Title: Human sex hormone-binding globulin binding affinities of 125 structurally diverse chemicals and comparison with their binding to androgen receptor, estrogen receptor, and α-fetoprotein.
Journal: Toxicological sciences : an official journal of the Society of Toxicology 20150201
Title: Synthesis of end-functionalized polyacetylenes that contain polar groups by employing well-defined palladium catalysts.
Journal: Chemistry (Weinheim an der Bergstrasse, Germany) 20121029
Title: Ormeloxifene inhibits osteoclast differentiation in parallel to downregulating RANKL-induced ROS generation and suppressing the activation of ERK and JNK in murine RAW264.7 cells.
Journal: Journal of molecular endocrinology 20120601
Title: Pharmacokinetic evaluation of toremifene and its clinical implications for the treatment of osteoporosis.
Journal: Expert opinion on drug metabolism & toxicology 20120401
Title: Evaluation of the OECD (Q)SAR Application Toolbox for the profiling of estrogen receptor binding affinities.
Journal: SAR and QSAR in environmental research 20120101
Title: Development, characterization, and in vitro evaluation of tamoxifen microemulsions.
Journal: Journal of drug delivery 20120101
Title: Lipophilic Pt(II) complexes with selective efficacy against cisplatin-resistant testicular cancer cells.
Journal: Journal of inorganic biochemistry 20111201
Title: Breast cancer medications and vision: effects of treatments for early-stage disease.
Journal: Current eye research 20111001
Title: Synthesis and characterization of triphenylethylene derivatives with aggregation-induced emission characteristics.
Journal: Journal of fluorescence 20110901
Title: Piezofluorochromic and aggregation-induced-emission compounds containing triphenylethylene and tetraphenylethylene moieties.
Journal: Chemistry, an Asian journal 20110606
Title: An integrated bioinformatics approach identifies elevated cyclin E2 expression and E2F activity as distinct features of tamoxifen resistant breast tumors.
Journal: PloS one 20110101
Title: Sensitization of glioma cells to tamoxifen-induced apoptosis by Pl3-kinase inhibitor through the GSK-3β/β-catenin signaling pathway.
Journal: PloS one 20110101
Title: Ficus platyphylla promotes fertility in female Rattus norvegicus Wistar strain: a preliminary study.
Journal: Reproductive biology and endocrinology : RB&E 20110101
Title: Tamoxifen and raloxifene modulate gap junction coupling during early phases of retinoic acid-dependent neuronal differentiation of NTera2/D1 cells.
Journal: Cell biology and toxicology 20101201
Title: Anti-breast cancer potential of SS1020, a novel antiestrogen lacking estrogenic and genotoxic actions.
Journal: International journal of cancer 20101001
Title: Estrogen antagonist and development of macular hole.
Journal: Korean journal of ophthalmology : KJO 20101001
Title: Structure-function relationships of estrogenic triphenylethylenes related to endoxifen and 4-hydroxytamoxifen.
Journal: Journal of medicinal chemistry 20100422
Title: Selective estrogen receptor modulator (SERM) for the treatment of osteoporosis in postmenopausal women: focus on lasofoxifene.
Journal: Clinical interventions in aging 20100101
Title: Granulosa cell tumor of the ovary and antecedent of adjuvant tamoxifen use for breast cancer.
Journal: World journal of surgical oncology 20100101
Title: Female sex hormones mediate the allergic lung reaction by regulating the release of inflammatory mediators and the expression of lung E-selectin in rats.
Journal: Respiratory research 20100101
Title: Ultrastructural effects of tamoxifen on uterus in rats.
Journal: The Tokai journal of experimental and clinical medicine 20090920
Title: Lasofoxifene: Evidence of its therapeutic value in osteoporosis.
Journal: Core evidence 20090101
Title: Bazedoxifene for the prevention of postmenopausal osteoporosis.
Journal: Therapeutics and clinical risk management 20081201
Title: Selective estrogen receptor modulators: an update on recent clinical findings.
Journal: Obstetrical & gynecological survey 20080301
Title: Nanoparticles loaded with ferrocenyl tamoxifen derivatives for breast cancer treatment.
Journal: International journal of pharmaceutics 20080122
Title: Optimizing high-performance liquid chromatography method with fluorescence detection for quantification of tamoxifen and two metabolites in human plasma: application to a clinical study.
Journal: Journal of pharmaceutical and biomedical analysis 20080122
Title: A mass spectrometric approach for the study of the metabolism of clomiphene, tamoxifen and toremifene by liquid chromatography time-of-flight spectroscopy.
Journal: European journal of mass spectrometry (Chichester, England) 20080101
Title: By looking back we can see the way forward: enhancing the gains achieved with antihormone therapy.
Journal: Breast cancer research : BCR 20080101
Title: Tamoxifen accelerates proteasomal degradation of O6-methylguanine DNA methyltransferase in human cancer cells.
Journal: International journal of cancer 20071115
Title: Practical synthesis of unsymmetrical tetraarylethylenes and their application for the preparation of [triphenylethylene-spacer-triphenylethylene] triads.
Journal: The Journal of organic chemistry 20071012
Title: Synthesis of 1,1,2-triphenylethylenes and their antiproliferative effect on human cancer cell lines.
Journal: Anti-cancer drugs 20071001
Title: Tamoxifen stimulates calcium entry into human platelets.
Journal: Journal of cardiovascular pharmacology 20071001
Title: The differential effects of bisphosphonates, SERMS (selective estrogen receptor modulators), and parathyroid hormone on bone remodeling in osteoporosis.
Journal: Clinical interventions in aging 20070301
Title: Medicinal chemistry and emerging strategies applied to the development of selective estrogen receptor modulators (SERMs).
Journal: Current medicinal chemistry 20070101
Title: Estrogenic or antiestrogenic therapies for multiple myeloma?
Journal: Molecular cancer 20070101
Title: Decursin and decursinol angelate inhibit estrogen-stimulated and estrogen-independent growth and survival of breast cancer cells.
Journal: Breast cancer research : BCR 20070101
Title: Prediction of estrogen receptor agonists and characterization of associated molecular descriptors by statistical learning methods.
Journal: Journal of molecular graphics & modelling 20061101
Title: Modulation of estrogen receptor transactivation and estrogen-induced gene expression by ormeloxifene-a triphenylethylene derivative.
Journal: Steroids 20061101
Title: Fragmentation of 2,2,2-triphenylethoxychlorocarbene: evidence for ultrafast fragmentation-rearrangement in excited diazirines.
Journal: Organic letters 20061012
Title: Functional inhibition of intestinal and uterine muscles by non-permeant triphenylethylene derivatives.
Journal: European journal of pharmacology 20060217
Title: Identification of covalent attachment site of antiestrogenic estradiol 11 beta-derivatives on human estrogen receptor alpha ligand-binding domain.
Journal: The Journal of steroid biochemistry and molecular biology 20060201
Title: [Interactions between radiation and hormonal therapy in breast cancer: simultaneous or sequential treatment].
Journal: Orvosi hetilap 20060122
Title: Additive growth inhibitory effects of ibandronate and antiestrogens in estrogen receptor-positive breast cancer cell lines.
Journal: Breast cancer research : BCR 20060101
Title: Effects of tamoxifen on vaginal blood flow and epithelial morphology in the rat.
Journal: BMC women's health 20060101
Title: Dielectric and shear mechanical alpha and beta relaxations in seven glass-forming liquids.
Journal: The Journal of chemical physics 20051215
Title: Investigation of radical cation in electrophilic fluorination by ESI-MS.
Journal: Organic letters 20050901
Title: Synthesis, structure-activity relationships and antagonistic effects in human MCF-7 breast cancer cells of flexible estrogen receptor modulators.
Journal: Medicinal chemistry (Shariqah (United Arab Emirates)) 20050701
Title: Endometrial K-ras mutations in postmenopausal breast cancer patients treated with adjuvant tamoxifen or toremifene.
Journal: Cancer chemotherapy and pharmacology 20050401
Title: K-ras mutation in the endometrium of tamoxifen-treated breast cancer patients, with a comparison of tamoxifen and toremifene.
Journal: British journal of cancer 20050328
Title: Recycling nanoparticles stabilized in water-in-CO2 microemulsions for catalytic hydrogenations.
Journal: Langmuir : the ACS journal of surfaces and colloids 20050301
Title: Endocrinology and hormone therapy in breast cancer: selective oestrogen receptor modulators and downregulators for breast cancer - have they lost their way?
Journal: Breast cancer research : BCR 20050101
Title: Selective estrogen receptor modulators inhibit growth and progression of premalignant lesions in a mouse model of ductal carcinoma in situ.
Journal: Breast cancer research : BCR 20050101
Title: Advances in estrogen receptor biology: prospects for improvements in targeted breast cancer therapy.
Journal: Breast cancer research : BCR 20040101
Title: Study of 202 natural, synthetic, and environmental chemicals for binding to the androgen receptor.
Journal: Chemical research in toxicology 20031001
Title: The effect of estradiol in the striatum is blocked by ICI 182,780 but not tamoxifen: pharmacological and behavioral evidence.
Journal: Neuroendocrinology 20030401
Title: Effects of tamoxifen on ischemia-induced angiogenesis in the mouse lung.
Journal: Angiogenesis 20030101
Title: Triphenylethylene antiestrogen-induced acute relaxation of mouse duodenal muscle. Possible involvement of Ca2+ channels.
Journal: European journal of pharmacology 20020612
Title: Tamoxifen and toremifene impair retrieval, but not acquisition, of spatial information processing in mice.
Journal: Pharmacology, biochemistry, and behavior 20020501
Title: Some coumarins and triphenylethene derivatives as inhibitors of human testes microsomal 17beta-hydroxysteroid dehydrogenase (17beta-HSD type 3): further studies with tamoxifen on the rat testes microsomal enzyme.
Journal: Journal of enzyme inhibition and medicinal chemistry 20020401
Title: [Selective estrogen receptor modulators (SERMs) in the practice].
Journal: Magyar onkologia 20020101
Title: The preparation of phenyl-stilbene derivatives using the safety catch linker.
Journal: Methods in molecular biology (Clifton, N.J.) 20020101
Title: Endocrine manipulation in advanced breast cancer: recent advances with SERM therapies.
Journal: Clinical cancer research : an official journal of the American Association for Cancer Research 20011201
Title: Future use of selective estrogen receptor modulators and aromatase inhibitors.
Journal: Clinical cancer research : an official journal of the American Association for Cancer Research 20011201
Title: Okadaic acid-sensitive activation of Maxi Cl(-) channels by triphenylethylene antioestrogens in C1300 mouse neuroblastoma cells.
Journal: The Journal of physiology 20011001
Title: Molecular classification of estrogens.
Journal: Cancer research 20010915
Title: Differential SERM activation of the estrogen receptors (ERalpha and ERbeta) at AP-1 sites.
Journal: Chemistry & biology 20010501
Title: Flexible estrogen receptor modulators: design, synthesis, and antagonistic effects in human MCF-7 breast cancer cells.
Journal: Journal of medicinal chemistry 20010329
Title: [Synthesis of triphenylethylene with aliphatic cyclic moiety and its antagonism on estrogen receptor].
Journal: Yao xue xue bao = Acta pharmaceutica Sinica 20010301
Title: Update on endocrine aspects of breast cancer: report from the 23rd San Antonio Breast Cancer Symposium, San Antonio, Texas, USA, 6-9 December 2000.
Journal: Breast cancer research : BCR 20010101
Title: Selective estrogen receptor modulation: the search for an ideal hormonal therapy for breast cancer.
Journal: Cancer investigation 20010101
Title: Cone voltage and collision cell collision-induced dissociation study of triphenylethylenes of pharmaceutical interest.
Journal: Rapid communications in mass spectrometry : RCM 20010101
Title: Estrogen receptor binding affinity and uterotrophic activity of triphenylhaloethylenes.
Journal: Journal of steroid biochemistry 19880601
