Title: Development and Characterization of a Potent Free Fatty Acid Receptor 1 (FFA1) Fluorescent Tracer.
Journal: Journal of medicinal chemistry 20160526
Title: Identification and pharmacological characterization of multiple allosteric binding sites on the free fatty acid 1 receptor.
Journal: Molecular pharmacology 20121101
Title: AMG 837: a potent, orally bioavailable GPR40 agonist.
Journal: Bioorganic & medicinal chemistry letters 20120115
Title: Identification of a potent and selective free fatty acid receptor 1 (FFA1/GPR40) agonist with favorable physicochemical and in vitro ADME properties.
Journal: Journal of medicinal chemistry 20111013
Title: Enantioselective synthesis of a GPR40 agonist AMG 837 via catalytic asymmetric conjugate addition of terminal alkyne to α,β-unsaturated thioamide.
Journal: Organic letters 20110304
Title: AMG 837: a novel GPR40/FFA1 agonist that enhances insulin secretion and lowers glucose levels in rodents.
Journal: PloS one 20110101
Title: Houze JB, et al. AMG 837: a potent, orally bioavailable GPR40 agonist. Bioorg Med Chem Lett. 2012 Jan 15;22(2):1267-70.
Title: Lin DC, et al. AMG 837: a novel GPR40/FFA1 agonist that enhances insulin secretion and lowers glucose levels in rodents. PLoS One. 2011;6(11):e27270.
