Title: Design, synthesis, and antibacterial activity of novel pleuromutilin derivatives bearing an amino thiazolyl ring.
Journal: Archiv der Pharmazie 20120801
Title: [Effect of different compatibility of tetramethylpyrazine on its pharmacokinetics in vivo].
Journal: Zhongguo Zhong yao za zhi = Zhongguo zhongyao zazhi = China journal of Chinese materia medica 20120501
Title: Pleuromutilin and its derivatives-the lead compounds for novel antibiotics.
Journal: Mini reviews in medicinal chemistry 20120101
Title: Determination of minimum inhibitory and minimum bactericidal concentrations of tiamulin against field isolates of Actinobacillus pleuropneumoniae.
Journal: Veterinary microbiology 20110805
Title: Decreased susceptibility of MRSA ST398 to tiamulin.
Journal: Veterinary microbiology 20110805
Title: Change in antimicrobial susceptibility of Mycoplasma gallisepticum field isolates.
Journal: Veterinary microbiology 20110602
Title: Assessment of the antihistomonal effect of paromomycin and tiamulin.
Journal: Tijdschrift voor diergeneeskunde 20110601
Title: Antimicrobial susceptibility of Actinobacillus pleuropneumoniae isolates from clinical outbreaks of porcine respiratory diseases.
Journal: Veterinary microbiology 20110512
Title: Recurrence of Chlamydiasuis infection in pigs after short-term antimicrobial treatment.
Journal: Veterinary journal (London, England : 1997) 20110301
Title: Simultaneous determination of three classes of antibiotics in the suspended solids of swine wastewater by ultrasonic extraction, solid-phase extraction and liquid chromatography-mass spectrometry.
Journal: Journal of environmental sciences (China) 20110101
Title: Mutations in 23S rRNA gene associated with decreased susceptibility to tiamulin and valnemulin in Mycoplasma gallisepticum.
Journal: FEMS microbiology letters 20100701
Title: Factors influencing the activity of tiamulin against Histomonas meleagridis in vitro.
Journal: Avian diseases 20100601
Title: Tiamulin hydrogen fumarate--veterinary uses and HPLC method of determination in premixes and medicated feeding stuffs.
Journal: Acta poloniae pharmaceutica 20100101
Title: The activity and compatibility of the antibiotic tiamulin with other drugs in poultry medicine--A review.
Journal: Poultry science 20091101
Title: Mutilins derivatives: from veterinary to human-used antibiotics.
Journal: Mini reviews in medicinal chemistry 20091001
Title: U2504 determines the species specificity of the A-site cleft antibiotics: the structures of tiamulin, homoharringtonine, and bruceantin bound to the ribosome.
Journal: Journal of molecular biology 20090529
Title: Spironucleosis in gamebirds.
Journal: The Veterinary record 20090321
Title: Single 23S rRNA mutations at the ribosomal peptidyl transferase centre confer resistance to valnemulin and other antibiotics in Mycobacterium smegmatis by perturbation of the drug binding pocket.
Journal: Molecular microbiology 20090301
Title: Tiamulin activity against Brachyspira hyodysenteriae.
Journal: The Veterinary record 20081206
Title: Compatibility of a combination of tiamulin and chlortetracycline with salinomycin in feed during a pulsed medication program coadministration in broilers.
Journal: Poultry science 20081201
Title: Tiamulin activity against Brachyspira hyodysenteriae.
Journal: The Veterinary record 20081201
Title: A click chemistry approach to pleuromutilin conjugates with nucleosides or acyclic nucleoside derivatives and their binding to the bacterial ribosome.
Journal: Journal of medicinal chemistry 20080828
Title: Simultaneous determination of sulfonamides, tetracyclines and tiamulin in swine wastewater by solid-phase extraction and liquid chromatography-mass spectrometry.
Journal: Journal of chromatography. A 20080822
Title: Compatibility of a combination of tiamulin plus chlortetracycline with salinomycin in feed during a long-term co-administration in broilers.
Journal: Poultry science 20080801
Title: [Multiresistant Brachyspira hyodysenteriae in a Dutch sow herd].
Journal: Tijdschrift voor diergeneeskunde 20080701
Title: Treatment of histomonosis in turkeys with tiamulin.
Journal: The Veterinary record 20071201
Title: The effect of medicated diets and level of feeding on caecal microbiota of lactating rabbit does.
Journal: Journal of applied microbiology 20071001
Title: Effects of tiamulin, neomycin, tetracycline, fluorophenicol, penicillin G, Linco-Spectin, erythromycin and oxytetracycline on controlling bacterial contaminations of the river buffalo (Buballus bubalis) semen.
Journal: Pakistan journal of biological sciences : PJBS 20070915
Title: The effect of lactating rabbit does on the development of the caecal microbial community in the pups they nurture.
Journal: Journal of applied microbiology 20070901
Title: Susceptibility of bacteria isolated from pigs to tiamulin and enrofloxacin metabolites.
Journal: Veterinary microbiology 20070331
Title: Persistence of antibiotics such as macrolides, tiamulin and salinomycin in soil.
Journal: Environmental pollution (Barking, Essex : 1987) 20061001
Title: Isolation and structural elucidation of tiamulin metabolites formed in liver microsomes of pigs.
Journal: Journal of pharmaceutical and biomedical analysis 20060918
Title: Elimination of macrolides, tiamulin, and salinomycin during manure storage.
Journal: Archives of environmental contamination and toxicology 20060701
Title: Treatment of a field case of avian intestinal spirochaetosis caused by Brachyspira pilosicoli with tiamulin.
Journal: Avian pathology : journal of the W.V.P.A 20060601
Title: Trace analysis of tiamulin in honey by liquid chromatography-diode array-electrospray ionization mass spectrometry detection.
Journal: Journal of chromatography. A 20060526
Title: Tiamulin and semduramicin: effects of simultaneous administration on performance and health of growing broiler chickens.
Journal: Poultry science 20060301
Title: Tiamulin resistance in porcine Brachyspira pilosicoli isolates.
Journal: Research in veterinary science 20060201
Title: Evaluation of the therapeutic activity of tulathromycin against swine respiratory disease on farms in Europe.
Journal: Veterinary therapeutics : research in applied veterinary medicine 20050101
Title: Inhibition of peptide bond formation by pleuromutilins: the structure of the 50S ribosomal subunit from Deinococcus radiodurans in complex with tiamulin.
Journal: Molecular microbiology 20041201
Title: Mutations in ribosomal protein L3 and 23S ribosomal RNA at the peptidyl transferase centre are associated with reduced susceptibility to tiamulin in Brachyspira spp. isolates.
Journal: Molecular microbiology 20041201
Title: Testing the efficacy of fermented wheat germ extract against Mycoplasma gallisepticum infection of chickens.
Journal: Poultry science 20041101
Title: Comparison of methods for antimicrobial susceptibility testing and MIC values for pleuromutilin drugs for Brachyspira hyodysenteriae isolated in Germany.
Journal: Veterinary microbiology 20040819
Title: Further characterization of porcine Brachyspira hyodysenteriae isolates with decreased susceptibility to tiamulin.
Journal: Journal of medical microbiology 20040401
Title: Decreased susceptibility to tiamulin and valnemulin among Czech isolates of Brachyspira hyodysenteriae.
Journal: Journal of medical microbiology 20040401
Title: Biochemical background of toxic interaction between tiamulin and monensin.
Journal: Chemico-biological interactions 20040315
Title: [The use of macrolides, lincomycin and tiamulin as animal feed drugs for pigs in Schleswig-Holstein].
Journal: Berliner und Munchener tierarztliche Wochenschrift 20040101
Title: Effects of the administration of spiramycin and tiamulin on in vivo complex formation and hepatic cytochrome P4503A (CYP3A)-dependent monooxygenases in rabbits.
Journal: Veterinary research communications 20030901
Title: Determination of antibiotics from soil by pressurized liquid extraction and liquid chromatography-tandem mass spectrometry.
Journal: Journal of chromatography. A 20030627
Title: Putative biomarkers for evaluating antibiotic treatment: an experimental model of porcine Actinobacillus pleuropneumoniae infection.
Journal: Research in veterinary science 20030601
Title: Determination of antibiotics such as macrolides, ionophores and tiamulin in liquid manure by HPLC-MS/MS.
Journal: Analytical and bioanalytical chemistry 20030401
Title: Effects of the antibacterial agents tiamulin, olanquindox and metronidazole and the anthelmintic ivermectin on the soil invertebrate species Folsomia fimetaria (Collembola) and Enchytraeus crypticus (Enchytraeidae).
Journal: Chemosphere 20030101
Title: Screening method for detecting cross-contamination residues of tiamulin in swine feeds.
Journal: Journal of AOAC International 20030101
Title: In vitro formation of metabolic-intermediate cytochrome P450 complexes in rabbit liver microsomes by tiamulin and various macrolides.
Journal: Veterinary research 20030101
Title: Reduction of economic losses caused by mycoplasmal pneumonia of pigs by vaccination with Respisure and by Tiamutin treatment.
Journal: Acta veterinaria Hungarica 20030101
Title: In vitro development of resistance to enrofloxacin, erythromycin, tylosin, tiamulin and oxytetracycline in Mycoplasma gallisepticum, Mycoplasma iowae and Mycoplasma synoviae.
Journal: Veterinary microbiology 20020802
Title: Influence of in-feed zinc bacitracin and tiamulin treatment on experimental avian intestinal spirochaetosis caused by Brachyspira intermedia.
Journal: Avian pathology : journal of the W.V.P.A 20020601
Title: Evaluation of tiamulin and lincomycin for the treatment of broiler breeders experimentally infected with the intestinal spirochaete Brachyspira pilosicoli.
Journal: Avian pathology : journal of the W.V.P.A 20020601
Title: Simultaneous determination of various macrolides by liquid chromatography/mass spectrometry.
Journal: Journal of veterinary science 20020601
Title: Determination of tiamulin in type C medicated swine feeds using high throughput extraction with liquid chromatography.
Journal: Journal of AOAC International 20020101
Title: An assessment of antimicrobial consumption in food producing animals in Kenya.
Journal: Journal of veterinary pharmacology and therapeutics 20011201
Title: The pleuromutilin drugs tiamulin and valnemulin bind to the RNA at the peptidyl transferase centre on the ribosome.
Journal: Molecular microbiology 20010901
Title: Eradication of endemic Brachyspira pilosicoli infection from a farrowing herd: a case report.
Journal: Animal health research reviews 20010601
Title: Susceptibility to pleuromutilins in Brachyspira (Serpulina) hyodysenteriae.
Journal: Animal health research reviews 20010601
Title: Intestinal spirochete infections of chickens: a review of disease associations, epidemiology and control.
Journal: Animal health research reviews 20010601
Title: Pleuromutilins. Part 1. The identification of novel mutilin 14-carbamates.
Journal: Bioorganic & medicinal chemistry 20010501
Title: An investigation of the etiology of a mild diarrhea observed in a group of grower/finisher pigs.
Journal: The Canadian veterinary journal = La revue veterinaire canadienne 20010101
Title: Proposed quality control guidelines for National Committee for Clinical Laboratory Standards Susceptibility Tests using the veterinary antimicrobial agent tiamulin.
Journal: Diagnostic microbiology and infectious disease 20010101
Title: Noa M, et al. Tiamulin-nitrovin interaction in pigs: a case report and experimental reproduction. Vet Hum Toxicol. 2000 Oct;42(5):286-8.
Title: Dreyfuss J, et al. Metabolism of tritium- and carbon-14-labeled tiamulin in dogs, rats, and pigs. J Antibiot (Tokyo). 1979 May;32(5):496-503.
Title: Islam KM, et al. The activity and compatibility of the antibiotic tiamulin with other drugs in poultry medicine--A review. Poult Sci. 2009 Nov;88(11):2353-9.