Title: Role of sigma-1 receptors in paclitaxel-induced neuropathic pain in mice.
Journal: The journal of pain : official journal of the American Pain Society 20121101
Title: Synthesis and biological evaluation of the 1-arylpyrazole class of σ(1) receptor antagonists: identification of 4-{2-[5-methyl-1-(naphthalen-2-yl)-1H-pyrazol-3-yloxy]ethyl}morpholine (S1RA, E-52862).
Journal: Journal of medicinal chemistry 20121011
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Title: Romero L, et al. Pharmacological properties of S1RA, a new sigma-1 receptor antagonist that inhibits neuropathic pain and activity-induced spinal sensitization. Br J Pharmacol. 2012 Aug;166(8):2289-306.
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