Title: A semi-quantitative translational pharmacology analysis to understand the relationship between in vitro ENT1 inhibition and the clinical incidence of dyspnoea and bronchospasm.
Journal: Toxicology and applied pharmacology 20170215
Title: Decreased extracellular adenosine levels lead to loss of hypoxia-induced neuroprotection after repeated episodes of exposure to hypoxia.
Journal: PloS one 20130101
Title: Cysteine residues in the transmembrane (TM) 9 to TM11 region of the human equilibrative nucleoside transporter subtype 1 play an important role in inhibitor binding and translocation function.
Journal: Molecular pharmacology 20121101
Title: Adenosine-mediated cardiovascular toxicity in amitriptyline-poisoned rats.
Journal: Drug and chemical toxicology 20121001
Title: Expression of A1 adenosine receptors in the developing avian retina: in vivo modulation by A(2A) receptors and endogenous adenosine.
Journal: Journal of neurochemistry 20121001
Title: On-pump inhibition of es-ENT1 nucleoside transporter and adenosine deaminase during aortic crossclamping entraps intracellular adenosine and protects against reperfusion injury: role of adenosine A1 receptor.
Journal: The Journal of thoracic and cardiovascular surgery 20120701
Title: Myocardial protection in beating heart cardiac surgery: I: pre- or postconditioning with inhibition of es-ENT1 nucleoside transporter and adenosine deaminase attenuates post-MI reperfusion-mediated ventricular fibrillation and regional contractile dysfunction.
Journal: The Journal of thoracic and cardiovascular surgery 20120701
Title: Microwave-promoted 'one-pot' synthesis of 4-nitrobenzylthioinosine analogues using thiourea as a sulfur precursor.
Journal: Chemistry, an Asian journal 20120102
Title: Inhibition of hippocampal synaptic activity by ATP, hypoxia or oxygen-glucose deprivation does not require CD73.
Journal: PloS one 20120101
Title: Insulin-increased L-arginine transport requires A(2A) adenosine receptors activation in human umbilical vein endothelium.
Journal: PloS one 20120101
Title: Adenosine negatively regulates duodenal motility in mice: role of A(1) and A(2A) receptors.
Journal: British journal of pharmacology 20111101
Title: Differential adenosine uptake in mixed neuronal/glial or purified glial cultures of avian retinal cells: modulation by adenosine metabolism and the ERK cascade.
Journal: Biochemical and biophysical research communications 20111014
Title: Behavioral effects of elevated expression of human equilibrative nucleoside transporter 1 in mice.
Journal: Behavioural brain research 20111010
Title: Expression of human equilibrative nucleoside transporter 1 in mouse neurons regulates adenosine levels in physiological and hypoxic-ischemic conditions.
Journal: Journal of neurochemistry 20110701
Title: Variability in transport and biotransformation of cytarabine is associated with its toxicity in peripheral blood mononuclear cells.
Journal: Pharmacogenomics 20110401
Title: Membrane transport of sepiapterin and dihydrobiopterin by equilibrative nucleoside transporters: a plausible gateway for the salvage pathway of tetrahydrobiopterin biosynthesis.
Journal: Molecular genetics and metabolism 20110101
Title: Antimutagenic, antigenotoxic and antioxidant activities of phenolic-enriched extracts from Teucrium ramosissimum: combination with their phytochemical composition.
Journal: Environmental toxicology and pharmacology 20110101
Title: Endogenous luminal surface adenosine signaling regulates duodenal bicarbonate secretion in rats.
Journal: The Journal of pharmacology and experimental therapeutics 20101201
Title: Testicular expression of Adora3i2 in Adora3 knockout mice reveals a role of mouse A3Ri2 and human A3Ri3 adenosine receptors in sperm.
Journal: The Journal of biological chemistry 20101029
Title: Differential expression of functional nucleoside transporters in non-differentiated and differentiated human endothelial progenitor cells.
Journal: Placenta 20101001
Title: Characterization of mammalian equilibrative nucleoside transporters (ENTs) by mass spectrometry.
Journal: Protein expression and purification 20100901
Title: Photoreactivity of carboxylated single-walled carbon nanotubes in sunlight: reactive oxygen species production in water.
Journal: Environmental science & technology 20100901
Title: Biodistribution and uptake of 3'-deoxy-3'-fluorothymidine in ENT1-knockout mice and in an ENT1-knockdown tumor model.
Journal: Journal of nuclear medicine : official publication, Society of Nuclear Medicine 20100901
Title: Improved syntheses of 5'-S-(2-aminoethyl)-6-N-(4-nitrobenzyl)-5'-thioadenosine (SAENTA), analogues, and fluorescent probe conjugates: analysis of cell-surface human equilibrative nucleoside transporter 1 (hENT1) levels for prediction of the antitumor efficacy of gemcitabine.
Journal: Journal of medicinal chemistry 20100826
Title: Excitatory synaptic transmission in the spinal substantia gelatinosa is under an inhibitory tone of endogenous adenosine.
Journal: Neuroscience letters 20100614
Title: Immunomodulatory effects of proanthocyanidin A-1 derived in vitro from Rhododendron spiciferum.
Journal: Fitoterapia 20100301
Title: Kinetic study of anti-viral ribavirin uptake mediated by hCNT3 and hENT1 in Xenopus laevis oocytes.
Journal: Biophysical chemistry 20100301
Title: Compensatory upregulation of the adenosine system following phenylephrine-induced hypertrophy in cultured rat ventricular myocytes.
Journal: American journal of physiology. Heart and circulatory physiology 20100201
Title: Expression and functional activity of nucleoside transporters in human choroid plexus.
Journal: Cerebrospinal fluid research 20100101
Title: Human erythrocyte nucleoside transporter ENT1 functions at ice-cold temperatures.
Journal: Drug metabolism and pharmacokinetics 20100101
Title: Genetic mapping of targets mediating differential chemical phenotypes in Plasmodium falciparum.
Journal: Nature chemical biology 20091001
Title: Synthesis of radiolabeled cytarabine conjugates.
Journal: Bioorganic & medicinal chemistry letters 20090815
Title: Negative crosstalk between M1 and M2 muscarinic autoreceptors involves endogenous adenosine activating A1 receptors at the rat motor endplate.
Journal: Neuroscience letters 20090814
Title: Prevention of early loss of transplanted islets in the liver of mice by adenosine.
Journal: Transplantation 20090715
Title: Inhibitory effect of nonsteroidal anti-inflammatory drugs on adenosine transport in vascular smooth muscle cells.
Journal: European journal of pharmacology 20090610
Title: TGF-beta1 inhibits expression and activity of hENT1 in a nitric oxide-dependent manner in human umbilical vein endothelium.
Journal: Cardiovascular research 20090601
Title: Metformin prevents myocardial reperfusion injury by activating the adenosine receptor.
Journal: Journal of cardiovascular pharmacology 20090501
Title: Ethanol blocks adenosine uptake via inhibiting the nucleoside transport system in bronchial epithelial cells.
Journal: Alcoholism, clinical and experimental research 20090501
Title: The role of the equilibrative nucleoside transporter 1 (ENT1) in transport and metabolism of ribavirin by human and wild-type or Ent1-/- mouse erythrocytes.
Journal: The Journal of pharmacology and experimental therapeutics 20090401
Title: Modulation of gamma oscillations by endogenous adenosine through A1 and A2A receptors in the mouse hippocampus.
Journal: Neuropharmacology 20090201
Title: Synthesis and biological evaluation of phloridzin analogs as human concentrative nucleoside transporter 3 (hCNT3) inhibitors.
Journal: Bioorganic & medicinal chemistry letters 20090201
Title: Identification of a novel point mutation in ENT1 that confers resistance to Ara-C in human T cell leukemia CCRF-CEM cells.
Journal: FEBS letters 20090122
Title: CoMFA and CoMSIA 3D-QSAR studies on S(6)-(4-nitrobenzyl)mercaptopurine riboside (NBMPR) analogs as inhibitors of human equilibrative nucleoside transporter 1 (hENT1).
Journal: Bioorganic & medicinal chemistry letters 20090115
Title: Activation of adenosine A2B receptors enhances ciliary beat frequency in mouse lateral ventricle ependymal cells.
Journal: Cerebrospinal fluid research 20090101
Title: Contribution of Na+-independent nucleoside transport to ribavirin uptake in the rat intestine and human epithelial LS180 cells.
Journal: European journal of pharmacology 20081228
Title: The role of ecto-5'-nucleotidase/CD73 in glioma cell line proliferation.
Journal: Molecular and cellular biochemistry 20081201
Title: Enhancing brain adenosine signaling with the nucleoside transport blocker NBTI (S-(4-nitrobenzyl)-6-theoinosine) mimics the effects of inescapable shock on later shuttle-escape performance in rats.
Journal: Behavioral neuroscience 20081201
Title: Imatinib inhibition of fludarabine uptake in T-lymphocytes.
Journal: Cancer chemotherapy and pharmacology 20080901
Title: Mutation of Trp29 of human equilibrative nucleoside transporter 1 alters affinity for coronary vasodilator drugs and nucleoside selectivity.
Journal: The Biochemical journal 20080901
Title: Inosine and equilibrative nucleoside transporter 2 contribute to hypoxic preconditioning in the murine cardiomyocyte HL-1 cell line.
Journal: American journal of physiology. Heart and circulatory physiology 20080601
Title: Uridine protects cortical neurons from glucose deprivation-induced death: possible role of uridine phosphorylase.
Journal: Journal of neurotrauma 20080601
Title: Cytotoxic activities of nucleoside and nucleobase analog drugs in malignant mesothelioma: characterization of a novel nucleobase transport activity.
Journal: Biochemical pharmacology 20080515
Title: Potential of various drugs to inhibit nucleoside uptake in rat syncytiotrophoblast cell line, TR-TBT 18d-1.
Journal: Placenta 20080501
Title: Constrained NBMPR analogue synthesis, pharmacophore mapping and 3D-QSAR modeling of equilibrative nucleoside transporter 1 (ENT1) inhibitory activity.
Journal: Bioorganic & medicinal chemistry 20080401
Title: Kinetics of nucleoside uptake by the basolateral side of the sheep choroid plexus epithelium perfused in situ.
Journal: Experimental physiology 20080301
Title: Cyclic ADP-ribose mediates formyl methionyl leucyl phenylalanine (fMLP)-induced intracellular Ca(2+) rise and migration of human neutrophils.
Journal: Journal of pharmacological sciences 20080301
Title: Generation of superoxide from reaction of 3H-1,2-dithiole-3-thione with thiols: implications for dithiolethione chemoprotection.
Journal: Molecular and cellular biochemistry 20080101
Title: Tuning adenosine A1 and A2A receptors activation mediates L-citrulline-induced inhibition of [3H]-acetylcholine release depending on nerve stimulation pattern.
Journal: Neurochemistry international 20080101
Title: Adenosine uptake-dependent C6 cell growth inhibition.
Journal: European journal of pharmacology 20071222
Title: Novel C2-purine position analogs of nitrobenzylmercaptopurine riboside as human equilibrative nucleoside transporter 1 inhibitors.
Journal: Bioorganic & medicinal chemistry 20071215
Title: Nucleoside and nucleobase transporters of primary human cardiac microvascular endothelial cells: characterization of a novel nucleobase transporter.
Journal: American journal of physiology. Heart and circulatory physiology 20071201
Title: Synthesis, flow cytometric evaluation, and identification of highly potent dipyridamole analogues as equilibrative nucleoside transporter 1 inhibitors.
Journal: Journal of medicinal chemistry 20070809
Title: Nucleoside transporter expression and activity is regulated during granulocytic differentiation of NB4 cells in response to all-trans-retinoic acid.
Journal: Leukemia research 20070701
Title: Localization of broadly selective equilibrative and concentrative nucleoside transporters, hENT1 and hCNT3, in human kidney.
Journal: American journal of physiology. Renal physiology 20070701
Title: Cardioprotective effects of novel tetrahydroisoquinoline analogs of nitrobenzylmercaptopurine riboside in an isolated perfused rat heart model of acute myocardial infarction.
Journal: American journal of physiology. Heart and circulatory physiology 20070601
Title: L-citrulline inhibits [3H]acetylcholine release from rat motor nerve terminals by increasing adenosine outflow and activation of A1 receptors.
Journal: British journal of pharmacology 20070601
Title: Temporal and mechanistic dissociation of ATP and adenosine release during ischaemia in the mammalian hippocampus.
Journal: Journal of neurochemistry 20070601
Title: Nucleoside transporter expression and adenosine uptake in the rat cochlea.
Journal: Neuroreport 20070212
Title: Characterization of resistance to cytosine arabinoside (Ara-C) in NALM-6 human B leukemia cells.
Journal: Clinica chimica acta; international journal of clinical chemistry 20070201
Title: A novel mechanism of vasoregulation: ADP-induced relaxation of the porcine isolated coronary artery is mediated via adenosine release.
Journal: FASEB journal : official publication of the Federation of American Societies for Experimental Biology 20070201
Title: Influence of hyperthyroidism on the effect of adenosine transport blockade assessed by a novel method in guinea pig atria.
Journal: Cell biochemistry and biophysics 20070101
Title: Human equilibrative nucleoside transporter 1, as a predictor of 5-fluorouracil resistance in human pancreatic cancer.
Journal: Anticancer research 20070101
Title: Insulin restores glucose inhibition of adenosine transport by increasing the expression and activity of the equilibrative nucleoside transporter 2 in human umbilical vein endothelium.
Journal: Journal of cellular physiology 20061201
Title: Insulin restores metabolic function in cultured cortical neurons subjected to oxidative stress.
Journal: Diabetes 20061001
Title: Uridine prevents the glucose deprivation-induced death of immunostimulated astrocytes via the action of uridine phosphorylase.
Journal: Neuroscience research 20060901
Title: In vitro synergistic cytotoxicity of gemcitabine and pemetrexed and pharmacogenetic evaluation of response to gemcitabine in bladder cancer patients.
Journal: British journal of cancer 20060807
Title: Alkyl-fluorinated thymidine derivatives for imaging cell proliferation I. The in vitro evaluation of some alkyl-fluorinated thymidine derivatives.
Journal: Nuclear medicine and biology 20060801
Title: The role of human nucleoside transporters in cellular uptake of 4'-thio-beta-D-arabinofuranosylcytosine and beta-D-arabinosylcytosine.
Journal: Molecular pharmacology 20060701
Title: Genetic interdependence of adenosine and dopamine receptors: evidence from receptor knockout mice.
Journal: Neuroscience 20060512
Title: Characterization of novel Na+-dependent nucleobase transport systems at the blood-testis barrier.
Journal: American journal of physiology. Endocrinology and metabolism 20060501
Title: Microsphere-based protease assays and screening application for lethal factor and factor Xa.
Journal: Cytometry. Part A : the journal of the International Society for Analytical Cytology 20060501
Title: Studies of nucleoside transporters using novel autofluorescent nucleoside probes.
Journal: Biochemistry 20060131
Title: In-vitro and in-vivo anti-cancer activity of a novel gemcitabine-cardiolipin conjugate.
Journal: Anti-cancer drugs 20060101
Title: Effect of nucleoside transport blockade on the interstitial adenosine level characterized by a novel method in guinea pig atria.
Journal: Journal of cardiovascular pharmacology 20060101
Title: 6-Benzylthioinosine analogues: promising anti-toxoplasmic agents as inhibitors of the mammalian nucleoside transporter ENT1 (es).
Journal: Biochemical pharmacology 20051219
Title: Effects on sleep of microdialysis of adenosine A1 and A2a receptor analogs into the lateral preoptic area of rats.
Journal: American journal of physiology. Regulatory, integrative and comparative physiology 20051201
Title: ATP- and adenosine-induced relaxation of the smooth muscle of the pig urethra.
Journal: BJU international 20051201
Title: Inosine infusion prevents mortality in endotoxic shock.
Journal: The Journal of trauma 20051201
Title: 2-n-Butyl-9-methyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine and analogues as A2A adenosine receptor antagonists. Design, synthesis, and pharmacological characterization.
Journal: Journal of medicinal chemistry 20051103
Title: Localization of the NBMPR-sensitive equilibrative nucleoside transporter, ENT1, in the rat dorsal root ganglion and lumbar spinal cord.
Journal: Brain research 20051019
Title: Adenosine down-regulates giant depolarizing potentials in the developing rat hippocampus by exerting a negative control on glutamatergic inputs.
Journal: Journal of neurophysiology 20051001
Title: Adenosine and deoxyadenosine induces apoptosis in oestrogen receptor-positive and -negative human breast cancer cells via the intrinsic pathway.
Journal: Cell proliferation 20051001
Title: Equilibrative nucleoside transporter 1 expression is downregulated by hypoxia in human umbilical vein endothelium.
Journal: Circulation research 20050708
Title: Adenosine and purine nucleosides prevent the disruption of mitochondrial transmembrane potential by peroxynitrite in rat primary astrocytes.
Journal: Archives of pharmacal research 20050701
Title: D-Glucose upregulates adenosine transport in cultured human aortic smooth muscle cells.
Journal: American journal of physiology. Heart and circulatory physiology 20050601
Title: 6-Benzylthioinosine analogues as subversive substrate of Toxoplasma gondii adenosine kinase: activities and selective toxicities.
Journal: Biochemical pharmacology 20050515
Title: Purine nucleosides stimulate Na/K ATPase, and prolong survival in hemorrhagic shock.
Journal: The Journal of trauma 20050501
Title: Subtype-specific regulation of equilibrative nucleoside transporters by protein kinase CK2.
Journal: The Biochemical journal 20050301
Title: Residues Met89 and Ser160 in the human equilibrative nucleoside transporter 1 affect its affinity for adenosine, guanosine, S6-(4-nitrobenzyl)-mercaptopurine riboside, and dipyridamole.
Journal: Molecular pharmacology 20050301
Title: Astrocytes and neurons: different roles in regulating adenosine levels.
Journal: Neurological research 20050301
Title: Nucleoside transport at the blood-testis barrier studied with primary-cultured sertoli cells.
Journal: The Journal of pharmacology and experimental therapeutics 20050201
Title: An investigation of binding sites for paracetamol in the mouse brain and spinal cord.
Journal: European journal of pharmacology 20050131
Title: Inhibition of nucleoside transport proteins by C8-alkylamine-substituted purines.
Journal: Journal of medicinal chemistry 20050113
Title: Protective effect of adenosine and purine nucleos(t)ides against the death by hydrogen peroxide and glucose deprivation in rat primary astrocytes.
Journal: Neuroscience research 20050101
Title: Adenosine kinase inhibitor attenuates the expression of inducible nitric oxide synthase in glial cells.
Journal: Neuropharmacology 20050101
Title: Brain penetration of synthetic adenosine A1 receptor agonists in situ: role of the rENT1 nucleoside transporter and binding to blood constituents.
Journal: European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences 20050101
Title: Equilibrative nucleoside transporter 2 is expressed in human umbilical vein endothelium, but is not involved in the inhibition of adenosine transport induced by hyperglycaemia.
Journal: Placenta 20050101
Title: Fine tuning of rabbit equilibrative nucleoside transporter activity by an alternatively spliced variant.
Journal: Journal of drug targeting 20050101
Title: Transport of endogenous nucleosides in guinea pig heart.
Journal: Canadian journal of physiology and pharmacology 20041201
Title: CPEC induces erythroid differentiation of human myeloid leukemia K562 cells through CTP depletion and p38 MAP kinase.
Journal: Leukemia 20041101
Title: Quantitative autoradiography of adenosine receptors and NBTI-sensitive adenosine transporters in the brains of mice deficient in the preproenkephalin gene.
Journal: Brain research 20041029
Title: Tetanic depression is overcome by tonic adenosine A(2A) receptor facilitation of L-type Ca(2+) influx into rat motor nerve terminals.
Journal: The Journal of physiology 20041001
Title: Nucleoside transporter subtype expression and function in rat skeletal muscle microvascular endothelial cells.
Journal: British journal of pharmacology 20040901
Title: Determinants of sensitivity and resistance to gemcitabine: the roles of human equilibrative nucleoside transporter 1 and deoxycytidine kinase in non-small cell lung cancer.
Journal: Cancer science 20040901
Title: Regulation by equilibrative nucleoside transporter of adenosine outward currents in adult rat spinal dorsal horn neurons.
Journal: Brain research bulletin 20040730
Title: Hypoxia induces adenosine release from the rat carotid body.
Journal: Journal of neurochemistry 20040601
Title: Renal secretion of the antiviral nucleoside analog AM188 is inhibited by probenecid, p-aminohippuric acid, and cimetidine in the isolated perfused rat kidney.
Journal: Pharmaceutical research 20040601
Title: Mutation of leucine-92 selectively reduces the apparent affinity of inosine, guanosine, NBMPR [S6-(4-nitrobenzyl)-mercaptopurine riboside] and dilazep for the human equilibrative nucleoside transporter, hENT1.
Journal: The Biochemical journal 20040515
Title: Novel halogenated nitrobenzylthioinosine analogs as es nucleoside transporter inhibitors.
Journal: Bioorganic & medicinal chemistry letters 20040503
Title: Pharmacological analysis and molecular cloning of the canine equilibrative nucleoside transporter 1.
Journal: European journal of pharmacology 20040426
Title: Synthesis, biological activity and molecular modeling of 6-benzylthioinosine analogues as subversive substrates of Toxoplasma gondii adenosine kinase.
Journal: Journal of medicinal chemistry 20040408
Title: Interaction of the novel adenosine uptake inhibitor 3-[1-(6,7-diethoxy-2-morpholinoquinazolin-4-yl)piperidin-4-yl]-1,6-dimethyl-2,4(1H,3H)-quinazolinedione hydrochloride (KF24345) with the es and ei subtypes of equilibrative nucleoside transporters.
Journal: The Journal of pharmacology and experimental therapeutics 20040301
Title: Inhibition of glucose uptake in murine cardiomyocyte cell line HL-1 by cardioprotective drugs dilazep and dipyridamole.
Journal: American journal of physiology. Heart and circulatory physiology 20040201
Title: Adenosine transport in peripheral blood lymphocytes from Lesch-Nyhan patients.
Journal: The Biochemical journal 20040201
Title: Glycine 154 of the equilibrative nucleoside transporter, hENT1, is important for nucleoside transport and for conferring sensitivity to the inhibitors nitrobenzylthioinosine, dipyridamole, and dilazep.
Journal: Biochemical pharmacology 20040201
Title: Extracellular inosine is modulated by H2O2 and protects sertoli cells against lipoperoxidation and cellular injury.
Journal: Free radical research 20040101
Title: Mechanism of ganciclovir uptake by rabbit retina and human retinal pigmented epithelium cell line ARPE-19.
Journal: Current eye research 20040101
Title: Nitrobenzylthioinosine (NBMPR) binding and nucleoside transporter ENT1 mRNA expression after prolonged wakefulness and recovery sleep in the cortex and basal forebrain of rat.
Journal: Journal of sleep research 20031201
Title: Positive inotropic effect of the inhibition of cyclic GMP-stimulated 3',5'-cyclic nucleotide phosphodiesterase (PDE2) on guinea pig left atria in eu- and hyperthyroidism.
Journal: General physiology and biophysics 20031201
Title: Blood-brain barrier transport of synthetic adenosine A1 receptor agonists in vitro: structure transport relationships.
Journal: European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences 20031101
Title: Modulation of GABA release during morphine withdrawal in midbrain neurons in vitro.
Journal: Neuropharmacology 20031001
Title: Endogenous adenosine modulation of 22Na uptake by rat brain synaptosomes.
Journal: Neurochemical research 20031001
Title: Role of endogenous adenosine in the acute and late response to allergen challenge in actively sensitized Brown Norway rats.
Journal: British journal of pharmacology 20030701
Title: Functional differences in nucleoside and nucleobase transporters expressed on the rabbit corneal epithelial cell line (SIRC) and isolated rabbit cornea.
Journal: AAPS pharmSci 20030601
Title: Characterization of the transport of nucleoside analog drugs by the human multidrug resistance proteins MRP4 and MRP5.
Journal: Molecular pharmacology 20030501
Title: Control of glutamatergic neurotransmission in the rat spinal dorsal horn by the nucleoside transporter ENT1.
Journal: The Journal of physiology 20030415
Title: Molecular and biochemical events during differentiation of the HD3 chicken erythroblastic cell line.
Journal: The international journal of biochemistry & cell biology 20030401
Title: Inhibition of nucleoside transport by new analogues of nitrobenzylthioinosine.
Journal: Bioorganic & medicinal chemistry 20030320
Title: 5-Aminoimidazole-4-carboxamide riboside induces apoptosis in Jurkat cells, but the AMP-activated protein kinase is not involved.
Journal: The Biochemical journal 20030315
Title: Diurnal regulation of arylalkylamine N-acetyltransferase activity in chicken retinal cells in vitro: analysis of culture conditions.
Journal: Molecular vision 20030305
Title: Extracellular purines from cells of seminiferous tubules.
Journal: Molecular and cellular biochemistry 20030301
Title: Synthesis and flow cytometric evaluation of novel 1,2,3,4-tetrahydroisoquinoline conformationally constrained analogues of nitrobenzylmercaptopurine riboside (NBMPR) designed for probing its conformation when bound to the es nucleoside transporter.
Journal: Journal of medicinal chemistry 20030227
Title: Functional expression of a sodium dependent nucleoside transporter on rabbit cornea: Role in corneal permeation of acyclovir and idoxuridine.
Journal: Current eye research 20030101
Title: 2'-Deoxyadenosine causes apoptotic cell death in a human colon carcinoma cell line.
Journal: Journal of biochemical and molecular toxicology 20030101
Title: Quantitative autoradiography of adenosine receptors and NBTI-sensitive adenosine transporters in the brains and spinal cords of mice deficient in the mu-opioid receptor gene.
Journal: Brain research 20020705
Title: Complex effects of sulfhydryl reagents on ligand interactions with nucleoside transporters: evidence for multiple populations of ENT1 transporters with differential sensitivities to N-ethylmaleimide.
Journal: Archives of biochemistry and biophysics 20020701
Title: Sustained ER Ca2+ depletion suppresses protein synthesis and induces activation-enhanced cell death in mast cells.
Journal: The Journal of biological chemistry 20020419
Title: Inhibition of nitrobenzylthioinosine-sensitive adenosine transport by elevated D-glucose involves activation of P2Y2 purinoceptors in human umbilical vein endothelial cells.
Journal: Circulation research 20020322
Title: Inhibition of shiga toxin cytotoxicity in human renal cortical epithelial cells by nitrobenzylthioinosine.
Journal: The Journal of infectious diseases 20020315
Title: The kinetics of hypoxanthine transport across the perfused choroid plexus of the sheep.
Journal: Brain research 20020125
Title: Mutation of residue 33 of human equilibrative nucleoside transporters 1 and 2 alters sensitivity to inhibition of transport by dilazep and dipyridamole.
Journal: The Journal of biological chemistry 20020104
Title: Immunohistochemical variation of human equilibrative nucleoside transporter 1 protein in primary breast cancers.
Journal: Clinical cancer research : an official journal of the American Association for Cancer Research 20020101
Title: Nucleoside transport inhibitors, dipyridamole and p-nitrobenzylthioinosine, selectively potentiate the antitumor activity of NB1011.
Journal: Anti-cancer drugs 20020101
Title: Transport characteristics of HL-1 cells: a new model for the study of adenosine physiology in cardiomyocytes.
Journal: Biochemistry and cell biology = Biochimie et biologie cellulaire 20020101
Title: Regulation of K(+) current in human airway epithelial cells by exogenous and autocrine adenosine.
Journal: American journal of physiology. Cell physiology 20011201
Title: Extracellular formation and uptake of adenosine during skeletal muscle contraction in the rat: role of adenosine transporters.
Journal: The Journal of physiology 20011201
Title: Topology of a human equilibrative, nitrobenzylthioinosine (NBMPR)-sensitive nucleoside transporter (hENT1) implicated in the cellular uptake of adenosine and anti-cancer drugs.
Journal: The Journal of biological chemistry 20011130
Title: Nucleoside transporter subtype expression: effects on potency of adenosine kinase inhibitors.
Journal: British journal of pharmacology 20011101
Title: Transport characteristics of the anti-human immunodeficiency virus nucleoside analog, abacavir, into brain and cerebrospinal fluid.
Journal: The Journal of pharmacology and experimental therapeutics 20010901
Title: Cloned blood-brain barrier adenosine transporter is identical to the rat concentrative Na+ nucleoside cotransporter CNT2.
Journal: Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism 20010801
Title: Equilibrative nucleoside transporters: mapping regions of interaction for the substrate analogue nitrobenzylthioinosine (NBMPR) using rat chimeric proteins.
Journal: Biochemistry 20010710
Title: Characterization of an NBTI-sensitive equilibrative nucleoside transporter in vascular smooth muscle.
Journal: Journal of molecular and cellular cardiology 20010601
Title: Developmental regulation of the concentrative nucleoside transporters CNT1 and CNT2 in rat liver.
Journal: Journal of hepatology 20010601
Title: Long-term activation of adenosine A(2a) receptors blocks glutamate excitotoxicity in cultures of avian retinal neurons.
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Title: Characterization of nucleoside transport systems in cultured rat epididymal epithelium.
Journal: American journal of physiology. Cell physiology 20010501
Title: Ontogenic and longitudinal activity of Na(+)-nucleoside transporters in the human intestine.
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Title: Synthesis using ring closure metathesis and effect on nucleoside transport of a (N)-methanocarba S-(4-nitrobenzyl)thioinosine derivative.
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Journal: The Journal of biological chemistry 20010126
Title: Identification of Cys140 in helix 4 as an exofacial cysteine residue within the substrate-translocation channel of rat equilibrative nitrobenzylthioinosine (NBMPR)-insensitive nucleoside transporter rENT2.
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Title: Cloning of a novel isoform of the mouse NBMPR-sensitive equilibrative nucleoside transporter (ENT1) lacking a putative phosphorylation site.
Journal: Gene 20010110
Title: Nitrobenzylthioinosine (NBT), a nucleoside transport inhibitor, protects against Shiga toxin cytotoxicity in human microvascular endothelial cells.
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Title: Molecular cloning and functional characterization of inhibitor-sensitive (mENT1) and inhibitor-resistant (mENT2) equilibrative nucleoside transporters from mouse brain.
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