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Title: Dual action molecules: bioassays of combined novel antioxidants and angiotensin II receptor antagonists.
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Title: Low-temperature loading of Cu+ species over porous metal-organic frameworks (MOFs) and adsorptive desulfurization with Cu+-loaded MOFs.
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Title: Synthesis and Anti-hyperlipidemic Activity of 3H-benzo [4, 5] thieno [2, 3-d] [1, 2, 3] triazin-4-ones: Possible Mechanism of Altered Lipid Metabolism.
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Title: Symmetrical approach of spiro-pyrazolidinediones as acetyl-CoA carboxylase inhibitors.
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Title: Management of singlet and triplet excitons in a single emission layer: a simple approach for a high-efficiency fluorescence/phosphorescence hybrid white organic light-emitting device.
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Title: (Z)-3-(1H-Indol-3-yl)-2-(3,4,5-tri-methoxy-phen-yl)acrylonitrile.
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Title: (Z)-3-(1-Benzofuran-2-yl)-2-(3,4,5-tri-meth-oxy-phen-yl)acrylonitrile.
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Title: Oxidative desulfurization of benzothiophene and thiophene with WOx/ZrO2 catalysts: effect of calcination temperature of catalysts.
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Title: Synthesis, docking studies and biological evaluation of benzo[b]thiophen-2-yl-3-(4-arylpiperazin-1-yl)-propan-1-one derivatives on 5-HT1A serotonin receptors.
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Title: (E)-3-[(2-Methyl-4-nitro-phen-yl)imino-meth-yl]-1-benzothio-phene.
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Title: Bacterial dioxygenase- and monooxygenase-catalysed sulfoxidation of benzo[b]thiophenes.
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Title: Remarkable adsorption capacity of CuCl2-loaded porous vanadium benzenedicarboxylate for benzothiophene.
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Title: Synthesis and characterization of nonsymmetric cyclopentene-based dithienylethenes.
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Title: Argentation chromatography for the separation of polycyclic aromatic compounds according to ring number.
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Title: Gynecologic effects of arzoxifene in postmenopausal women with osteoporosis or low bone mass.
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Title: Benzothiophene carboxamide derivatives as inhibitors of Plasmodium falciparum enoyl-ACP reductase.
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Title: Benzothiophene carboxamide derivatives as novel antimalarials.
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Title: Pharmacophore-based discovery of FXR-agonists. Part II: identification of bioactive triterpenes from Ganoderma lucidum.
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Title: Importance of heterocylic aromatic compounds in monitored natural attenuation for coal tar contaminated aquifers: A review.
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Title: Synthesis of benzothiophene derivatives by Pd-catalyzed or radical-promoted heterocyclodehydration of 1-(2-mercaptophenyl)-2-yn-1-ols.
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Title: Conformationally constrained farnesoid X receptor (FXR) agonists: alternative replacements of the stilbene.
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Title: A practical, one-pot synthesis of highly substituted thiophenes and benzo[b]thiophenes from bromoenynes and o-alkynylbromobenzenes.
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Title: Breast cancer medications and vision: effects of treatments for early-stage disease.
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Title: (E)-2-[1-(1-Benzothio-phen-2-yl)ethyl-idene]-N-phenyl-hydrazinecarboxamide.
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Title: Design and synthesis of 1,3-biarylsulfanyl derivatives as new anti-breast cancer agents.
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Title: Novel cyclopalladated imino-thiophenes: synthesis and reactivity toward alkynes and carbon monoxide.
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Title: Structural features determining the intestinal epithelial permeability and efflux of novel HIV-1 protease inhibitors.
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Title: Synthesis, structure and cytotoxicity of 3-C, N, S, Se substituted benzo[b]selenophene derivatives.
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Title: Benzimidazolone as potent chymase inhibitor: modulation of reactive metabolite formation in the hydrophobic (P1) region.
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Title: Palladium-catalyzed three-component domino reaction for the preparation of benzo[b]thiophene and related compounds.
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Title: Multimetal Fischer carbene complexes of Group VI transition metals: synthesis, structure and substituent effect investigation.
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Title: 7-Methyl-5,6,7,8-tetra-hydro-1-benzo-thieno[2,3-d]pyrimidin-4-amine.
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Title: 3'-(4-Meth-oxy-phen-yl)-4'-phenyl-3H,4'H-spiro-[1-benzothio-phene-2,5'-isoxazol]-3-one.
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Title: Effect of carbohydrate amino group modifications on the cytotoxicity of glycosylated 2-phenyl-benzo[b]thiophenes and 2-phenyl-benzo[b]furans.
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Title: 5-Methyl-phenanthro[2,3-b]thio-phene.
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Title: Novel benzo[b]thiophene derivatives as new potential antidepressants with rapid onset of action.
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Title: Ring-closure reactions of 1,2-diaza-4,5-benzoheptatrienyl metal compounds: experiment and theory.
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Title: Synthesis, evaluation and structural studies of antiproliferative tubulin-targeting azetidin-2-ones.
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Title: 2-Phenyl-8,9,10,11-tetra-hydro-1-benzo-thieno[3,2-e][1,2,4]triazolo[1,5-c]pyrimidine.
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Title: Carbon-sulfur bond cleavage and hydrodesulfurization of thiophenes by tungsten.
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Title: Oxidative desulfurization of fuels catalyzed by Fenton-like ionic liquids at room temperature.
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Title: Synthesis, photophysical characterization, and enzymatic incorporation of a microenvironment-sensitive fluorescent uridine analog.
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Title: Ruthenium-catalyzed oxidative vinylation of heteroarene carboxylic acids with alkenes via regioselective C-H bond cleavage.
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Title: Photon-quantitative reaction of a dithiazolylarylene in solution.
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Title: Remarkable adsorptive performance of a metal-organic framework, vanadium-benzenedicarboxylate (MIL-47), for benzothiophene.
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Title: Solution-processable organic single crystals with bandlike transport in field-effect transistors.
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Title: The identification of substituted benzothiophene derivatives as PGE(2) subtype 4 receptor antagonists: From acid to non-acid.
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Title: Benzothieno[3,2-b]quinolinium and 3-(phenylthio)quinolinium compounds: Synthesis and evaluation against opportunistic fungal pathogens.
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Title: Synthesis of benzothiophene carboxamide derivatives and their pharmacological evaluation as potent antihypertriglyceridemic agents in rats.
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Title: Crystal structure prediction and isostructurality of three small molecules.
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Title: Synthesis of regioselectively functionalized benzo[b]thiophenes by combined ortho-lithiation-halocyclization strategies.
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Title: Indole- and benzothiophene-based histamine H3 antagonists.
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Title: Synthesis of benzofuran, benzothiophene, and benzothiazole-based thioamides and their evaluation as K(ATP) channel openers.
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Title: Rotary molecular motors: a large increase in speed through a small change in design.
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Title: Ladder-type pi-conjugated 4-hetero-1,4-dihydrophosphinines: a structure-property study.
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Title: Benzo[b]thiophene-6-carboxamide 1,1-dioxides: inhibitors of human cancer cell growth at nanomolar concentrations.
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Title: Di(hetero)arylamines in the benzo[b]thiophene series as novel potent antioxidants.
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Title: Polymer-bound oxidovanadium(IV) and dioxidovanadium(V) complexes as catalysts for the oxidative desulfurization of model fuel diesel.
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Title: QSAR analysis of antitumor active amides and quinolones from thiophene series.
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Title: Synthesis and characterization of selective dopamine D2 receptor antagonists. 2. Azaindole, benzofuran, and benzothiophene analogs of L-741,626.
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Title: Substituted 2-(3',4',5'-trimethoxybenzoyl)-benzo[b]thiophene derivatives as potent tubulin polymerization inhibitors.
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Title: Toward the discovery of new agents able to inhibit the expression of microsomal prostaglandin E synthase-1 enzyme as promising tools in drug development.
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Title: New cyclopalladated benzothiophenes: a catalyst precursor for the Suzuki coupling of deactivated aryl chlorides.
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Title: Ester-directed regioselective borylation of heteroarenes catalyzed by a silica-supported iridium complex.
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Title: A benzothiophene inhibitor of mitogen-activated protein kinase-activated protein kinase 2 inhibits tumor necrosis factor alpha production and has oral anti-inflammatory efficacy in acute and chronic models of inflammation.
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Title: Benzothiophene containing Rho kinase inhibitors: Efficacy in an animal model of glaucoma.
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Title: 3-(4-Methoxy-benz-yl)-1-benzothio-phene.
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Title: The effect of substituted thiophene and benzothiophene derivates on PPARgamma expression and glucose metabolism.
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Title: Synthesis and study of some new 1,3-isoindoledione derivatives as potential antibacterial agents.
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Title: Novel benzothiophene H1-antihistamines for the treatment of insomnia.
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Title: 1-(Phenyl-sulfon-yl)benzo[1,2:2',3']thieno[5',4'-b]carbazole.
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Title: Substituted benzothiophene or benzofuran derivatives as a novel class of bone morphogenetic protein-2 up-regulators: synthesis, structure-activity relationships, and preventive bone loss efficacies in senescence accelerated mice (SAMP6) and ovariectomized rats.
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Title: Structure based drug design: development of potent and selective factor IXa (FIXa) inhibitors.
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Title: Studies of benzothiophene template as potent factor IXa (FIXa) inhibitors in thrombosis.
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Title: Raloxifene inhibits bone loss and improves bone strength through an Opg-independent mechanism.
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Title: Modulation on C- and N-terminal moieties of a series of potent and selective linear tachykinin NK(2) receptor antagonists.
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Title: Immunogenetics and the Pathological Mechanisms of Human T-Cell Leukemia VirusType 1- (HTLV-1-)Associated Myelopathy/Tropical Spastic Paraparesis (HAM/TSP).
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Title: Novel protein kinase D inhibitors cause potent arrest in prostate cancer cell growth and motility.
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Title: QSAR studies of benzofuran/benzothiophene biphenyl derivatives as inhibitors of PTPase-1B.
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Title: As many as six tandem reactions in one step! Unprecedented formation of highly functionalized benzothiophenes.
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Title: Ethyl 2-(3,3-dibutyl-thio-ureido)-4,5,6,7-tetra-hydro-benzo[b]thio-phene-3-carboxyl-ate.
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Title: Novel reactivity of dibenzothiophene monooxygenase from Bacillus subtilis WU-S2B.
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Title: Biodegradation of thiodiglycol, a hydrolyzate of the chemical weapon Yperite, by benzothiophene-desulfurizing bacteria.
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Title: Benzothiophene inhibitors of MK2. Part 2: improvements in kinase selectivity and cell potency.
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Title: Benzothiophene inhibitors of MK2. Part 1: structure-activity relationships, assessments of selectivity and cellular potency.
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Title: Effects of arzoxifene on bone mineral density and endometrium in postmenopausal women with normal or low bone mass.
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Title: Raloxifene, a selective estrogen receptor modulator, induces mitochondria-mediated apoptosis in human endometrial carcinoma cells.
Journal: Medical molecular morphology 20080901
Title: alpha,alpha-Cyclopentaneglycine dipeptides capped with biaryls as tachykinin NK(2) receptor antagonists.
Journal: ChemMedChem 20080701
Title: Liquid phase adsorption by microporous coordination polymers: removal of organosulfur compounds.
Journal: Journal of the American Chemical Society 20080604
Title: Desulfurization of various organic sulfur compounds and the mixture of DBT + 4,6-DMDBT by Mycobacterium sp. ZD-19.
Journal: Bioresource technology 20080601
Title: 5,7-Bis(1-benzothio-phen-2-yl)-2,3-dihydro-thieno[3,4-b][1,4]dioxine.
Journal: Acta crystallographica. Section E, Structure reports online 20080601
Title: (11R,11aS)-11-Hydr-oxy-1,5,11,11a-tetra-hydro-1-benzothieno[2,3-f]indolizin-3(2H)-one.
Journal: Acta crystallographica. Section E, Structure reports online 20080601
Title: New thermally irreversible and fluorescent photochromic diarylethenes.
Journal: The journal of physical chemistry. A 20080529
Title: Raloxifene in breast cancer prevention.
Journal: Expert opinion on drug safety 20080501
Title: Preventing breast cancer in high-risk women, 2008.
Journal: Oncology (Williston Park, N.Y.) 20080501
Title: Screening for antidepressant, sedative and analgesic activities of novel fused thiophene derivatives.
Journal: Acta pharmaceutica (Zagreb, Croatia) 20080301
Title: Comparison of effects of alendronate and raloxifene on lumbar bone mineral density, bone turnover, and lipid metabolism in elderly women with osteoporosis.
Journal: Yonsei medical journal 20080227
Title: Deprotonative metalation of five-membered aromatic heterocycles using mixed lithium-zinc species.
Journal: The Journal of organic chemistry 20080104
Title: Amino acid derivatives as histone deacetylase inhibitors.
Journal: Bioorganic & medicinal chemistry letters 20080101
Title: Carbonic anhydrase IX in oligodendroglial brain tumors.
Journal: BMC cancer 20080101
Title: S35225 is a direct inhibitor of Plasminogen Activator Inhibitor type-1 activity in the blood.
Journal: Thrombosis research 20080101
Title: [Synthetic estrogens: some new pharmacological actions and mechanisms].
Journal: Nihon rinsho. Japanese journal of clinical medicine 20080101
Title: Efficacy of tibolone and raloxifene for the maintenance of skeletal muscle strength, bone mineral density, balance, body composition, cognitive function, mood/depression, anxiety and quality of life/well-being in late postmenopausal women >/= 70 years: study design of a randomized, double-blind, double-dummy, placebo-controlled, single-center trial.
Journal: Trials 20080101
Title: Human genetics branches out in Barcelona.
Journal: Genome biology 20080101
Title: Synthesis of thienyl analogues of PCBM and investigation of morphology of mixtures in P3HT.
Journal: Beilstein journal of organic chemistry 20080101
Title: Development of a groundwater biobarrier for the removal of polycyclic aromatic hydrocarbons, BTEX, and heterocyclic hydrocarbons.
Journal: Water science and technology : a journal of the International Association on Water Pollution Research 20080101
Title: S,C-sulfonium ylides from thiophenes: potential carbene precursors.
Journal: Journal of the American Chemical Society 20071226
Title: Synthesis of benzo[b]thiophenes by cyclization of arylketene dithioacetal monoxides under pummerer-like conditions.
Journal: Organic letters 20071220
Title: (Z)-3-(Benzo[b]thiophen-2-yl)-2-(3,4,5-trimethoxyphenyl)acrylonitrile and (E)-3-(benzo[b]thiophen-2-yl)-2-(3,4-dimethoxyphenyl)acrylonitrile. [corrected].
Journal: Acta crystallographica. Section C, Crystal structure communications 20071201
Title: Zipper-mode double C-H activation: palladium-catalyzed direct construction of highly-fused heterocyclic systems.
Journal: Organic letters 20071108
Title: Discovery of a new series of potent and selective linear tachykinin NK2 receptor antagonists.
Journal: Journal of medicinal chemistry 20071004
Title: Sulfur from benzothiophene and alkylbenzothiophenes supports growth of Rhodococcus sp. strain JVH1.
Journal: Biodegradation 20071001
Title: Structure-activity relationships for a family of benzothiophene selective estrogen receptor modulators including raloxifene and arzoxifene.
Journal: ChemMedChem 20071001
Title: Synthesis and evaluation of dual wavelength fluorescent benzo[b]thiophene boronic acid derivatives for sugar sensing.
Journal: Chemical biology & drug design 20071001
Title: Structural modulation of reactivity/activity in design of improved benzothiophene selective estrogen receptor modulators: induction of chemopreventive mechanisms.
Journal: Molecular cancer therapeutics 20070901
Title: Effect of estrogens on skin aging and the potential role of SERMs.
Journal: Clinical interventions in aging 20070901
Title: Update on bazedoxifene: a novel selective estrogen receptor modulator.
Journal: Clinical interventions in aging 20070901
Title: Benzo[b]thiophene-based histone deacetylase inhibitors.
Journal: Bioorganic & medicinal chemistry letters 20070815
Title: Chromatographic methods applied in the monitoring of biodesulfurization processes--state of the art.
Journal: Talanta 20070815
Title: Selectivity among organic sulfur compounds in one- and two-liquid-phase cultures of Rhodococcus sp. strain JVH1.
Journal: Biodegradation 20070801
Title: Nonconjugated dendritic iridium(III) complexes with tunable pyridine-based ligands: synthesis, photophysical, electrochemical, and electroluminescent properties.
Journal: Inorganic chemistry 20070709
Title: Synthesis and SAR of selective benzothiophene, benzofuran, and indole-based peroxisome proliferator-activated receptor delta agonists.
Journal: Bioorganic & medicinal chemistry letters 20070701
Title: Benzothiophene selective estrogen receptor modulators with modulated oxidative activity and receptor affinity.
Journal: Journal of medicinal chemistry 20070531
Title: Environmental factors influencing sorption of heterocyclic aromatic compounds to soil.
Journal: Environmental science & technology 20070501
Title: [Determination and distribution of sulfur compounds in coked gasoline by gas chromatography-sulfur chemiluminescence detection].
Journal: Se pu = Chinese journal of chromatography 20070501
Title: Raloxifene blocks estradiol induction of the serotonin transporter and 5-hydroxytryptamine2A receptor in female rat brain.
Journal: Neuroscience letters 20070424
Title: Desulfurization of liquid fuels by adsorption on carbon-based sorbents and ultrasound-assisted sorbent regeneration.
Journal: Langmuir : the ACS journal of surfaces and colloids 20070327
Title: Does aromaticity in a reaction product increase or decrease the intrinsic barrier? Kinetics of the reversible deprotonation of benzofuran-3(2H)-one and benzothiophene-3(2H)-one.
Journal: Journal of the American Chemical Society 20070307
Title: Chiral helicenoid diarylethene with large change in specific optical rotation by photochromism.
Journal: The Journal of organic chemistry 20070302
Title: The differential effects of bisphosphonates, SERMS (selective estrogen receptor modulators), and parathyroid hormone on bone remodeling in osteoporosis.
Journal: Clinical interventions in aging 20070301
Title: Potential sialyltransferase inhibitors based on neuraminyl substitution by hetaryl rings.
Journal: Carbohydrate research 20070226
Title: Medicinal chemistry and emerging strategies applied to the development of selective estrogen receptor modulators (SERMs).
Journal: Current medicinal chemistry 20070101
Title: Interactions of the human cytosolic sulfotransferases and steroid sulfatase in the metabolism of tibolone and raloxifene.
Journal: The Journal of steroid biochemistry and molecular biology 20070101
Title: Estrogenic or antiestrogenic therapies for multiple myeloma?
Journal: Molecular cancer 20070101
Title: Transition-metal/Lewis acid free synthesis of acyl benzothiophenes via C-C bond forming reaction.
Journal: Beilstein journal of organic chemistry 20070101
Title: GABA A/Bz receptor subtypes as targets for selective drugs.
Journal: Current medicinal chemistry 20070101
Title: Arzoxifene: the evidence for its development in the management of breast cancer.
Journal: Core evidence 20070101
Title: The cardiovascular effects of selective estrogen receptor modulators.
Journal: Annals of the New York Academy of Sciences 20061201
Title: A systematic resolution of sulfur in reticulated vitreous carbon using X-ray absorption spectroscopy.
Journal: Inorganic chemistry 20061127
Title: Syntheses and structures of novel heteroarene-fused coplanar pi-conjugated chromophores.
Journal: Organic letters 20061026
Title: Solid-phase synthesis of tetrahydro-beta-carbolines and tetrahydroisoquinolines by stereoselective intramolecular N-carbamyliminium Pictet-Spengler reactions.
Journal: Chemistry (Weinheim an der Bergstrasse, Germany) 20061025
Title: Synthesis and antimicrobial activity studies of ortho-chlorodiarylamines and heteroaromatic tetracyclic systems in the benzo[b]thiophene series.
Journal: Bioorganic & medicinal chemistry 20061015
Title: Sorption of heterocyclic organic compounds to reference soils: column studies for process identification.
Journal: Environmental science & technology 20061001
Title: Effect of ormeloxifene on ovariectomy-induced bone resorption, osteoclast differentiation and apoptosis and TGF beta-3 expression.
Journal: The Journal of steroid biochemistry and molecular biology 20060801
Title: Synthesis and evaluation of benzothiophene derivatives as ligands for imaging beta-amyloid plaques in Alzheimer's disease.
Journal: Nuclear medicine and biology 20060801
Title: The reaction of o-alkynylarene and heteroarene carboxaldehyde derivatives with iodonium ions and nucleophiles: a versatile and regioselective synthesis of 1H-isochromene, naphthalene, indole, benzofuran, and benzothiophene compounds.
Journal: Chemistry (Weinheim an der Bergstrasse, Germany) 20060724
Title: Gold-catalyzed intramolecular carbothiolation of alkynes: synthesis of 2,3-disubstituted benzothiophenes from (alpha-alkoxy alkyl) (ortho-alkynyl phenyl) sulfides.
Journal: Angewandte Chemie (International ed. in English) 20060703
Title: New HIV-1 reverse transcriptase inhibitors based on a tricyclic benzothiophene scaffold: synthesis, resolution, and inhibitory activity.
Journal: Bioorganic & medicinal chemistry letters 20060601
Title: Novel combretastatin analogues endowed with antitumor activity.
Journal: Journal of medicinal chemistry 20060601
Title: Chemical modification modulates estrogenic activity, oxidative reactivity, and metabolic stability in 4'F-DMA, a new benzothiophene selective estrogen receptor modulator.
Journal: Chemical research in toxicology 20060601
Title: [Isolation and characterization of a benzothiophene-desulfurizing bacterium].
Journal: Huan jing ke xue= Huanjing kexue 20060601
Title: Biodesulfurization of alkylated forms of dibenzothiophene and benzothiophene by Sphingomonas subarctica T7b.
Journal: Journal of bioscience and bioengineering 20060401
Title: Liquid-phase adsorption of multi-ring thiophenic sulfur compounds on carbon materials with different surface properties.
Journal: The journal of physical chemistry. B 20060316
Title: Evaluation of the antioxidant properties of diarylamines in the benzo[b]thiophene series by free radical scavenging activity and reducing power.
Journal: Bioorganic & medicinal chemistry letters 20060301
Title: Raloxifene: a selective estrogen-receptor modulator for postmenopausal osteoporosis - a clinical update on efficacy and safety.
Journal: Women's health (London, England) 20060301
Title: Characteristics of sulfur response in a micro-flame photometric detector.
Journal: Journal of chromatography. A 20060210
Title: Induction of apoptosis by photoexcited tetracyclic compounds derivatives of benzo[b]thiophenes and pyridines.
Journal: Journal of photochemistry and photobiology. B, Biology 20060201
Title: CFTR chloride channel drug discovery--inhibitors as antidiarrheals and activators for therapy of cystic fibrosis.
Journal: Current pharmaceutical design 20060101
Title: Benzothieno and benzofurano annelated estranes.
Journal: Steroids 20051201
Title: One-electron reduction potential for oxygen- and sulfur-centered organic radicals in protic and aprotic solvents.
Journal: Journal of the American Chemical Society 20051116
Title: Synthesis, characterization, and structure of cyclopenta[c]thiophenes and their manganese complexes.
Journal: Journal of the American Chemical Society 20051102
Title: Synthesis and biological activity of alpha-bromoacryloyl lexitropsin conjugates.
Journal: European journal of medicinal chemistry 20051101
Title: Carbonic anhydrase inhibitors: inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, and IX with benzo[b]thiophene 1,1-dioxide sulfonamides.
Journal: Bioorganic & medicinal chemistry letters 20051101
Title: Synthesis of oxadiazoles, thiadiazoles and triazoles derived from benzo[b]thiophene.
Journal: Molecules (Basel, Switzerland) 20050930
Title: Decoys for docking.
Journal: Journal of medicinal chemistry 20050602
Title: Hydroxylation activity of P450 BM-3 mutant F87V towards aromatic compounds and its application to the synthesis of hydroquinone derivatives from phenolic compounds.
Journal: Applied microbiology and biotechnology 20050601
Title: Biodesulfurization of dibenzothiophene and other organic sulfur compounds by a newly isolated Microbacterium strain ZD-M2.
Journal: FEMS microbiology letters 20050601
Title: Prediction of genotoxicity of chemical compounds by statistical learning methods.
Journal: Chemical research in toxicology 20050601
Title: Triplet-triplet energy transfer controlled by the donor-acceptor distance in rigidly held palladium-containing cofacial bisporphyrins.
Journal: Chemistry (Weinheim an der Bergstrasse, Germany) 20050520
Title: Selective adsorption of thiophene and 1-benzothiophene on metal-ion-exchanged zeolites in organic medium.
Journal: Journal of colloid and interface science 20050515
Title: Efficient access to 2-aryl-3-substituted benzo[b]thiophenes.
Journal: The Journal of organic chemistry 20050429
Title: Synthesis and binding affinities of novel SRIF-mimicking beta-D-glucosides satisfying the requirement for a pi-cloud at C1.
Journal: Organic letters 20050317
Title: Poly(thiaheterohelicene): a stiff conjugated helical polymer comprised of fused benzothiophene rings.
Journal: Organic letters 20050303
Title: Benzothiophenes containing a piperazine side chain as selective ligands for the estrogen receptor alpha and their bioactivities in vivo.
Journal: Bioorganic & medicinal chemistry letters 20050301
Title: Desulfurization of dibenzothiophene, benzothiophene, and other thiophene analogs by a newly isolated bacterium, Gordonia alkanivorans strain 1B.
Journal: Applied biochemistry and biotechnology 20050301
Title: Benzo[b]thiophenesulphonamide 1,1-dioxide derivatives inhibit tNOX activity in a redox state-dependent manner.
Journal: British journal of cancer 20050227
Title: In vitro metabolic fate of a novel structural class: evidence for the formation of a reactive intermediate on a benzothiophene moiety.
Journal: Chemico-biological interactions 20050227
Title: Design, synthesis, and biological evaluation of novel potent and selective alphavbeta3/alphavbeta5 integrin dual inhibitors with improved bioavailability. Selection of the molecular core.
Journal: Journal of medicinal chemistry 20050224
Title: Simultaneous determination of NSO-heterocycles, homocycles and their metabolites in groundwater of tar oil contaminated sites using LC with diode array UV and fluorescence detection.
Journal: Journal of chromatography. A 20050218
Title: Organoboron compounds with an 8-hydroxyquinolato chelate and its derivatives: substituent effects on structures and luminescence.
Journal: Inorganic chemistry 20050207
Title: Thermophilic biodesulfurization of various heterocyclic sulfur compounds and crude straight-run light gas oil fraction by a newly isolated strain Mycobacterium phlei WU-0103.
Journal: Current microbiology 20050201
Title: Endocrinology and hormone therapy in breast cancer: selective oestrogen receptor modulators and downregulators for breast cancer - have they lost their way?
Journal: Breast cancer research : BCR 20050101
Title: Benefit-risk assessment of raloxifene in postmenopausal osteoporosis.
Journal: Drug safety 20050101
Title: Adsorption, desorption, and conversion of thiophene on H-ZSM5.
Journal: Langmuir : the ACS journal of surfaces and colloids 20041207
Title: Screening of antimicrobial activity of diarylamines in the 2,3,5-trimethylbenzo[b]thiophene series: a structure-activity evaluation study.
Journal: Bioorganic & medicinal chemistry letters 20041206
Title: Synthesis and NMR spectroscopic studies of allylsulfanyl-N1-alkyl-N4-phenyl-1,4-phenylenediamines and their cyclization products, 2,3-dihydro-1-benzothiophenes and thiochromans.
Journal: Magnetic resonance in chemistry : MRC 20041201
Title: Palladium-catalyzed tandem reaction of yne-propargylic carbonates with boronic acids: a simple method for the synthesis of fused aromatic rings through allene-mediated electrocyclization.
Journal: Chemistry (Weinheim an der Bergstrasse, Germany) 20041025
Title: Benzothiophene and naphthalene derived constrained SERMs.
Journal: Bioorganic & medicinal chemistry letters 20041018
Title: Phenylpiperazinylmethylheterocycle derivatives: synthesis and dopamine receptor binding profiles.
Journal: Archiv der Pharmazie 20040701
Title: New 3-[4-(2,3-dihydro-14-benzodioxin-5-yl)piperazin-1-yl]-1-(5-substituted benzo[b]thiophen-3-yl)propanol derivatives with dual action at 5-HT(1A) serotonin receptors and serotonin transporter as a new class of antidepressants.
Journal: Die Pharmazie 20040701
Title: C17,20-lyase inhibitors I. Structure-based de novo design and SAR study of C17,20-lyase inhibitors.
Journal: Bioorganic & medicinal chemistry 20040501
Title: [Determination of sulfur compounds in fluid catalytic cracking gasoline by gas chromatography with a sulfur chemiluminescence detector].
Journal: Se pu = Chinese journal of chromatography 20040501
Title: Synthesis and serotonergic activity of variously substituted (3-amido)phenylpiperazine derivatives and benzothiophene-4-piperazine derivatives: novel antagonists for the vascular 5-HT1B receptor.
Journal: European journal of medicinal chemistry 20040401
Title: Discovery of novel heteroaryl-substituted chalcones as inhibitors of TNF-alpha-induced VCAM-1 expression.
Journal: Bioorganic & medicinal chemistry letters 20040322
Title: Design, synthesis and structure-activity relationship of novel RXR-selective modulators.
Journal: Bioorganic & medicinal chemistry letters 20040322
Title: Efficient isomer-pure synthesis of a benzo[b]thiophene analogue of pentacene.
Journal: The Journal of organic chemistry 20040319
Title: Synthesis and cytotoxic activity of lipophilic sulphonamide derivatives of the benzo[b]thiophene 1,1-dioxide.
Journal: Bioorganic & medicinal chemistry 20040301
Title: Synthesis of new thiophene and benzo[b]thiophene hydrazide derivatives as human NPY Y(5) antagonists.
Journal: Bioorganic & medicinal chemistry letters 20040209
Title: A synthesis of heteroaromatic analogues of 1-methyl-1,2,3,4-tetrahydroisoquinoline using the Pummerer-type cyclization reaction: observation of tandem cyclization reaction.
Journal: Chemical & pharmaceutical bulletin 20040201
Title: Elimination of sulfur from aromatic heterocycles by a water-soluble arene ruthenium cluster: synthesis and molecular structure of [H2S2Ru4(C6H6)4]Cl2.
Journal: Chemical communications (Cambridge, England) 20040121
Title: Modulation of selective serotonin reuptake inhibitor and 5-HT1A antagonist activity in 8-aza-bicyclo[3.2.1]octane derivatives of 2,3-dihydro-1,4-benzodioxane.
Journal: Bioorganic & medicinal chemistry letters 20040119
Title: Combined application of stable carbon isotope analysis and specific metabolites determination for assessing in situ degradation of aromatic hydrocarbons in a tar oil-contaminated aquifer.
Journal: Environmental science & technology 20040115
Title: Advances in estrogen receptor biology: prospects for improvements in targeted breast cancer therapy.
Journal: Breast cancer research : BCR 20040101
Title: Potent inhibition of human liver aldehyde oxidase by raloxifene.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20040101
Title: NH2-SEP-PAK cartridges for enrichment of Aromatic Sulfur Compounds from sea water: determination by GC-FID and GC-MS.
Journal: Annali di chimica 20040101
Title: Monitoring toxicity of industrial wastewater and specific chemicals to a green alga, nitrifying bacteria and an aquatic bacterium.
Journal: Water science and technology : a journal of the International Association on Water Pollution Research 20040101
Title: Structure-activity relationship of benzo[b]thiophene-2-sulfonamide derivatives as novel human chymase inhibitors.
Journal: Bioorganic & medicinal chemistry letters 20031117
Title: Reactions that generate aromatic molecules: is aromatic stabilization less or more advanced than bond changes at the transition state? Kinetic and thermodynamic acidities of rhenium carbene complexes.
Journal: Journal of the American Chemical Society 20031008
Title: Nitrosation, nitration, and autoxidation of the selective estrogen receptor modulator raloxifene by nitric oxide, peroxynitrite, and reactive nitrogen/oxygen species.
Journal: Chemical research in toxicology 20031001
Title: 2,6-disubstituted pyran-4-one and thiopyran-4-one inhibitors of DNA-Dependent protein kinase (DNA-PK).
Journal: Bioorganic & medicinal chemistry letters 20030915
Title: 2-(2'-Hydroxyphenyl)benzene sulfinate desulfinase from the thermophilic desulfurizing bacterium Paenibacillus sp. strain A11-2: purification and characterization.
Journal: Applied microbiology and biotechnology 20030901
Title: Synthesis and binding affinities of fluoroalkylated raloxifenes.
Journal: Bioorganic & medicinal chemistry 20030815
Title: Target specificity of selective estrogen receptor modulators within human endometrial cancer cells.
Journal: The Journal of steroid biochemistry and molecular biology 20030701
Title: Diastereoselective photochromism of a bisbenzothienylethene governed by steric as well as electronic interactions.
Journal: Journal of the American Chemical Society 20030618
Title: Preparation and characterization of organotin-oxomolybdate coordination polymers and their use in sulfoxidation catalysis.
Journal: Chemistry (Weinheim an der Bergstrasse, Germany) 20030616
Title: New benzo(b)thiophenesulphonamide 1,1-dioxide derivatives induce a reactive oxygen species-mediated process of apoptosis in tumour cells.
Journal: Oncogene 20030612
Title: Anaerobic desulphurisation of thiophenes by mixed microbial communities from oilfields.
Journal: Biodegradation 20030601
Title: The effect of minor-groove hydrogen-bond acceptors and donors on the stability and replication of four unnatural base pairs.
Journal: Journal of the American Chemical Society 20030521
Title: New fibrinolytic agents: benzothiophene derivatives as inhibitors of the t-PA-PAI-1 complex formation.
Journal: Bioorganic & medicinal chemistry letters 20030519
Title: Discovery and characterization of a potent and selective non-amidine inhibitor of human factor Xa.
Journal: Biochemical pharmacology 20030501
Title: Selective estrogen receptor modulators.
Journal: Southern medical journal 20030501
Title: Hydrogenation and carbon-sulfur bond hydrogenolysis of benzothiophene promoted by Re2(CO)10 and H4Re4(CO)12.
Journal: Inorganic chemistry 20030407
Title: Effect of treatment with the selective oestrogen receptor modulator LY117018-HCl on pituitary sensitivity to GnRH and subsequent ovulation.
Journal: Reproduction (Cambridge, England) 20030401
Title: Design, synthesis and in vitro evaluation of novel benzo[b]thiophene derivatives as serotonin N-acetyltransferase (AANAT) inhibitors.
Journal: Journal of enzyme inhibition and medicinal chemistry 20030401
Title: Photochemistry and photophysics of thienocarbazoles.
Journal: Photochemistry and photobiology 20030201
Title: Advances in breast cancer treatment and prevention: preclinical studies on aromatase inhibitors and new selective estrogen receptor modulators (SERMs).
Journal: Breast cancer research : BCR 20030101
Title: Crystal structures of two potent nonamidine inhibitors bound to factor Xa.
Journal: Biochemistry 20021231
Title: [Determination of sulfur compounds in catalytic diesel oil by gas chromatography with atomic emission detector and its applications].
Journal: Se pu = Chinese journal of chromatography 20021101
Title: Recombinant Rhodococcus sp. strain T09 can desulfurize DBT in the presence of inorganic sulfate.
Journal: Current microbiology 20021001
Title: Purification and characterization of the monooxygenase catalyzing sulfur-atom specific oxidation of dibenzothiophene and benzothiophene from the thermophilic bacterium Paenibacillus sp. strain A11-2.
Journal: Applied microbiology and biotechnology 20021001
Title: 4-Substituted D-glutamic acid analogues: the first potent inhibitors of glutamate racemase (MurI) enzyme with antibacterial activity.
Journal: Journal of medicinal chemistry 20020926
Title: Synthesis and molecular modeling of new 1-aryl-3-[4-arylpiperazin-1-yl]-1-propane derivatives with high affinity at the serotonin transporter and at 5-HT(1A) receptors.
Journal: Journal of medicinal chemistry 20020912
Title: Isolation and characterization of a moderate thermophile, Mycobacterium phlei GTIS10, capable of dibenzothiophene desulfurization.
Journal: Applied microbiology and biotechnology 20020901
Title: Synthesis of fluoren-9-ones by the palladium-catalyzed cyclocarbonylation of o-halobiaryls.
Journal: The Journal of organic chemistry 20020809
Title: Geochemical and physiological evidence for mixed aerobic and anaerobic field biodegradation of coal tar waste by subsurface microbial communities.
Journal: Microbial ecology 20020801
Title: Biodesulfurization of naphthothiophene and benzothiophene through selective cleavage of carbon-sulfur bonds by Rhodococcus sp. strain WU-K2R.
Journal: Applied and environmental microbiology 20020801
Title: Analysis of aromatic sulfur compounds in gas oils using GC with sulfur chemiluminescence detection and high-resolution MS.
Journal: Analytical chemistry 20020801
Title: Biodesulfurization of benzothiophene and dibenzothiophene by a newly isolated Rhodococcus strain.
Journal: Applied microbiology and biotechnology 20020701
Title: Cytochrome P450 3A4-mediated bioactivation of raloxifene: irreversible enzyme inhibition and thiol adduct formation.
Journal: Chemical research in toxicology 20020701
Title: One-pot synthesis of benzo[b]furan and indole inhibitors of tubulin polymerization.
Journal: Journal of medicinal chemistry 20020606
Title: New 3-[4-(aryl)piperazin-1-yl]-1-(benzo[b]thiophen-2-yl)propane derivatives with dual action at 5-HT1A serotonin receptors and serotonin transporter as a new class of antidepressants.
Journal: Die Pharmazie 20020601
Title: Benzoyl and cinnamoyl nitrogen mustard derivatives of benzoheterocyclic analogues of the tallimustine: synthesis and antitumour activity.
Journal: Bioorganic & medicinal chemistry 20020501
Title: Macrophage inducible nitric oxide synthase gene expression is blocked by a benzothiophene derivative with anti-HIV properties.
Journal: Molecular genetics and metabolism 20020401
Title: Toward selective ERbeta agonists for central nervous system disorders: synthesis and characterization of aryl benzthiophenes.
Journal: Journal of medicinal chemistry 20020328
Title: Metabolic response against sulfur-containing heterocyclic compounds by the lignin-degrading basidiomycete Coriolus versicolor.
Journal: Applied microbiology and biotechnology 20020301
Title: Re(2)(CO)(10)-promoted S-binding, C-S bond cleavage, and hydrogenation of benzothiophenes: organometallic models for the hydrodesulfurization of thiophenes.
Journal: Journal of the American Chemical Society 20020227
Title: Aerobic co-metabolism of sulfur, nitrogen and oxygen heterocycles by three marine bacterial consortia.
Journal: Journal of basic microbiology 20020101
Title: Isolation and characterization of thermophilic benzothiophene-degrading Mycobacterium sp.
Journal: Applied biochemistry and biotechnology 20020101
Title: Physical organic chemistry of transition metal carbene complexes. 23. Kinetic and thermodynamic acidities of cationic benzothienyl- and selenylcarbene complexes of rhenium in aqueous acetonitrile.
Journal: Journal of the American Chemical Society 20011205
Title: Raloxifene.
Journal: Current drug targets 20011201
Title: Effects of the new selective estrogen receptor modulator LY353381.HCl (Arzoxifene) on human endometrial cancer growth in athymic mice.
Journal: Clinical cancer research : an official journal of the American Association for Cancer Research 20011201
Title: Synthesis and studies on spectroscopic as well as electron donating properties of the two alkoxy benzo[b]thiophenes.
Journal: Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy 20011201
Title: Selective estrogen receptor modulator effects on serum lipoproteins and vascular function in postmenopausal women and in hypercholesterolemic men.
Journal: Annals of the New York Academy of Sciences 20011201
Title: New cytotoxic benzo(b)thiophenilsulfonamide 1,1-dioxide derivatives inhibit a NADH oxidase located in plasma membranes of tumour cells.
Journal: British journal of cancer 20011101
Title: Benzo[b]thiophene desulfurization by Gordonia rubropertinctus strain T08.
Journal: Applied microbiology and biotechnology 20011001
Title: Desulfurization of benzothiophene by the Gram-negative bacterium, Sinorhizobium sp. KT55.
Journal: Current microbiology 20010901
Title: 1-(2-[4-[6-Hydroxy-2-(4-hydroxyphenyl)benzo[b]thiol-3-ylcarbonyl]phenoxy]ethyl)piperidinium chloride.
Journal: Acta crystallographica. Section C, Crystal structure communications 20010901
Title: Effect of raloxifene on serum triglycerides in postmenopausal women: influence of predisposing factors for hypertriglyceridemia.
Journal: Clinical therapeutics 20010901
Title: Identification and characterization of a benzothiophene inhibitor of herpes simplex virus type 1 replication which acts at the immediate early stage of infection.
Journal: Antiviral research 20010801
Title: Analysis of cross-resistance of the selective estrogen receptor modulators arzoxifene (LY353381) and LY117018 in tamoxifen-stimulated breast cancer xenografts.
Journal: Clinical cancer research : an official journal of the American Association for Cancer Research 20010801
Title: Microbial desulfurization of alkylated dibenzothiophene and alkylated benzothiophene by recombinant Rhodococcus sp. strain T09.
Journal: Applied microbiology and biotechnology 20010701
Title: Phase I study of a third-generation selective estrogen receptor modulator, LY353381.HCL, in metastatic breast cancer.
Journal: Journal of clinical oncology : official journal of the American Society of Clinical Oncology 20010401
Title: A novel palladium-mediated coupling approach to 2,3-disubstituted benzo(b)thiophenes and its application to the synthesis of tubulin binding agents.
Journal: Organic letters 20010308
Title: Electron transfer compatible molecular design of benzothiophene-acetophenone bichromophores: a theoretical approach.
Journal: Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy 20010301
Title: Update on endocrine aspects of breast cancer: report from the 23rd San Antonio Breast Cancer Symposium, San Antonio, Texas, USA, 6-9 December 2000.
Journal: Breast cancer research : BCR 20010101
Title: Selective estrogen receptor modulators: mechanism of action and clinical experience. Focus on raloxifene.
Journal: Reproduction, fertility, and development 20010101
Title: Raloxifene: another selective estrogen modulator.
Journal: In vivo (Athens, Greece) 20010101
Title: Isolation of a unique benzothiophene-desulphurizing bacterium, Gordona sp. strain 213E (NCIMB 40816), and characterization of the desulphurization pathway.
Journal: Microbiology (Reading, England) 19980901
Title: Synthesis and in vitro LTD4 antagonist activity of bicyclic and monocyclic cyclopentylurethane and cyclopentylacetamide N-arylsulfonyl amides.
Journal: Journal of medicinal chemistry 19900901
