative physiology 20020601
Title: Roles for both cyclic GMP and cyclic AMP in the inhibition of collagen-induced platelet aggregation by nitroprusside.
Journal: British journal of haematology 20020601
Title: Extracellular superoxide dismutase and glomerular mesangial cells: its production and regulation.
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Title: Cyclosporine inhibition of vascular endothelial growth factor production in rheumatoid synovial fibroblasts.
Journal: Arthritis and rheumatism 20020501
Title: Peptides interact in gonadotrophin regulation.
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Title: Interactions of diol dehydrase and 3',4'-anhydroadenosylcobalamin: suicide inactivation by electron transfer.
Journal: Biochemistry 20020205
Title: mAChRs in the grasshopper brain mediate excitation by activation of the AC/PKA and the PLC second-messenger pathways.
Journal: Journal of neurophysiology 20020201
Title: Modulation by 5-hydroxytryptamine of nicotinic acetylcholine responses recorded from an identified cockroach (Periplaneta americana) motoneuron.
Journal: The European journal of neuroscience 20020201
Title: Cyclosporine differentially regulates interleukin-10, interleukin-15, and tumor necrosis factor a production by rheumatoid synoviocytes.
Journal: Arthritis and rheumatism 20020101
Title: Synthesis of novel 8-substituted carbocyclic analogs of 2',3'-dideoxyadenosine with activity against hepatitis B virus.
Journal: Nucleosides, nucleotides & nucleic acids 20020101
Title: Rapid and non-genomic reduction of intracellular [Ca(2+)] induced by aldosterone in human bronchial epithelium.
Journal: The Journal of physiology 20011115
Title: Synthesis of 9-(2,3-dideoxy-2-fluoro-beta-D-threo-pentofuranosyl)adenine (FddA) via a purine 3'-deoxynucleoside.
Journal: The Journal of organic chemistry 20011102
Title: Stereoselective synthesis of a novel carbocyclic nucleoside.
Journal: The Journal of organic chemistry 20011102
Title: The cAMP-mediated protein kinase signal transduction pathway is involved in the pyrogenic effect of CRH in rats.
Journal: Chinese medical journal 20011001
Title: Differential effects of nucleoside analogs on oxidative phosphorylation in human pancreatic cells.
Journal: Digestive diseases and sciences 20010901
Title: Enhanced oral bioavailability of 2'- beta-fluoro-2',3'-dideoxyadenosine (F-ddA) through local inhibition of intestinal adenosine deaminase.
Journal: Pharmaceutical research 20010901
Title: Comparison of the antiviral activity of hydrophobic amino acid phosphoramidate monoesters of 2'3'-dideoxyadenosine (DDA) and 3'-azido-3'-deoxythymidine (AZT).
Journal: Nucleosides, nucleotides & nucleic acids 20010801
Title: Helicobacter pylori induces pepsinogen secretion by rat gastric cells in culture via a cAMP signal pathway.
Journal: International journal of molecular medicine 20010601
Title: Crystal structures of a ddATP-, ddTTP-, ddCTP, and ddGTP- trapped ternary complex of Klentaq1: insights into nucleotide incorporation and selectivity.
Journal: Protein science : a publication of the Protein Society 20010601
Title: High performance liquid chromatography analysis of 9-(2',3'-dideoxy-2'beta-fluoro-D-threo-penta furanosyl) adenine and its metabolite in human plasma using solid-phase extraction on a polyfluorinated reversed stationary phase.
Journal: Biomedical chromatography : BMC 20010601
Title: Evaluation of a fluorogenic derivatization method for the reversed-phase HPLC analysis of 2'-beta-fluoro-2',3'-dideoxyadenosine, a new anti-AIDS drug.
Journal: Journal of pharmaceutical and biomedical analysis 20010501
Title: Evaluation of the mutagenic and genotoxic activities of anti-hepatitis B analogs of beta-L-adenosine by the Ames test and the Comet assay.
Journal: Antiviral research 20010501
Title: cAMP-independent phosphorylation activation of CFTR by G proteins in native human sweat duct.
Journal: American journal of physiology. Cell physiology 20010301
Title: 3',5'-cyclic adenosine monophosphate regulates expression of synaptotagmin in neonatal sympathetic ganglia in vitro.
Journal: Journal of neurobiology 20010301
Title: The peptide TRH uncovers the presence of presynaptic 5-HT1A receptors via activation of a second messenger pathway in the rat dorsal vagal complex.
Journal: The Journal of physiology 20010301
Title: Antiviral activity and intracellular metabolism of bis(tButylSATE) phosphotriester of beta-L-2',3'dideoxyadenosine, a potent inhibitor of HIV and HBV replication.
Journal: Antiviral chemistry & chemotherapy 20010301
Title: Potentiation of thromboxane A2-induced platelet secretion by Gi signaling through the phosphoinositide-3 kinase pathway.
Journal: Thrombosis and haemostasis 20010201
Title: Fluorometric determination of 2'-beta-fluoro-2',3'-dideoxyadenosine 5'-triphosphate, the active metabolite of a new anti-human immunodeficiency virus drug, in human lymphocytes.
Journal: Analytical biochemistry 20010101
Title: Synthesis and in vitro antiviral activity evaluation of 9-(2-azido-2,3-dideoxy-beta-D-threo-pentofuranosyl)adenine derivatives.
Journal: Nucleosides, nucleotides & nucleic acids 20010101
Title: Synthesis and antiviral evaluation of 3'-C-trifluoromethyl nucleoside derivatives bearing adenine as the base.
Journal: Nucleosides, nucleotides & nucleic acids 20010101
Title: Anti-HIV activity of novel phosphonate derivatives of AZT, d4T, and ddA.
Journal: Nucleosides, nucleotides & nucleic acids 20010101
Title: Phosphorylation of the anti-HIV compound (S,S)-isodideoxyadenosine by human recombinant deoxycytidine kinase.
Journal: Biochemical pharmacology 20001115
Title: Correlation between intracellular pharmacological activation of nucleoside analogues and HIV suppression in vitro.
Journal: Antiviral chemistry & chemotherapy 20001101
Title: Interactions of conformationally biased north and south 2'-fluoro-2', 3'-dideoxynucleoside 5'-triphosphates with the active site of HIV-1 reverse transcriptase.
Journal: Biochemistry 20000919
Title: Intracellular metabolism of beta-L-2',3'-dideoxyadenosine: relevance to its limited antiviral activity.
Journal: Antimicrobial agents and chemotherapy 20000401
Title: Activities of masked 2',3'-dideoxynucleoside monophosphate derivatives against human immunodeficiency virus in resting macrophages.
Journal: Antimicrobial agents and chemotherapy 20000101
Title: cycloSal-Pronucleotides of 2',3'-dideoxyadenosine and 2', 3'-dideoxy-2',3'-didehydroadenosine: synthesis and antiviral evaluation of a highly efficient nucleotide delivery system.
Journal: Journal of medicinal chemistry 19990506
Title: cycloSal-Pronucleotides of 2'-fluoro-ara- and 2'-fluoro-ribo-2',3'- dideoxyadenosine as a strategy to bypass a metabolic blockade.
Journal: Journal of medicinal chemistry 19990506
Title: A new class of anti-HIV agents: synthesis and activity of conjugates of HIV protease inhibitors with a reverse transcriptase inhibitor.
Journal: Bioorganic & medicinal chemistry letters 19990322
Title: Effect of acyclic nucleoside phosphonates on the HIV-1 integrase in vitro.
Journal: Nucleosides & nucleotides 19990101
Title: CycloSal-2'-ara(ribo)-fluoro-2',3'-dideoxyadenosine monophosphates--an effort to solve the structure-activity relationship of 2'-fluoro-ddA.
Journal: Nucleosides & nucleotides 19990101
Title: Synthesis and biological activity of 2',5'-oligoadenylate trimers containing 5'-terminal 5'-amino-5'-deoxy- and 5'-amino-3',5'-dideoxyadenosine derivatives.
Journal: Nucleosides & nucleotides 19990101
Title: Conversion of 2',3'-dideoxyadenosine (ddA) and 2',3'-didehydro-2',3'-dideoxyadenosine (d4A) to their corresponding aryloxyphosphoramidate derivatives markedly potentiates their activity against human immunodeficiency virus and hepatitis B virus.
Journal: FEBS letters 19970630
Title: In vitro induction of human immunodeficiency virus type 1 variants resistant to 2'-beta-Fluoro-2',3'-dideoxyadenosine.
Journal: Antimicrobial agents and chemotherapy 19970601
Title: Decomposition pathways and in vitro HIV inhibitory effects of isoddA pronucleotides: toward a rational approach for intracellular delivery of nucleoside 5'-monophosphates.
Journal: Journal of medicinal chemistry 19960510
Title: Sensitization of C-fibres by prostaglandin E2 in the rat is inhibited by guanosine 5'-O-(2-thiodiphosphate), 2',5'-dideoxyadenosine and Walsh inhibitor peptide.
Journal: Neuroscience 19960301
Title: Selective pressure of a quinoxaline nonnucleoside inhibitor of human immunodeficiency virus type 1 (HIV-1) reverse transcriptase (RT) on HIV-1 replication results in the emergence of nucleoside RT-inhibitor-specific (RT Leu-74-->Val or Ile and Val-75-->Leu or Ile) HIV-1 mutants.
Journal: Proceedings of the National Academy of Sciences of the United States of America 19960109
Title: Synthesis and biological evaluation of N6-cycloalkyl derivatives of 1-deazaadenine nucleosides: a new class of anti-human immunodeficiency virus agents.
Journal: Journal of medicinal chemistry 19950929
Title: Enhancement by hydroxyurea of the anti-human immunodeficiency virus type 1 potency of 2'-beta-fluoro-2',3'-dideoxyadenosine in peripheral blood mononuclear cells.
Journal: Biochemical pharmacology 19950717
Title: Enhancement by 2'-deoxycoformycin of the 5'-phosphorylation and anti-human immunodeficiency virus activity of 2',3'-dideoxyadenosine and 2'-beta-fluoro-2',3'-dideoxyadenosine.
Journal: Molecular pharmacology 19941101
Title: Synthesis and evaluation of the anti-HIV activity of aza and deaza analogues of isoddA and their phosphates as prodrugs.
Journal: Journal of medicinal chemistry 19941014
Title: Equal inhibition of the replication of human immunodeficiency virus in human T-cell culture by ddA bis(SATE)phosphotriester and 3'-azido-2',3'-dideoxythymidine.
Journal: Biochemical pharmacology 19940705
Title: Inhibitory effect of 9-(2-phosphonylmethoxyethyl)-adenine (PMEA) on human and duck hepatitis B virus infection.
Journal: Antiviral research 19930601
Title: Acute cardiotoxicity of nucleoside analogs FddA and FddI in rats.
Journal: Fundamental and applied toxicology : official journal of the Society of Toxicology 19930401
Title: Potential prodrug derivatives of 2',3'-didehydro-2',3'-dideoxynucleosides. Preparations and antiviral activities.
Journal: Journal of medicinal chemistry 19920724
Title: Use of a standardized cell culture assay to assess activities of nucleoside analogs against hepatitis B virus replication.
Journal: Antiviral research 19920701
Title: Synthesis and anti-HIV activity of isonucleosides.
Journal: Journal of medicinal chemistry 19920626
Title: Substrate specificity of human deoxycytidine kinase toward antiviral 2',3'-dideoxynucleoside analogs.
Journal: Biochemical pharmacology 19920122
Title: Potential anti-AIDS drugs. Lipophilic, adenosine deaminase-activated prodrugs.
Journal: Journal of medicinal chemistry 19910501
Title: Synthesis and anti-HIV activity of 2-, 3-, and 4-substituted analogues of 1-[(2-hydroxyethoxy)methyl]-6-(phenylthio)thymine (HEPT).
Journal: Journal of medicinal chemistry 19910401
Title: Inhibitory effects of selected antiviral compounds on human hepatitis B virus DNA synthesis.
Journal: Antimicrobial agents and chemotherapy 19910201
Title: A new class of HIV-1-specific 6-substituted acyclouridine derivatives: synthesis and anti-HIV-1 activity of 5- or 6-substituted analogues of 1-[(2-hydroxyethoxy)methyl]-6-(phenylthio)thymine (HEPT).
Journal: Journal of medicinal chemistry 19910101
Title: Lipophilic halogenated congeners of 2',3'-dideoxypurine nucleosides active against human immunodeficiency virus in vitro.
Journal: Proceedings of the National Academy of Sciences of the United States of America 19901201
Title: Comparative activities of several nucleoside analogs against duck hepatitis B virus in vitro.
Journal: Antimicrobial agents and chemotherapy 19900701
Title: Synthesis and structure-activity relationships of 6-substituted 2',3'-dideoxypurine nucleosides as potential anti-human immunodeficiency virus agents.
Journal: Journal of medicinal chemistry 19900601
Title: Activities of 3'-azido-3'-deoxythymidine nucleotide dimers in primary lymphocytes infected with human immunodeficiency virus type 1.
Journal: Antimicrobial agents and chemotherapy 19900601
Title: Cyclobut-A and cyclobut-G: broad-spectrum antiviral agents with potential utility for the therapy of AIDS.
Journal: Journal of medicinal chemistry 19900501
Title: Acid-stable 2'-fluoro purine dideoxynucleosides as active agents against HIV.
Journal: Journal of medicinal chemistry 19900301
Title: Muramyl dipeptide inhibits replication of human immunodeficiency virus in vitro.
Journal: AIDS research and human retroviruses 19900301
Title: Cyclobut-A and cyclobut-G, carbocyclic oxetanocin analogs that inhibit the replication of human immunodeficiency virus in T cells and monocytes and macrophages in vitro.
Journal: Antimicrobial agents and chemotherapy 19900201
Title: Exacerbation of human immunodeficiency virus infection in promonocytic cells by bacterial immunomodulators.
Journal: Journal of acquired immune deficiency syndromes 19900101
Title: Potentiating effect of ribavirin on the in vitro and in vivo antiretrovirus activities of 2',3'-dideoxyinosine and 2',3'-dideoxy-2,6-diaminopurine riboside.
Journal: Journal of acquired immune deficiency syndromes 19900101
Title: Synthesis and anti-HIV activity of carbocyclic 2',3'-didehydro-2',3'-dideoxy 2,6-disubstituted purine nucleosides.
Journal: Journal of medicinal chemistry 19900101
Title: A novel lead for specific anti-HIV-1 agents: 1-[(2-hydroxyethoxy)methyl]-6-(phenylthio)thymine.
Journal: Journal of medicinal chemistry 19891201
Title: 3'-Fluoro-2',3'-dideoxy-5-chlorouridine: most selective anti-HIV-1 agent among a series of new 2'- and 3'-fluorinated 2',3'-dideoxynucleoside analogues.
Journal: Journal of medicinal chemistry 19890801
Title: Nucleic acid related compounds. 57. Synthesis, x-ray crystal structure, lipophilic partition properties, and antiretroviral activities of anomeric 3'-azido-2',3'-dideoxy-2,6-diaminopurine ribosides.
Journal: Journal of medicinal chemistry 19890801
Title: Synthesis of the 2-chloro analogues of 3'-deoxyadenosine, 2',3'-dideoxyadenosine, and 2',3'-didehydro-2',3'-dideoxyadenosine as potential antiviral agents.
Journal: Journal of medicinal chemistry 19890501
Title: Inhibition of infectivity of human immunodeficiency virus by a novel nucleoside, oxetanocin, and related compounds.
Journal: Antimicrobial agents and chemotherapy 19890501
Title: Anti-HIV compound assessment by two novel high capacity assays.
Journal: Journal of virological methods 19890301
Title: Replication of human immunodeficiency virus in monocytes. Granulocyte/macrophage colony-stimulating factor (GM-CSF) potentiates viral production yet enhances the antiviral effect mediated by 3'-azido-2'3'-dideoxythymidine (AZT) and other dideoxynucleoside congeners of thymidine.
Journal: The Journal of experimental medicine 19890301
Title: Potentiating effect of ribavirin on the anti-retrovirus activity of 3'-azido-2,6-diaminopurine-2',3'-dideoxyriboside in vitro and in vivo.
Journal: Antiviral research 19890101
Title: 1',2'-seco-dideoxynucleosides as potential anti-HIV agents.
Journal: Journal of medicinal chemistry 19890101
Title: Marked in vivo antiretrovirus activity of 9-(2-phosphonylmethoxyethyl)adenine, a selective anti-human immunodeficiency virus agent.
Journal: Proceedings of the National Academy of Sciences of the United States of America 19890101
Title: Nucleotide dimers suppress HIV expression in vitro.
Journal: AIDS research and human retroviruses 19881201
Title: Comparative activity of 2',3'-saturated and unsaturated pyrimidine and purine nucleosides against human immunodeficiency virus type 1 in peripheral blood mononuclear cells.
Journal: Biochemical pharmacology 19881001
Title: Inhibition of human immunodeficiency virus (HIV-1/HTLV-IIIBa-L) replication in fresh and cultured human peripheral blood monocytes/macrophages by azidothymidine and related 2',3'-dideoxynucleosides.
Journal: The Journal of experimental medicine 19880901
Title: Adenallene and cytallene: acyclic-nucleoside analogues that inhibit replication and cytopathic effect of human immunodeficiency virus in vitro.
Journal: Proceedings of the National Academy of Sciences of the United States of America 19880801
Title: Dextran sulfate suppression of viruses in the HIV family: inhibition of virion binding to CD4+ cells.
Journal: Science (New York, N.Y.) 19880429
Title: Metabolism and anti-human immunodeficiency virus-1 activity of 2-halo-2',3'-dideoxyadenosine derivatives.
Journal: The Journal of biological chemistry 19880425
Title: Investigations on the anti-HIV activity of 2',3'-dideoxyadenosine analogues with modifications in either the pentose or purine moiety. Potent and selective anti-HIV activity of 2,6-diaminopurine 2',3'-dideoxyriboside.
Journal: Biochemical pharmacology 19880401
Title: Potent and selective activity of 3'-azido-2,6-diaminopurine-2',3'-dideoxyriboside, 3'-fluoro-2,6-diaminopurine-2',3'-dideoxyriboside, and 3'-fluoro-2',3'-dideoxyguanosine against human immunodeficiency virus.
Journal: Molecular pharmacology 19880301
Title: Dideoxynucleosides are less inhibitory in vitro against human immunodeficiency virus type 2 (HIV-2) than against HIV-1.
Journal: Antimicrobial agents and chemotherapy 19871201
Title: Synthesis and anti-HIV activity of various 2'- and 3'-substituted 2',3'-dideoxyadenosines: a structure-activity analysis.
Journal: Journal of medicinal chemistry 19871101
Title: Ribavirin antagonizes inhibitory effects of pyrimidine 2',3'-dideoxynucleosides but enhances inhibitory effects of purine 2',3'-dideoxynucleosides on replication of human immunodeficiency virus in vitro.
Journal: Antimicrobial agents and chemotherapy 19871001
Title: 2',3'-Dideoxy-2'-fluoro-ara-A. An acid-stable purine nucleoside active against human immunodeficiency virus (HIV).
Journal: Biochemical pharmacology 19870901
Title: 3'-substituted 2',3'-dideoxynucleoside analogues as potential anti-HIV (HTLV-III/LAV) agents.
Journal: Journal of medicinal chemistry 19870801
Title: The anti-HTLV-III (anti-HIV) and cytotoxic activity of 2',3'-didehydro-2',3'-dideoxyribonucleosides: a comparison with their parental 2',3'-dideoxyribonucleosides.
Journal: Molecular pharmacology 19870701
Title: The 2',3'-dideoxyriboside of 2,6-diaminopurine selectively inhibits human immunodeficiency virus (HIV) replication in vitro.
Journal: Biochemical and biophysical research communications 19870529
Title: Potential anti-AIDS drugs. 2',3'-Dideoxycytidine analogues.
Journal: Journal of medicinal chemistry 19870501
Title: Both 2',3'-dideoxythymidine and its 2',3'-unsaturated derivative (2',3'-dideoxythymidinene) are potent and selective inhibitors of human immunodeficiency virus replication in vitro.
Journal: Biochemical and biophysical research communications 19870115
Title: Inhibition of the in vitro infectivity and cytopathic effect of human T-lymphotrophic virus type III/lymphadenopathy-associated virus (HTLV-III/LAV) by 2',3'-dideoxynucleosides.
Journal: Proceedings of the National Academy of Sciences of the United States of America 19860301
Title: Balzarini J, et al. Conversion of 2',3'-dideoxyadenosine (ddA) and 2',3'-didehydro-2',3'-dideoxyadenosine (d4A) to their corresponding aryloxyphosphoramidate derivatives markedly potentiates their activity against human immunodeficiency virus and hepatitis B virus. FEBS Lett. 1997 Jun 30;410(2-3):324-8.
